1IBL
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![BU of 1ibl by Molmil](/molmil-images/mine/1ibl) | STRUCTURE OF THE THERMUS THERMOPHILUS 30S RIBOSOMAL SUBUNIT IN COMPLEX WITH A MESSENGER RNA FRAGMENT AND COGNATE TRANSFER RNA ANTICODON STEM-LOOP BOUND AT THE A SITE AND WITH THE ANTIBIOTIC PAROMOMYCIN | 分子名称: | 16S RIBOSOMAL RNA, 30S RIBOSOMAL PROTEIN S10, 30S RIBOSOMAL PROTEIN S11, ... | 著者 | Ogle, J.M, Brodersen, D.E, Clemons Jr, W.M, Tarry, M.J, Carter, A.P, Ramakrishnan, V. | 登録日 | 2001-03-28 | 公開日 | 2001-05-04 | 最終更新日 | 2022-12-21 | 実験手法 | X-RAY DIFFRACTION (3.11 Å) | 主引用文献 | Recognition of cognate transfer RNA by the 30S ribosomal subunit. Science, 292, 2001
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2N7B
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![BU of 2n7b by Molmil](/molmil-images/mine/2n7b) | Solution structure of the human Siglec-8 lectin domain in complex with 6'sulfo sialyl Lewisx | 分子名称: | 3-aminopropan-1-ol, N-acetyl-alpha-neuraminic acid-(2-3)-6-O-sulfo-beta-D-galactopyranose-(1-4)-[alpha-L-fucopyranose-(1-3)]2-acetamido-2-deoxy-beta-D-glucopyranose, Sialic acid-binding Ig-like lectin 8 | 著者 | Proepster, J.M, Yang, F, Rabbani, S, Ernst, B, Allain, F.H.-T, Schubert, M. | 登録日 | 2015-09-07 | 公開日 | 2016-07-06 | 最終更新日 | 2020-07-29 | 実験手法 | SOLUTION NMR | 主引用文献 | Structural basis for sulfation-dependent self-glycan recognition by the human immune-inhibitory receptor Siglec-8. Proc.Natl.Acad.Sci.USA, 113, 2016
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1HJG
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![BU of 1hjg by Molmil](/molmil-images/mine/1hjg) | Alteration of the co-substrate selectivity of deacetoxycephalosporin C synthase: The role of arginine-258 | 分子名称: | 3-METHYL-2-OXOBUTANOIC ACID, DEACETOXYCEPHALOSPORIN C SYNTHASE, FE (II) ION | 著者 | Lee, H.J, Lloyd, M.D, Clifton, I.J, Harlos, K, Dubus, A, Baldwin, J.E, Frere, J.M, Schofield, C.J. | 登録日 | 2001-01-15 | 公開日 | 2001-06-01 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Alteration of the 2-Oxoacid Cosubstrate Selectivity in Deacetoxycephalosporin C Synthase: The Role of Arginine-258 J.Biol.Chem., 276, 2001
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1HJF
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![BU of 1hjf by Molmil](/molmil-images/mine/1hjf) | Alteration of the co-substrate selectivity of deacetoxycephalosporin C synthase: The role of arginine-258 | 分子名称: | 2-OXO-4-METHYLPENTANOIC ACID, DEACETOXYCEPHALOSPORIN C SYNTHASE, FE (II) ION | 著者 | Lee, H.J, Lloyd, M.D, Clifton, I.J, Harlos, K, Dubus, A, Baldwin, J.E, Frere, J.M, Schofield, C.J. | 登録日 | 2001-01-15 | 公開日 | 2001-06-01 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Alteration of the 2-Oxoacid Cosubstrate Selectivity in Deacetoxycephalosporin C Synthase: The Role of Arginine-258 J.Biol.Chem., 276, 2001
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6BN1
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![BU of 6bn1 by Molmil](/molmil-images/mine/6bn1) | Salvador Hippo SARAH domain complex | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, NICKEL (II) ION, Scaffold protein salvador, ... | 著者 | Cairns, L, Kavran, J.M. | 登録日 | 2017-11-15 | 公開日 | 2018-03-14 | 最終更新日 | 2018-04-25 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Salvador has an extended SARAH domain that mediates binding to Hippo kinase. J. Biol. Chem., 293, 2018
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6C79
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![BU of 6c79 by Molmil](/molmil-images/mine/6c79) | Conformational Changes in a Class A Beta lactamase that Prime it for Catalysis | 分子名称: | (6R,7R)-3-(acetyloxymethyl)-7-[[(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-methoxyimino-ethanoyl]amino]-8-oxo-5-thia-1-azabicy clo[4.2.0]oct-2-ene-2-carboxylic acid, Beta-lactamase Toho-1, SULFATE ION | 著者 | Coates, L, Langan, P.S, Vandavasi, V.G, Cooper, S.J, Weiss, K.L, Ginell, S.L, Parks, J.M. | 登録日 | 2018-01-22 | 公開日 | 2018-03-21 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (1.1 Å) | 主引用文献 | Substrate Binding Induces Conformational Changes in a Class A Beta-lactamase That Prime It for Catalysis Acs Catalysis, 8, 2018
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6C7Y
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![BU of 6c7y by Molmil](/molmil-images/mine/6c7y) | Crystal structure of inhibitory protein SOCS1 in complex with JAK1 kinase domain | 分子名称: | 1,2-ETHANEDIOL, ACETATE ION, ADENOSINE-5'-DIPHOSPHATE, ... | 著者 | Liau, N.P.D, Laktyushin, A, Lucet, I.S, Murphy, J.M, Yao, S, Callaghan, K, Nicola, N.A, Kershaw, N.J, Babon, J.J. | 登録日 | 2018-01-23 | 公開日 | 2018-05-02 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.499 Å) | 主引用文献 | The molecular basis of JAK/STAT inhibition by SOCS1. Nat Commun, 9, 2018
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6CC9
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![BU of 6cc9 by Molmil](/molmil-images/mine/6cc9) | NMR data-driven model of GTPase KRas-GMPPNP:Cmpd2 complex tethered to a nanodisc | 分子名称: | (2R,4S)-4-[(5-bromo-1H-indole-3-carbonyl)amino]-2-[(4-chlorophenyl)methyl]piperidin-1-ium, 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, Apolipoprotein A-I, ... | 著者 | Fang, Z, Marshall, C.B, Nishikawa, T, Gossert, A.D, Jansen, J.M, Jahnke, W, Ikura, M. | 登録日 | 2018-02-06 | 公開日 | 2018-09-05 | 最終更新日 | 2024-05-01 | 実験手法 | SOLUTION NMR | 主引用文献 | Inhibition of K-RAS4B by a Unique Mechanism of Action: Stabilizing Membrane-Dependent Occlusion of the Effector-Binding Site. Cell Chem Biol, 25, 2018
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6CNX
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![BU of 6cnx by Molmil](/molmil-images/mine/6cnx) | Crystal Structure of the Human vaccinia-related kinase 1 (VRK1) bound to an N-propynyl-N-isopentyl-dihydropteridin inhibitor | 分子名称: | (7R)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5H)-one, (7S)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5H)-one, ACETATE ION, ... | 著者 | Counago, R.M, dos Reis, C.V, de Souza, G.P, Azevedo, A, Guimaraes, C, Mascarello, A, Gama, F, Ferreira, M, Massirer, K.B, Arruda, P, Edwards, A.M, Elkins, J.M, Structural Genomics Consortium (SGC) | 登録日 | 2018-03-09 | 公開日 | 2018-04-04 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Crystal Structure of the Human Vaccinia-Related Kinase 1 (VRK1) bound to a N-propynyl-N-isopentil-dihydropteridine inhibitor To Be Published
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1KSI
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![BU of 1ksi by Molmil](/molmil-images/mine/1ksi) | CRYSTAL STRUCTURE OF A EUKARYOTIC (PEA SEEDLING) COPPER-CONTAINING AMINE OXIDASE AT 2.2A RESOLUTION | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, COPPER (II) ION, ... | 著者 | Wilce, M.C.J, Kumar, V, Freeman, H.C, Guss, J.M. | 登録日 | 1996-07-20 | 公開日 | 1997-12-24 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Crystal structure of a eukaryotic (pea seedling) copper-containing amine oxidase at 2.2 A resolution. Structure, 4, 1996
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6C7A
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![BU of 6c7a by Molmil](/molmil-images/mine/6c7a) | Conformational Changes in a Class A Beta lactamase that Prime it for Catalysis | 分子名称: | Beta-lactamase Toho-1, SULFATE ION | 著者 | Coates, L, Langan, P.S, Vandavasi, V.G, Cooper, S.J, Weiss, K.L, Ginell, S.L, Parks, J.M. | 登録日 | 2018-01-22 | 公開日 | 2018-03-21 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (1.05 Å) | 主引用文献 | Substrate Binding Induces Conformational Changes in a Class A Beta-lactamase That Prime It for Catalysis Acs Catalysis, 8, 2018
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6C78
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![BU of 6c78 by Molmil](/molmil-images/mine/6c78) | Substrate Binding Induces Conformational Changes In A Class A Beta Lactamase That Primes It For Catalysis | 分子名称: | Beta-lactamase Toho-1 | 著者 | Langan, P.S, Vandavasi, V.G, Cooper, S.J, Weiss, K.L, Ginell, S.L, Parks, J.M, Coates, L. | 登録日 | 2018-01-22 | 公開日 | 2018-03-21 | 最終更新日 | 2024-03-13 | 実験手法 | NEUTRON DIFFRACTION (1.75 Å) | 主引用文献 | Substrate Binding Induces Conformational Changes in a Class A Beta-lactamase That Prime It for Catalysis Acs Catalysis, 8, 2018
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1JU4
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![BU of 1ju4 by Molmil](/molmil-images/mine/1ju4) | BACTERIAL COCAINE ESTERASE COMPLEX WITH PRODUCT | 分子名称: | BENZOIC ACID, cocaine esterase | 著者 | Larsen, N.A, Turner, J.M, Stevens, J, Rosser, S.J, Basran, A, Lerner, R.A, Bruce, N.C, Wilson, I.A. | 登録日 | 2001-08-23 | 公開日 | 2001-12-21 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.63 Å) | 主引用文献 | Crystal structure of a bacterial cocaine esterase. Nat.Struct.Biol., 9, 2002
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1ICA
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6CY2
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![BU of 6cy2 by Molmil](/molmil-images/mine/6cy2) | RNA octamer containing 2'-OMe, 4'Calpha-OMe U. | 分子名称: | RNA (5'-R(*(CBV)P*GP*AP*AP*(UOA)P*UP*CP*G)-3') | 著者 | Harp, J.M, Egli, M. | 登録日 | 2018-04-04 | 公開日 | 2018-08-29 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | Structural basis for the synergy of 4'- and 2'-modifications on siRNA nuclease resistance, thermal stability and RNAi activity. Nucleic Acids Res., 46, 2018
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1I1J
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![BU of 1i1j by Molmil](/molmil-images/mine/1i1j) | STRUCTURE OF MELANOMA INHIBITORY ACTIVITY PROTEIN: A MEMBER OF A NEW FAMILY OF SECRETED PROTEINS | 分子名称: | MELANOMA DERIVED GROWTH REGULATORY PROTEIN | 著者 | Lougheed, J.C, Holton, J.M, Alber, T, Bazan, J.F, Handel, T.M. | 登録日 | 2001-02-02 | 公開日 | 2001-05-16 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.39 Å) | 主引用文献 | Structure of melanoma inhibitory activity protein, a member of a recently identified family of secreted proteins. Proc.Natl.Acad.Sci.USA, 98, 2001
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6CJN
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![BU of 6cjn by Molmil](/molmil-images/mine/6cjn) | Crystal Structure of Chalcone Isomerase from Medicago Sativa with the G95T mutation | 分子名称: | Chalcone--flavonone isomerase 1, SULFATE ION | 著者 | Burke, J.R, La Clair, J.J, Philippe, R.N, Pabis, A, Jez, J.M, Cortina, G, Kaltenbach, M, Bowman, M.E, Woods, K.B, Nelson, A.T, Tawfik, D.S, Kamerlin, S.C.L, Noel, J.P. | 登録日 | 2018-02-26 | 公開日 | 2019-03-13 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Bifunctional Substrate Activation via an Arginine Residue Drives Catalysis in Chalcone Isomerases Acs Catalysis, 2019
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1I86
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![BU of 1i86 by Molmil](/molmil-images/mine/1i86) | |
1I89
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![BU of 1i89 by Molmil](/molmil-images/mine/1i89) | Chalcone synthase (G256L) | 分子名称: | CHALCONE SYNTHASE 2 | 著者 | Jez, J.M, Bowman, M.E, Noel, J.P. | 登録日 | 2001-03-12 | 公開日 | 2001-12-12 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.86 Å) | 主引用文献 | Structure-guided programming of polyketide chain-length determination in chalcone synthase. Biochemistry, 40, 2001
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1I8B
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![BU of 1i8b by Molmil](/molmil-images/mine/1i8b) | Chalcone synthase (G256F) | 分子名称: | CHALCONE SYNTHASE 2 | 著者 | Jez, J.M, Bowman, M.E, Noel, J.P. | 登録日 | 2001-03-12 | 公開日 | 2001-12-12 | 最終更新日 | 2021-10-27 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Structure-guided programming of polyketide chain-length determination in chalcone synthase. Biochemistry, 40, 2001
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6BQL
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![BU of 6bql by Molmil](/molmil-images/mine/6bql) | Crystal Structure of the Human CAMKK2B in complex with TAE-226 | 分子名称: | 1,2-ETHANEDIOL, 2-({5-CHLORO-2-[(2-METHOXY-4-MORPHOLIN-4-YLPHENYL)AMINO]PYRIMIDIN-4-YL}AMINO)-N-METHYLBENZAMIDE, ACETATE ION, ... | 著者 | Counago, R.M, de Souza, G.P, dos Reis, C.V, Ramos, P.Z, Drewry, D, Massirer, K.B, Arruda, P, Edwards, A.M, Elkins, J.M, Structural Genomics Consortium (SGC) | 登録日 | 2017-11-28 | 公開日 | 2017-12-13 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Crystal Structure of the Human CAMKK2B in complex with TAE-226 To Be Published
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2N7A
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![BU of 2n7a by Molmil](/molmil-images/mine/2n7a) | Solution structure of the human Siglec-8 lectin domain | 分子名称: | Sialic acid-binding Ig-like lectin 8 | 著者 | Proepster, J.M, Yang, F, Rabbani, S, Ernst, B, Allain, F.H.-T, Schubert, M. | 登録日 | 2015-09-07 | 公開日 | 2016-07-06 | 最終更新日 | 2023-06-14 | 実験手法 | SOLUTION NMR | 主引用文献 | Structural basis for sulfation-dependent self-glycan recognition by the human immune-inhibitory receptor Siglec-8. Proc.Natl.Acad.Sci.USA, 113, 2016
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1KUF
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![BU of 1kuf by Molmil](/molmil-images/mine/1kuf) | High-resolution Crystal Structure of a Snake Venom Metalloproteinase from Taiwan Habu | 分子名称: | CADMIUM ION, metalloproteinase | 著者 | Huang, K.F, Chiou, S.H, Ko, T.P, Yuann, J.M, Wang, A.H.J. | 登録日 | 2002-01-21 | 公開日 | 2002-07-03 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.35 Å) | 主引用文献 | The 1.35 A structure of cadmium-substituted TM-3, a snake-venom metalloproteinase from Taiwan habu: elucidation of a TNFalpha-converting enzyme-like active-site structure with a distorted octahedral geometry of cadmium. Acta Crystallogr.,Sect.D, 58, 2002
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6CI1
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6CFM
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![BU of 6cfm by Molmil](/molmil-images/mine/6cfm) | Crystal Structure of the Human vaccinia-related kinase bound to a propynyl-pteridinone inhibitor | 分子名称: | (7R)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7,8-dimethyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5H)-one, CHLORIDE ION, GLYCEROL, ... | 著者 | Counago, R.M, dos Reis, C.V, de Souza, G.P, Azevedo, A, Guimaraes, C, Mascarello, A, Gama, F, Ferreira, M, Massirer, K.B, Arruda, P, Edwards, A.M, Elkins, J.M, Structural Genomics Consortium (SGC) | 登録日 | 2018-02-15 | 公開日 | 2018-03-07 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.45 Å) | 主引用文献 | Crystal Structure of the Human vaccinia-related kinase bound to a propynyl-pteridinone inhibitor To Be Published
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