7Y4G
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![BU of 7y4g by Molmil](/molmil-images/mine/7y4g) | sit-bound btDPP4 | 分子名称: | (2R)-4-OXO-4-[3-(TRIFLUOROMETHYL)-5,6-DIHYDRO[1,2,4]TRIAZOLO[4,3-A]PYRAZIN-7(8H)-YL]-1-(2,4,5-TRIFLUOROPHENYL)BUTAN-2-A MINE, btDPP4 | 著者 | Hang, J, Jiang, C, Wang, K, Zhang, Z, Guo, F, Liu, J, Wang, G, Lei, X, Gonzalez, F, Qiao, J. | 登録日 | 2022-06-14 | 公開日 | 2023-06-14 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.97 Å) | 主引用文献 | Microbial-host-isozyme analyses reveal microbial DPP4 as a potential antidiabetic target. Science, 381, 2023
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5BTX
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![BU of 5btx by Molmil](/molmil-images/mine/5btx) | Structure of the N-terminal domain of lpg1496 from Legionella pneumophila in complex with nucleotide | 分子名称: | ADENOSINE-3',5'-CYCLIC-MONOPHOSPHATE, lpg1496 | 著者 | Wong, K, Kozlov, G, Gehring, K, Montreal-Kingston Bacterial Structural Genomics Initiative (BSGI) | 登録日 | 2015-06-03 | 公開日 | 2015-08-26 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structure of the Legionella Effector, lpg1496, Suggests a Role in Nucleotide Metabolism. J.Biol.Chem., 290, 2015
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6A04
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![BU of 6a04 by Molmil](/molmil-images/mine/6a04) | Structure of pSTING complex | 分子名称: | 9,9'-[(2R,3R,3aS,5S,7aR,9R,10R,10aS,12S,14aR)-3,5,10,12-tetrahydroxy-5,12-dioxidooctahydro-2H,7H-difuro[3,2-d:3',2'-j][1,3,7,9,2,8]tetraoxadiphosphacyclododecine-2,9-diyl]bis(2-amino-1,9-dihydro-6H-purin-6-one), SULFATE ION, Stimulator of interferon genes protein | 著者 | Yuan, Z.L, Shang, G.J, Cong, X.Y, Gu, L.C. | 登録日 | 2018-06-05 | 公開日 | 2019-06-19 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Crystal structures of porcine STINGCBD-CDN complexes reveal the mechanism of ligand recognition and discrimination of STING proteins. J.Biol.Chem., 294, 2019
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5BU0
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![BU of 5bu0 by Molmil](/molmil-images/mine/5bu0) | Structure of the C-terminal domain of lpg1496 from Legionella pneumophila | 分子名称: | lpg1496 | 著者 | Wong, K, Kozlov, G, Gehring, K, Montreal-Kingston Bacterial Structural Genomics Initiative (BSGI) | 登録日 | 2015-06-03 | 公開日 | 2015-08-26 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (2.35 Å) | 主引用文献 | Structure of the Legionella Effector, lpg1496, Suggests a Role in Nucleotide Metabolism. J.Biol.Chem., 290, 2015
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3ED0
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![BU of 3ed0 by Molmil](/molmil-images/mine/3ed0) | Crystal structure of (3R)-Hydroxyacyl-Acyl Carrier Protein Dehydratase (FabZ) from Helicobacter pylori in complex with emodin | 分子名称: | (3R)-hydroxymyristoyl-acyl carrier protein dehydratase, 3-METHYL-1,6,8-TRIHYDROXYANTHRAQUINONE, BENZAMIDINE, ... | 著者 | Zhang, L, Zhang, H, Liu, W, Guo, Y, Shen, X, Jiang, H. | 登録日 | 2008-09-02 | 公開日 | 2009-07-21 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Emodin targets the beta-hydroxyacyl-acyl carrier protein dehydratase from Helicobacter pylori: enzymatic inhibition assay with crystal structural and thermodynamic characterization BMC MICROBIOL., 9, 2009
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4FFC
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![BU of 4ffc by Molmil](/molmil-images/mine/4ffc) | |
5BTZ
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![BU of 5btz by Molmil](/molmil-images/mine/5btz) | Structure of the middle domain of lpg1496 from Legionella pneumophila in P212121 space group | 分子名称: | lpg1496 | 著者 | Wong, K, Kozlov, G, Gehring, K, Montreal-Kingston Bacterial Structural Genomics Initiative (BSGI) | 登録日 | 2015-06-03 | 公開日 | 2015-08-26 | 最終更新日 | 2020-01-08 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Structure of the Legionella Effector, lpg1496, Suggests a Role in Nucleotide Metabolism. J.Biol.Chem., 290, 2015
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4ZPV
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![BU of 4zpv by Molmil](/molmil-images/mine/4zpv) | Structure of MERS-Coronavirus Spike Receptor-binding Domain (England1 Strain) in Complex with Vaccine-Elicited Murine Neutralizing Antibody D12 (Crystal Form 2) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, D12 Fab Heavy chain, D12 Fab light chain, ... | 著者 | Joyce, M.G, Mascola, J.R, Graham, B.S, Kwong, P.D. | 登録日 | 2015-05-08 | 公開日 | 2015-10-21 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | Evaluation of candidate vaccine approaches for MERS-CoV. Nat Commun, 6, 2015
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1AX8
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![BU of 1ax8 by Molmil](/molmil-images/mine/1ax8) | Human obesity protein, leptin | 分子名称: | OBESITY PROTEIN | 著者 | Zhang, F, Beals, J.M, Briggs, S.L, Clawson, D.K, Wery, J.-P, Schevitz, R.W. | 登録日 | 1997-10-31 | 公開日 | 1998-11-25 | 最終更新日 | 2012-05-09 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Crystal structure of the obese protein leptin-E100. Nature, 387, 1997
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7CVA
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![BU of 7cva by Molmil](/molmil-images/mine/7cva) | RNA methyltransferase METTL4 | 分子名称: | Methyltransferase-like protein 2 | 著者 | Luo, Q, Ma, J. | 登録日 | 2020-08-25 | 公開日 | 2021-09-01 | 最終更新日 | 2022-10-12 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Structural insights into molecular mechanism for N6-adenosine methylation by MT-A70 family methyltransferase METTL4 Nat Commun, 13, 2022
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7CV9
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![BU of 7cv9 by Molmil](/molmil-images/mine/7cv9) | RNA methyltransferase METTL4 | 分子名称: | GLYCEROL, Methyltransferase-like protein 2, S-ADENOSYL-L-HOMOCYSTEINE | 著者 | Luo, Q, Ma, J. | 登録日 | 2020-08-25 | 公開日 | 2021-09-01 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (2.455 Å) | 主引用文献 | Structural insights into molecular mechanism for N6-adenosine methylation by MT-A70 family methyltransferase METTL4 Nat Commun, 13, 2022
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7CV6
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![BU of 7cv6 by Molmil](/molmil-images/mine/7cv6) | RNA methyltransferase METTL4 | 分子名称: | 2'-O-methyladenosine 5'-(dihydrogen phosphate), Methyltransferase-like protein 2, S-ADENOSYL-L-HOMOCYSTEINE | 著者 | Luo, Q, Ma, J. | 登録日 | 2020-08-25 | 公開日 | 2021-09-01 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (3.01 Å) | 主引用文献 | Structural insights into molecular mechanism for N6-adenosine methylation by MT-A70 family methyltransferase METTL4 Nat Commun, 13, 2022
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7CV7
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![BU of 7cv7 by Molmil](/molmil-images/mine/7cv7) | RNA methyltransferase METTL4 | 分子名称: | Methyltransferase-like protein 2, S-ADENOSYLMETHIONINE | 著者 | Luo, Q, Ma, J. | 登録日 | 2020-08-25 | 公開日 | 2021-09-01 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structural insights into molecular mechanism for N6-adenosine methylation by MT-A70 family methyltransferase METTL4 Nat Commun, 13, 2022
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7CV8
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![BU of 7cv8 by Molmil](/molmil-images/mine/7cv8) | RNA methyltransferase METTL4 | 分子名称: | GLYCEROL, Methyltransferase-like protein 2, SINEFUNGIN | 著者 | Luo, Q, Ma, J. | 登録日 | 2020-08-25 | 公開日 | 2021-09-01 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (2.37 Å) | 主引用文献 | Structural insights into molecular mechanism for N6-adenosine methylation by MT-A70 family methyltransferase METTL4 Nat Commun, 13, 2022
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5UQW
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![BU of 5uqw by Molmil](/molmil-images/mine/5uqw) | Crystal structure of human KRAS G12V mutant in complex with GDP | 分子名称: | GTPase KRas, GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION | 著者 | Huang, C.S, Kaplan, A, Stockwell, B.R, Tong, L. | 登録日 | 2017-02-08 | 公開日 | 2017-03-22 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Multivalent Small-Molecule Pan-RAS Inhibitors. Cell, 168, 2017
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3GVG
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![BU of 3gvg by Molmil](/molmil-images/mine/3gvg) | |
3GWC
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![BU of 3gwc by Molmil](/molmil-images/mine/3gwc) | |
4ZPW
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![BU of 4zpw by Molmil](/molmil-images/mine/4zpw) | Structure of unbound MERS-CoV spike receptor-binding domain (England1 strain). | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, PHOSPHATE ION, Spike glycoprotein | 著者 | Joyce, M.G, Mascola, J.R, Graham, B.S, Kwong, P.D. | 登録日 | 2015-05-08 | 公開日 | 2015-08-12 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (3.023 Å) | 主引用文献 | Evaluation of candidate vaccine approaches for MERS-CoV. Nat Commun, 6, 2015
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5E29
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![BU of 5e29 by Molmil](/molmil-images/mine/5e29) | Crystal Structure of Deoxygenated Hemoglobin in Complex with an Allosteric Effector and Nitric Oxide | 分子名称: | 2-(nitrooxy)ethyl 2-(4-{2-[(3,5-dimethylphenyl)amino]-2-oxoethyl}phenoxy)-2-methylpropanoate, 2-{4-[(3,5-DIMETHYLANILINO)-CARBONYL-METHYL]-PHENOXY}-2-METHYLPROPIONIC ACID, CACODYLATE ION, ... | 著者 | Safo, M.K, Deshpande, T.M. | 登録日 | 2015-09-30 | 公開日 | 2015-10-14 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Design, Synthesis, and Investigation of Novel Nitric Oxide (NO)-Releasing Prodrugs as Drug Candidates for the Treatment of Ischemic Disorders: Insights into NO-Releasing Prodrug Biotransformation and Hemoglobin-NO Biochemistry. Biochemistry, 54, 2015
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4F47
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![BU of 4f47 by Molmil](/molmil-images/mine/4f47) | |
5TDR
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![BU of 5tdr by Molmil](/molmil-images/mine/5tdr) | Set3 PHD finger in complex with histone H3K4me2 | 分子名称: | Histone H3, SET domain-containing protein 3, SODIUM ION, ... | 著者 | Andrews, F.H, Ali, M, Kutateladze, T.G. | 登録日 | 2016-09-19 | 公開日 | 2016-11-02 | 最終更新日 | 2017-06-28 | 実験手法 | X-RAY DIFFRACTION (1.42 Å) | 主引用文献 | Structural Insight into Recognition of Methylated Histone H3K4 by Set3. J. Mol. Biol., 429, 2017
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5DJN
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![BU of 5djn by Molmil](/molmil-images/mine/5djn) | |
3H81
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![BU of 3h81 by Molmil](/molmil-images/mine/3h81) | |
2L0K
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![BU of 2l0k by Molmil](/molmil-images/mine/2l0k) | NMR solution structure of a transcription factor SpoIIID in complex with DNA | 分子名称: | Stage III sporulation protein D | 著者 | Chen, B, Himes, P, Lu, Z, Liu, A, Yan, H, Kroos, L. | 登録日 | 2010-07-08 | 公開日 | 2011-08-17 | 最終更新日 | 2024-05-01 | 実験手法 | SOLUTION NMR | 主引用文献 | Novel Mode of DNA Binding by Bacterial Transcription Factor SpoIIID To be Published
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4FF5
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![BU of 4ff5 by Molmil](/molmil-images/mine/4ff5) | |