9C1W
Structure of AKT2 with compound 3
Summary for 9C1W
Entry DOI | 10.2210/pdb9c1w/pdb |
Related | 8UVY 8UW2 8UW7 8UW9 |
Descriptor | RAC-beta serine/threonine-protein kinase, 4-{2-[({4-[(2P)-2-(2-aminopyridin-3-yl)-5-phenyl-3H-imidazo[4,5-b]pyridin-3-yl]phenyl}methyl)amino]ethyl}-2-hydroxybenzaldehyde, 1,2-ETHANEDIOL, ... (4 entities in total) |
Functional Keywords | inhibitor, kinase, transferase, transferase-inhibitor complex, transferase/inhibitor |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 1 |
Total formula weight | 52662.13 |
Authors | |
Primary citation | Craven, G.B.,Ma, X.,Taunton, J. Mutant-selective AKT1 inhibitors via lysine targeting and neo-zinc chelation To Be Published, |
Experimental method | X-RAY DIFFRACTION (2 Å) |
Structure validation
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