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6PDP

Human PIM1 bound to benzothiophene inhibitor 379

Summary for 6PDP
Entry DOI10.2210/pdb6pdp/pdb
Related6PCW 6PDI 6PDN 6PDO
DescriptorSerine/threonine-protein kinase pim-1, Peptide, SULFATE ION, ... (5 entities in total)
Functional Keywordsproto-oncogene serine/threonine-protein kinase pim-1, structural genomics, structural genomics consortium, sgc, transferase, transferase-transferase inhibitor complex, transferase/transferase inhibitor
Biological sourceHomo sapiens (Human)
More
Total number of polymer chains2
Total formula weight37635.88
Authors
Primary citationGodoi, P.H.C.,Santiago, A.S.,Fala, A.M.,Ramos, P.Z.,Sriranganadane, D.,Mascarello, A.,Segretti, N.,Azevedo, H.,Guimaraes, C.R.W.,Arruda, P.,Elkins, J.M.,Counago, R.M.
Human PIM1
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.5 Å)
Structure validation

218500

数据于2024-04-17公开中

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