6PDP
Human PIM1 bound to benzothiophene inhibitor 379
Summary for 6PDP
Entry DOI | 10.2210/pdb6pdp/pdb |
Related | 6PCW 6PDI 6PDN 6PDO |
Descriptor | Serine/threonine-protein kinase pim-1, Peptide, SULFATE ION, ... (5 entities in total) |
Functional Keywords | proto-oncogene serine/threonine-protein kinase pim-1, structural genomics, structural genomics consortium, sgc, transferase, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Homo sapiens (Human) More |
Total number of polymer chains | 2 |
Total formula weight | 37635.88 |
Authors | Godoi, P.H.C.,Sriranganadane, D.,Santiago, A.S.,Fala, A.M.,Ramos, P.Z.,Mascarello, A.,Segretti, N.,Azevedo, H.,Guimaraes, C.R.W.,Arruda, P.,Elkins, J.M.,Counago, R.M.,Structural Genomics Consortium (SGC) (deposition date: 2019-06-19, release date: 2019-07-24, Last modification date: 2024-03-13) |
Primary citation | Godoi, P.H.C.,Santiago, A.S.,Fala, A.M.,Ramos, P.Z.,Sriranganadane, D.,Mascarello, A.,Segretti, N.,Azevedo, H.,Guimaraes, C.R.W.,Arruda, P.,Elkins, J.M.,Counago, R.M. Human PIM1 To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.5 Å) |
Structure validation
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