6PCW

Human PIM1 bound to benzothiophene inhibitor 213

Summary for 6PCW

• Entry DOI: 10.2210/pdb6pcw/pdb
• Descriptor: Serine/threonine-protein kinase pim-1, Peptide, 4-[5-(cyclopropylcarbamoyl)thiophen-2-yl]-1-benzothiophene-2-carboxamide, ... (5 entities in total)
• Functional Keywords: proto-oncogene serine/threonine-protein kinase pim-1, structural genomics, structural genomics consortium, sgc, transferase, transferase-transferase inhibitor complex, transferase/transferase inhibitor
• Biological source: Homo sapiens (Human); More
• Total number of polymer chains: 2
• Total formula weight: 37709.97

Authors

Godoi, P.H.C.,Santiago, A.S.,Fala, A.M.,Ramos, P.Z.,Sriranganadane, D.,Mascarello, A.,Segretti, N.,Azevedo, H.,Guimaraes, C.R.W.,Arruda, P.,Elkins, J.M.,Counago, R.M.,Structural Genomics Consortium (SGC) (deposition date: 2019-06-18, release date: 2019-07-24, Last modification date: 2023-10-11)

• Primary citation: Godoi, P.H.C.,Santiago, A.S.,Fala, A.M.,Ramos, P.Z.,Sriranganadane, D.,Mascarello, A.,Segretti, N.,Azevedo, H.,Guimaraes, C.R.W.,Arruda, P.,Elkins, J.M.,Counago, R.M.; PIM1 bound to benzothiophene inhibitor; To Be Published,

Experimental method

X-RAY DIFFRACTION (2.2 Å)