6PDN

Human PIM1 bound to benzothiophene inhibitor 292

Summary for 6PDN

• Entry DOI: 10.2210/pdb6pdn/pdb
• Related: 6PCW 6PDI
• Descriptor: Serine/threonine-protein kinase pim-1, peptide, 4-{5-[(3-aminopropyl)carbamoyl]thiophen-2-yl}-1-benzothiophene-2-carboxylic acid, ... (5 entities in total)
• Functional Keywords: proto-oncogene serine/threonine-protein kinase pim-1, structural genomics, structural genomics consortium, sgc, transferase, transferase-transferase inhibitor complex, transferase/transferase inhibitor
• Biological source: Homo sapiens (Human); More
• Total number of polymer chains: 2
• Total formula weight: 37715.87

Authors

Godoi, P.H.C.,Santiago, A.S.,Fala, A.M.,Ramos, P.Z.,Sriranganadane, D.,Mascarello, A.,Segretti, N.,Azevedo, H.,Guimaraes, C.R.W.,Arruda, P.,Elkins, J.M.,Counago, R.M.,Structural Genomics Consortium (SGC) (deposition date: 2019-06-19, release date: 2019-07-24, Last modification date: 2024-10-23)

• Primary citation: Godoi, P.H.C.,Santiago, A.S.,Fala, A.M.,Ramos, P.Z.,Sriranganadane, D.,Mascarello, A.,Segretti, N.,Azevedo, H.,Guimaraes, C.R.W.,Arruda, P.,Elkins, J.M.,Counago, R.M.; Human PIM1; To Be Published,

Experimental method

X-RAY DIFFRACTION (2.4 Å)