5VQK

X-ray co-structure of nuclear receptor ROR-gammat Ligand Binding Domain with a inverse agonist and SRC2 peptide

Summary for 5VQK

• Entry DOI: 10.2210/pdb5vqk/pdb
• Related: 5VB3 5VB5 5VB6 5VB7 5VQL
• Descriptor: Nuclear receptor ROR-gamma, SRC2 chimera, 1-(4-fluorophenyl)-7-methoxy-N-{[4-(methylsulfamoyl)phenyl]methyl}-1H-pyrazolo[3,4-c]pyridine-4-carboxamide (3 entities in total)
• Functional Keywords: nuclear receptor, nuclear hormone receptor, transcription
• Biological source: Homo sapiens (Human); More
• Total number of polymer chains: 1
• Total formula weight: 32911.93

Authors

Li, X. (deposition date: 2017-05-09, release date: 2018-05-16, Last modification date: 2024-03-13)

• Primary citation: Li, X.; X-ray co-structure of nuclear receptor ROR-gammat Ligand Binding Domain with a inverse agonist and SRC2 peptide; To Be Published,

Experimental method

X-RAY DIFFRACTION (3.1 Å)