5VQL

X-ray co-structure of nuclear receptor ROR-gammat Ligand Binding Domain with a inverse agonist and SRC2 peptide

Summary for 5VQL

• Entry DOI: 10.2210/pdb5vql/pdb
• Related: 5VB3 5VB5 5VB6 5VB7 5VQK
• Descriptor: Nuclear receptor ROR-gamma, SRC2 chimera, SODIUM ION, 5'-(4-cyclopropyl-6-methoxypyrimidin-5-yl)-N-{[4-(ethylsulfonyl)phenyl]methyl}spiro[cyclopentane-1,3'-pyrrolo[3,2-b]pyridine]-1'(2'H)-carboxamide, ... (4 entities in total)
• Functional Keywords: nuclear receptor, nuclear hormone receptor, transcription
• Biological source: Homo sapiens (Human); More
• Total number of polymer chains: 1
• Total formula weight: 33013.09

Authors

Li, X. (deposition date: 2017-05-09, release date: 2018-05-16, Last modification date: 2024-03-13)

• Primary citation: Li, X.; X-ray co-structure of nuclear receptor ROR-gammat Ligand Binding Domain with a inverse agonist and SRC2 peptide; To Be Published,

Experimental method

X-RAY DIFFRACTION (2.7 Å)