4DM6
Crystal structure of RARb LBD homodimer in complex with TTNPB
Summary for 4DM6
Entry DOI | 10.2210/pdb4dm6/pdb |
Related | 1XAP 4DM8 4DMA |
Descriptor | Retinoic acid receptor beta, Nuclear receptor coactivator 1, 4-[(1E)-2-(5,5,8,8-TETRAMETHYL-5,6,7,8-TETRAHYDRONAPHTHALEN-2-YL)PROP-1-ENYL]BENZOIC ACID, ... (4 entities in total) |
Functional Keywords | transcription, nuclear receptor, retinoic acid, alpha helical sandwich, transcription regulator, retinoic acid binding, nucleus - cytoplasm, transcription-protein binding complex, transcription/protein binding |
Biological source | Homo sapiens (human) More |
Cellular location | Isoform Beta-1: Nucleus. Isoform Beta-2: Nucleus. Isoform Beta-4: Cytoplasm: P10826 Nucleus (By similarity): Q15788 |
Total number of polymer chains | 4 |
Total formula weight | 66667.20 |
Authors | Osz, J.,Brelivet, Y.,Peluso-Iltis, C.,Cura, V.,Eiler, S.,Ruff, M.,Bourguet, W.,Rochel, N.,Moras, D. (deposition date: 2012-02-07, release date: 2012-03-07, Last modification date: 2024-02-28) |
Primary citation | Osz, J.,Brelivet, Y.,Peluso-Iltis, C.,Cura, V.,Eiler, S.,Ruff, M.,Bourguet, W.,Rochel, N.,Moras, D. Structural basis for a molecular allosteric control mechanism of cofactor binding to nuclear receptors. Proc.Natl.Acad.Sci.USA, 109:E588-E594, 2012 Cited by PubMed: 22355136DOI: 10.1073/pnas.1118192109 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.9 Å) |
Structure validation
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