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4DM6

Crystal structure of RARb LBD homodimer in complex with TTNPB

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
A0048384biological_processretinoic acid receptor signaling pathway
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0005634cellular_componentnucleus
B0006355biological_processregulation of DNA-templated transcription
B0048384biological_processretinoic acid receptor signaling pathway
Functional Information from PDB Data
site_idAC1
Number of Residues14
DetailsBINDING SITE FOR RESIDUE TTB A 501
ChainResidue
APHE201
ASER289
AGLY393
AVAL397
ALEU416
AHOH617
APHE230
ALEU233
AALA234
ALEU271
AILE272
AILE275
AARG278
APHE288

site_idAC2
Number of Residues18
DetailsBINDING SITE FOR RESIDUE TTB B 1501
ChainResidue
BPHE1201
BPHE1230
BLEU1233
BALA1234
BCYS1237
BLEU1271
BILE1272
BILE1275
BARG1278
BPHE1288
BSER1289
BGLY1303
BPHE1304
BGLY1393
BVAL1397
BLEU1400
BILE1412
BHOH1628

site_idAC3
Number of Residues12
DetailsBINDING SITE FOR CHAIN E OF NUCLEAR RECEPTOR COACTIVATOR 1
ChainResidue
ALYS246
AGLN259
AILE260
ALYS264
APRO410
ALEU411
AGLU414
AMET415
AGLU417
AHOH650
BMET1182
BGLU1185

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues8
DetailsMotif: {"description":"LXXLL motif 4"}
ChainResidueDetails

246031

PDB entries from 2025-12-10

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