3RNN
Crystal Structure of iGluR2 Ligand Binding Domain with Symmetric Sulfonamide Containing Potentiator
Summary for 3RNN
Entry DOI | 10.2210/pdb3rnn/pdb |
Related | 1FTJ 1FTK 1FTL 1LB9 1LBC 3RN8 |
Descriptor | Glutamate receptor 2, N,N'-(benzene-1,4-diyldiethane-2,1-diyl)dipropane-2-sulfonamide, GLUTAMIC ACID, ... (5 entities in total) |
Functional Keywords | iglur2 ligand binding domain, membrane, transport protein |
Biological source | Homo sapiens (human) More |
Total number of polymer chains | 3 |
Total formula weight | 97628.46 |
Authors | Timm, D.E. (deposition date: 2011-04-22, release date: 2011-05-25, Last modification date: 2019-07-17) |
Primary citation | Timm, D.E.,Benveniste, M.,Weeks, A.M.,Nisenbaum, E.S.,Partin, K.M. Structural and functional analysis of two new positive allosteric modulators of GluA2 desensitization and deactivation. Mol.Pharmacol., 80:267-280, 2011 Cited by PubMed: 21543522DOI: 10.1124/mol.110.070243 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.75 Å) |
Structure validation
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