3RNN
Crystal Structure of iGluR2 Ligand Binding Domain with Symmetric Sulfonamide Containing Potentiator
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A, B, C | Glutamate receptor 2 | polymer | 292 | 32035.7 | 3 | UniProt (P42262) Pfam (PF10613) Pfam (PF00060) In PDB | Homo sapiens (human) | GluR-2, AMPA-selective glutamate receptor 2, GluR-B, GluR-K2, Glutamate receptor ionotropic, AMPA 2, GluA2 |
2 | A, B | N,N'-(benzene-1,4-diyldiethane-2,1-diyl)dipropane-2-sulfonamide | non-polymer | 376.5 | 2 | Chemie (RNN) | |||
3 | A, B, C | GLUTAMIC ACID | non-polymer | 147.1 | 3 | Chemie (GLU) | |||
4 | A, B, C | ZINC ION | non-polymer | 65.4 | 5 | Chemie (ZN) | |||
5 | water | water | 18.0 | 835 | Chemie (HOH) |
Sequence modifications
A, B, C: 3 - 117 (UniProt: P42262)
A, B, C: 120 - 279 (UniProt: P42262)
PDB | External Database | Details |
---|---|---|
Arg -12 | - | EXPRESSION TAG |
Gly -11 | - | EXPRESSION TAG |
Ser -10 | - | EXPRESSION TAG |
Ala -9 | - | EXPRESSION TAG |
Met -8 | - | EXPRESSION TAG |
Gly -7 | - | EXPRESSION TAG |
Ser -6 | - | EXPRESSION TAG |
Gly -5 | - | EXPRESSION TAG |
Asn -4 | - | EXPRESSION TAG |
Asp -3 | - | EXPRESSION TAG |
Thr -2 | - | EXPRESSION TAG |
Ser -1 | - | EXPRESSION TAG |
Arg 0 | - | EXPRESSION TAG |
Gly 1 | - | EXPRESSION TAG |
Ala 2 | - | EXPRESSION TAG |
PDB | External Database | Details |
---|---|---|
Gly 118 | - | LINKER |
Thr 119 | - | LINKER |
Gly 231 | Arg 764 | SEE REMARK 999 |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 3 |
Total formula weight | 96107.0 | |
Non-Polymers* | Number of molecules | 10 |
Total formula weight | 1521.5 | |
All* | Total formula weight | 97628.5 |