3FSK
P38 kinase crystal structure in complex with RO6257
Summary for 3FSK
Entry DOI | 10.2210/pdb3fsk/pdb |
Related | 3FLN 3FLS 3FLW 3FLY 3FLZ 3FMH 3FMJ 3FMK 3FML 3FMM 3FMN |
Descriptor | Mitogen-activated protein kinase 14, 3-(2-chlorophenyl)-7-[(trans-4-hydroxycyclohexyl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one (3 entities in total) |
Functional Keywords | p38; map kinase; serine/threonine kinase, alternative splicing, atp-binding, cytoplasm, kinase, nucleotide-binding, nucleus, phosphoprotein, polymorphism, serine/threonine-protein kinase, transferase, signaling protein |
Biological source | Homo sapiens (human) |
Cellular location | Cytoplasm (By similarity): Q16539 |
Total number of polymer chains | 1 |
Total formula weight | 43122.55 |
Authors | Kuglstatter, A.,Bertrand, J.,Takahara, P.,Villasenor, A. (deposition date: 2009-01-09, release date: 2009-12-22, Last modification date: 2023-09-06) |
Primary citation | Arora, N.,Williams, C.,Delano, W.,Will, D.,Kuglstatter, A. Mapping Binding Pocket Volume: Potential Applications towards Ligand Design and Selectivity To be Published, |
Experimental method | X-RAY DIFFRACTION (2 Å) |
Structure validation
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