3FMN
P38 kinase crystal structure in complex with RO2530
Summary for 3FMN
Entry DOI | 10.2210/pdb3fmn/pdb |
Related | 3FLN 3FLS 3FLW 3FLY 3FLZ 3FMH 3FMJ 3FMK 3FML 3FMM |
Descriptor | Mitogen-activated protein kinase 14, 6-(2,4-difluorophenoxy)-N-(tetrahydro-2H-pyran-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-3-amine (3 entities in total) |
Functional Keywords | p38; map kinase; serine/threonine kinase, atp-binding, kinase, nucleotide-binding, nucleus, phosphoprotein, serine/threonine-protein kinase, transferase, signaling protein |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 1 |
Total formula weight | 43096.03 |
Authors | Kuglstatter, A.,Ghate, M. (deposition date: 2008-12-22, release date: 2009-12-22, Last modification date: 2023-09-06) |
Primary citation | Soth, M.,Kuglstatter, A.,Gabriel, T. P38 kinase crystal structure in complex with RO2530 To be Published, |
Experimental method | X-RAY DIFFRACTION (1.9 Å) |
Structure validation
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