3ADX
Human PPARgamma ligand-binding domain in complex with indomethacin and nitro-233
Summary for 3ADX
Entry DOI | 10.2210/pdb3adx/pdb |
Related | 3ADS 3ADT 3ADU 3ADV 3ADW |
Descriptor | Peroxisome proliferator-activated receptor gamma, 3-[5-(2-nitropent-1-en-1-yl)furan-2-yl]benzoic acid, INDOMETHACIN, ... (4 entities in total) |
Functional Keywords | nuclear receptor, ligand-dependent transcription factor, ligand-binding domain, activator, diabetes mellitus, disease mutation, dna-binding, metal-binding, nucleus, obesity, phosphoprotein, receptor, transcription, transcription regulation, zinc-finger |
Biological source | Homo sapiens (human) |
Cellular location | Nucleus: P37231 |
Total number of polymer chains | 2 |
Total formula weight | 66404.52 |
Authors | Waku, T.,Shiraki, T.,Oyama, T.,Morikawa, K. (deposition date: 2010-01-29, release date: 2010-12-22, Last modification date: 2023-11-01) |
Primary citation | Waku, T.,Shiraki, T.,Oyama, T.,Maebara, K.,Nakamori, R.,Morikawa, K. The nuclear receptor PPARgamma individually responds to serotonin- and fatty acid-metabolites Embo J., 29:3395-3407, 2010 Cited by PubMed: 20717101DOI: 10.1038/emboj.2010.197 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.95 Å) |
Structure validation
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