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3FSK

P38 kinase crystal structure in complex with RO6257

Summary for 3FSK
Entry DOI10.2210/pdb3fsk/pdb
Related3FLN 3FLS 3FLW 3FLY 3FLZ 3FMH 3FMJ 3FMK 3FML 3FMM 3FMN
DescriptorMitogen-activated protein kinase 14, 3-(2-chlorophenyl)-7-[(trans-4-hydroxycyclohexyl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one (3 entities in total)
Functional Keywordsp38; map kinase; serine/threonine kinase, alternative splicing, atp-binding, cytoplasm, kinase, nucleotide-binding, nucleus, phosphoprotein, polymorphism, serine/threonine-protein kinase, transferase, signaling protein
Biological sourceHomo sapiens (human)
Cellular locationCytoplasm (By similarity): Q16539
Total number of polymer chains1
Total formula weight43122.55
Authors
Kuglstatter, A.,Bertrand, J.,Takahara, P.,Villasenor, A. (deposition date: 2009-01-09, release date: 2009-12-22, Last modification date: 2023-09-06)
Primary citationArora, N.,Williams, C.,Delano, W.,Will, D.,Kuglstatter, A.
Mapping Binding Pocket Volume: Potential Applications towards Ligand Design and Selectivity
To be Published,
Experimental method
X-RAY DIFFRACTION (2 Å)
Structure validation

217705

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