1GQR
ACETYLCHOLINESTERASE (E.C. 3.1.1.7) COMPLEXED WITH RIVASTIGMINE
Summary for 1GQR
Entry DOI | 10.2210/pdb1gqr/pdb |
Related | 1ACJ 1ACL 1AMN 1AX9 1CFJ 1DX6 1E3Q 1E66 1EA5 1EEA 1EVE 1FSS 1GPK 1GPN 1GQS 1HBJ 1OCE 1QID 1QIE 1QIF 1QIG 1QIH 1QII 1QIJ 1QIK 1QIM 1QTI 1SOM 1VOT 1VXO 1VXR 2ACE 2ACK 2DFP 3ACE 4ACE |
Descriptor | ACETYLCHOLINESTERASE, 2-acetamido-2-deoxy-beta-D-glucopyranose, 3-[(1S)-1-(DIMETHYLAMINO)ETHYL]PHENOL, ... (5 entities in total) |
Functional Keywords | hydrolase, neurotransmitter cleavage |
Biological source | TORPEDO CALIFORNICA (PACIFIC ELECTRIC RAY) |
Cellular location | Isoform H: Cell membrane; Lipid-anchor, GPI- anchor. Isoform T: Cell membrane; Peripheral membrane protein: P04058 |
Total number of polymer chains | 1 |
Total formula weight | 60902.73 |
Authors | Raves, M.L.,Harel, M.,Silman, I.,Sussman, J.L. (deposition date: 2001-12-04, release date: 2002-03-15, Last modification date: 2023-12-13) |
Primary citation | Bar-on, P.,Millard, C.B.,Harel, M.,Dvir, H.,Enz, A.,Sussman, J.L.,Silman, I. Kinetic and Structural Studies on the Interaction of Cholinesterases with the Anti-Alzheimer Drug Rivastigmine Biochemistry, 41:3555-, 2002 Cited by PubMed: 11888271DOI: 10.1021/BI020016X PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.2 Å) |
Structure validation
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