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7S11
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BU of 7s11 by Molmil
Crystal structure of Fab in complex with mouse CD96 monomer
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, Fab heavy chain, Fab light chain, ...
Authors:Lee, P.S, Chau, B, Strop, P.
Deposit date:2021-08-31
Release date:2021-11-03
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (2.58 Å)
Cite:Antibody blockade of CD96 by distinct molecular mechanisms.
Mabs, 13, 2021
5KW2
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BU of 5kw2 by Molmil
The extra-helical binding site of GPR40 and the structural basis for allosteric agonism and incretin stimulation
Descriptor: (3~{S})-3-cyclopropyl-3-[2-[1-[2-[2,2-dimethylpropyl-(6-methylpyridin-2-yl)carbamoyl]-5-methoxy-phenyl]piperidin-4-yl]-1-benzofuran-6-yl]propanoic acid, Free fatty acid receptor 1,Lysozyme,Free fatty acid receptor 1
Authors:Ho, J.D, Chau, B, Rodgers, L, Lu, F, Wilbur, K.L, Otto, K.A, Chen, Y, Song, M, Riley, J.P, Yang, H.-C, Reynolds, N.A, Kahl, S.D, Lewis, A.P, Groshong, C, Madsen, R.E, Conners, K, Linswala, J.P, Gheyi, T, Saflor, M.D, Lee, M.R, Benach, J, Baker, K.A, Montrose-Rafizadeh, C, Genin, M.J, Miller, A.R, Hamdouchi, C.
Deposit date:2016-07-15
Release date:2018-05-02
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (2.76 Å)
Cite:Structural basis for GPR40 allosteric agonism and incretin stimulation.
Nat Commun, 9, 2018
7KHD
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BU of 7khd by Molmil
Human GITR-GITRL complex
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, Tumor necrosis factor ligand superfamily member 18, Tumor necrosis factor receptor superfamily member 18
Authors:Wang, F, Chau, B, West, S.M, Strop, P.
Deposit date:2020-10-21
Release date:2021-03-03
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (2.956102 Å)
Cite:Structures of mouse and human GITR-GITRL complexes reveal unique TNF superfamily interactions.
Nat Commun, 12, 2021
7KHX
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BU of 7khx by Molmil
Mouse GITR-GITRL complex
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Tumor necrosis factor ligand superfamily member 18, ...
Authors:Wang, F, Chau, B, West, S.M, Strop, P.
Deposit date:2020-10-22
Release date:2021-03-03
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (3.20569849 Å)
Cite:Structures of mouse and human GITR-GITRL complexes reveal unique TNF superfamily interactions.
Nat Commun, 12, 2021
7SU1
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BU of 7su1 by Molmil
Crystal structure of an acidic pH-selective Ipilimumab variant Ipi.106 in complex with CTLA-4
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, Cytotoxic T-lymphocyte protein 4, Fab heavy chain, ...
Authors:Lee, P.S, Chau, B, Strop, P.
Deposit date:2021-11-15
Release date:2022-03-02
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (2.53 Å)
Cite:Improved therapeutic index of an acidic pH-selective antibody.
Mabs, 14, 2022
7SU0
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BU of 7su0 by Molmil
Crystal structure of an acidic pH-selective Ipilimumab variant Ipi.105 in complex with CTLA-4
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, CITRATE ANION, Cytotoxic T-lymphocyte protein 4, ...
Authors:Lee, P.S, Chau, B, Strop, P.
Deposit date:2021-11-15
Release date:2022-03-02
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (2.41 Å)
Cite:Improved therapeutic index of an acidic pH-selective antibody.
Mabs, 14, 2022
5UZB
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BU of 5uzb by Molmil
Cryo-EM structure of the MAL TIR domain filament
Descriptor: Toll/interleukin-1 receptor domain-containing adapter protein
Authors:Ve, T, Vajjhala, P.R, Hedger, A, Croll, T, DiMaio, F, Horsefield, S, Yu, X, Lavrencic, P, Hassan, Z, Morgan, G.P, Mansell, A, Mobli, M, O'Carrol, A, Chauvin, B, Gambin, Y, Sierecki, E, Landsberg, M.J, Stacey, K.J, Egelman, E.H, Kobe, B.
Deposit date:2017-02-25
Release date:2017-07-26
Last modified:2020-01-15
Method:ELECTRON MICROSCOPY (7 Å)
Cite:Structural basis of TIR-domain-assembly formation in MAL- and MyD88-dependent TLR4 signaling.
Nat. Struct. Mol. Biol., 24, 2017
6CTS
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BU of 6cts by Molmil
PROPOSED MECHANISM FOR THE CONDENSATION REACTION OF CITRATE SYNTHASE. 1.9-ANGSTROMS STRUCTURE OF THE TERNARY COMPLEX WITH OXALOACETATE AND CARBOXYMETHYL COENZYME A
Descriptor: CITRATE SYNTHASE, CITRYL-THIOETHER-COENZYME *A
Authors:Karpusas, M, Branchaud, B, Remington, S.J.
Deposit date:1989-11-16
Release date:1990-10-15
Last modified:2024-03-13
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:Proposed mechanism for the condensation reaction of citrate synthase: 1.9-A structure of the ternary complex with oxaloacetate and carboxymethyl coenzyme A.
Biochemistry, 29, 1990
1XAE
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BU of 1xae by Molmil
Crystal structure of wild type yellow fluorescent protein zFP538 from Zoanthus
Descriptor: BETA-MERCAPTOETHANOL, fluorescent protein FP538
Authors:Remington, S.J, Wachter, R.M, Yarbrough, D.K, Branchaud, B, Anderson, D.C, Kallio, K, Lukyanov, K.A.
Deposit date:2004-08-25
Release date:2005-02-08
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (2.7 Å)
Cite:zFP538, a yellow-fluorescent protein from Zoanthus, contains a novel three-ring chromophore.
Biochemistry, 44, 2005
1XA9
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BU of 1xa9 by Molmil
Crystal structure of yellow fluorescent protein zFP538 K66M green mutant
Descriptor: BETA-MERCAPTOETHANOL, fluorescent protein FP538
Authors:Remington, S.J, Wachter, R.M, Yarbrough, D.K, Branchaud, B, Anderson, D.C, Kallio, K, Lukyanov, K.A.
Deposit date:2004-08-25
Release date:2005-02-08
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:zFP538, a yellow-fluorescent protein from Zoanthus, contains a novel three-ring chromophore.
Biochemistry, 44, 2005
5CTS
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BU of 5cts by Molmil
PROPOSED MECHANISM FOR THE CONDENSATION REACTION OF CITRATE SYNTHASE. 1.9-ANGSTROMS STRUCTURE OF THE TERNARY COMPLEX WITH OXALOACETATE AND CARBOXYMETHYL COENZYME A
Descriptor: CARBOXYMETHYL COENZYME *A, CITRATE SYNTHASE, OXALOACETATE ION
Authors:Karpusas, M, Branchaud, B, Remington, S.J.
Deposit date:1989-11-16
Release date:1990-10-15
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Proposed mechanism for the condensation reaction of citrate synthase: 1.9-A structure of the ternary complex with oxaloacetate and carboxymethyl coenzyme A.
Biochemistry, 29, 1990
2CBS
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BU of 2cbs by Molmil
CELLULAR RETINOIC ACID BINDING PROTEIN II IN COMPLEX WITH A SYNTHETIC RETINOIC ACID (RO-13 6307)
Descriptor: 3-METHYL-7-(5,5,8,8-TETRAMETHYL-5,6,7,8-TETRAHYDRO-NAPHTHALEN-2-YL) -OCTA-2,4,6-TRIENOIC ACID, PROTEIN (CRABP-II)
Authors:Chaudhuri, B, Kleywegt, G.J, Bergfors, T, Jones, T.A.
Deposit date:1999-02-22
Release date:1999-12-22
Last modified:2023-08-23
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:Structures of cellular retinoic acid binding proteins I and II in complex with synthetic retinoids.
Acta Crystallogr.,Sect.D, 55, 1999
2CBR
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BU of 2cbr by Molmil
CELLULAR RETINOIC ACID BINDING PROTEIN I IN COMPLEX WITH A RETINOBENZOIC ACID (AM80)
Descriptor: 4-[(5,5,8,8-tetramethyl-5,6,7,8-tetrahydronaphthalen-2-yl)carbamoyl]benzoic acid, PROTEIN (CRABP-I)
Authors:Chaudhuri, B, Kleywegt, G.J, Bergfors, T, Jones, T.A.
Deposit date:1999-02-22
Release date:1999-12-21
Last modified:2023-08-23
Method:X-RAY DIFFRACTION (2.8 Å)
Cite:Structures of cellular retinoic acid binding proteins I and II in complex with synthetic retinoids.
Acta Crystallogr.,Sect.D, 55, 1999
3CBS
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BU of 3cbs by Molmil
CELLULAR RETINOIC ACID BINDING PROTEIN II IN COMPLEX WITH A SYNTHETIC RETINOIC ACID (RO-12 7310)
Descriptor: (2E,4E,6E,8E)-9-(4-hydroxy-2,3,6-trimethylphenyl)-3,7-dimethylnona-2,4,6,8-tetraenoic acid, PROTEIN (CRABP-II)
Authors:Chaudhuri, B, Kleywegt, G.J, Bergfors, T, Jones, T.A.
Deposit date:1999-02-22
Release date:1999-12-22
Last modified:2023-08-30
Method:X-RAY DIFFRACTION (2 Å)
Cite:Structures of cellular retinoic acid binding proteins I and II in complex with synthetic retinoids.
Acta Crystallogr.,Sect.D, 55, 1999
1RPJ
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BU of 1rpj by Molmil
CRYSTAL STRUCTURE OF D-ALLOSE BINDING PROTEIN FROM ESCHERICHIA COLI
Descriptor: PROTEIN (PRECURSOR OF PERIPLASMIC SUGAR RECEPTOR), SULFATE ION, ZINC ION, ...
Authors:Chaudhuri, B, Jones, T.A, Mowbray, S.L.
Deposit date:1999-02-04
Release date:1999-02-16
Last modified:2023-08-23
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Structure of D-allose binding protein from Escherichia coli bound to D-allose at 1.8 A resolution.
J.Mol.Biol., 286, 1999
7S13
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BU of 7s13 by Molmil
Crystal structure of Fab in complex with mouse CD96 dimer
Descriptor: 1,2-ETHANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, CITRATE ANION, ...
Authors:Lee, P.S, Barman, I, Strop, P.
Deposit date:2021-08-31
Release date:2021-10-20
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (2.12 Å)
Cite:Antibody blockade of CD96 by distinct molecular mechanisms.
Mabs, 13, 2021
6VCB
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BU of 6vcb by Molmil
Cryo-EM structure of the Glucagon-like peptide-1 receptor in complex with G protein, GLP-1 peptide and a positive allosteric modulator
Descriptor: 1-[(1R)-1-(2,6-dichloro-3-methoxyphenyl)ethyl]-6-{2-[(2R)-piperidin-2-yl]phenyl}-1H-benzimidazole, Glucagon-like peptide 1, Glucagon-like peptide 1 receptor, ...
Authors:Sun, B, Feng, D, Bueno, A, Kobilka, B, Sloop, K.
Deposit date:2019-12-20
Release date:2020-07-22
Last modified:2020-09-30
Method:ELECTRON MICROSCOPY (3.3 Å)
Cite:Structural insights into probe-dependent positive allosterism of the GLP-1 receptor.
Nat.Chem.Biol., 16, 2020
6UQC
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BU of 6uqc by Molmil
Mouse IgG2a Bispecific Fc
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-3)-[2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-3)-[alpha-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Wang, F, Tsai, J.C, Davis, J.H, West, S.M, Strop, P.
Deposit date:2019-10-18
Release date:2020-01-01
Last modified:2023-10-11
Method:X-RAY DIFFRACTION (1.87 Å)
Cite:Design and characterization of mouse IgG1 and IgG2a bispecific antibodies for use in syngeneic models.
Mabs, 12, 2019
1AMZ
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BU of 1amz by Molmil
CHICKEN CITRATE SYNTHASE COMPLEX WITH NITROMETHYLDE-COA AND MALATE
Descriptor: CITRATE SYNTHASE, D-MALATE, NITROMETHYLDETHIA COENZYME A
Authors:Usher, K.C, Remington, S.J.
Deposit date:1997-06-19
Release date:1997-12-24
Last modified:2023-08-02
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Mechanisms of Enzyme-Catalyzed Deprotonation of Acetyl-Coenzyme A
To be Published
1AL6
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BU of 1al6 by Molmil
CHICKEN CITRATE SYNTHASE COMPLEX WITH N-HYDROXYAMIDO-COA AND OXALOACETATE
Descriptor: CITRATE SYNTHASE, N-HYDROXYAMIDOCARBOXYMETHYLDETHIA COENZYME *A, OXALOACETATE ION
Authors:Usher, K.C, Remington, S.J.
Deposit date:1997-06-12
Release date:1997-12-24
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (1.85 Å)
Cite:Mechanisms of Enzyme-Catalyzed Deprotonation of Acetyl-Coenzyme A
To be Published
1CSS
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BU of 1css by Molmil
ALPHA-FLUORO ACID AND ALPHA-FLUORO AMIDE ANALOGS OF ACETYL-COA AS INHIBITORS OF OF CITRATE SYNTHASE: EFFECT OF PKA MATCHING ON BINDING AFFINITY AND HYDROGEN BOND LENGTH
Descriptor: ALPHA-FLUORO-CARBOXYMETHYLDETHIA COENZYME A COMPLEX, CITRATE SYNTHASE, OXALOACETATE ION
Authors:Usher, K.C, Remington, S.J.
Deposit date:1995-08-04
Release date:1995-10-15
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (1.7 Å)
Cite:alpha-Fluoro acid and alpha-fluoro amide analogs of acetyl-CoA as inhibitors of citrate synthase: effect of pKa matching on binding affinity and hydrogen bond length.
Biochemistry, 34, 1995
1CSR
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BU of 1csr by Molmil
Alpha-fluoro acid and alpha-fluoro amide analogs of acetyl-coa as inhibitors of of citrate synthase: effect of pka matching on binding affinity and hydrogen bond length
Descriptor: ALPHA-FLUORO-AMIDOCARBOXYMETHYLDETHIA COENZYME A COMPLEX, CITRATE SYNTHASE, OXALOACETATE ION
Authors:Usher, K.C, Remington, S.J.
Deposit date:1995-08-04
Release date:1995-10-15
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (1.7 Å)
Cite:alpha-Fluoro acid and alpha-fluoro amide analogs of acetyl-CoA as inhibitors of citrate synthase: effect of pKa matching on binding affinity and hydrogen bond length.
Biochemistry, 34, 1995
6CSC
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BU of 6csc by Molmil
CHICKEN CITRATE SYNTHASE COMPLEX WITH TRIFLUOROACETONYL-COA AND CITRATE
Descriptor: CITRATE SYNTHASE, CITRIC ACID, TRIFLUOROACETONYL COENZYME A
Authors:Usher, K.C, Remington, S.J.
Deposit date:1997-06-19
Release date:1997-12-24
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (2.25 Å)
Cite:Trifluoroacetonyl Coenzyme A, an Inhibitor of Citrate Synthase, Binds in a Combination of Productive and Nonproductive Modes
To be Published
1BCS
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BU of 1bcs by Molmil
COMPLEX OF THE WHEAT SERINE CARBOXYPEPTIDASE, CPDW-II, WITH THE MICROBIAL PEPTIDE ALDEHYDE INHIBITOR, CHYMOSTATIN, AND ARGININE AT 100 DEGREES KELVIN
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ACETATE ION, ...
Authors:Bullock, T.L, Remington, S.J.
Deposit date:1995-11-03
Release date:1996-03-08
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (2.08 Å)
Cite:Peptide aldehyde complexes with wheat serine carboxypeptidase II: implications for the catalytic mechanism and substrate specificity.
J.Mol.Biol., 255, 1996
1BCR
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BU of 1bcr by Molmil
COMPLEX OF THE WHEAT SERINE CARBOXYPEPTIDASE, CPDW-II, WITH THE MICROBIAL PEPTIDE ALDEHYDE INHIBITOR, ANTIPAIN, AND ARGININE AT ROOM TEMPERATURE
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ANTIPAIN, ...
Authors:Bullock, T.L, Remington, S.J.
Deposit date:1995-11-03
Release date:1996-03-08
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:Peptide aldehyde complexes with wheat serine carboxypeptidase II: implications for the catalytic mechanism and substrate specificity.
J.Mol.Biol., 255, 1996

 

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