1THG
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1CRL
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1ACJ
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1ACL
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1TRH
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1LPS
| A STRUCTURAL BASIS FOR THE CHIRAL PREFERENCES OF LIPASES | 分子名称: | (1S)-MENTHYL HEXYL PHOSPHONATE GROUP, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Grochulski, P.G, Cygler, M.C. | 登録日 | 1995-01-05 | 公開日 | 1995-02-14 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.18 Å) | 主引用文献 | A Structural Basis for the Chiral Preferences of Lipases J.Am.Chem.Soc., 116, 1994
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1LPM
| A STRUCTURAL BASIS FOR THE CHIRAL PREFERENCES OF LIPASES | 分子名称: | (1R)-MENTHYL HEXYL PHOSPHONATE GROUP, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Grochulski, P.G, Cygler, M.C. | 登録日 | 1995-01-06 | 公開日 | 1995-04-20 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.18 Å) | 主引用文献 | A Structural Basis for the Chiral Preferences of Lipases J.Am.Chem.Soc., 116, 1994
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1LPN
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1LPO
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1LPP
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1CLE
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1FSS
| ACETYLCHOLINESTERASE (E.C. 3.1.1.7) COMPLEXED WITH FASCICULIN-II | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, ACETYLCHOLINESTERASE, FASCICULIN II, ... | 著者 | Harel, M, Kleywegt, G.J, Silman, I, Sussman, J.L. | 登録日 | 1995-10-25 | 公開日 | 1996-03-08 | 最終更新日 | 2021-06-02 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Crystal structure of an acetylcholinesterase-fasciculin complex: interaction of a three-fingered toxin from snake venom with its target. Structure, 3, 1995
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1MAH
| FASCICULIN2-MOUSE ACETYLCHOLINESTERASE COMPLEX | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, ACETYLCHOLINESTERASE, FASCICULIN 2 | 著者 | Bourne, Y, Taylor, P, Marchot, P. | 登録日 | 1995-11-21 | 公開日 | 1996-04-03 | 最終更新日 | 2021-03-31 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | Acetylcholinesterase inhibition by fasciculin: crystal structure of the complex. Cell(Cambridge,Mass.), 83, 1995
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1AMN
| TRANSITION STATE ANALOG: ACETYLCHOLINESTERASE COMPLEXED WITH M-(N,N,N-TRIMETHYLAMMONIO)TRIFLUOROACETOPHENONE | 分子名称: | ACETYLCHOLINESTERASE, M-(N,N,N-TRIMETHYLAMMONIO)-2,2,2-TRIFLUORO-1,1-DIHYDROXYETHYLBENZENE, SULFATE ION | 著者 | Harel, M, Silman, I, Sussman, J.L. | 登録日 | 1996-02-13 | 公開日 | 1996-04-03 | 最終更新日 | 2021-06-02 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | The X-ray structure of a transition state analog complex reveals the molecular origins of the catalytic power and substrate specificity of acetylcholinesterase. J.Am.Chem.Soc., 118, 1996
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2ACE
| NATIVE ACETYLCHOLINESTERASE (E.C. 3.1.1.7) FROM TORPEDO CALIFORNICA | 分子名称: | ACETYLCHOLINE, ACETYLCHOLINESTERASE | 著者 | Harel, M, Raves, M.L, Silman, I, Sussman, J.L. | 登録日 | 1996-06-23 | 公開日 | 1996-11-08 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Structure of acetylcholinesterase complexed with the nootropic alkaloid, (-)-huperzine A. Nat.Struct.Biol., 4, 1997
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1VOT
| ACETYLCHOLINESTERASE (E.C. 3.1.1.7) COMPLEXED WITH HUPERZINE A | 分子名称: | ACETYLCHOLINESTERASE, Huperzine A | 著者 | Raves, M.L, Harel, M, Silman, I, Sussman, J.L. | 登録日 | 1996-06-23 | 公開日 | 1997-06-16 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Structure of acetylcholinesterase complexed with the nootropic alkaloid, (-)-huperzine A. Nat.Struct.Biol., 4, 1997
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1AKN
| STRUCTURE OF BILE-SALT ACTIVATED LIPASE | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, BILE-SALT ACTIVATED LIPASE | 著者 | Wang, X, Zhang, X. | 登録日 | 1997-05-23 | 公開日 | 1998-05-27 | 最終更新日 | 2023-08-02 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | The crystal structure of bovine bile salt activated lipase: insights into the bile salt activation mechanism. Structure, 5, 1997
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1AQL
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2ACK
| ACETYLCHOLINESTERASE COMPLEXED WITH EDROPHONIUM, MONOCHROMATIC DATA | 分子名称: | ACETYLCHOLINESTERASE, EDROPHONIUM ION | 著者 | Raves, M.L, Sussman, J.L, Harel, M, Silman, I. | 登録日 | 1997-10-29 | 公開日 | 1998-02-11 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Static Laue diffraction studies on acetylcholinesterase. Acta Crystallogr.,Sect.D, 54, 1998
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1AX9
| ACETYLCHOLINESTERASE COMPLEXED WITH EDROPHONIUM, LAUE DATA | 分子名称: | ACETYLCHOLINESTERASE, EDROPHONIUM ION | 著者 | Raves, M.L, Ravelli, R.B.G, Sussman, J.L, Harel, M, Silman, I. | 登録日 | 1997-11-03 | 公開日 | 1998-02-11 | 最終更新日 | 2023-08-02 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Static Laue diffraction studies on acetylcholinesterase. Acta Crystallogr.,Sect.D, 54, 1998
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2BCE
| CHOLESTEROL ESTERASE FROM BOS TAURUS | 分子名称: | CHOLESTEROL ESTERASE | 著者 | Chen, J.C.-H, Miercke, L.J.W, Krucinski, J, Starr, J.R, Saenz, G, Wang, X, Spilburg, C.A, Lange, L.G, Ellsworth, J.L, Stroud, R.M. | 登録日 | 1998-01-28 | 公開日 | 1999-02-02 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Structure of bovine pancreatic cholesterol esterase at 1.6 A: novel structural features involved in lipase activation. Biochemistry, 37, 1998
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1EVE
| THREE DIMENSIONAL STRUCTURE OF THE ANTI-ALZHEIMER DRUG, E2020 (ARICEPT), COMPLEXED WITH ITS TARGET ACETYLCHOLINESTERASE | 分子名称: | 1-BENZYL-4-[(5,6-DIMETHOXY-1-INDANON-2-YL)METHYL]PIPERIDINE, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Kryger, G, Silman, I, Sussman, J.L. | 登録日 | 1998-03-04 | 公開日 | 1999-01-20 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Structure of acetylcholinesterase complexed with E2020 (Aricept): implications for the design of new anti-Alzheimer drugs. Structure Fold.Des., 7, 1999
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1OCE
| ACETYLCHOLINESTERASE (E.C. 3.1.1.7) COMPLEXED WITH MF268 | 分子名称: | ACETYLCHOLINESTERASE, CIS-2,6-DIMETHYLMORPHOLINOOCTYLCARBAMYLESEROLINE | 著者 | Bartolucci, C, Perola, E, Cellai, L, Brufani, M, Lamba, D. | 登録日 | 1998-06-12 | 公開日 | 1999-05-18 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | "Back door" opening implied by the crystal structure of a carbamoylated acetylcholinesterase. Biochemistry, 38, 1999
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1MAA
| MOUSE ACETYLCHOLINESTERASE CATALYTIC DOMAIN, GLYCOSYLATED PROTEIN | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[beta-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ACETYLCHOLINESTERASE, ... | 著者 | Bourne, Y, Taylor, P, Bougis, P.E, Marchot, P. | 登録日 | 1998-11-04 | 公開日 | 1999-04-20 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Crystal structure of mouse acetylcholinesterase. A peripheral site-occluding loop in a tetrameric assembly. J.Biol.Chem., 274, 1999
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2DFP
| X-RAY STRUCTURE OF AGED DI-ISOPROPYL-PHOSPHORO-FLUORIDATE (DFP) BOUND TO ACETYLCHOLINESTERASE | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Kryger, G, Millard, C.B, Silman, I, Sussman, J.L. | 登録日 | 1998-12-07 | 公開日 | 1999-06-28 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Crystal structures of aged phosphonylated acetylcholinesterase: nerve agent reaction products at the atomic level. Biochemistry, 38, 1999
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