7OM1
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![BU of 7om1 by Molmil](/molmil-images/mine/7om1) | Tankyrase 2 in complex with an inhibitor (OUL220) | Descriptor: | 8-methoxy-4~{H}-thieno[2,3-c]isoquinolin-5-one, GLYCEROL, Poly [ADP-ribose] polymerase tankyrase-2, ... | Authors: | Sowa, S.T, Lehtio, L. | Deposit date: | 2021-05-21 | Release date: | 2021-12-08 | Last modified: | 2024-01-31 | Method: | X-RAY DIFFRACTION (1.7 Å) | Cite: | Analogs of TIQ-A as inhibitors of human mono-ADP-ribosylating PARPs. Bioorg.Med.Chem., 52, 2021
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4DFR
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![BU of 4dfr by Molmil](/molmil-images/mine/4dfr) | CRYSTAL STRUCTURES OF ESCHERICHIA COLI AND LACTOBACILLUS CASEI DIHYDROFOLATE REDUCTASE REFINED AT 1.7 ANGSTROMS RESOLUTION. I. GENERAL FEATURES AND BINDING OF METHOTREXATE | Descriptor: | CALCIUM ION, CHLORIDE ION, DIHYDROFOLATE REDUCTASE, ... | Authors: | Filman, D.J, Matthews, D.A, Bolin, J.T, Kraut, J. | Deposit date: | 1982-06-25 | Release date: | 1982-10-21 | Last modified: | 2024-02-28 | Method: | X-RAY DIFFRACTION (1.7 Å) | Cite: | Crystal structures of Escherichia coli and Lactobacillus casei dihydrofolate reductase refined at 1.7 A resolution. I. General features and binding of methotrexate. J.Biol.Chem., 257, 1982
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7P49
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![BU of 7p49 by Molmil](/molmil-images/mine/7p49) | HLA-E*01:03 in complex with Mtb14 | Descriptor: | Beta-2-microglobulin, GLYCEROL, HLA class I histocompatibility antigen, ... | Authors: | Walters, L.C, Gillespie, G.M. | Deposit date: | 2021-07-10 | Release date: | 2022-06-22 | Last modified: | 2024-01-31 | Method: | X-RAY DIFFRACTION (2.05 Å) | Cite: | Primary and secondary functions of HLA-E are determined by stability and conformation of the peptide-bound complexes. Cell Rep, 39, 2022
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7OVX
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![BU of 7ovx by Molmil](/molmil-images/mine/7ovx) | E3 RING ligase binding domain | Descriptor: | E3 ubiquitin-protein ligase TRIM7, Peptide G | Authors: | James, L.C. | Deposit date: | 2021-06-15 | Release date: | 2022-06-22 | Last modified: | 2024-01-31 | Method: | X-RAY DIFFRACTION (1.7 Å) | Cite: | E3 ligase targeting domain To Be Published
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7P0U
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![BU of 7p0u by Molmil](/molmil-images/mine/7p0u) | ORF virus encoded Bcl-2 homolog ORFV125 in complex with Puma BH3 peptide | Descriptor: | 1,2-ETHANEDIOL, Activator of apoptosis harakiri, Apoptosis inhibitor, ... | Authors: | Suraweera, C.D, Hinds, M.G, Kvansakul, M. | Deposit date: | 2021-06-30 | Release date: | 2022-07-13 | Last modified: | 2024-01-31 | Method: | X-RAY DIFFRACTION (1.99374259 Å) | Cite: | Structural Investigation of Orf Virus Bcl-2 Homolog ORFV125 Interactions with BH3-Motifs from BH3-Only Proteins Puma and Hrk. Viruses, 13, 2021
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7OW2
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![BU of 7ow2 by Molmil](/molmil-images/mine/7ow2) | E3 RING ligase binding domain with peptide | Descriptor: | CHLORIDE ION, E3 ubiquitin-protein ligase RNF187 peptide, E3 ubiquitin-protein ligase TRIM7, ... | Authors: | James, L.C. | Deposit date: | 2021-06-16 | Release date: | 2022-07-13 | Last modified: | 2024-01-31 | Method: | X-RAY DIFFRACTION (2.17 Å) | Cite: | E3 ligase targeting domain To Be Published
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7P4B
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![BU of 7p4b by Molmil](/molmil-images/mine/7p4b) | HLA-E*01:03 in complex with IL9 | Descriptor: | Beta-2-microglobulin, ESAT-6-like protein EsxH, GLYCEROL, ... | Authors: | Walters, L.C, Gillespie, G.M. | Deposit date: | 2021-07-10 | Release date: | 2022-07-27 | Last modified: | 2024-01-31 | Method: | X-RAY DIFFRACTION (1.72 Å) | Cite: | Primary and secondary functions of HLA-E are determined by stability and conformation of the peptide-bound complexes. Cell Rep, 39, 2022
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7Q2U
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![BU of 7q2u by Molmil](/molmil-images/mine/7q2u) | The crystal structure of the HINT1 Q62A mutant. | Descriptor: | CACODYLATE ION, HEXAETHYLENE GLYCOL, Histidine triad nucleotide-binding protein 1, ... | Authors: | Dolot, R.M, Strom, A.M, Wagner, C.R. | Deposit date: | 2021-10-26 | Release date: | 2021-11-03 | Last modified: | 2024-02-07 | Method: | X-RAY DIFFRACTION (2.27 Å) | Cite: | Dynamic Long-Range Interactions Influence Substrate Binding and Catalysis by Human Histidine Triad Nucleotide-Binding Proteins (HINTs), Key Regulators of Multiple Cellular Processes and Activators of Antiviral ProTides. Biochemistry, 61, 2022
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7Q1E
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![BU of 7q1e by Molmil](/molmil-images/mine/7q1e) | CPAP:TUBULIN:IIH5 ALPHAREP COMPLEX | Descriptor: | Centromere protein J, GLYCEROL, GUANOSINE-5'-TRIPHOSPHATE, ... | Authors: | Campanacci, V, Gigant, b. | Deposit date: | 2021-10-19 | Release date: | 2022-04-13 | Last modified: | 2024-01-31 | Method: | X-RAY DIFFRACTION (2.7 Å) | Cite: | Structural convergence for tubulin binding of CPAP and vinca domain microtubule inhibitors. Proc.Natl.Acad.Sci.USA, 119, 2022
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7POX
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![BU of 7pox by Molmil](/molmil-images/mine/7pox) | TNKS2 in complex with OM-1700, treated with H2O2 | Descriptor: | N-[3-[5-(5-ethoxypyridin-2-yl)-4-(2-fluorophenyl)-1,2,4-triazol-3-yl]cyclobutyl]pyridine-2-carboxamide, Poly [ADP-ribose] polymerase tankyrase-2 | Authors: | Sowa, S.T, Lehtio, L. | Deposit date: | 2021-09-10 | Release date: | 2022-05-04 | Last modified: | 2024-01-31 | Method: | X-RAY DIFFRACTION (2.5 Å) | Cite: | The zinc-binding motif in tankyrases is required for the structural integrity of the catalytic ADP-ribosyltransferase domain. Open Biology, 12, 2022
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7Q4L
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![BU of 7q4l by Molmil](/molmil-images/mine/7q4l) | |
7PFX
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7PEW
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![BU of 7pew by Molmil](/molmil-images/mine/7pew) | |
7PFC
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![BU of 7pfc by Molmil](/molmil-images/mine/7pfc) | |
7PEY
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![BU of 7pey by Molmil](/molmil-images/mine/7pey) | |
7PEX
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7PEZ
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![BU of 7pez by Molmil](/molmil-images/mine/7pez) | |
7PET
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![BU of 7pet by Molmil](/molmil-images/mine/7pet) | The 4x177 nucleosome array containing H1 | Descriptor: | DNA (702-MER), Histone H1.4, Histone H2A type 1-B/E, ... | Authors: | Dombrowski, M, Cramer, P. | Deposit date: | 2021-08-11 | Release date: | 2022-08-03 | Method: | ELECTRON MICROSCOPY (9.5 Å) | Cite: | Histone H1 binding to nucleosome arrays depends on linker DNA length and trajectory. Nat.Struct.Mol.Biol., 29, 2022
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7PF3
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7PF5
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![BU of 7pf5 by Molmil](/molmil-images/mine/7pf5) | |
7PF4
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![BU of 7pf4 by Molmil](/molmil-images/mine/7pf4) | |
7PFU
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7PF6
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![BU of 7pf6 by Molmil](/molmil-images/mine/7pf6) | |
7PEV
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![BU of 7pev by Molmil](/molmil-images/mine/7pev) | |
7PF2
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![BU of 7pf2 by Molmil](/molmil-images/mine/7pf2) | |