3U9S
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3u9s by Molmil](/molmil-images/mine/3u9s) | Crystal structure of P. aeruginosa 3-methylcrotonyl-CoA carboxylase (MCC) 750 kD holoenzyme, CoA complex | Descriptor: | 5-(HEXAHYDRO-2-OXO-1H-THIENO[3,4-D]IMIDAZOL-6-YL)PENTANAL, COENZYME A, Methylcrotonyl-CoA carboxylase, ... | Authors: | Huang, C.S, Tong, L. | Deposit date: | 2011-10-19 | Release date: | 2011-12-14 | Last modified: | 2013-01-23 | Method: | X-RAY DIFFRACTION (3.5 Å) | Cite: | An unanticipated architecture of the 750-kDa {alpha}6{beta}6 holoenzyme of 3-methylcrotonyl-CoA carboxylase Nature, 481, 2012
|
|
8GK8
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 8gk8 by Molmil](/molmil-images/mine/8gk8) | R21A Staphylococcus aureus pyruvate carboxylase | Descriptor: | 5-(HEXAHYDRO-2-OXO-1H-THIENO[3,4-D]IMIDAZOL-6-YL)PENTANAL, ACETYL COENZYME *A, COENZYME A, ... | Authors: | Laseke, A.J, St.Maurice, M. | Deposit date: | 2023-03-17 | Release date: | 2023-08-30 | Last modified: | 2024-03-13 | Method: | X-RAY DIFFRACTION (2.68 Å) | Cite: | Allosteric Site at the Biotin Carboxylase Dimer Interface Mediates Activation and Inhibition in Staphylococcus aureus Pyruvate Carboxylase. Biochemistry, 62, 2023
|
|
8HZ5
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 8hz5 by Molmil](/molmil-images/mine/8hz5) | |
8HZ4
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 8hz4 by Molmil](/molmil-images/mine/8hz4) | |
8HWL
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 8hwl by Molmil](/molmil-images/mine/8hwl) | Human Pyruvate Carboxylase | Descriptor: | 5-(HEXAHYDRO-2-OXO-1H-THIENO[3,4-D]IMIDAZOL-6-YL)PENTANAL, Pyruvate carboxylase, mitochondrial | Authors: | Liu, D.S, Su, J.Y. | Deposit date: | 2022-12-30 | Release date: | 2024-01-31 | Method: | ELECTRON MICROSCOPY (5.63 Å) | Cite: | Human Pyruvate Carboxylase To Be Published
|
|
8J4Z
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 8j4z by Molmil](/molmil-images/mine/8j4z) | |
8J7O
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 8j7o by Molmil](/molmil-images/mine/8j7o) | |
8J78
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 8j78 by Molmil](/molmil-images/mine/8j78) | Human 3-methylcrotonyl-CoA carboxylase in BCCP-H2 state | Descriptor: | 5-(HEXAHYDRO-2-OXO-1H-THIENO[3,4-D]IMIDAZOL-6-YL)PENTANAL, Methylcrotonoyl-CoA carboxylase beta chain, mitochondrial, ... | Authors: | Liu, D.S, Su, J.Y. | Deposit date: | 2023-04-27 | Release date: | 2024-05-08 | Method: | ELECTRON MICROSCOPY (3.88 Å) | Cite: | Human 3-methylcrotonyl-CoA carboxylase in BCCP-H2 state To Be Published
|
|
8J99
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 8j99 by Molmil](/molmil-images/mine/8j99) | Human 3-methylcrotonyl-CoA carboxylase in BCS-mcoa state | Descriptor: | Methylcrotonoyl-CoA carboxylase beta chain, mitochondrial, Methylcrotonoyl-CoA carboxylase subunit alpha, ... | Authors: | Liu, D.S, Su, J.Y. | Deposit date: | 2023-05-02 | Release date: | 2024-05-08 | Method: | ELECTRON MICROSCOPY (2.87 Å) | Cite: | Human 3-methylcrotonyl-CoA carboxylase in BCS-mcoa state To Be Published
|
|
8J7D
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 8j7d by Molmil](/molmil-images/mine/8j7d) | Human 3-methylcrotonyl-CoA carboxylase in BCCP-H1 state | Descriptor: | 5-(HEXAHYDRO-2-OXO-1H-THIENO[3,4-D]IMIDAZOL-6-YL)PENTANAL, Methylcrotonoyl-CoA carboxylase beta chain, mitochondrial, ... | Authors: | Liu, D.S, Su, J.Y. | Deposit date: | 2023-04-27 | Release date: | 2024-05-08 | Method: | ELECTRON MICROSCOPY (2.7 Å) | Cite: | Human 3-methylcrotonyl-CoA carboxylase in BCCP-H1 state To Be Published
|
|
8JAK
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 8jak by Molmil](/molmil-images/mine/8jak) | Human MCC in MCCU state | Descriptor: | 5-(HEXAHYDRO-2-OXO-1H-THIENO[3,4-D]IMIDAZOL-6-YL)PENTANAL, Methylcrotonoyl-CoA carboxylase beta chain, mitochondrial, ... | Authors: | Liu, D.S, Su, J.Y, Tian, X.Y. | Deposit date: | 2023-05-06 | Release date: | 2024-05-15 | Method: | ELECTRON MICROSCOPY (2.52 Å) | Cite: | Human MCC in BCCP-BCS state To Be Published
|
|
8JAW
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 8jaw by Molmil](/molmil-images/mine/8jaw) | Human MCC in MCCD state | Descriptor: | 5-(HEXAHYDRO-2-OXO-1H-THIENO[3,4-D]IMIDAZOL-6-YL)PENTANAL, Methylcrotonoyl-CoA carboxylase beta chain, mitochondrial, ... | Authors: | Liu, D.S, Su, J.Y, Tian, X.Y. | Deposit date: | 2023-05-07 | Release date: | 2024-05-15 | Method: | ELECTRON MICROSCOPY (2.51 Å) | Cite: | Human MCC in BCCP-CTS state To Be Published
|
|
2QF7
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2qf7 by Molmil](/molmil-images/mine/2qf7) | Crystal structure of a complete multifunctional pyruvate carboxylase from Rhizobium etli | Descriptor: | CHLORIDE ION, COENZYME A, FORMIC ACID, ... | Authors: | St Maurice, M, Surinya, K.H, Rayment, I. | Deposit date: | 2007-06-27 | Release date: | 2007-09-04 | Last modified: | 2012-02-15 | Method: | X-RAY DIFFRACTION (2 Å) | Cite: | Domain architecture of pyruvate carboxylase, a biotin-dependent multifunctional enzyme Science, 317, 2007
|
|
2W6O
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2w6o by Molmil](/molmil-images/mine/2w6o) | Crystal structure of Biotin carboxylase from E. coli in complex with 4-Amino-7,7-dimethyl-7,8-dihydro-quinazolinone fragment | Descriptor: | 4-amino-7,7-dimethyl-7,8-dihydroquinazolin-5(6H)-one, BIOTIN CARBOXYLASE, CHLORIDE ION | Authors: | Mochalkin, I, Miller, J.R. | Deposit date: | 2008-12-18 | Release date: | 2009-05-19 | Last modified: | 2023-12-13 | Method: | X-RAY DIFFRACTION (2.5 Å) | Cite: | Discovery of Antibacterial Biotin Carboxylase Inhibitors by Virtual Screening and Fragment-Based Approaches. Acs Chem.Biol., 4, 2009
|
|
2W70
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2w70 by Molmil](/molmil-images/mine/2w70) | |
2W6Q
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2w6q by Molmil](/molmil-images/mine/2w6q) | Crystal structure of Biotin carboxylase from E. coli in complex with the triazine-2,4-diamine fragment | Descriptor: | 6-(2-phenoxyethoxy)-1,3,5-triazine-2,4-diamine, BIOTIN CARBOXYLASE, CHLORIDE ION | Authors: | Mochalkin, I, Miller, J.R. | Deposit date: | 2008-12-18 | Release date: | 2009-05-19 | Last modified: | 2023-12-13 | Method: | X-RAY DIFFRACTION (2.05 Å) | Cite: | Discovery of Antibacterial Biotin Carboxylase Inhibitors by Virtual Screening and Fragment-Based Approaches. Acs Chem.Biol., 4, 2009
|
|
2W71
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2w71 by Molmil](/molmil-images/mine/2w71) | |
2W6Z
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2w6z by Molmil](/molmil-images/mine/2w6z) | |
2VQD
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2vqd by Molmil](/molmil-images/mine/2vqd) | |
2W6P
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2w6p by Molmil](/molmil-images/mine/2w6p) | |
2W6M
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2w6m by Molmil](/molmil-images/mine/2w6m) | |
2V59
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2v59 by Molmil](/molmil-images/mine/2v59) | |
2V58
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2v58 by Molmil](/molmil-images/mine/2v58) | CRYSTAL STRUCTURE OF BIOTIN CARBOXYLASE FROM E.COLI IN COMPLEX WITH POTENT INHIBITOR 1 | Descriptor: | 6-(2,6-dibromophenyl)pyrido[2,3-d]pyrimidine-2,7-diamine, BIOTIN CARBOXYLASE, CHLORIDE ION | Authors: | Mochalkin, I, Miller, J.R. | Deposit date: | 2008-10-02 | Release date: | 2009-01-13 | Last modified: | 2023-12-13 | Method: | X-RAY DIFFRACTION (2.1 Å) | Cite: | A Class of Selective Antibacterials Derived from a Protein Kinase Inhibitor Pharmacophore. Proc.Natl.Acad.Sci.USA, 106, 2009
|
|
2W6N
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2w6n by Molmil](/molmil-images/mine/2w6n) | |
2VPQ
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2vpq by Molmil](/molmil-images/mine/2vpq) | |