5WC7
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![BU of 5wc7 by Molmil](/molmil-images/mine/5wc7) | CypA Mutant - I97V S99T C115S | 分子名称: | Peptidyl-prolyl cis-trans isomerase A | 著者 | Fraser, J.S. | 登録日 | 2017-06-29 | 公開日 | 2018-04-18 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.43 Å) | 主引用文献 | Rescue of conformational dynamics in enzyme catalysis by directed evolution. Nat Commun, 9, 2018
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3CYS
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![BU of 3cys by Molmil](/molmil-images/mine/3cys) | DETERMINATION OF THE NMR SOLUTION STRUCTURE OF THE CYCLOPHILIN A-CYCLOSPORIN A COMPLEX | 分子名称: | CYCLOSPORIN A, PEPTIDYL-PROLYL CIS-TRANS ISOMERASE A | 著者 | Spitzfaden, C, Braun, W, Wider, G, Widmer, H, Wuthrich, K. | 登録日 | 1994-02-28 | 公開日 | 1994-08-31 | 最終更新日 | 2017-11-01 | 実験手法 | SOLUTION NMR | 主引用文献 | Determination of the NMR Solution Structure of the Cyclophilin A-Cyclosporin a Complex. J.Biomol.NMR, 4, 1994
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2FU0
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![BU of 2fu0 by Molmil](/molmil-images/mine/2fu0) | Plasmodium falciparum cyclophilin PFE0505w putative cyclosporin-binding domain | 分子名称: | cyclophilin, putative | 著者 | Dong, A, Lew, J, Sundararajan, E, Zhao, Y, Wasney, G, Vedadi, M, Koeieradzki, I, Edwards, A.M, Arrowsmith, C.H, Weigelt, J, Sundstrom, M, Bochkarev, A, Hui, R, Hills, T, Structural Genomics Consortium (SGC) | 登録日 | 2006-01-25 | 公開日 | 2006-02-07 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Genome-scale protein expression and structural biology of Plasmodium falciparum and related Apicomplexan organisms. Mol.Biochem.Parasitol., 151, 2007
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2R99
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![BU of 2r99 by Molmil](/molmil-images/mine/2r99) | Crystal structure of cyclophilin ABH-like domain of human peptidylprolyl isomerase E isoform 1 | 分子名称: | Peptidyl-prolyl cis-trans isomerase E | 著者 | Walker, J.R, Davis, T, Newman, E.M, Mackenzie, F, Sundstrom, M, Arrowsmith, C.H, Edwards, A.M, Bochkarev, A, Dhe-Paganon, S, Structural Genomics Consortium (SGC) | 登録日 | 2007-09-12 | 公開日 | 2007-09-25 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.61 Å) | 主引用文献 | Structural and biochemical characterization of the human cyclophilin family of peptidyl-prolyl isomerases. PLoS Biol., 8, 2010
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5LUD
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![BU of 5lud by Molmil](/molmil-images/mine/5lud) | Structure of Cyclophilin A in complex with 2,3-Diaminopyridine | 分子名称: | Peptidyl-prolyl cis-trans isomerase, pyridine-2,3-diamine | 著者 | McNae, I.W, Nowicki, M.W, Blackburn, E.A, Wear, M.A, Walkinshaw, M.D. | 登録日 | 2016-09-08 | 公開日 | 2017-04-05 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.25 Å) | 主引用文献 | Thermo-kinetic analysis space expansion for cyclophilin-ligand interactions - identification of a new nonpeptide inhibitor using BiacoreTM T200. FEBS Open Bio, 7, 2017
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6U5C
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![BU of 6u5c by Molmil](/molmil-images/mine/6u5c) | |
8EJX
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![BU of 8ejx by Molmil](/molmil-images/mine/8ejx) | |
3EOV
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![BU of 3eov by Molmil](/molmil-images/mine/3eov) | Crystal structure of cyclophilin from Leishmania donovani ligated with cyclosporin A | 分子名称: | CYCLOSPORIN A, PEPTIDYL-PROLYL CIS-TRANS ISOMERASE | 著者 | Venugopal, V, Dasgupta, D, Datta, A.K, Banerjee, R. | 登録日 | 2008-09-29 | 公開日 | 2008-11-11 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Structure of Cyclophilin from Leishmania Donovani Bound to Cyclosporin at 2.6 A Resolution: Correlation between Structure and Thermodynamic Data. Acta Crystallogr.,Sect.D, 65, 2009
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5T9W
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![BU of 5t9w by Molmil](/molmil-images/mine/5t9w) | Discovery of a Potent Cyclophilin Inhibitor (Compound 5) based on Structural Simplification of Sanglifehrin A | 分子名称: | 3-[(3-hydroxyphenyl)methyl]-6-(propan-2-yl)-19-oxa-1,4,7,25-tetraazabicyclo[19.3.1]pentacosa-13,15-diene-2,5,8,20-tetrone, Peptidyl-prolyl cis-trans isomerase A | 著者 | Appleby, T.C, Steadman, V, Pettit, P, Schmitz, U, Mackman, R.L, Schultz, B. | 登録日 | 2016-09-09 | 公開日 | 2017-01-25 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Discovery of Potent Cyclophilin Inhibitors Based on the Structural Simplification of Sanglifehrin A. J. Med. Chem., 60, 2017
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1J2A
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![BU of 1j2a by Molmil](/molmil-images/mine/1j2a) | Structure of E. coli cyclophilin B K163T mutant | 分子名称: | cyclophilin B | 著者 | Konno, M, Sano, Y, Okudaira, K, Kawaguchi, Y, Yamagishi-Ohmori, Y, Fushinobu, S, Matsuzawa, H. | 登録日 | 2002-12-26 | 公開日 | 2004-02-10 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Escherichia coli cyclophilin B binds a highly distorted form of trans-prolyl peptide isomer Eur.J.Biochem., 271, 2004
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1IIP
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![BU of 1iip by Molmil](/molmil-images/mine/1iip) | Bovine Cyclophilin 40, Tetragonal Form | 分子名称: | Cyclophilin 40, GLYCEROL | 著者 | Taylor, P, Dornan, J, Carrello, A, Minchin, R.F, Ratajczak, T, Walkinshaw, M.D. | 登録日 | 2001-04-24 | 公開日 | 2001-05-16 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Two structures of cyclophilin 40: folding and fidelity in the TPR domains. Structure, 9, 2001
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7ZFM
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![BU of 7zfm by Molmil](/molmil-images/mine/7zfm) | Engineered Protein Targeting the Zika Viral Envelope Fusion Loop | 分子名称: | 1,2-ETHANEDIOL, ACETIC ACID, HEXAETHYLENE GLYCOL, ... | 著者 | Athayde, D, Archer, M, Viana, I.F.T, Adan, W.C.S, Xavier, L.S.S, Lins, R.D. | 登録日 | 2022-04-01 | 公開日 | 2022-08-17 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.711 Å) | 主引用文献 | In Vitro Neutralisation of Zika Virus by an Engineered Protein Targeting the Viral Envelope Fusion Loop SSRN, 2022
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7ZDN
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![BU of 7zdn by Molmil](/molmil-images/mine/7zdn) | Human Cyclophilin D in complex with fragment | 分子名称: | (1~{R},9~{R},10~{S})-12-oxa-8-azatricyclo[7.3.1.0^{2,7}]trideca-2(7),3,5-trien-10-ol, Peptidyl-prolyl cis-trans isomerase F, mitochondrial | 著者 | Silva, D.O, Graedler, U, Bandeiras, T.M. | 登録日 | 2022-03-29 | 公開日 | 2023-04-19 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Human Cyclophilin D in complex with fragment To Be Published
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6BTA
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![BU of 6bta by Molmil](/molmil-images/mine/6bta) | CypA Mutant - S99T C115S | 分子名称: | Peptidyl-prolyl cis-trans isomerase A | 著者 | Fraser, J.S, Kenner, L.R, Liu, L. | 登録日 | 2017-12-06 | 公開日 | 2018-04-18 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Rescue of conformational dynamics in enzyme catalysis by directed evolution. Nat Commun, 9, 2018
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7PCJ
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![BU of 7pcj by Molmil](/molmil-images/mine/7pcj) | X-ray structure of CypA-C52AK125C/CsA/aromatic foldamer complex | 分子名称: | 8-azanyl-4-(2-methylpropoxy)quinoline-2-carboxylic acid, 8-azanyl-4-(3-azanylpropoxy)quinoline-2-carboxylic acid, 8-azanyl-4-oxidanyl-quinoline-2-carboxylic acid, ... | 著者 | Vallade, M, Langlois d'Estaintot, B, Fischer, L, Buratto, J, Savko, M, Huc, I. | 登録日 | 2021-08-03 | 公開日 | 2022-07-13 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.91 Å) | 主引用文献 | X-ray structure of a cystein mutant of Cyclophilin A tethered to an aromatic oligoamide foldamer complexed with Cyclosporin A To Be Published
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7N3J
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7PMT
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![BU of 7pmt by Molmil](/molmil-images/mine/7pmt) | Human Cyclophilin D in complex with N-[(5-ethyl-4-oxo-1,2,3,4,5,6- hexahydro-1,5-benzodiazocin-8-yl)methyl]-7-methyl-2-oxo-1H,2H-pyrazolo[1,5-a]pyrimidine-6-carboxamide | 分子名称: | DIMETHYL SULFOXIDE, Peptidyl-prolyl cis-trans isomerase F, mitochondrial, ... | 著者 | Silva, D.O, Graedler, U, Bandeiras, T.M. | 登録日 | 2021-09-02 | 公開日 | 2022-09-14 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (0.98 Å) | 主引用文献 | Human Cyclophilin D in complex with N-[(4-aminophenyl)methyl]-7-methyl-2-oxo-1H,2H-pyrazolo[1,5-a]pyrimidine-6-carboxamide To Be Published
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7L6Y
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7L6Z
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![BU of 7l6z by Molmil](/molmil-images/mine/7l6z) | Crystal Structure of Peptidyl-Prolyl Cis-Trans Isomerasefrom (PpiB) Streptococcus pneumoniae R6 | 分子名称: | 1,2-ETHANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CHLORIDE ION, ... | 著者 | Minasov, G, Shuvalova, L, Kiryukhina, O, Dubrovska, I, Satchell, K.J.F, Center for Structural Genomics of Infectious Diseases (CSGID) | 登録日 | 2020-12-24 | 公開日 | 2021-12-01 | 実験手法 | X-RAY DIFFRACTION (1.88 Å) | 主引用文献 | Crystal Structure of Peptidyl-Prolyl Cis-Trans Isomerasefrom (PpiB) Streptococcus pneumoniae R6 To Be Published
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7OGI
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![BU of 7ogi by Molmil](/molmil-images/mine/7ogi) | Human Cyclophilin D in complex with N-(5-ethyl-4-oxo-1,2,3,4,5,6-hexahydro-1,5-benzodiazocin-8-yl)-7methyl-2-oxo-1H,2H-pyrazolo[1,5-a]pyrimidine-6-carboxamide | 分子名称: | DIMETHYL SULFOXIDE, N-(5-ethyl-4-oxidanylidene-1,2,3,6-tetrahydro-1,5-benzodiazocin-8-yl)-7-methyl-2-oxidanylidene-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide, Peptidyl-prolyl cis-trans isomerase F, ... | 著者 | Silva, D.O, Graedler, U, Bandeiras, T.M. | 登録日 | 2021-05-06 | 公開日 | 2022-06-01 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.01 Å) | 主引用文献 | Human Cyclophilin D in complex with N-(5-ethyl-4-oxo-1,2,3,4,5,6-hexahydro-1,5-benzodiazocin-8-yl)-7methyl-2-oxo-1H,2H-pyrazolo[1,5-a]pyrimidine-6-carboxamide To Be Published
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7Q6P
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6FK1
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![BU of 6fk1 by Molmil](/molmil-images/mine/6fk1) | Cyclophilin A | 分子名称: | 1,2-ETHANEDIOL, Peptidyl-prolyl cis-trans isomerase A | 著者 | Lisboa, J, dos Santos, N.M.S. | 登録日 | 2018-01-23 | 公開日 | 2019-02-06 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.299 Å) | 主引用文献 | Production, crystallization and structure determination of cyclophilin A from Mus musculus To Be Published
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3O7T
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![BU of 3o7t by Molmil](/molmil-images/mine/3o7t) | Crystal Structure of Cyclophilin A from Moniliophthora perniciosa | 分子名称: | Cyclophilin A | 著者 | Monzani, P.S, Pereira, H.M, Gramacho, K.P, Meirelles, F.V, Oliva, G, Cascardo, J.C.M. | 登録日 | 2010-07-31 | 公開日 | 2011-08-10 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Crystal Structures of apo-cyclophilin and bounded cyclosporine A from Moniliophthora perniciosa To be Published
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3ODL
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![BU of 3odl by Molmil](/molmil-images/mine/3odl) | Crystal structure of cyclophilin A in complex with Voclosporin Z-ISA247 | 分子名称: | Cyclophilin A, Voclosporin | 著者 | Kuglstatter, A, Stihle, M, Benz, J, Hennig, M. | 登録日 | 2010-08-11 | 公開日 | 2011-02-16 | 最終更新日 | 2023-12-06 | 実験手法 | X-RAY DIFFRACTION (2.31 Å) | 主引用文献 | Structural basis for the cyclophilin A binding affinity and immunosuppressive potency of E-ISA247 (voclosporin). Acta Crystallogr.,Sect.D, 67, 2011
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8B58
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![BU of 8b58 by Molmil](/molmil-images/mine/8b58) | |