Loading
PDBj
メニューPDBj@FacebookPDBj@X(formerly Twitter)PDBj@BlueSkyPDBj@YouTubewwPDB FoundationwwPDBDonate
RCSB PDBPDBeBMRBAdv. SearchSearch help

8REF
DownloadVisualize
BU of 8ref by Molmil
Crystal structure of HLA B*13:01 in complex with SVLNDILARL, an 10-mer epitope from SARS-CoV-2 Spike (S975-984)
分子名称: 1,2-ETHANEDIOL, Beta-2-microglobulin, DI(HYDROXYETHYL)ETHER, ...
著者Ahn, Y.M, Maddumage, J.C, Szeto, C, Gras, S.
登録日2023-12-11
公開日2024-05-15
最終更新日2024-11-20
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献The impact of SARS-CoV-2 spike mutation on peptide presentation is HLA allomorph-specific.
Curr Res Struct Biol, 7, 2024
7QSX
DownloadVisualize
BU of 7qsx by Molmil
Non-obligately L8S8-complex forming RubisCO derived from ancestral sequence reconstruction and rational engineering in L8 complex
分子名称: 2-CARBOXYARABINITOL-1,5-DIPHOSPHATE, MAGNESIUM ION, RubisCO large subunit
著者Zarzycki, J, Schulz, L, Erb, T.J, Hochberg, G.K.A.
登録日2022-01-14
公開日2022-10-12
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Evolution of increased complexity and specificity at the dawn of form I Rubiscos.
Science, 378, 2022
8JNK
DownloadVisualize
BU of 8jnk by Molmil
Crystal structure of human ALKBH3 bound to ssDNA through active site crosslink
分子名称: Alpha-ketoglutarate-dependent dioxygenase alkB homolog 3, DNA, MANGANESE (II) ION, ...
著者Zhang, L.
登録日2023-06-06
公開日2024-01-24
最終更新日2024-11-13
実験手法X-RAY DIFFRACTION (2.69 Å)
主引用文献The Molecular Basis of Human ALKBH3 Mediated RNA N 1 -methyladenosine (m 1 A) Demethylation.
Angew.Chem.Int.Ed.Engl., 63, 2024
7MYR
DownloadVisualize
BU of 7myr by Molmil
BACE-1 in complex with compound #18
分子名称: (4aR,7aR)-6-(5-fluoropyrimidin-2-yl)-7a-(1,2-thiazol-5-yl)-4,4a,5,6,7,7a-hexahydropyrrolo[3,4-d][1,3]thiazin-2-amine, Beta-secretase 1, GLYCEROL, ...
著者Hendle, J, Timm, D.E, Stout, S.L.
登録日2021-05-21
公開日2021-07-14
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (1.72 Å)
主引用文献Discovery and Early Clinical Development of LY3202626, a Low-Dose, CNS-Penetrant BACE Inhibitor.
J.Med.Chem., 64, 2021
7CNY
DownloadVisualize
BU of 7cny by Molmil
Crystal structure of 8PE bound PSD from E. coli (2.12 A)
分子名称: 1,2-Dioctanoyl-SN-Glycero-3-Phosphoethanolamine, DODECYL-BETA-D-MALTOSIDE, Phosphatidylserine decarboxylase alpha chain, ...
著者Kim, J, Cho, G.
登録日2020-08-03
公開日2021-03-24
最終更新日2024-11-13
実験手法X-RAY DIFFRACTION (2.12 Å)
主引用文献Structural insights into phosphatidylethanolamine formation in bacterial membrane biogenesis.
Sci Rep, 11, 2021
7QSW
DownloadVisualize
BU of 7qsw by Molmil
L8S8-complex forming RubisCO derived from ancestral sequence reconstruction of the last common ancestor of SSU-bearing Form I RubisCOs
分子名称: 2-CARBOXYARABINITOL-1,5-DIPHOSPHATE, MAGNESIUM ION, RubisCO large subunit, ...
著者Zarzycki, J, Schulz, L, Erb, T.J, Hochberg, G.K.A.
登録日2022-01-14
公開日2022-10-12
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Evolution of increased complexity and specificity at the dawn of form I Rubiscos.
Science, 378, 2022
7QSV
DownloadVisualize
BU of 7qsv by Molmil
L8-complex forming RubisCO derived from ancestral sequence reconstruction of the last common ancestor of Form I'' and Form I RubisCOs
分子名称: 2-CARBOXYARABINITOL-1,5-DIPHOSPHATE, MAGNESIUM ION, RubisCO large subunit
著者Zarzycki, J, Schulz, L, Erb, T.J, Hochberg, G.K.A.
登録日2022-01-14
公開日2022-10-12
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Evolution of increased complexity and specificity at the dawn of form I Rubiscos.
Science, 378, 2022
8VFU
DownloadVisualize
BU of 8vfu by Molmil
The Fab Crystal Structure of the PAN IL-1 Family Inhibitor Antibody 3G5
分子名称: 3G5 Heavy Chain, 3G5 Light Chain
著者Fields, J.K, Sundberg, E.J.
登録日2023-12-22
公開日2024-02-21
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献Antibodies targeting the shared cytokine receptor IL-1 receptor accessory protein invoke distinct mechanisms to block all cytokine signaling.
Cell Rep, 43, 2024
1E5M
DownloadVisualize
BU of 1e5m by Molmil
Beta ketoacyl acyl carrier protein synthase II (KASII) from Synechocystis sp.
分子名称: BETA KETOACYL ACYL CARRIER PROTEIN SYNTHASE II
著者Moche, M, Edwards, P, Dehesh, K, Lindqvist, Y.
登録日2000-07-27
公開日2001-01-16
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.54 Å)
主引用文献The Crystal Structure of Beta-Ketoacyl-Acyl Carrier Protein Synthase II from Synechocystis Sp. At 1.54 A Resolution and its Relationship to Other Condensing Enzymes
J.Mol.Biol., 305, 2001
1EAJ
DownloadVisualize
BU of 1eaj by Molmil
DIMERIC STRUCTURE OF THE COXSACKIE VIRUS AND ADENOVIRUS RECEPTOR D1 DOMAIN AT 1.35 ANGSTROM RESOLUTION
分子名称: COXSACKIE VIRUS AND ADENOVIRUS RECEPTOR, SULFATE ION
著者van Raaij, M.J, Cusack, S.
登録日2001-07-12
公開日2001-07-13
最終更新日2024-10-09
実験手法X-RAY DIFFRACTION (1.35 Å)
主引用文献Dimeric structure of the coxsackievirus and adenovirus receptor D1 domain at 1.7 A resolution.
Structure, 8, 2000
9BZ7
DownloadVisualize
BU of 9bz7 by Molmil
Pannexin 1 lacking C-terminal activating domain
分子名称: Pannexin
著者Ehrlich, J.J, Kawate, T.
登録日2024-05-24
公開日2024-12-11
最終更新日2024-12-25
実験手法ELECTRON MICROSCOPY (2.9 Å)
主引用文献The C-terminal activating domain promotes pannexin 1 channel opening.
Proc.Natl.Acad.Sci.USA, 121, 2024
4XEB
DownloadVisualize
BU of 4xeb by Molmil
The structure of P. funicolosum Cel7A
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, CHLORIDE ION, Glucanase, ...
著者Alahuhta, P.M, Lunin, V.V.
登録日2014-12-23
公開日2016-06-22
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Engineering enhanced cellobiohydrolase activity
Nat Commun, 9(1), 2018
6CUM
DownloadVisualize
BU of 6cum by Molmil
Crystal structure of a C-terminal proteolytic fragment of a protein annotated as an LAO/AO transport system ATPase but likely MeaB and MMAA-like GTPase from Mycobacterium smegmatis
分子名称: 1,2-ETHANEDIOL, LAO/AO transport system ATPase
著者Seattle Structural Genomics Center for Infectious Disease (SSGCID)
登録日2018-03-26
公開日2018-04-11
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Ab initio structure solution of a proteolytic fragment using ARCIMBOLDO.
Acta Crystallogr F Struct Biol Commun, 74, 2018
1ELP
DownloadVisualize
BU of 1elp by Molmil
GAMMA-D CRYSTALLIN STRUCTURE AT 1.95 A RESOLUTION
分子名称: GAMMA-D CRYSTALLIN
著者Chirgadze, Yu.N, Driessen, H.P.C, Wright, G, Slingsby, C, Hay, R.E, Lindley, P.F.
登録日1995-12-20
公開日1996-06-10
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Structure of bovine eye lens gammaD (gammaIIIb)-crystallin at 1.95 A.
Acta Crystallogr.,Sect.D, 52, 1996
6VGI
DownloadVisualize
BU of 6vgi by Molmil
Crystal Structures of FLAP bound to MK-866
分子名称: 3-[3-(tert-butylsulfanyl)-1-[(4-chlorophenyl)methyl]-5-(propan-2-yl)-1H-indol-2-yl]-2,2-dimethylpropanoic acid, 5-lipoxygenase-activating protein, SULFATE ION
著者Ho, J.D, Lee, M.R, Rauch, C.T, Aznavour, K, Park, J.S, Luz, J.G, Antonysamy, S, Condon, B, Maletic, M, Zhang, A, Hickey, M.J, Hughes, N.E, Chandrasekhar, S, Sloan, A.V, Gooding, K, Harvey, A, Yu, X.P, Kahl, S.D, Norman, B.H.
登録日2020-01-08
公開日2020-12-02
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.61 Å)
主引用文献Structure-based, multi-targeted drug discovery approach to eicosanoid inhibition: Dual inhibitors of mPGES-1 and 5-lipoxygenase activating protein (FLAP).
Biochim Biophys Acta Gen Subj, 1865, 2020
5I0B
DownloadVisualize
BU of 5i0b by Molmil
Structure of PAK4
分子名称: 6-bromo-2-[1-methyl-3-(propan-2-yl)-1H-pyrazol-4-yl]-1H-imidazo[4,5-b]pyridine, Serine/threonine-protein kinase PAK 4
著者Park, S.Y.
登録日2016-02-03
公開日2016-12-14
最終更新日2024-10-23
実験手法X-RAY DIFFRACTION (3.09 Å)
主引用文献The discovery and the structural basis of an imidazo[4,5-b]pyridine-based p21-activated kinase 4 inhibitor
Bioorg. Med. Chem. Lett., 26, 2016
8E05
DownloadVisualize
BU of 8e05 by Molmil
Structure of dimeric LRRK1
分子名称: GUANOSINE-5'-DIPHOSPHATE, Leucine-rich repeat serine/threonine-protein kinase 1
著者Reimer, J.M, Lin, Y.X, Leschziner, A.E.
登録日2022-08-08
公開日2023-08-30
最終更新日2025-05-28
実験手法ELECTRON MICROSCOPY (4.6 Å)
主引用文献Structure of LRRK1 and mechanisms of autoinhibition and activation.
Nat.Struct.Mol.Biol., 30, 2023
8Q18
DownloadVisualize
BU of 8q18 by Molmil
The Crystal Structure of Human Carbonic Anhydrase IX in Complex with Sulfonamide
分子名称: 1,1,3-tris(oxidanylidene)-2-(2-phenylethyl)-1,2-benzothiazole-6-sulfonamide, Carbonic anhydrase 9, GLYCEROL, ...
著者Leitans, J, Tars, K.
登録日2023-07-31
公開日2023-11-08
最終更新日2024-11-20
実験手法X-RAY DIFFRACTION (2.13 Å)
主引用文献Structural Basis of Saccharin Derivative Inhibition of Carbonic Anhydrase IX.
Chemmedchem, 18, 2023
5L6O
DownloadVisualize
BU of 5l6o by Molmil
EphB3 kinase domain covalently bound to an irreversible inhibitor (compound 3)
分子名称: 1,4-DIETHYLENE DIOXIDE, 1-(4-phenylazanylquinazolin-7-yl)ethanone, Ephrin type-B receptor 3
著者Schimpl, M, Overman, R, Kung, A, Chen, Y.-C, Ni, F, Zhu, J, Turner, M, Molina, H, Zhang, C.
登録日2016-05-30
公開日2016-08-10
最終更新日2024-11-13
実験手法X-RAY DIFFRACTION (1.88 Å)
主引用文献Development of Specific, Irreversible Inhibitors for a Receptor Tyrosine Kinase EphB3.
J.Am.Chem.Soc., 138, 2016
8Q1A
DownloadVisualize
BU of 8q1a by Molmil
The Crystal Structure of Human Carbonic Anhydrase IX in Complex with inhibitor
分子名称: 1,1,3-tris(oxidanylidene)-2-pentyl-1,2-benzothiazole-6-sulfonamide, Carbonic anhydrase 9, GLYCEROL, ...
著者Leitans, J, Tars, K.
登録日2023-07-31
公開日2023-11-08
最終更新日2024-11-06
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Structural Basis of Saccharin Derivative Inhibition of Carbonic Anhydrase IX.
Chemmedchem, 18, 2023
4TV1
DownloadVisualize
BU of 4tv1 by Molmil
Crystal structure of hERa-LBD (Y537S) in complex with propylparaben
分子名称: 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, Estrogen receptor, ...
著者Delfosse, V, Grimaldi, M, Bourguet, W.
登録日2014-06-25
公開日2015-01-28
最終更新日2024-10-23
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献A structural perspective on nuclear receptors as targets of environmental compounds.
Acta Pharmacol.Sin., 36, 2015
7NXG
DownloadVisualize
BU of 7nxg by Molmil
Wax synthase 1 from Acinetobacter baylyi (AbWSD1) co-crystallized with myristic acid
分子名称: MYRISTIC ACID, O-acyltransferase WSD
著者Vollheyde, K, Kuehnel, K, Lambrecht, F, Kawelke, S, Herrfurth, C, Feussner, I.
登録日2021-03-18
公開日2022-03-30
最終更新日2024-06-19
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Crystal Structure of the Bifunctional Wax Synthase 1 from Acinetobacter baylyi Suggests a Conformational Change upon Substrate Binding and Formation of Additional Substrate Binding Sites
Acs Catalysis, 12, 2022
7RQQ
DownloadVisualize
BU of 7rqq by Molmil
Structure of chimeric antibody F10heavy_L9light with PfCSP peptide NANPNVDP
分子名称: 1,2-ETHANEDIOL, F10 Heavy Chain, L9 Kappa Chain, ...
著者Hurlburt, N.K, Pancera, M.
登録日2021-08-06
公開日2022-03-02
最終更新日2024-10-30
実験手法X-RAY DIFFRACTION (1.89 Å)
主引用文献The light chain of the L9 antibody is critical for binding circumsporozoite protein minor repeats and preventing malaria.
Cell Rep, 38, 2022
1MHH
DownloadVisualize
BU of 1mhh by Molmil
Structure of P. magnus protein L mutant bound to a mouse Fab
分子名称: 1,2-ETHANEDIOL, Fab, heavy chain, ...
著者Graille, M, Stura, E.A.
登録日2002-08-20
公開日2003-01-14
最終更新日2025-03-26
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Evidence for plasticity and structural mimicry at the immunoglobulin light chain-protein L interface
J.Biol.Chem., 277, 2002
7NS5
DownloadVisualize
BU of 7ns5 by Molmil
Structure of yeast Fbp1 (Fructose-1,6-bisphosphatase 1)
分子名称: Fructose-1,6-bisphosphatase, MAGNESIUM ION, PHOSPHATE ION
著者Sherpa, D, Chrustowicz, J, Prabu, J.R, Schulman, B.A.
登録日2021-03-05
公開日2021-05-05
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献GID E3 ligase supramolecular chelate assembly configures multipronged ubiquitin targeting of an oligomeric metabolic enzyme.
Mol.Cell, 81, 2021

242842

件を2025-10-08に公開中

PDB statisticsPDBj update infoContact PDBjnumon