1DCY
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![BU of 1dcy by Molmil](/molmil-images/mine/1dcy) | |
1DB4
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![BU of 1db4 by Molmil](/molmil-images/mine/1db4) | HUMAN S-PLA2 IN COMPLEX WITH INDOLE 8 | 分子名称: | CALCIUM ION, PHOSPHOLIPASE A2, [3-(1-BENZYL-3-CARBAMOYLMETHYL-2-METHYL-1H-INDOL-5-YLOXY)-PROPYL-]-PHOSPHONIC ACID | 著者 | Chirgadze, N.Y, Schevitz, R.W, Wery, J.-P. | 登録日 | 1999-11-02 | 公開日 | 1999-11-12 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Structure-based design of the first potent and selective inhibitor of human non-pancreatic secretory phospholipase A2. Nat.Struct.Biol., 2, 1995
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1BBC
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![BU of 1bbc by Molmil](/molmil-images/mine/1bbc) | STRUCTURE OF RECOMBINANT HUMAN RHEUMATOID ARTHRITIC SYNOVIAL FLUID PHOSPHOLIPASE A2 AT 2.2 ANGSTROMS RESOLUTION | 分子名称: | PHOSPHOLIPASE A2 | 著者 | Wery, J.-P, Schevitz, R.W, Clawson, D.K, Bobbitt, J.L, Dow, E.R, Gamboa, G, Goodsonjunior, T, Hermann, R.B, Kramer, R.M, Mcclure, D.B, Mihelich, E.D, Putnam, J.E, Sharp, J.D, Stark, D.H, Teater, C, Warrick, M.W, Jones, N.D. | 登録日 | 1992-05-04 | 公開日 | 1993-10-31 | 最終更新日 | 2019-08-14 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Structure of recombinant human rheumatoid arthritic synovial fluid phospholipase A2 at 2.2 A resolution. Nature, 352, 1991
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1AE7
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![BU of 1ae7 by Molmil](/molmil-images/mine/1ae7) | NOTEXIN, A PRESYNAPTIC NEUROTOXIC PHOSPHOLIPASE A2 | 分子名称: | PHOSPHOLIPASE A2, SULFATE ION | 著者 | Westerlund, B, Nordlund, P, Uhlin, U, Eaker, D, Eklund, H. | 登録日 | 1997-03-06 | 公開日 | 1997-05-15 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | The three-dimensional structure of notexin, a presynaptic neurotoxic phospholipase A2 at 2.0 A resolution. FEBS Lett., 301, 1992
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1BK9
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![BU of 1bk9 by Molmil](/molmil-images/mine/1bk9) | PHOSPHOLIPASE A2 MODIFIED BY PBPB | 分子名称: | 1,4-BUTANEDIOL, CALCIUM ION, PHOSPHOLIPASE A2, ... | 著者 | Zhao, H, Tang, L, Wang, X, Lin, Z, Zhou, Y. | 登録日 | 1998-07-16 | 公開日 | 1999-03-02 | 最終更新日 | 2023-08-02 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structure of a snake venom phospholipase A2 modified by p-bromo-phenacyl-bromide. Toxicon, 36, 1998
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1J1A
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![BU of 1j1a by Molmil](/molmil-images/mine/1j1a) | PANCREATIC SECRETORY PHOSPHOLIPASE A2 (IIa) WITH ANTI-INFLAMMATORY ACTIVITY | 分子名称: | (S)-5-(4-BENZYLOXY-PHENYL)-4-(7-PHENYL-HEPTANOYLAMINO)-PENTANOIC ACID, CALCIUM ION, Phospholipase A2 | 著者 | Hansford, K.A, Reid, R.C, Clark, C.I, Tyndall, J.D.A, Whitehouse, M.W, Guthrie, T, McGeary, R.P, Schafer, K, Martin, J.L, Fairlie, D.P. | 登録日 | 2002-12-03 | 公開日 | 2003-03-18 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | D-Tyrosine as a Chiral Precusor to Potent Inhibitors of Human Nonpancreatic Secretory Phospholipase A2 (IIa) with Antiinflammatory Activity Chembiochem, 4, 2003
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1IJL
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![BU of 1ijl by Molmil](/molmil-images/mine/1ijl) | Crystal structure of acidic phospholipase A2 from deinagkistrodon acutus | 分子名称: | CALCIUM ION, PHOSPHOLIPASE A2, ZINC ION | 著者 | Gu, L, Zhang, H, Song, S, Zhou, Y, Lin, Z. | 登録日 | 2001-04-27 | 公開日 | 2001-12-28 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Structure of an acidic phospholipase A2 from the venom of Deinagkistrodon acutus. Acta Crystallogr.,Sect.D, 58, 2002
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1IRB
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![BU of 1irb by Molmil](/molmil-images/mine/1irb) | CARBOXYLIC ESTER HYDROLASE | 分子名称: | CALCIUM ION, PHOSPHOLIPASE A2 | 著者 | Sundaralingam, M. | 登録日 | 1997-08-13 | 公開日 | 1997-12-24 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Phospholipase A2 engineering. Deletion of the C-terminus segment changes substrate specificity and uncouples calcium and substrate binding at the zwitterionic interface. Biochemistry, 35, 1996
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1JIA
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![BU of 1jia by Molmil](/molmil-images/mine/1jia) | |
1JLT
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![BU of 1jlt by Molmil](/molmil-images/mine/1jlt) | Vipoxin Complex | 分子名称: | (4R)-2-METHYLPENTANE-2,4-DIOL, (4S)-2-METHYL-2,4-PENTANEDIOL, PHOSPHOLIPASE A2, ... | 著者 | Banumathi, S, Rajashankar, K.R, Notzel, C, Aleksiev, B, Singh, T.P, Genov, N, Betzel, C. | 登録日 | 2001-07-16 | 公開日 | 2001-10-31 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | Structure of the neurotoxic complex vipoxin at 1.4 A resolution. Acta Crystallogr.,Sect.D, 57, 2001
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1JQ8
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![BU of 1jq8 by Molmil](/molmil-images/mine/1jq8) | Design of specific inhibitors of phospholipase A2: Crystal structure of a complex formed between phospholipase A2 from Daboia russelli pulchella and a designed pentapeptide Leu-Ala-Ile-Tyr-Ser at 2.0 resolution | 分子名称: | ACETIC ACID, Peptide inhibitor, Phospholipase A2, ... | 著者 | Chandra, V, Jasti, J, Kaur, P, Dey, S, Betzel, C, Singh, T.P. | 登録日 | 2001-08-04 | 公開日 | 2002-11-06 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Design of specific peptide inhibitors of phospholipase A2: structure of a complex formed between Russell's viper phospholipase A2 and a designed peptide Leu-Ala-Ile-Tyr-Ser (LAIYS). ACTA CRYSTALLOGR.,SECT.D, 58, 2002
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1KPM
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![BU of 1kpm by Molmil](/molmil-images/mine/1kpm) | First Structural Evidence of a Specific Inhibition of Phospholipase A2 by Vitamin E and its Implications in Inflammation: Crystal Structure of the Complex Formed between Phospholipase A2 and Vitamin E at 1.8 A Resolution. | 分子名称: | ACETIC ACID, Phospholipase A2, VITAMIN E | 著者 | Chandra, V, Jasti, J, Kaur, P, Betzel, C, Srinivasan, A, Singh, T.P. | 登録日 | 2002-01-01 | 公開日 | 2002-07-10 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | First Structural Evidence of a Specific Inhibition of Phospholipase A2 by alpha-Tocopherol (Vitamin E) and its
Implications in Inflammation: Crystal Structure of the Complex Formed Between Phospholipase A2 and
alpha-Tocopherol at 1.8 A Resolution J.Mol.Biol., 320, 2002
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1KVW
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![BU of 1kvw by Molmil](/molmil-images/mine/1kvw) | |
1KVO
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![BU of 1kvo by Molmil](/molmil-images/mine/1kvo) | |
1KVX
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![BU of 1kvx by Molmil](/molmil-images/mine/1kvx) | |
1L8S
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![BU of 1l8s by Molmil](/molmil-images/mine/1l8s) | |
1KQU
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![BU of 1kqu by Molmil](/molmil-images/mine/1kqu) | Human phospholipase A2 complexed with a substrate anologue | 分子名称: | 6-PHENYL-4(R)-(7-PHENYL-HEPTANOYLAMINO)-HEXANOIC ACID, CALCIUM ION, Phospholipase A2, ... | 著者 | Tyndall, J.D, Martin, J.L. | 登録日 | 2002-01-07 | 公開日 | 2003-11-11 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | D-Tyrosine as a chiral precusor to potent inhibitors of human nonpancreatic secretory phospholipase A2 (IIa) with antiinflammatory activity. Chembiochem, 4, 2003
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2OSN
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![BU of 2osn by Molmil](/molmil-images/mine/2osn) | |
2OTH
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![BU of 2oth by Molmil](/molmil-images/mine/2oth) | Crystal structure of a ternary complex of phospholipase A2 with indomethacin and nimesulide at 2.9 A resolution | 分子名称: | 4-NITRO-2-PHENOXYMETHANESULFONANILIDE, ACETONITRILE, INDOMETHACIN, ... | 著者 | Kumar, S, Singh, N, Sharma, S, Kaur, P, Singh, T.P. | 登録日 | 2007-02-08 | 公開日 | 2007-02-27 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Crystal structure of a ternary complex of phospholipase A2 with indomethacin and nimesulide at 2.9 A resolution To be Published
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2PB8
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![BU of 2pb8 by Molmil](/molmil-images/mine/2pb8) | Crystal structure of the complex formed between phospholipase A2 and peptide Ala-Val-Tyr-Ser at 2.0 A resolution | 分子名称: | ACETATE ION, AVYS, Phospholipase A2 VRV-PL-VIIIa | 著者 | Kumar, S, Singh, N, Sharma, S, Kaur, P, Singh, T.P. | 登録日 | 2007-03-28 | 公開日 | 2007-04-17 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Crystal structure of the complex formed between phospholipase A2 and peptide Ala-Val-Tyr-Ser at 2.0 A resolution To be Published
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2OQD
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![BU of 2oqd by Molmil](/molmil-images/mine/2oqd) | Crystal Structure of BthTX-II | 分子名称: | Phospholipase A2 | 著者 | Correa, L.C, Marchi-Salvador, D.P, Cintra, A.C.O, Soares, A.M, Fontes, M.R.M. | 登録日 | 2007-01-31 | 公開日 | 2008-02-12 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.19 Å) | 主引用文献 | Crystal structure of a myotoxic Asp49-phospholipase A(2) with low catalytic activity: Insights into Ca(2+)-independent catalytic mechanism. Biochim.Biophys.Acta, 1784, 2008
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2OUB
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![BU of 2oub by Molmil](/molmil-images/mine/2oub) | Crystal structure of the complex formed between phospholipase A2 and atenolol at 2.75 A resolution | 分子名称: | 2-(4-(2-HYDROXY-3-(ISOPROPYLAMINO)PROPOXY)PHENYL)ETHANAMIDE, Phospholipase A2 VRV-PL-VIIIa | 著者 | Kumar, S, Singh, N, Sharma, S, Kaur, P, Singh, T.P. | 登録日 | 2007-02-10 | 公開日 | 2007-02-27 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.75 Å) | 主引用文献 | Crystal structure of the complex formed between phospholipase A2 and atenolol at 2.75 A resolution To be Published
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1LE6
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![BU of 1le6 by Molmil](/molmil-images/mine/1le6) | CARBOXYLIC ESTER HYDROLASE, P 1 21 1 SPACE GROUP | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, CALCIUM ION, Group X Secretory Phospholipase A2 | 著者 | Pan, Y.H, Jain, M.K, Bahnson, B.J. | 登録日 | 2002-04-09 | 公開日 | 2002-08-14 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (1.97 Å) | 主引用文献 | Crystal structure of human group X secreted phospholipase A2. Electrostatically neutral interfacial surface targets zwitterionic membranes. J.Biol.Chem., 277, 2002
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2O1N
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![BU of 2o1n by Molmil](/molmil-images/mine/2o1n) | Crystal structure of a complex of phospholipase A2 with a peptide Ala-Ile-Ala-Ser at 2.8 A resolution | 分子名称: | Ala-Ile-Ala-Ser peptide, Phospholipase A2 VRV-PL-VIIIa | 著者 | Kumar, S, Singh, N, Sharma, S, Kaur, P, Singh, T.P. | 登録日 | 2006-11-29 | 公開日 | 2006-12-19 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Crystal structure of a complex of phospholipase A2 with a peptide Ala-Ile-Ala-Ser at 2.8 A resolution To be Published
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2OK9
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![BU of 2ok9 by Molmil](/molmil-images/mine/2ok9) | PrTX-I-BPB | 分子名称: | ISOPROPYL ALCOHOL, Phospholipase A2 homolog 1, p-Bromophenacyl bromide | 著者 | Marchi-Salvador, D.P, Fernandes, C.A.H, Soares, A.M, Fontes, M.R. | 登録日 | 2007-01-16 | 公開日 | 2008-09-23 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.34 Å) | 主引用文献 | Crystal structure of a phospholipase A(2) homolog complexed with p-bromophenacyl bromide reveals important structural changes associated with the inhibition of myotoxic activity. Biochim.Biophys.Acta, 1794, 2009
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