6ZEJ
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![BU of 6zej by Molmil](/molmil-images/mine/6zej) | Structure of PP1-Phactr1 chimera [PP1(7-304) + linker (SGSGS) + Phactr1(526-580)] | 分子名称: | 1,2-ETHANEDIOL, GLYCEROL, MANGANESE (II) ION, ... | 著者 | Mouilleron, S, Treisman, R, Fedoryshchak, R, Lee, R, Butler, A.M, Prechova, M. | 登録日 | 2020-06-16 | 公開日 | 2020-09-30 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.78 Å) | 主引用文献 | Molecular basis for substrate specificity of the Phactr1/PP1 phosphatase holoenzyme. Elife, 9, 2020
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6ZEI
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![BU of 6zei by Molmil](/molmil-images/mine/6zei) | Structure of PP1-IRSp53 S455E chimera [PP1(7-304) + linker (G/S)x9 + IRSp53(449-465)] bound to Phactr1 (516-580) | 分子名称: | GLYCEROL, MANGANESE (II) ION, PHOSPHATE ION, ... | 著者 | Mouilleron, S, Treisman, R, Fedoryshchak, R, Lee, R, Butler, A.M, Prechova, M. | 登録日 | 2020-06-16 | 公開日 | 2020-09-30 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.39 Å) | 主引用文献 | Molecular basis for substrate specificity of the Phactr1/PP1 phosphatase holoenzyme. Elife, 9, 2020
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6ZEH
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![BU of 6zeh by Molmil](/molmil-images/mine/6zeh) | Structure of PP1-spectrin alpha II chimera [PP1(7-304) + linker (G/S)x9 + spectrin alpha II (1025-1039)] bound to Phactr1 (516-580) | 分子名称: | MANGANESE (II) ION, PHOSPHATE ION, Phosphatase and actin regulator, ... | 著者 | Mouilleron, S, Treisman, R, Fedoryshchak, R, Lee, R, Butler, A.M, Prechova, M. | 登録日 | 2020-06-16 | 公開日 | 2020-09-30 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | Molecular basis for substrate specificity of the Phactr1/PP1 phosphatase holoenzyme. Elife, 9, 2020
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6Z9D
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6ZEE
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![BU of 6zee by Molmil](/molmil-images/mine/6zee) | Structure of PP1(7-300) bound to Phactr1 (507-580) at pH8.4 | 分子名称: | 1,2-ETHANEDIOL, 3,6,9,12,15,18-HEXAOXAICOSANE, GLYCEROL, ... | 著者 | Mouilleron, S, Treisman, R, Fedoryshchak, R, Lee, R, Butler, A.M, Prechova, M. | 登録日 | 2020-06-16 | 公開日 | 2020-09-30 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Molecular basis for substrate specificity of the Phactr1/PP1 phosphatase holoenzyme. Elife, 9, 2020
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6ZEG
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![BU of 6zeg by Molmil](/molmil-images/mine/6zeg) | Structure of PP1-IRSp53 chimera [PP1(7-304) + linker (G/S)x9 + IRSp53(449-465)] bound to Phactr1 (516-580) | 分子名称: | 1,2-ETHANEDIOL, 3,6,9,12,15,18-HEXAOXAICOSANE, MANGANESE (II) ION, ... | 著者 | Mouilleron, S, Treisman, R, Fedoryshchak, R, Lee, R, Butler, A.M, Prechova, M. | 登録日 | 2020-06-16 | 公開日 | 2020-09-30 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.09 Å) | 主引用文献 | Molecular basis for substrate specificity of the Phactr1/PP1 phosphatase holoenzyme. Elife, 9, 2020
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6ZK6
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![BU of 6zk6 by Molmil](/molmil-images/mine/6zk6) | Protein Phosphatase 1 (PP1) T320E mutant | 分子名称: | FE (III) ION, MANGANESE (II) ION, PHOSPHATE ION, ... | 著者 | Salvi, F, Barabas, O, Koehn, M. | 登録日 | 2020-06-29 | 公開日 | 2020-11-18 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Towards Dissecting the Mechanism of Protein Phosphatase-1 Inhibition by Its C-Terminal Phosphorylation. Chembiochem, 22, 2021
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1U32
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![BU of 1u32 by Molmil](/molmil-images/mine/1u32) | Crystal structure of a Protein Phosphatase-1: Calcineurin Hybrid Bound to Okadaic Acid | 分子名称: | BETA-MERCAPTOETHANOL, MANGANESE (II) ION, OKADAIC ACID, ... | 著者 | Maynes, J.T, Perreault, K.R, Cherney, M.M, Luu, H.A, James, M.N.G, Holmes, C.F.B. | 登録日 | 2004-07-20 | 公開日 | 2004-08-17 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Crystal Structure and Mutagenesis of a Protein Phosphatase-1:Calcineurin Hybrid Elucidate the Role of the {beta}12-{beta}13 Loop in Inhibitor Binding J.Biol.Chem., 279, 2004
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6XUE
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4JA9
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![BU of 4ja9 by Molmil](/molmil-images/mine/4ja9) | Rat PP5 apo | 分子名称: | MAGNESIUM ION, Serine/threonine-protein phosphatase 5 | 著者 | Haslbeck, V, Helmuth, M, Alte, F, Popowicz, G, Schmidt, W, Weiwad, M, Fischer, G, Gemmecker, G, Sattler, M, Striggow, F, Groll, M, Richter, K. | 登録日 | 2013-02-18 | 公開日 | 2014-02-19 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Selective activators of protein phosphatase 5 target the auto-inhibitory mechanism. Biosci.Rep., 35, 2015
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4KBP
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![BU of 4kbp by Molmil](/molmil-images/mine/4kbp) | KIDNEY BEAN PURPLE ACID PHOSPHATASE | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, FE (III) ION, PHOSPHATE ION, ... | 著者 | Klabunde, T, Strater, N, Krebs, B. | 登録日 | 1995-10-02 | 公開日 | 1996-12-07 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Mechanism of Fe(III)-Zn(II) purple acid phosphatase based on crystal structures. J.Mol.Biol., 259, 1996
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6XUG
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6XUQ
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6ZEF
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![BU of 6zef by Molmil](/molmil-images/mine/6zef) | Structure of PP1(7-300) bound to Phactr1 (516-580) at pH 5.25 | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, MANGANESE (II) ION, ... | 著者 | Mouilleron, S, Treisman, R, Fedoryshchak, R, Lee, R, Butler, A.M, Prechova, M. | 登録日 | 2020-06-16 | 公開日 | 2020-09-30 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.94 Å) | 主引用文献 | Molecular basis for substrate specificity of the Phactr1/PP1 phosphatase holoenzyme. Elife, 9, 2020
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1FJM
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![BU of 1fjm by Molmil](/molmil-images/mine/1fjm) | Protein serine/threonine phosphatase-1 (alpha isoform, type 1) complexed with microcystin-LR toxin | 分子名称: | BETA-MERCAPTOETHANOL, MANGANESE (II) ION, PROTEIN SERINE/THREONINE PHOSPHATASE-1 (ALPHA ISOFORM, ... | 著者 | Goldberg, J, Nairn, A.C, Kuriyan, J. | 登録日 | 1995-12-17 | 公開日 | 1996-06-20 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Three-dimensional structure of the catalytic subunit of protein serine/threonine phosphatase-1. Nature, 376, 1995
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1HO5
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1HPU
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![BU of 1hpu by Molmil](/molmil-images/mine/1hpu) | 5'-NUCLEOTIDASE (CLOSED FORM), COMPLEX WITH AMPCP | 分子名称: | 5'-NUCLEOTIDASE, MANGANESE (II) ION, PHOSPHOMETHYLPHOSPHONIC ACID ADENOSYL ESTER | 著者 | Knoefel, T, Straeter, N. | 登録日 | 2000-12-13 | 公開日 | 2002-03-20 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Mechanism of hydrolysis of phosphate esters by the dimetal center of 5'-nucleotidase based on crystal structures. J.Mol.Biol., 309, 2001
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1WAO
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![BU of 1wao by Molmil](/molmil-images/mine/1wao) | PP5 structure | 分子名称: | MANGANESE (II) ION, SERINE/THREONINE PROTEIN PHOSPHATASE 5 | 著者 | Barford, D. | 登録日 | 2004-10-27 | 公開日 | 2005-02-22 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Molecular Basis for Tpr Domain-Mediated Regulation of Protein Phosphatase 5 Embo J., 24, 2005
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7ZR1
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![BU of 7zr1 by Molmil](/molmil-images/mine/7zr1) | Chaetomium thermophilum Mre11-Rad50-Nbs1 complex bound to ATPyS (composite structure) | 分子名称: | DH domain-containing protein, Double-strand break repair protein, FHA domain-containing protein, ... | 著者 | Bartho, J.D, Rotheneder, M, Stakyte, K, Lammens, K, Hopfner, K.P. | 登録日 | 2022-05-03 | 公開日 | 2023-01-11 | 最終更新日 | 2023-12-13 | 実験手法 | ELECTRON MICROSCOPY (4 Å) | 主引用文献 | Cryo-EM structure of the Mre11-Rad50-Nbs1 complex reveals the molecular mechanism of scaffolding functions. Mol.Cell, 83, 2023
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4I5L
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![BU of 4i5l by Molmil](/molmil-images/mine/4i5l) | Structural mechanism of trimeric PP2A holoenzyme involving PR70: insight for Cdc6 dephosphorylation | 分子名称: | CALCIUM ION, DI(HYDROXYETHYL)ETHER, MALONATE ION, ... | 著者 | Wlodarchak, N, Satyshur, K.A, Guo, F, Xing, Y. | 登録日 | 2012-11-28 | 公開日 | 2013-05-08 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.43 Å) | 主引用文献 | Structure of the Ca(2+)-dependent PP2A heterotrimer and insights into Cdc6 dephosphorylation. Cell Res., 23, 2013
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1HP1
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![BU of 1hp1 by Molmil](/molmil-images/mine/1hp1) | 5'-NUCLEOTIDASE (OPEN FORM) COMPLEX WITH ATP | 分子名称: | 5'-NUCLEOTIDASE, ADENOSINE-5'-TRIPHOSPHATE, CARBONATE ION, ... | 著者 | Knoefel, T, Straeter, N. | 登録日 | 2000-12-12 | 公開日 | 2002-03-20 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Mechanism of hydrolysis of phosphate esters by the dimetal center of 5'-nucleotidase based on crystal structures. J.Mol.Biol., 309, 2001
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6YE1
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![BU of 6ye1 by Molmil](/molmil-images/mine/6ye1) | Human Ecto-5'-nucleotidase (CD73) in complex with the AMPCP derivative A894 (compound 2n in publication) in the closed form (crystal form IV) | 分子名称: | 5'-nucleotidase, ZINC ION, [(2~{R},3~{S},4~{R},5~{R})-5-[2-chloranyl-6-(cyclopentylamino)purin-9-yl]-3,4-bis(oxidanyl)oxolan-2-yl]methoxymethylphosphonic acid | 著者 | Scaletti, E, Strater, N. | 登録日 | 2020-03-23 | 公開日 | 2021-01-20 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.66 Å) | 主引用文献 | Discovery of Potent and Selective Methylenephosphonic Acid CD73 Inhibitors. J.Med.Chem., 64, 2021
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4JA7
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![BU of 4ja7 by Molmil](/molmil-images/mine/4ja7) | Rat PP5 co-crystallized with P5SA-2 | 分子名称: | MAGNESIUM ION, Serine/threonine-protein phosphatase 5 | 著者 | Haslbeck, V, Helmuth, M, Alte, F, Popowicz, G, Schmidt, W, Weiwad, M, Fischer, G, Gemmecker, G, Sattler, M, Striggow, F, Groll, M, Richter, K. | 登録日 | 2013-02-18 | 公開日 | 2014-02-19 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Selective activators of protein phosphatase 5 target the auto-inhibitory mechanism. Biosci.Rep., 35, 2015
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4LAC
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![BU of 4lac by Molmil](/molmil-images/mine/4lac) | Crystal Structure of Protein Phosphatase 2A (PP2A) and PP2A phosphatase activator (PTPA) complex with ATPgammaS | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, DI(HYDROXYETHYL)ETHER, MANGANESE (II) ION, ... | 著者 | Guo, F, Stanevich, V, Wlodarchak, N, Satyshur, K.A, Xing, Y. | 登録日 | 2013-06-19 | 公開日 | 2013-10-09 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.82 Å) | 主引用文献 | Structural basis of PP2A activation by PTPA, an ATP-dependent activation chaperone. Cell Res., 24, 2014
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6YE2
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