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1QLL
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Piratoxin-II (Prtx-II) - a K49 PLA2 from Bothrops pirajai
分子名称: N-TRIDECANOIC ACID, PHOSPHOLIPASE A2
著者Lee, W.-H, Polikarpov, I.
登録日1999-09-01
公開日2000-09-07
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.04 Å)
主引用文献Structural Basis for Low Catalytic Activity in Lys49 Phospholipases A2-A Hypothesis: The Crystal Structure of Piratoxin II Complexed to Fatty Acid
Biochemistry, 40, 2001
2PH4
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Crystal structure of a novel Arg49 phospholipase A2 homologue from Zhaoermia mangshanensis venom
分子名称: DI(HYDROXYETHYL)ETHER, SULFATE ION, Zhaoermiatoxin
著者Murakami, M.T, Kuch, U, Mebs, D, Arni, R.K.
登録日2007-04-10
公開日2008-03-18
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Crystal structure of a novel myotoxic Arg49 phospholipase A(2) homolog (zhaoermiatoxin) from Zhaoermia mangshanensis snake venom: Insights into Arg49 coordination and the role of Lys122 in the polarization of the C-terminus.
Toxicon, 51, 2008
5VFM
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Crystal structure of BnSP-7 from Bothrops pauloensis complexed with p-coumaric acid
分子名称: 1-ETHOXY-2-(2-METHOXYETHOXY)ETHANE, 4'-HYDROXYCINNAMIC ACID, Basic phospholipase A2 homolog BnSP-7, ...
著者De Lima, L.F.G, Fontes, M.R.M.
登録日2017-04-08
公開日2017-12-20
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.058 Å)
主引用文献Structural studies with BnSP-7 reveal an atypical oligomeric conformation compared to phospholipases A2-like toxins.
Biochimie, 142, 2017
4NTW
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Structure of acid-sensing ion channel in complex with snake toxin
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Acid-sensing ion channel 1, Basic phospholipase A2 homolog Tx-beta, ...
著者Baconguis, I, Bohlen, C.J, Goehring, A, Julius, D, Gouaux, E.
登録日2013-12-02
公開日2014-02-19
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.07 Å)
主引用文献X-ray structure of Acid-sensing ion channel 1-snake toxin complex reveals open state of a na(+)-selective channel.
Cell(Cambridge,Mass.), 156, 2014
2AOZ
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Crystal structure of the myotoxin-II from Atropoides nummifer venom
分子名称: Phospholipase A2 homolog, SULFATE ION
著者Melo, C.C, Murakami, M.T, Angulo, Y, Lomonte, B, Arni, R.K.
登録日2005-08-15
公開日2006-07-25
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2.08 Å)
主引用文献Structure of myotoxin II, a catalytically inactive Lys49 phospholipase A2 homologue from Atropoides nummifer venom.
Acta Crystallogr.,Sect.F, 62, 2006
4K06
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Crystal structure of MTX-II from Bothrops brazili venom complexed with polyethylene glycol
分子名称: 2-(2-(2-(2-(2-(2-ETHOXYETHOXY)ETHOXY)ETHOXY)ETHOXY)ETHOXY)ETHANOL, 2-{2-[2-(2-{2-[2-(2-ETHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHOXY]-ETHOXY}-ETHANOL, MTX-II, ...
著者Fernandes, C.A.H, Comparetti, E.J, Borges, R.J, Fontes, M.R.M.
登録日2013-04-03
公開日2013-11-13
最終更新日2013-11-27
実験手法X-RAY DIFFRACTION (2.08 Å)
主引用文献Structural bases for a complete myotoxic mechanism: Crystal structures of two non-catalytic phospholipases A2-like from Bothrops brazili venom.
Biochim.Biophys.Acta, 1834, 2013
2QU9
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Crystal structure of the complex of group II phospholipase A2 with Eugenol
分子名称: 2-methoxy-4-[(1E)-prop-1-en-1-yl]phenol, Phospholipase A2 VRV-PL-VIIIa, SULFATE ION
著者Kumar, S, Vikram, G, Singh, N, Sinha, M, Sharma, S, Kaur, P, Srinivasan, A, Singh, T.P.
登録日2007-08-04
公開日2007-08-14
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.08 Å)
主引用文献Crystal structure of the complex of group II phospholipase A2 with Eugenol
To be Published
5VFJ
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Crystal structure of BnSP-7 from bothrops pauloensis complexed with caffeic acid
分子名称: Basic phospholipase A2 homolog BnSP-7, CAFFEIC ACID, SULFATE ION
著者De Lima, L.F.G, Fontes, M.R.M.
登録日2017-04-07
公開日2017-12-20
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.084 Å)
主引用文献Structural studies with BnSP-7 reveal an atypical oligomeric conformation compared to phospholipases A2-like toxins.
Biochimie, 142, 2017
1LE7
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CARBOXYLIC ESTER HYDROLASE, C 2 2 21 space group
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, CALCIUM ION, Group X Secretory Phospholipase A2
著者Pan, Y.H, Jain, M.K, Bahnson, B.J.
登録日2002-04-09
公開日2002-08-14
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.09 Å)
主引用文献Crystal structure of human group X secreted phospholipase A2. Electrostatically neutral interfacial surface targets zwitterionic membranes.
J.Biol.Chem., 277, 2002
1POE
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STRUCTURES OF FREE AND INHIBITED HUMAN SECRETORY PHOSPHOLIPASE A2 FROM INFLAMMATORY EXUDATE
分子名称: 1-O-OCTYL-2-HEPTYLPHOSPHONYL-SN-GLYCERO-3-PHOSPHOETHANOLAMINE, CALCIUM ION, PHOSPHOLIPASE A2
著者Scott, D.L, White, S.P, Sigler, P.B.
登録日1992-09-07
公開日1993-10-31
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Structures of free and inhibited human secretory phospholipase A2 from inflammatory exudate.
Science, 254, 1991
1M8T
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Structure of an acidic Phospholipase A2 from the venom of Ophiophagus hannah at 2.1 resolution from a hemihedrally twinned crystal form
分子名称: CALCIUM ION, HEXANE-1,6-DIOL, Phospholipase a2
著者Xu, S, Gu, L, Wang, Q, Shu, Y, Lin, Z.
登録日2002-07-26
公開日2003-09-02
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Structure of a king cobra phospholipase A2 determined from a hemihedrally twinned crystal.
Acta Crystallogr.,Sect.D, 59, 2003
2DPZ
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Structure of the complex of phospholipase A2 with N-(4-hydroxyphenyl)- acetamide at 2.1 A resolution
分子名称: N-(4-HYDROXYPHENYL)ACETAMIDE (TYLENOL), Phospholipase A2 VRV-PL-VIIIa, SULFATE ION
著者Singh, N, Sharma, S, Singh, T.P.
登録日2006-05-18
公開日2006-06-06
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Phospholipase A2 as a target protein for non-steroidal anti-inflammatory drugs (NSAIDs): Crystal structure of the complex formed between a group II phospholipase A2 and N-(4-hydroxyphenyl) - acetamide at 2.1 resolution
To be Published
3P2P
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ENHANCED ACTIVITY AND ALTERED SPECIFICITY OF PHOSPHOLIPASE A2 BY DELETION OF A SURFACE LOOP
分子名称: CALCIUM ION, PHOSPHOLIPASE A2
著者Dijkstra, B.W, Thunnissen, M.M.G.M, Kalk, K.H, Drenth, J.
登録日1989-11-29
公開日1990-01-15
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Enhanced activity and altered specificity of phospholipase A2 by deletion of a surface loop.
Science, 244, 1989
3BP2
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BU of 3bp2 by Molmil
ROLE OF THE N-TERMINUS IN THE INTERACTION OF PANCREATIC PHOSPHOLIPASE A2 WITH AGGREGATED SUBSTRATES. PROPERTIES AND CRYSTAL STRUCTURE OF TRANSAMINATED PHOSPHOLIPASE A2
分子名称: CALCIUM ION, PHOSPHOLIPASE A2
著者Dijkstra, B.W, Drenth, J.
登録日1983-06-27
公開日1983-09-15
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Role of the N-terminus in the interaction of pancreatic phospholipase A2 with aggregated substrates. Properties and crystal structure of transaminated phospholipase A2
Biochemistry, 23, 1984
3JR8
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Crystal Structure of BthTX-II (Asp49-PLA2 from Bothrops jararacussu snake venom) with calcium ions
分子名称: CALCIUM ION, Phospholipase A2 bothropstoxin-2
著者Borges, R.J, dos Santos, J.I, Fontes, M.R.M.
登録日2009-09-08
公開日2010-09-08
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Structural, functional, and bioinformatics studies reveal a new snake venom homologue phospholipase A2 class.
Proteins, 79, 2011
2PVT
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Crystal structure of a new isoform of phospholipase A2 from russells viper at 2.1 A resolution
分子名称: phospholipase A2
著者Kumar, S, Singh, N, Sharma, S, Kaur, P, Singh, T.P.
登録日2007-05-10
公開日2007-05-22
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Crystal structure of a new isoform of phospholipase A2 from russells viper at 2.1 A resolution
To be Published
1POD
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BU of 1pod by Molmil
STRUCTURES OF FREE AND INHIBITED HUMAN SECRETORY PHOSPHOLIPASE A2 FROM INFLAMMATORY EXUDATE
分子名称: CALCIUM ION, PHOSPHOLIPASE A2
著者Scott, D.L, White, S.P, Sigler, P.B.
登録日1992-09-07
公開日1993-10-31
最終更新日2019-08-14
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Structures of free and inhibited human secretory phospholipase A2 from inflammatory exudate.
Science, 254, 1991
7ROX
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BU of 7rox by Molmil
BthTX-I complexed with inhibitor MMV
分子名称: 12-methoxy-Nb-methylvoachalotine, Basic phospholipase A2 homolog bothropstoxin-I
著者Borges, R.J, De Marino, I, Uson, I, Fontes, M.R.M.
登録日2021-08-02
公開日2022-11-09
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Structural and functional studies of a snake venom phospholipase A 2 -like protein complexed to an inhibitor from Tabernaemontana catharinensis.
Biochimie, 206, 2023
1KQU
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Human phospholipase A2 complexed with a substrate anologue
分子名称: 6-PHENYL-4(R)-(7-PHENYL-HEPTANOYLAMINO)-HEXANOIC ACID, CALCIUM ION, Phospholipase A2, ...
著者Tyndall, J.D, Martin, J.L.
登録日2002-01-07
公開日2003-11-11
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献D-Tyrosine as a chiral precusor to potent inhibitors of human nonpancreatic secretory phospholipase A2 (IIa) with antiinflammatory activity.
Chembiochem, 4, 2003
4K09
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Crystal structure of BbTX-II from Bothrops brazili venom
分子名称: BbTX-II
著者Fernandes, C.A.H, Comparetti, E.J, Borges, R.J, Fontes, M.R.M.
登録日2013-04-03
公開日2013-11-20
最終更新日2013-11-27
実験手法X-RAY DIFFRACTION (2.107 Å)
主引用文献Structural bases for a complete myotoxic mechanism: Crystal structures of two non-catalytic phospholipases A2-like from Bothrops brazili venom.
Biochim.Biophys.Acta, 1834, 2013
1JIA
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STRUCTURE OF A BASIC PHOSPHOLIPASE A2 FROM AGKISTRODON HALYS PALLAS AT 2.13A RESOLUTION
分子名称: CALCIUM ION, PHOSPHOLIPASE A2
著者Zhao, K, Lin, Z.
登録日1997-06-09
公開日1998-06-10
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.13 Å)
主引用文献Structure of a basic phospholipase A2 from Agkistrodon halys Pallas at 2.13 A resolution.
Acta Crystallogr.,Sect.D, 54, 1998
6CE2
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Crystal structure of Myotoxin I (MjTX-I) from Bothrops moojeni complexed to inhibitor suramin
分子名称: 2-{2-[2-(2-{2-[2-(2-ETHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHOXY]-ETHOXY}-ETHANOL, 8,8'-[CARBONYLBIS[IMINO-3,1-PHENYLENECARBONYLIMINO(4-METHYL-3,1-PHENYLENE)CARBONYLIMINO]]BIS-1,3,5-NAPHTHALENETRISULFON IC ACID, Basic phospholipase A2 homolog 1
著者Salvador, G.H.M, Fontes, M.R.M.
登録日2018-02-10
公開日2018-07-25
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Structural and functional characterization of suramin-bound MjTX-I from Bothrops moojeni suggests a particular myotoxic mechanism.
Sci Rep, 8, 2018
3VC0
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Crystal structure of Taipoxin beta subunit isoform 1
分子名称: Phospholipase A2 homolog, taipoxin beta chain
著者Cendron, L, Micetic, I, Polverino de Laureto, P, Beltramini, M, Paoli, M.
登録日2012-01-03
公開日2012-07-25
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Structural analysis of trimeric phospholipase A(2) neurotoxin from the Australian taipan snake venom.
Febs J., 279, 2012
4WTB
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BthTX-I, a svPLA2s-like toxin, complexed with zinc ions
分子名称: Basic phospholipase A2 homolog bothropstoxin-1, CHLORIDE ION, SULFATE ION, ...
著者Borges, R.J, Fontes, M.R.M.
登録日2014-10-29
公開日2015-11-11
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.16 Å)
主引用文献Functional and structural studies of a Phospholipase A2-like protein complexed to zinc ions: Insights on its myotoxicity and inhibition mechanism.
Biochim. Biophys. Acta, 1861, 2017
3I3H
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Crystal structure of Bothropstoxin-I crystallized at 291K
分子名称: Phospholipase A2 homolog bothropstoxin-1
著者Salvador, G.H.M, Marchi-Salvador, D.P, Soares, A.M, Fontes, M.R.M.
登録日2009-06-30
公開日2010-08-11
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.17 Å)
主引用文献Structural Studies with a BthTX-I a Lys49 PLA2 from Bothrops jararacussu Snake Venom Crystallized at Different Temperatures
To be Published

221716

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