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2WZ6
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G93A SOD1 mutant complexed with Quinazoline.
分子名称: 4-(4-METHYL-1,4-DIAZEPAN-1-YL)-2-(TRIFLUOROMETHYL)QUINAZOLINE, COPPER (II) ION, SULFATE ION, ...
著者Antonyuk, S.V, Strange, R.W, Hasnain, S.S.
登録日2009-11-23
公開日2010-12-08
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献Structural Discovery of Small Molecule Binding Sites in Cu-Zn Human Superoxide Dismutase Familial Amyotrophic Lateral Sclerosis Mutants Provides Insights for Lead Optimization.
J.Med.Chem., 53, 2010
2X7Y
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P450 BM3 F87A in complex with DMSO
分子名称: BIFUNCTIONAL P-450/NADPH-P450 REDUCTASE, DIMETHYL SULFOXIDE, PROTOPORPHYRIN IX CONTAINING FE, ...
著者Kuper, J, Wong, T.S, Roccatano, D, Wilmanns, M, Schwaneberg, U.
登録日2010-03-04
公開日2011-03-23
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献The Role of Active-Site Phe87 in Modulating the Organic Co-Solvent Tolerance of Cytochrome P450 Bm3 Monooxygenase.
Acta Crystallogr.,Sect.F, 68, 2012
2WRX
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Semi-synthetic analogue of human insulin NMeAlaB26-insulin at pH 3.0
分子名称: INSULIN A CHAIN, INSULIN B CHAIN, SODIUM ION
著者Brzozowski, A.M, Jiracek, J, Zakova, L, Antolikova, E, Watson, C.J, Turkenburg, J.P, Dodson, G.G.
登録日2009-09-02
公開日2010-02-09
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Implications for the Active Form of Human Insulin Based on the Structural Convergence of Highly Active Hormone Analogues.
Proc.Natl.Acad.Sci.USA, 107, 2010
2X1V
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Crystal Structure of the activating H-Ras I163F mutant in Costello Syndrome, bound to MG-GDP
分子名称: GTPASE HRAS, GUANOSINE-5'-DIPHOSPHATE
著者Anand, K.
登録日2010-01-04
公開日2010-01-12
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Crystal Structure of the Activating H-Ras I163F Mutant in Costello Syndrome, Bound to Mg-Gdp
To be Published
2WUT
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Crystal structure of human myelin protein P2 in complex with palmitate
分子名称: CHLORIDE ION, GLYCEROL, MYELIN P2 PROTEIN, ...
著者Majava, V, Nanekar, R, Kursula, P.
登録日2009-10-09
公開日2010-05-12
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Structural and Functional Characterization of Human Peripheral Nervous System Myelin Protein P2.
Plos One, 5, 2010
2XKR
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Crystal Structure of Mycobacterium tuberculosis CYP142: A novel cholesterol oxidase
分子名称: PROTOPORPHYRIN IX CONTAINING FE, PUTATIVE CYTOCHROME P450 142, TETRAETHYLENE GLYCOL
著者Driscoll, M, McLean, K.J, Levy, C.W, Lafite, P, Mast, N, Pikuleva, I.A, Rigby, S.E.J, Leys, D, Munro, A.W.
登録日2010-07-12
公開日2010-09-29
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.601 Å)
主引用文献Structural and Biochemical Characterization of Mycobacterium Tuberculosis Cyp142: Evidence for Multiple Cholesterol 27-Hydroxylase Activities in a Human Pathogen.
J.Biol.Chem., 285, 2010
2XMF
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Myosin 1e SH3
分子名称: MYOSIN 1E SH3, OCTANE 1,8-DIAMINE
著者Edwards, T, Allsop, G, Peckham, M.
登録日2010-07-27
公開日2011-08-10
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Myosin 1E SH3
To be Published
2XFJ
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Human BACE-1 in complex with N-((1S,2R)-3-(((1S)-2-(cyclohexylamino)- 1-methyl-2-oxoethyl)amino)-2-hydroxy-1-(phenylmethyl)propyl)-3-(ethylamino)-5-(2-oxo-1-pyrrolidinyl)benzamide
分子名称: BETA-SECRETASE 1, N-[(1S,2R)-1-benzyl-3-{[(1S)-2-(cyclohexylamino)-1-methyl-2-oxoethyl]amino}-2-hydroxypropyl]-3-(ethylamino)-5-(2-oxopyrrolidin-1-yl)benzamide
著者Clarke, B, Cutler, L, Demont, E, Dingwall, C, Dunsdon, R, Hawkins, J, Howes, C, Hussain, I, Maile, G, Matico, R, Mosley, J, Naylor, A, O'Brien, A, Redshaw, S, Rowland, P, Soleil, V, Smith, K.J, Sweitzer, S, Theobald, P, Vesey, D, Walter, D.S, Wayne, G.
登録日2010-05-24
公開日2010-07-07
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Bace-1 Inhibitors Using Novel Edge-to-Face Interaction with Arg-296
Bioorg.Med.Chem.Lett., 20, 2010
2XJW
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Lysozyme-CO releasing molecule adduct
分子名称: CARBON MONOXIDE, CHLORIDE ION, LYSOZYME C, ...
著者Santos-Silva, T, Mukhopadhyay, A, Romao, M.J.
登録日2010-07-06
公開日2011-01-26
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.67 Å)
主引用文献Corm-3 Reactivity Toward Proteins: The Crystal Structure of a Ru(II) Dicarbonyl-Lysozyme Complex.
J.Am.Chem.Soc., 133, 2011
2Y04
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TURKEY BETA1 ADRENERGIC RECEPTOR WITH STABILISING MUTATIONS AND BOUND PARTIAL AGONIST SALBUTAMOL
分子名称: BETA-1 ADRENERGIC RECEPTOR, CHOLESTEROL HEMISUCCINATE, HEGA-10, ...
著者Warne, A, Moukhametzianov, R, Baker, J.G, Nehme, R, Edwards, P.C, Leslie, A.G.W, Schertler, G.F.X, Tate, C.G.
登録日2010-11-30
公開日2011-01-12
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (3.05 Å)
主引用文献The Structural Basis for Agonist and Partial Agonist Action on a Beta1-Adrenergic Receptor
Nature, 469, 2011
2XR5
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Crystal structure of the complex of the carbohydrate recognition domain of human DC-SIGN with pseudo dimannoside mimic.
分子名称: CALCIUM ION, CD209 ANTIGEN, CHLORIDE ION, ...
著者Thepaut, M, Suitkeviciute, I, Sattin, S, Reina, J, Bernardi, A, Fieschi, F.
登録日2010-09-10
公開日2011-10-19
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.42 Å)
主引用文献Structure of a Glycomimetic Ligand in the Carbohydrate Recognition Domain of C-Type Lectin Dc-Sign. Structural Requirements for Selectivity and Ligand Design.
J.Am.Chem.Soc., 135, 2013
2XST
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Crystal Structure of the Human Lipocalin 15
分子名称: 1,2-ETHANEDIOL, LIPOCALIN 15
著者Muniz, J.R.C, Gileadi, C, Yue, W.W, Krojer, T, Ugochukwu, E, Phillips, C, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Weigelt, J, Bountra, C, Kavanagh, K.L, Oppermann, U.
登録日2010-09-30
公開日2010-10-13
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.63 Å)
主引用文献Crystal Structure of the Human Lipocalin 15
To be Published
2YZ2
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Crystal structure of the ABC transporter in the cobalt transport system
分子名称: Putative ABC transporter ATP-binding protein TM_0222
著者Ethayathullah, A.S, Bessho, Y, Padmanabhan, B, Singh, T.P, Kaur, P, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2007-05-02
公開日2007-11-06
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal structure of the ABC transporter in the cobalt transport system
To be Published
2YZU
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Crystal structure of oxidized thioredoxin from Thermus thermophilus HB8
分子名称: Thioredoxin
著者Ebihara, A, Yanai, H, Yokoyama, S, Kuramitsu, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2007-05-06
公開日2007-11-06
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystal structure of oxidized thioredoxin from Thermus thermophilus HB8
To be Published
2Y83
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Actin filament pointed end
分子名称: ACTIN, ALPHA SKELETAL MUSCLE, ADENOSINE-5'-DIPHOSPHATE, ...
著者Narita, A, Oda, T, Maeda, Y.
登録日2011-02-02
公開日2011-03-30
最終更新日2024-05-08
実験手法ELECTRON MICROSCOPY (22.9 Å)
主引用文献Structural Basis for the Slow Dynamics of the Actin Filament Pointed End.
Embo J., 30, 2011
2YCY
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TURKEY BETA1 ADRENERGIC RECEPTOR WITH STABILISING MUTATIONS AND BOUND ANTAGONIST CYANOPINDOLOL
分子名称: 4-{[(2S)-3-(tert-butylamino)-2-hydroxypropyl]oxy}-3H-indole-2-carbonitrile, BETA-1 ADRENERGIC RECEPTOR, SODIUM ION, ...
著者Moukhametzianov, R, Warne, T, Edwards, P.C, Serrano-Vega, M.J, Leslie, A.G.W, Tate, C.G, Schertler, G.F.X.
登録日2011-03-17
公開日2011-06-08
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (3.15 Å)
主引用文献Two Distinct Conformations of Helix 6 Observed in Antagonist-Bound Structures of a {Beta}1- Adrenergic Receptor.
Proc.Natl.Acad.Sci.USA, 108, 2011
2YCZ
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TURKEY BETA1 ADRENERGIC RECEPTOR WITH STABILISING MUTATIONS AND BOUND ANTAGONIST IODOCYANOPINDOLOL
分子名称: 4-{[(2S)-3-(tert-butylamino)-2-hydroxypropyl]oxy}-3-iodo-1H-indole-2-carbonitrile, BETA-1 ADRENERGIC RECEPTOR, octyl 1-thio-beta-D-glucopyranoside
著者Moukhametzianov, R, Warne, T, Edwards, P.C, Serrano-Vega, M.J, Leslie, A.G.W, Tate, C.G, Schertler, G.F.X.
登録日2011-03-17
公開日2011-06-01
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (3.65 Å)
主引用文献Two Distinct Conformations of Helix 6 Observed in Antagonist-Bound Structures of a {Beta}1- Adrenergic Receptor.
Proc.Natl.Acad.Sci.USA, 108, 2011
2YSV
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Solution structure of C2H2 type Zinc finger domain 17 in Zinc finger protein 473
分子名称: ZINC ION, Zinc finger protein 473
著者Tsuda, K, Muto, Y, Inoue, M, Kigawa, T, Terada, T, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2007-04-04
公開日2007-10-09
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of C2H2 type Zinc finger domain 17 in Zinc finger protein 473
To be Published
2YTM
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Solution structure of the C2H2 type zinc finger (region 696-728) of human Zinc finger protein 28 homolog
分子名称: ZINC ION, Zinc finger protein 28 homolog
著者Tochio, N, Tomizawa, T, Abe, H, Saito, K, Li, H, Sato, M, Koshiba, S, Kobayashi, N, Kigawa, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2007-04-05
公開日2007-10-09
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of the C2H2 type zinc finger (region 696-728) of human Zinc finger protein 28 homolog
To be Published
2YSS
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Crystal structure of Humanized HYHEL-10 FV mutant(HQ39KW47Y)-HEN lysozyme complex
分子名称: ANTI-LYSOZYME ANTIBODY FV REGION, Lysozyme C
著者Nakanishi, T, Tsumoto, K, Yokota, A, Kondo, H, Kumagai, I.
登録日2007-04-03
公開日2008-04-08
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Critical contribution of VH-VL interaction to reshaping of an antibody: the case of humanization of anti-lysozyme antibody, HyHEL-10
Protein Sci., 17, 2008
2Z12
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Structure of the transformed monoclinic lysozyme by controlled dehydration
分子名称: CHLORIDE ION, Lysozyme C, SODIUM ION
著者Harata, K, Akiba, T.
登録日2007-05-07
公開日2008-03-18
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (1.15 Å)
主引用文献Effect of a sodium ion on the dehydration-induced phase transition of monoclinic lysozyme crystals.
Acta Crystallogr.,Sect.D, 63, 2007
2YRJ
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Solution structure of the C2H2-type zinc finger domain (781-813) from zinc finger protein 473
分子名称: ZINC ION, Zinc finger protein 473
著者Qin, X.R, Izumi, K, Yoshida, M, Hayashi, F, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2007-04-02
公開日2007-10-02
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of the C2H2-type zinc finger domain (781-813) from zinc finger protein 473
To be Published
2YRZ
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Solution structure of the fibronectin type III domain of human Integrin beta-4
分子名称: Integrin beta-4
著者Abe, H, Sasagawa, A, Tochio, N, Koshiba, S, Inoue, M, Kigawa, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2007-04-03
公開日2008-04-08
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of the fibronectin type III domain of human Integrin beta-4
To be Published
2YSX
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Solution structure of the human SHIP SH2 domain
分子名称: Signaling inositol polyphosphate phosphatase SHIP II
著者Kasai, T, Koshiba, S, Watanabe, S, Harada, T, Kigawa, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2007-04-04
公開日2008-04-08
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of the human SHIP SH2 domain
To be Published
2YTJ
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Solution structure of the C2H2 type zinc finger (region 771-803) of human Zinc finger protein 484
分子名称: ZINC ION, Zinc finger protein 484
著者Tomizawa, T, Tochio, N, Abe, H, Saito, K, Li, H, Sato, M, Koshiba, S, Kobayashi, N, Kigawa, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2007-04-05
公開日2007-10-09
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of the C2H2 type zinc finger (region 771-803) of human Zinc finger protein 484
To be Published

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