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3W6A
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BU of 3w6a by Molmil
Crystal structure of cross-linked tetragonal hen egg white lysozyme soaked wiht 5mM [Ru(benzene)Cl2]2
分子名称: ACETATE ION, Benzeneruthenium(II) chloride, CHLORIDE ION, ...
著者Tabe, H, Abe, S, Hikage, T, Kitagawa, S, Ueno, T.
登録日2013-02-13
公開日2014-02-19
実験手法X-RAY DIFFRACTION (1.77 Å)
主引用文献Solid Artificial Metalloenzymes: Post-Engineering of Porous Protein Crystals by Organometallic Complexes
To be Published
2G0H
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BU of 2g0h by Molmil
Structure-based drug design of a novel family of PPAR partial agonists: virtual screening, x-ray crystallography and in vitro/in vivo biological activities
分子名称: N-[1-(4-FLUOROPHENYL)-3-(2-THIENYL)-1H-PYRAZOL-5-YL]-3,5-BIS(TRIFLUOROMETHYL)BENZENESULFONAMIDE, Peroxisome proliferator-activated receptor gamma
著者Lu, I.L, Peng, Y.H, Huang, C.F, Lin, Y.T, Hsu, J.T.A, Wu, S.Y.
登録日2006-02-13
公開日2006-05-16
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structure-Based Drug Design of a Novel Family of PPARgamma Partial Agonists: Virtual Screening, X-ray Crystallography, and in Vitro/in Vivo Biological Activities
J.Med.Chem., 49, 2006
1UYP
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BU of 1uyp by Molmil
The three-dimensional structure of beta-fructosidase (invertase) from Thermotoga maritima
分子名称: BETA-FRUCTOSIDASE, CITRIC ACID, GLYCEROL, ...
著者Alberto, F, Bignon, C, Sulzenbacher, G, Henrissat, B, Czjzek, M.
登録日2004-03-02
公開日2004-03-22
最終更新日2018-06-13
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献The three-dimensional structure of invertase (beta-fructosidase) from Thermotoga maritima reveals a bimodular arrangement and an evolutionary relationship between retaining and inverting glycosidases.
J. Biol. Chem., 279, 2004
1TZ7
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BU of 1tz7 by Molmil
Aquifex aeolicus amylomaltase
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, 4-alpha-glucanotransferase
著者Barends, T.R.M, Korf, H, Kaper, T, van der Maarel, M.J.E.C, Dijkhuizen, L, Dijkstra, B.W.
登録日2004-07-09
公開日2005-08-02
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Structural influences on product specificity in amylomaltase from Aquifex aeolicus
TO BE PUBLISHED
1V5Y
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BU of 1v5y by Molmil
Binding of coumarins to NAD(P)H:FMN oxidoreductase
分子名称: 4-HYDROXY-2H-CHROMEN-2-ONE, FLAVIN MONONUCLEOTIDE, Major NAD(P)H-flavin oxidoreductase
著者Kobori, T, Koike, H, Sasaki, H, Zenno, S, Saigo, K, Tanokura, M.
登録日2003-11-26
公開日2005-03-08
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Binding of coumarins to NAD(P)H:FMN oxidoreductase
To be Published
1V5Z
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BU of 1v5z by Molmil
Binding of coumarins to NAD(P)H:FMN oxidoreductase
分子名称: (2E)-3-(2-HYDROXYPHENYL)ACRYLIC ACID, FLAVIN MONONUCLEOTIDE, Major NAD(P)H-flavin oxidoreductase
著者Kobori, T, Koike, H, Sasaki, H, Zenno, S, Saigo, K, Tanokura, M.
登録日2003-11-26
公開日2005-03-08
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Binding of coumarins to NAD(P)H:FMN oxidoreductase
To be Published
5JVG
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BU of 5jvg by Molmil
The large ribosomal subunit from Deinococcus radiodurans in complex with avilamycin
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, 23S ribosomal RNA, 50S ribosomal protein L11, ...
著者Krupkin, M, Wekselman, I, Matzov, D, Eyal, Z, Diskin Posner, Y, Rozenberg, H, Zimmerman, E, Bashan, A, Yonath, A.
登録日2016-05-11
公開日2016-11-09
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (3.428 Å)
主引用文献Avilamycin and evernimicin induce structural changes in rProteins uL16 and CTC that enhance the inhibition of A-site tRNA binding.
Proc.Natl.Acad.Sci.USA, 113, 2016
6MXT
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BU of 6mxt by Molmil
Crystal structure of human beta2 adrenergic receptor bound to salmeterol and Nb71
分子名称: (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, 3,6,9,12,15,18-HEXAOXAICOSANE-1,20-DIOL, Endolysin, ...
著者Masureel, M, Zou, Y, Picard, L.P, van der Westhuizen, E, Mahoney, J.P, Rodrigues, J.P.G.L.M, Mildorf, T.J, Dror, R.O, Shaw, D.E, Bouvier, M, Pardon, E, Steyaert, J, Sunahara, R.K, Weis, W.I, Zhang, C, Kobilka, B.K.
登録日2018-10-31
公開日2018-11-14
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.95934224 Å)
主引用文献Structural insights into binding specificity, efficacy and bias of a beta2AR partial agonist.
Nat. Chem. Biol., 14, 2018
6FTF
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BU of 6ftf by Molmil
Regulatory subunit of a cAMP-independent protein kinase A from Trypanosoma cruzi at 1.09 A resolution
分子名称: 1,2-ETHANEDIOL, 7-cyano-7-deazainosine, Protein kinase A regulatory subunit, ...
著者Volpato Santos, Y, Lorentzen, E, Basquin, J, Boshart, M.
登録日2018-02-21
公開日2019-04-03
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.09151936 Å)
主引用文献Nucleoside analogue activators of cyclic AMP-independent protein kinase A of Trypanosoma.
Nat Commun, 10, 2019
2KM6
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BU of 2km6 by Molmil
NMR structure of the NLRP7 Pyrin domain
分子名称: NACHT, LRR and PYD domains-containing protein 7
著者Pinheiro, A, Proell, M, Schwarzenbacher, R, Peti, W.
登録日2009-07-21
公開日2010-06-09
最終更新日2024-05-08
実験手法SOLUTION NMR
主引用文献Three-dimensional structure of the NLRP7 pyrin domain: insight into pyrin-pyrin-mediated effector domain signaling in innate immunity.
J.Biol.Chem., 285, 2010
2L87
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BU of 2l87 by Molmil
The 27-residue N-terminus CCR5-peptide in a ternary complex with HIV-1 gp120 and a CD4-mimic peptide
分子名称: C-C chemokine receptor type 5
著者Schnur, E, Noah, E, Ayzenshtat, I, Sargsyan, H, Inui, T, Ding, F.X, Arshava, B, Sagi, Y, Kessler, N, Levy, R, Scherf, T, Naider, F, Anglister, J.
登録日2011-01-06
公開日2011-07-27
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献The Conformation and Orientation of a 27-Residue CCR5 Peptide in a Ternary Complex with HIV-1 gp120 and a CD4-Mimic Peptide.
J.Mol.Biol., 410, 2011
5KI9
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BU of 5ki9 by Molmil
Crystal structure of human beta-defensin 4 (HBD4)
分子名称: Beta-defensin 104, SULFATE ION, trifluoroacetic acid
著者Jacek, L, Adam, P, Marzenam, P.
登録日2016-06-16
公開日2017-06-28
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Human beta-Defensin 4: defensin without the "twist"
To Be Published
6FLO
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BU of 6flo by Molmil
Regulatory subunit of a cAMP-independent protein kinase A from Trypanosoma brucei at 2.1 Angstrom resolution
分子名称: GLYCEROL, INOSINE, Protein kinase A regulatory subunit
著者Volpato Santos, Y, Lorentzen, E, Basquin, J, Boshart, M.
登録日2018-01-26
公開日2019-08-14
最終更新日2024-04-10
実験手法X-RAY DIFFRACTION (2.13868666 Å)
主引用文献Purine nucleosides replace cAMP in allosteric regulation of PKA in trypanosomatid pathogens.
Elife, 12, 2024
6MRX
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BU of 6mrx by Molmil
Sialidase26 apo
分子名称: Sialidase26
著者Zaramela, L.S, Martino, C, Alisson-Silva, F, Rees, S.D, Diaz, S.L, Chuzel, L, Ganatra, M.B, Taron, C.H, Zuniga, C, Chang, G, Varki, A, Zengler, K.
登録日2018-10-15
公開日2019-10-02
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Gut bacteria responding to dietary change encode sialidases that exhibit preference for red meat-associated carbohydrates.
Nat Microbiol, 4, 2019
2LMJ
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BU of 2lmj by Molmil
Itk-sh3
分子名称: Tyrosine-protein kinase ITK/TSK
著者Kristiansen, P, Bie Andersen, T, Huszenicza, Z, Andreotti, A.H, Spurkland, A.
登録日2011-12-05
公開日2012-12-05
最終更新日2024-05-01
実験手法SOLUTION NMR
主引用文献The SH3 domains of the Tec family kinase Itk and the Src family kinase Lck compete for adjacent sites on T-cell specific adapter protein
To be Published
3P3H
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BU of 3p3h by Molmil
Human carbonic anhydrase II in complex with p-(5-ferrocenyl-1H-1,2,3-triazol-1-yl)benzenesulfonamide
分子名称: Carbonic anhydrase 2, GLYCEROL, ZINC ION, ...
著者Salmon, A.J.
登録日2010-10-04
公開日2011-09-28
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Protein crystal structures with ferrocene and ruthenocene-based enzyme inhibitors.
Chem.Commun.(Camb.), 48, 2012
3P55
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BU of 3p55 by Molmil
Human carbonic anhydrase II in complex with p-(4-ferrocenyl-1H-1,2,3-triazol-1-yl)benzenesulfonamide
分子名称: Carbonic anhydrase 2, GLYCEROL, ZINC ION, ...
著者Salmon, A.J.
登録日2010-10-07
公開日2011-10-12
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Protein crystal structures with ferrocene and ruthenocene-based enzyme inhibitors.
Chem.Commun.(Camb.), 48, 2012
2LPX
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BU of 2lpx by Molmil
Solution Structure of Strawberry Allergen Fra a 1e
分子名称: Major strawberry allergen Fra a 1-E
著者Seutter von Loetzen, C, Hartl-Spiegelhauer, O, Schweimer, K, Schwab, W, Roesch, P.
登録日2012-02-20
公開日2012-03-07
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Solution structure of the strawberry allergen Fra a 1.
Biosci.Rep., 32, 2012
3P26
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Crystal structure of S. cerevisiae Hbs1 protein (apo-form), a translational GTPase involved in RNA quality control pathways and interacting with Dom34/Pelota
分子名称: Elongation factor 1 alpha-like protein
著者van den Elzen, A, Henri, J, Lazar, N, Gas, M.E, Durand, D, Lacroute, F, Nicaise, M, van Tilbeurgh, H, Sraphin, B, Graille, M, Paris-Sud Yeast Structural Genomics (YSG)
登録日2010-10-01
公開日2010-11-17
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Dissection of Dom34-Hbs1 reveals independent functions in two RNA quality control pathways.
Nat.Struct.Mol.Biol., 17, 2010
2LJA
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Solution Structure of a putative thiol-disulfide oxidoreductase from Bacteroides vulgatus
分子名称: Putative thiol-disulfide oxidoreductase
著者Harris, R, Seidel, R.D, Hillerich, B, Gizzi, A, Kar, A, Lafleur, J, Chamala, S, Foti, R, Villegas, G, Evans, B, Zencheck, W, Girvin, M.E, Almo, S.C, New York Structural Genomics Research Consortium (NYSGRC)
登録日2011-09-09
公開日2011-10-05
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Solution Structure of a putative thiol-disulfide oxidoreductase from Bacteroides vulgatus
To be Published
6MYV
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BU of 6myv by Molmil
Sialidase26 co-crystallized with DANA-Gc
分子名称: 2,6-anhydro-3,5-dideoxy-5-[(hydroxyacetyl)amino]-D-glycero-L-altro-non-2-enonic acid, Sialidase26
著者Zaramela, L.S, Martino, C, Alisson-Silva, F, Rees, S.D, Diaz, S.L, Chuzel, L, Ganatra, M.B, Taron, C.H, Zuniga, C, Huang, J, Siegel, D, Chang, G, Varki, A, Zengler, K.
登録日2018-11-02
公開日2019-10-02
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Gut bacteria responding to dietary change encode sialidases that exhibit preference for red meat-associated carbohydrates.
Nat Microbiol, 4, 2019
4O8Q
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BU of 4o8q by Molmil
Crystal structure of bovine MHD domain of the COPI delta subunit at 2.15 A resolution
分子名称: Coatomer subunit delta, FORMIC ACID
著者Lahav, A, Rozenberg, H, Cassel, D, Adir, N.
登録日2013-12-29
公開日2015-01-07
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Structure of the bovine COPI delta subunit mu homology domain at 2.15 angstrom resolution.
Acta Crystallogr.,Sect.D, 71, 2015
3P27
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Crystal structure of S. cerevisiae Hbs1 protein (GDP-bound form), a translational GTPase involved in RNA quality control pathways and interacting with Dom34/Pelota
分子名称: Elongation factor 1 alpha-like protein, GUANOSINE-5'-DIPHOSPHATE
著者van den Elzen, A, Henri, J, Lazar, N, Gas, M.E, Durand, D, Lacroute, F, Nicaise, M, van Tilbeurgh, H, Sraphin, B, Graille, M, Paris-Sud Yeast Structural Genomics (YSG)
登録日2010-10-01
公開日2010-11-17
最終更新日2012-03-14
実験手法X-RAY DIFFRACTION (2.95 Å)
主引用文献Dissection of Dom34-Hbs1 reveals independent functions in two RNA quality control pathways.
Nat.Struct.Mol.Biol., 17, 2010
2LRD
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BU of 2lrd by Molmil
The solution structure of the monomeric Acanthaporin
分子名称: Acanthaporin
著者Michalek, M, Soennichsen, F.D, Wechselberger, R, Dingley, A.J, Wienk, H, Simanski, M, Herbst, R, Lorenzen, I, Marciano-Cabral, F, Gelhaus, C, Groetzinger, J, Leippe, M.
登録日2012-03-28
公開日2012-05-02
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Structure and function of a unique pore-forming protein from a pathogenic acanthamoeba.
Nat.Chem.Biol., 9, 2013
3P44
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Human carbonic anhydrase II in complex with p-(4-ruthenocenyl-1H-1,2,3-triazol-1-yl)benzenesulfonamide
分子名称: Carbonic anhydrase 2, GLYCEROL, ZINC ION, ...
著者Salmon, A.J.
登録日2010-10-06
公開日2011-10-12
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Protein crystal structures with ferrocene and ruthenocene-based enzyme inhibitors.
Chem.Commun.(Camb.), 48, 2012

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件を2024-08-07に公開中

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