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4FWL
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Crystal structure of Salmonella typhimurium propionate kinase (TdcD) in complex with Phosphate (PO4)
分子名称: 1,2-ETHANEDIOL, PHOSPHATE ION, Propionate kinase
著者Chittori, S, Savithri, H.S, Murthy, M.R.N.
登録日2012-07-01
公開日2013-06-19
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Mechanistic features of Salmonella typhimurium propionate kinase (TdcD): insights from kinetic and crystallographic studies.
Biochim.Biophys.Acta, 1834, 2013
4FSC
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BU of 4fsc by Molmil
Crystal Structure of Bacillus thuringiensis PlcR in its apo form
分子名称: Transcriptional activator PlcR protein
著者Grenha, R, Slamti, L, Bouillaut, L, Lereclus, D, Nessler, S.
登録日2012-06-27
公開日2013-03-13
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (3.65 Å)
主引用文献Structural basis for the activation mechanism of the PlcR virulence regulator by the quorum-sensing signal peptide PapR.
Proc.Natl.Acad.Sci.USA, 110, 2013
6DW7
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BU of 6dw7 by Molmil
SAMHD1 without Catalytic Nucleotides
分子名称: 2'-DEOXYADENOSINE 5'-TRIPHOSPHATE, Deoxynucleoside triphosphate triphosphohydrolase SAMHD1, GLYCINE, ...
著者Knecht, K.M, Buzovetsky, O, Schneider, C, Thomas, D, Srikanth, V, Kaderali, L, Tofoleanu, F, Reiss, K, Ferreiros, N, Geisslinger, G, Batista, V.S, Ji, X, Cinatl, J, Keppler, O.T, Xiong, Y.
登録日2018-06-26
公開日2018-10-10
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献The structural basis for cancer drug interactions with the catalytic and allosteric sites of SAMHD1.
Proc. Natl. Acad. Sci. U.S.A., 115, 2018
7D3F
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BU of 7d3f by Molmil
Cryo-EM structure of human DUOX1-DUOXA1 in high-calcium state
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, Dual oxidase 1, ...
著者Chen, L, Wu, J.X.
登録日2020-09-19
公開日2020-12-09
最終更新日2021-06-23
実験手法ELECTRON MICROSCOPY (2.3 Å)
主引用文献Structures of human dual oxidase 1 complex in low-calcium and high-calcium states.
Nat Commun, 12, 2021
3QE3
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BU of 3qe3 by Molmil
Sheep liver sorbitol dehydrogenase
分子名称: ACETIC ACID, GLYCEROL, Sorbitol dehydrogenase, ...
著者Yennawar, N.H, Yennawar, H.P.
登録日2011-01-19
公開日2011-04-27
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献X-ray crystal structure and small-angle X-ray scattering of sheep liver sorbitol dehydrogenase.
Acta Crystallogr.,Sect.D, 67, 2011
4FXO
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BU of 4fxo by Molmil
Zinc-mediated allosteric inhibiton of caspase-6
分子名称: Caspase-6, ZINC ION
著者Velazquez-Delgado, E.M, Hardy, J.A.
登録日2012-07-03
公開日2012-08-22
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.85 Å)
主引用文献Zinc-mediated Allosteric Inhibition of Caspase-6.
J.Biol.Chem., 287, 2012
5VOL
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BU of 5vol by Molmil
Bacint_04212 ferulic acid esterase
分子名称: CALCIUM ION, ISOPROPYL ALCOHOL, Putative esterase
著者Koropatkin, N.M, Cann, I, Mackie, R.I.
登録日2017-05-03
公開日2017-07-19
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.98 Å)
主引用文献Biochemical and Structural Analyses of Two Cryptic Esterases in Bacteroides intestinalis and their Synergistic Activities with Cognate Xylanases.
J. Mol. Biol., 429, 2017
4FZB
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BU of 4fzb by Molmil
Structure of thymidylate synthase ThyX complexed to a new inhibitor
分子名称: 2-hydroxy-3-(4-methoxybenzyl)naphthalene-1,4-dione, DIMETHYL SULFOXIDE, FLAVIN-ADENINE DINUCLEOTIDE, ...
著者Basta, T, Boum, Y, Briffotaux, J, Becker, H.F, Lamarre-Jouenne, I, Lambry, J.C, Skouloubris, S, Liebl, U, van Tilbeurgh, H, Graille, M, Myllylkallio, H.
登録日2012-07-06
公開日2013-05-22
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.59 Å)
主引用文献Mechanistic and structural basis for inhibition of thymidylate synthase ThyX.
Open Biology, 2, 2012
7RZ8
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BU of 7rz8 by Molmil
Structure of the complex of LBD-TMD part of AMPA receptor GluA2 with auxiliary subunit TARP gamma-5 bound to agonist quisqualate
分子名称: (S)-2-AMINO-3-(3,5-DIOXO-[1,2,4]OXADIAZOLIDIN-2-YL)-PROPIONIC ACID, 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, Glutamate receptor 2
著者Klykov, O.V, Gangwar, S.P, Yelshanskaya, M.V, Sobolevsky, A.I.
登録日2021-08-27
公開日2021-10-27
最終更新日2022-02-16
実験手法ELECTRON MICROSCOPY (4.1 Å)
主引用文献Structure and desensitization of AMPA receptor complexes with type II TARP gamma 5 and GSG1L.
Mol.Cell, 81, 2021
7RZA
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Structure of the complex of AMPA receptor GluA2 with auxiliary subunit GSG1L bound to agonist quisqualate
分子名称: (S)-2-AMINO-3-(3,5-DIOXO-[1,2,4]OXADIAZOLIDIN-2-YL)-PROPIONIC ACID, Glutamate receptor 2
著者Gangwar, S.P, Klykov, O.V, Yelshanskaya, M.V, Sobolevsky, A.I.
登録日2021-08-27
公開日2021-10-27
最終更新日2022-02-16
実験手法ELECTRON MICROSCOPY (4.26 Å)
主引用文献Structure and desensitization of AMPA receptor complexes with type II TARP gamma 5 and GSG1L.
Mol.Cell, 81, 2021
7RZ6
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Structure of the complex of AMPA receptor GluA2 with auxiliary subunit TARP gamma-5 bound to agonist glutamate
分子名称: 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, GLUTAMIC ACID, Glutamate receptor 2
著者Klykov, O.V, Gangwar, S.P, Yelshanskaya, M.V, Sobolevsky, A.I.
登録日2021-08-27
公開日2021-10-27
最終更新日2022-02-16
実験手法ELECTRON MICROSCOPY (4.4 Å)
主引用文献Structure and desensitization of AMPA receptor complexes with type II TARP gamma 5 and GSG1L.
Mol.Cell, 81, 2021
7RYZ
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BU of 7ryz by Molmil
Structure of the complex of LBD-TMD part of AMPA receptor GluA2 with auxiliary subunit GSG1L bound to agonist quisqualate
分子名称: (S)-2-AMINO-3-(3,5-DIOXO-[1,2,4]OXADIAZOLIDIN-2-YL)-PROPIONIC ACID, Glutamate receptor 2
著者Gangwar, S.P, Klykov, O.V, Yelshanskaya, M.V, Sobolevsky, A.I.
登録日2021-08-26
公開日2021-10-27
最終更新日2022-02-16
実験手法ELECTRON MICROSCOPY (4.15 Å)
主引用文献Structure and desensitization of AMPA receptor complexes with type II TARP gamma 5 and GSG1L.
Mol.Cell, 81, 2021
7RZ5
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Structure of the complex of LBD-TMD part of AMPA receptor GluA2 with auxiliary subunit TARP gamma-5 bound to competitive antagonist ZK 200775
分子名称: 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, Glutamate receptor 2, {[7-morpholin-4-yl-2,3-dioxo-6-(trifluoromethyl)-3,4-dihydroquinoxalin-1(2H)-yl]methyl}phosphonic acid
著者Gangwar, S.P, Klykov, O.V, Yelshanskaya, M.V, Sobolevsky, A.I.
登録日2021-08-27
公開日2021-10-27
最終更新日2022-02-16
実験手法ELECTRON MICROSCOPY (3.3 Å)
主引用文献Structure and desensitization of AMPA receptor complexes with type II TARP gamma 5 and GSG1L.
Mol.Cell, 81, 2021
7RYY
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BU of 7ryy by Molmil
Structure of the complex of LBD-TMD part of AMPA receptor GluA2 with auxiliary subunit TARP gamma-5 bound to agonist glutamate
分子名称: 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, GLUTAMIC ACID, Glutamate receptor 2
著者Klykov, O.V, Gangwar, S.P, Yelshanskaya, M.V, Sobolevsky, A.I.
登録日2021-08-26
公開日2021-10-27
最終更新日2022-02-16
実験手法ELECTRON MICROSCOPY (4.4 Å)
主引用文献Structure and desensitization of AMPA receptor complexes with type II TARP gamma 5 and GSG1L.
Mol.Cell, 81, 2021
6DTT
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BU of 6dtt by Molmil
Apo T. maritima MalE2
分子名称: maltose-binding protein MalE2
著者Cuneo, M.J, Shukla, S.
登録日2018-06-18
公開日2018-09-19
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Differential Substrate Recognition by Maltose Binding Proteins Influenced by Structure and Dynamics.
Biochemistry, 57, 2018
7RZ9
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BU of 7rz9 by Molmil
Structure of the complex of AMPA receptor GluA2 with auxiliary subunit GSG1L in the apo state
分子名称: Glutamate receptor 2
著者Gangwar, S.P, Klykov, O.V, Yelshanskaya, M.V, Sobolevsky, A.I.
登録日2021-08-27
公開日2021-10-27
最終更新日2022-02-16
実験手法ELECTRON MICROSCOPY (4.15 Å)
主引用文献Structure and desensitization of AMPA receptor complexes with type II TARP gamma 5 and GSG1L.
Mol.Cell, 81, 2021
7RZ4
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BU of 7rz4 by Molmil
Structure of the complex of AMPA receptor GluA2 with auxiliary subunit TARP gamma-5 bound to competitive antagonist ZK 200775
分子名称: 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 2-acetamido-2-deoxy-beta-D-glucopyranose, Glutamate receptor 2, ...
著者Gangwar, S.P, Klykov, O.V, Yelshanskaya, M.V, Sobolevsky, A.I.
登録日2021-08-27
公開日2021-10-27
最終更新日2022-02-16
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献Structure and desensitization of AMPA receptor complexes with type II TARP gamma 5 and GSG1L.
Mol.Cell, 81, 2021
7DCL
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BU of 7dcl by Molmil
Crystal structure of the Zn-directed tetramer of the engineered cyt cb 562 variant, C96I/A38S AB5
分子名称: CHLORIDE ION, HEME C, ZINC ION, ...
著者Song, W.J, Yu, J.
登録日2020-10-26
公開日2021-03-03
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献Symmetry-related residues as promising hotspots for the evolution of de novo oligomeric enzymes.
Chem Sci, 12, 2021
7RZ7
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Structure of the complex of AMPA receptor GluA2 with auxiliary subunit TARP gamma-5 bound to agonist Quisqualate
分子名称: (S)-2-AMINO-3-(3,5-DIOXO-[1,2,4]OXADIAZOLIDIN-2-YL)-PROPIONIC ACID, Glutamate receptor 2
著者Klykov, O.V, Gangwar, S.P, Yelshanskaya, M.V, Sobolevsky, A.I.
登録日2021-08-27
公開日2021-10-27
最終更新日2022-02-16
実験手法ELECTRON MICROSCOPY (4.2 Å)
主引用文献Structure and desensitization of AMPA receptor complexes with type II TARP gamma 5 and GSG1L.
Mol.Cell, 81, 2021
6DW3
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SAMHD1 Bound to Cytarabine-TP in the Catalytic Pocket
分子名称: 2'-DEOXYADENOSINE 5'-TRIPHOSPHATE, 4-amino-1-{5-O-[(S)-hydroxy{[(R)-hydroxy(phosphonooxy)phosphoryl]oxy}phosphoryl]-beta-D-arabinofuranosyl}pyrimidin-2(1H)-one, Deoxynucleoside triphosphate triphosphohydrolase SAMHD1, ...
著者Knecht, K.M, Buzovetsky, O, Schneider, C, Thomas, D, Srikanth, V, Kaderali, L, Tofoleanu, F, Reiss, K, Ferreiros, N, Geisslinger, G, Batista, V.S, Ji, X, Cinatl, J, Keppler, O.T, Xiong, Y.
登録日2018-06-26
公開日2018-10-10
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献The structural basis for cancer drug interactions with the catalytic and allosteric sites of SAMHD1.
Proc. Natl. Acad. Sci. U.S.A., 115, 2018
7DCO
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BU of 7dco by Molmil
Cryo-EM structure of the activated spliceosome (Bact complex) at an atomic resolution of 2.5 angstrom
分子名称: BJ4_G0014900.mRNA.1.CDS.1, BJ4_G0027490.mRNA.1.CDS.1, BJ4_G0037700.mRNA.1.CDS.1, ...
著者Bai, R, Wan, R, Yan, C, Qi, J, Zhang, P, Lei, J, Shi, Y.
登録日2020-10-26
公開日2021-03-17
最終更新日2024-03-27
実験手法ELECTRON MICROSCOPY (2.5 Å)
主引用文献Mechanism of spliceosome remodeling by the ATPase/helicase Prp2 and its coactivator Spp2.
Science, 371, 2021
7KCB
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BU of 7kcb by Molmil
Symmetry in Yeast Alcohol Dehydrogenase 1 -Closed Form with NAD+ and Trifluoroethanol
分子名称: ADH1 isoform 1, NICOTINAMIDE-ADENINE-DINUCLEOTIDE, TRIFLUOROETHANOL, ...
著者Subramanian, R, Chang, L, Li, Z, Plapp, B.V.
登録日2020-10-05
公開日2021-03-31
実験手法ELECTRON MICROSCOPY (2.77 Å)
主引用文献Cryo-Electron Microscopy Structures of Yeast Alcohol Dehydrogenase.
Biochemistry, 60, 2021
7KCQ
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Symmetry in Yeast Alcohol Dehydrogenase 1 -Open Form of Apoenzyme
分子名称: Alcohol dehydrogenase, ZINC ION
著者Subramanian, R, Chang, L, Li, Z, Plapp, B.V.
登録日2020-10-07
公開日2021-03-31
実験手法ELECTRON MICROSCOPY (3.2 Å)
主引用文献Cryo-Electron Microscopy Structures of Yeast Alcohol Dehydrogenase.
Biochemistry, 60, 2021
2J21
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BU of 2j21 by Molmil
Human p53 core domain mutant M133L-V203A-N239Y-N268D-R282W
分子名称: CELLULAR TUMOR ANTIGEN P53, ZINC ION
著者Joerger, A.C, Fersht, A.R.
登録日2006-08-15
公開日2006-09-20
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structural Basis for Understanding Oncogenic P53 Mutations and Designing Rescue Drugs.
Proc.Natl.Acad.Sci.USA, 103, 2006
2J1Y
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Human p53 core domain mutant M133L-V203A-N239Y-G245S-N268D
分子名称: CALCIUM ION, CELLULAR TUMOR ANTIGEN P53, ZINC ION
著者Joerger, A.C, Fersht, A.R.
登録日2006-08-15
公開日2006-09-20
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.69 Å)
主引用文献Structural Basis for Understanding Oncogenic P53 Mutations and Designing Rescue Drugs.
Proc.Natl.Acad.Sci.USA, 103, 2006

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