7MU5
| Human DCTPP1 bound to Triptolide | 分子名称: | MAGNESIUM ION, dCTP pyrophosphatase 1, triptolide | 著者 | Hauk, G, Berger, J.M. | 登録日 | 2021-05-14 | 公開日 | 2022-08-24 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Triptolide sensitizes cancer cells to nucleoside DNA methyltransferase inhibitors through inhibition of DCTPP1 mediated cell-intrinsic resistance To Be Published
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7AKW
| Crystal structure of the viral rhodopsins chimera O1O2 | 分子名称: | EICOSANE, RETINAL, chimera of viral rhodopsins OLPVR1 and OLPVRII | 著者 | Kovalev, K, Zabelskii, D, Alekseev, A, Astashkin, R, Gordeliy, V. | 登録日 | 2020-10-02 | 公開日 | 2020-11-25 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.96 Å) | 主引用文献 | Viral rhodopsins 1 are an unique family of light-gated cation channels. Nat Commun, 11, 2020
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7AKY
| Crystal structure of the viral rhodopsin OLPVR1 in P21212 space group | 分子名称: | (2S)-2,3-dihydroxypropyl (9Z)-hexadec-9-enoate, EICOSANE, viral rhodopsin OLPVR1 | 著者 | Kovalev, K, Zabelskii, D, Alekseev, A, Astashkin, R, Gordeliy, V. | 登録日 | 2020-10-02 | 公開日 | 2020-11-25 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | Viral rhodopsins 1 are an unique family of light-gated cation channels. Nat Commun, 11, 2020
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7AKX
| Crystal structure of the viral rhodopsin OLPVR1 in P1 space group | 分子名称: | (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, EICOSANE, OLEIC ACID, ... | 著者 | Kovalev, K, Zabelskii, D, Alekseev, A, Astashkin, R, Gordeliy, V. | 登録日 | 2020-10-02 | 公開日 | 2020-11-25 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Viral rhodopsins 1 are an unique family of light-gated cation channels. Nat Commun, 11, 2020
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7EDB
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5HGO
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7E8I
| Structural insight into BRCA1-BARD1 complex recruitment to damaged chromatin | 分子名称: | BRCA1-associated RING domain protein 1, DNA (145-MER), Histone H2A, ... | 著者 | Dai, Y, Dai, L, Zhou, Z. | 登録日 | 2021-03-01 | 公開日 | 2021-06-30 | 最終更新日 | 2024-03-27 | 実験手法 | ELECTRON MICROSCOPY (3.1 Å) | 主引用文献 | Structural insight into BRCA1-BARD1 complex recruitment to damaged chromatin. Mol.Cell, 81, 2021
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5HGK
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5D7D
| Crystal structure of the ATP binding domain of S. aureus GyrB complexed with a ligand | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, 7-propyl-3-[2-(pyridin-3-yl)-1,3-thiazol-5-yl]-1,7-dihydro-6H-pyrazolo[3,4-b]pyridin-6-one, CHLORIDE ION, ... | 著者 | Zhang, J, Yang, Q, Cross, J.B, Romero, J.A.C, Ryan, M.D, Lippa, B, Dolle, R.E, Andersen, O.A, Barker, J, Cheng, R.K, Kahmann, J, Felicetti, B, Wood, M, Scheich, C. | 登録日 | 2015-08-13 | 公開日 | 2015-11-11 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Discovery of Indazole Derivatives as a Novel Class of Bacterial Gyrase B Inhibitors. Acs Med.Chem.Lett., 6, 2015
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5HGM
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1HT7
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5HGN
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5HGL
| Hexameric HIV-1 CA, open conformation | 分子名称: | CHLORIDE ION, Capsid protein P24, N-METHYL-NALPHA-[(2-METHYL-1H-INDOL-3-YL)ACETYL]-N-PHENYL-L-PHENYLALANINAMIDE | 著者 | Price, A.J, Jacques, D.A, James, L.C. | 登録日 | 2016-01-08 | 公開日 | 2016-08-10 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | HIV-1 uses dynamic capsid pores to import nucleotides and fuel encapsidated DNA synthesis. Nature, 536, 2016
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5D7R
| Crystal structure of the ATP binding domain of S. aureus GyrB complexed with a ligand | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, 3-hydroxy-5-[5-(6-hydroxy-7-propyl-2H-indazol-3-yl)-1,3-thiazol-2-yl]pyridine-2-carboxylic acid, CHLORIDE ION, ... | 著者 | Zhang, J, Yang, Q, Cross, J.B, Romero, J.A.C, Ryan, M.D, Lippa, B, Dolle, R.E, Andersen, O.A, Barker, J, Cheng, R.K, Kahmann, J, Felicetti, B, Wood, M, Scheich, C. | 登録日 | 2015-08-14 | 公開日 | 2015-11-18 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Discovery of Indazole Derivatives as a Novel Class of Bacterial Gyrase B Inhibitors. Acs Med.Chem.Lett., 6, 2015
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1K8J
| NMR STRUCTURE OF THE CK14 DNA DUPLEX: A PORTION OF THE KNOWN NF-kB SEQUENCE CK1 | 分子名称: | FIRST STRAND OF CK14 DNA DUPLEX, SECOND STRAND OF CK14 DNA DUPLEX | 著者 | Volk, D.E, Yang, X, Fennewald, S.M, King, D.J, Bassett, S.E, Venkitachalam, S, Herzog, N, Luxon, B.A, Gorenstein, D.G. | 登録日 | 2001-10-24 | 公開日 | 2003-04-15 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure and design of dithiophosphate backbone aptamers targeting transcription factor NF-kappaB Bioorg.Chem., 30, 2002
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1OYW
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1OYY
| Structure of the RecQ Catalytic Core bound to ATP-gamma-S | 分子名称: | ATP-dependent DNA helicase, MANGANESE (II) ION, PHOSPHOTHIOPHOSPHORIC ACID-ADENYLATE ESTER, ... | 著者 | Bernstein, D.A, Zittel, M.C, Keck, J.L. | 登録日 | 2003-04-07 | 公開日 | 2003-10-07 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | High-resolution structure of the E. coli RecQ helicase catalytic core Embo J., 22, 2003
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5HGP
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4CYB
| DpsC from Streptomyces coelicolor | 分子名称: | FE (III) ION, PUTATIVE DNA PROTECTION PROTEIN, SODIUM ION | 著者 | Townsend, P.D, Hitchings, M.D, Del Sol, R, Pohl, E. | 登録日 | 2014-04-10 | 公開日 | 2014-06-25 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.78 Å) | 主引用文献 | A Tale of Tails: Deciphering the Contribution of Terminal Tails to the Biochemical Properties of Two Dps Proteins from Streptomyces Coelicolor Cell.Mol.Life Sci., 71, 2014
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4BAE
| Optimisation of pyrroleamides as mycobacterial GyrB ATPase inhibitors: Structure Activity Relationship and in vivo efficacy in the mouse model of tuberculosis | 分子名称: | 2-[(3S,4R)-4-[(3-bromanyl-4-chloranyl-5-methyl-1H-pyrrol-2-yl)carbonylamino]-3-methoxy-piperidin-1-yl]-4-(2-methyl-1,2,4-triazol-3-yl)-1,3-thiazole-5-carboxylic acid, CALCIUM ION, DNA GYRASE SUBUNIT B, ... | 著者 | Read, J.A, Gingell, H.G, Madhavapeddi, P. | 登録日 | 2012-09-13 | 公開日 | 2013-10-30 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.35 Å) | 主引用文献 | Optimization of Pyrrolamides as Mycobacterial Gyrb ATPase Inhibitors: Structure Activity Relationship and in Vivo Efficacy in the Mouse Model of Tuberculosis. Antimicrob.Agents Chemother., 58, 2014
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4DA2
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2ETX
| Crystal Structure of MDC1 Tandem BRCT Domains | 分子名称: | Mediator of DNA damage checkpoint protein 1 | 著者 | Wasielewski, E, Kim, Y, Joachimiak, A, Thompson, J.R, Mer, G. | 登録日 | 2005-10-27 | 公開日 | 2005-11-15 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.33 Å) | 主引用文献 | Molecular Basis for the Association of Microcephalin (MCPH1) Protein with the Cell Division Cycle Protein 27 (Cdc27) Subunit of the Anaphase-promoting Complex. J.Biol.Chem., 287, 2012
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1KG6
| Crystal structure of the K142R mutant of E.coli MutY (core fragment) | 分子名称: | A/G-specific adenine glycosylase, GLYCEROL, IRON/SULFUR CLUSTER, ... | 著者 | Gilboa, R, Kilshtein, A, Zharkov, D.O, Kycia, J.H, Gerchman, S.E, Grollman, A.P, Shoham, G. | 登録日 | 2001-11-26 | 公開日 | 2002-11-26 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Analysis of the E.coli MutY DNA glycosylase structure and function by site-directed mutagenesis To be Published
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1KG4
| Crystal structure of the K142A mutant of E. coli MutY (core fragment) | 分子名称: | A/G-specific adenine glycosylase, GLYCEROL, IRON/SULFUR CLUSTER, ... | 著者 | Gilboa, R, Kilshtein, A, Zharkov, D.O, Kycia, J.H, Gerchman, S.E, Grollman, A.P, Shoham, G. | 登録日 | 2001-11-26 | 公開日 | 2002-11-26 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Analysis of the E.coli MutY DNA glycosylase structure and function by site-directed mutagenesis To be Published
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1KG3
| Crystal structure of the core fragment of MutY from E.coli at 1.55A resolution | 分子名称: | A/G-specific adenine glycosylase, GLYCEROL, IRON/SULFUR CLUSTER, ... | 著者 | Gilboa, R, Kilshtein, A, Zharkov, D.O, Kycia, J.H, Gerchman, S.E, Grollman, A.P, Shoham, G. | 登録日 | 2001-11-26 | 公開日 | 2002-11-26 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Analysis of the E.coli MutY DNA glycosylase structure and function by site-directed mutagenesis To be Published
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