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2GV2
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MDM2 in complex with an 8-mer p53 peptide analogue
分子名称: 8-MER P53 PEPTIDE ANALOGUE, E3 ubiquitin-protein ligase Mdm2
著者Schubert, C, Sakurai, K.
登録日2006-05-02
公開日2006-09-05
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Crystallographic Analysis of an 8-mer p53 Peptide Analogue Complexed with MDM2.
J.Am.Chem.Soc., 128, 2006
2HBD
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BU of 2hbd by Molmil
HIGH RESOLUTION X-RAY STRUCTURES OF MYOGLOBIN-AND HEMOGLOBIN-ALKYL ISOCYANIDE COMPLEXES
分子名称: HEMOGLOBIN A (METHYL ISOCYANIDE) (ALPHA CHAIN), HEMOGLOBIN A (METHYL ISOCYANIDE) (BETA CHAIN), METHYL ISOCYANIDE, ...
著者Johnson, K.A, Olson, J.S, Phillips Jr, G.N.
登録日1994-08-31
公開日1995-02-07
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献High Resolution X-Ray Structures of Myoglobin-and Hemoglobin-Alkyl Isocyanide Complexes
Thesis, 1, 1993
2GWX
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MOLECULAR RECOGNITION OF FATTY ACIDS BY PEROXISOME PROLIFERATOR-ACTIVATED RECEPTORS
分子名称: PROTEIN (PPAR-DELTA)
著者Xu, H.E, Lambert, M.H, Montana, V.G, Park, D.J, Blanchard, S, Brown, P, Sternbach, D, Lehmann, J, Bruce, G.W, Willson, T.M, Kliewer, S.A, Milburn, M.V.
登録日1999-03-11
公開日2000-03-11
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Molecular recognition of fatty acids by peroxisome proliferator-activated receptors.
Mol.Cell, 3, 1999
2HMG
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REFINEMENT OF THE INFLUENZA VIRUS HEMAGGLUTININ BY SIMULATED ANNEALING
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, HEMAGGLUTININ (HA1 CHAIN), HEMAGGLUTININ (HA2 CHAIN), ...
著者Weis, W.I, Bruenger, A.T, Skehel, J.J, Wiley, D.C.
登録日1989-09-11
公開日1991-01-15
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Refinement of the influenza virus hemagglutinin by simulated annealing.
J.Mol.Biol., 212, 1990
2PWG
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Crystal Structure of the Trehalulose Synthase MutB From Pseudomonas Mesoacidophila MX-45 Complexed to the Inhibitor Castanospermine
分子名称: CALCIUM ION, CASTANOSPERMINE, Sucrose isomerase
著者Ravaud, S, Robert, X, Haser, R, Aghajari, N.
登録日2007-05-11
公開日2007-06-26
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Trehalulose synthase native and carbohydrate complexed structures provide insights into sucrose isomerization.
J.Biol.Chem., 61, 2007
4CLA
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ALTERNATIVE BINDING MODES FOR CHLORAMPHENICOL AND 1-SUBSTITUTED CHLORAMPHENICOL ANALOGUES REVEALED BY SITE-DIRECTED MUTAGENESIS AND X-RAY CRYSTALLOGRAPHY OF CHLORAMPHENICOL ACETYLTRANSFERASE
分子名称: CHLORAMPHENICOL, COBALT (II) ION, TYPE III CHLORAMPHENICOL ACETYLTRANSFERASE
著者Leslie, A.G.W.
登録日1990-10-23
公開日1992-01-15
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Alternative binding modes for chloramphenicol and 1-substituted chloramphenicol analogues revealed by site-directed mutagenesis and X-ray crystallography of chloramphenicol acetyltransferase.
Biochemistry, 30, 1991
2HP2
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Inter-subunit signaling in GSAM
分子名称: (4R)-5-AMINO-4-[({3-HYDROXY-2-METHYL-5-[(PHOSPHONOOXY)METHYL]PYRIDIN-4-YL}METHYL)AMINO]PENTANOIC ACID, (4S)-4,5-DIAMINOPENTANOIC ACID, Glutamate-1-semialdehyde 2,1-aminomutase (GSAM) hybrid-form, ...
著者Stetefeld, J.
登録日2006-07-17
公開日2006-08-22
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Intersubunit signaling in glutamate-1-semialdehyde-aminomutase.
Proc.Natl.Acad.Sci.Usa, 103, 2006
2HOL
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Crystal structure of an E. coli thi-box riboswitch bound to thiamine pyrophosphate, barium ions
分子名称: BARIUM ION, CALCIUM ION, MAGNESIUM ION, ...
著者Edwards, T.E, Ferre-D'Amare, A.R.
登録日2006-07-14
公開日2006-09-19
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Crystal Structures of the Thi-Box Riboswitch Bound to Thiamine Pyrophosphate Analogs Reveal Adaptive RNA-Small Molecule Recognition
Structure, 14, 2006
2HOW
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Dipeptidase (PH0974) from Pyrococcus horikoshii OT3
分子名称: 356aa long hypothetical dipeptidase
著者Jeyakanthan, J, Yokoyama, S, Shiro, Y, Yutani, K, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2006-07-17
公開日2007-09-11
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Dipeptidase (PH0974) from Pyrococcus Horikoshii Ot3
To be Published
4OAR
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BU of 4oar by Molmil
Progesterone receptor with bound ulipristal acetate and a peptide from the co-repressor SMRT
分子名称: Peptide from Nuclear receptor corepressor 2, Progesterone receptor, [(8S,11R,13S,14S,17R)-17-acetyl-11-[4-(dimethylamino)phenyl]-13-methyl-3-oxo-1,2,6,7,8,11,12,14,15,16-decahydrocyclopen ta[a]phenanthren-17-yl] acetate
著者Petit-Topin, I, Fay, M.R, Resche-Rigon, M, Ulmann, A, Gainer, E, Rafestin-Oblin, M.-E, Fagart, J.
登録日2014-01-06
公開日2014-10-08
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.41 Å)
主引用文献Molecular determinants of the recognition of ulipristal acetate by oxo-steroid receptors.
J.Steroid Biochem.Mol.Biol., 144PB, 2014
4F9M
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BU of 4f9m by Molmil
Crystal structure of the PPARgamma-LBD complexed with a cercosporamide derivative modulator
分子名称: (9aS)-8-acetyl-N-[(2-ethyl-4-fluoronaphthalen-1-yl)methyl]-1,7-dihydroxy-3-methoxy-9a-methyl-9-oxo-9,9a-dihydrodibenzo[b,d]furan-4-carboxamide, Peroxisome proliferator-activated receptor gamma, peptide from Nuclear receptor coactivator 1
著者Matsui, Y, Hanzawa, H.
登録日2012-05-19
公開日2012-08-08
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Synthesis and biological evaluation of novel (-)-cercosporamide derivatives as potent selective PPARg modulators
Eur.J.Med.Chem., 54, 2012
2HOZ
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Inter-subunit signaling in GSAM
分子名称: (4S)-4,5-DIAMINOPENTANOIC ACID, 4'-DEOXY-4'-AMINOPYRIDOXAL-5'-PHOSPHATE, Glutamate-1-semialdehyde 2,1-aminomutase (GSAM) pmp-form
著者Stetefeld, J.
登録日2006-07-17
公開日2006-08-22
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Intersubunit signaling in glutamate-1-semialdehyde-aminomutase.
Proc.Natl.Acad.Sci.Usa, 103, 2006
2HNZ
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Crystal Structure of E138K Mutant HIV-1 Reverse Transcriptase in Complex with PETT-2
分子名称: 1-[2-(4-ETHOXY-3-FLUOROPYRIDIN-2-YL)ETHYL]-3-(5-METHYLPYRIDIN-2-YL)THIOUREA, PHOSPHATE ION, Reverse transcriptase/ribonuclease H
著者Ren, J, Nichols, C.E, Stamp, A, Chamberlain, P.P, Stammers, D.K.
登録日2006-07-13
公開日2006-09-05
最終更新日2021-10-20
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Structural insights into mechanisms of non-nucleoside drug resistance for HIV-1 reverse transcriptases mutated at codons 101 or 138.
Febs J., 273, 2006
2HMI
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BU of 2hmi by Molmil
HIV-1 REVERSE TRANSCRIPTASE/FRAGMENT OF FAB 28/DNA COMPLEX
分子名称: DNA (5'-D(*AP*TP*GP*GP*CP*GP*CP*CP*CP*GP*AP*AP*CP*AP*GP*GP*GP*AP*C)-3'), DNA (5'-D(*GP*TP*CP*CP*CP*TP*GP*TP*TP*CP*GP*GP*GP*CP*GP*CP*CP*A)-3'), FAB FRAGMENT OF MONOCLONAL ANTIBODY 28, ...
著者Ding, J, Arnold, E.
登録日1998-04-10
公開日1998-10-14
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structure and functional implications of the polymerase active site region in a complex of HIV-1 RT with a double-stranded DNA template-primer and an antibody Fab fragment at 2.8 A resolution.
J.Mol.Biol., 284, 1998
2HOO
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Crystal structure of an E. coli thi-box riboswitch bound to benfotiamine
分子名称: CALCIUM ION, S-BENZOYLTHIAMINE O-MONOPHOSPHATE, thi-box riboswitch
著者Edwards, T.E, Ferre-D'Amare, A.R.
登録日2006-07-14
公開日2006-09-19
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Crystal Structures of the Thi-Box Riboswitch Bound to Thiamine Pyrophosphate Analogs Reveal Adaptive RNA-Small Molecule Recognition
Structure, 14, 2006
2HOY
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BU of 2hoy by Molmil
Inter-subunit signaling in GSAM
分子名称: Glutamate-1-semialdehyde 2,1-aminomutase (GSAM) apo-form, PHOSPHATE ION
著者Stetefeld, J.
登録日2006-07-17
公開日2006-08-22
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Intersubunit signaling in glutamate-1-semialdehyde-aminomutase.
Proc.Natl.Acad.Sci.Usa, 103, 2006
2HPA
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BU of 2hpa by Molmil
STRUCTURAL ORIGINS OF L(+)-TARTRATE INHIBITION OF HUMAN PROSTATIC ACID PHOSPHATASE
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, N-PROPYL-TARTRAMIC ACID, ...
著者Lacount, M.W, Handy, G, Lebioda, L.
登録日1998-09-11
公開日1998-09-16
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Structural origins of L(+)-tartrate inhibition of human prostatic acid phosphatase.
J.Biol.Chem., 273, 1998
2HQL
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BU of 2hql by Molmil
Crystal structure of a small single-stranded DNA binding protein from Mycoplasma pneumoniae
分子名称: Hypothetical protein MG376 homolog
著者Das, D, Berkeley Structural Genomics Center (BSGC)
登録日2006-07-18
公開日2007-05-01
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal structure of a novel single-stranded DNA binding protein from Mycoplasma pneumoniae.
Proteins, 67, 2007
2HW8
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BU of 2hw8 by Molmil
Structure of ribosomal protein L1-mRNA complex at 2.1 resolution.
分子名称: 1,4-BUTANEDIOL, 36-MER, 50S ribosomal protein L1, ...
著者Tishchenko, S, Nikonova, E, Nikulin, A, Nevskaya, N, Volchkov, S, Piendl, W, Garber, M, Nikonov, S.
登録日2006-08-01
公開日2006-12-19
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Structure of the ribosomal protein L1-mRNA complex at 2.1 A resolution: common features of crystal packing of L1-RNA complexes.
ACTA CRYSTALLOGR.,SECT.D, 62, 2006
4DKN
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BU of 4dkn by Molmil
Crystal structure of amphioxus green fluorescent protein, GFPA1
分子名称: AMPHIOXUS GREEN FLUORESCENT PROTEIN, GFPA1
著者Bomati, E.K, Deheyn, D.D.
登録日2012-02-03
公開日2013-05-15
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (1.35 Å)
主引用文献Fluorescent proteins in Amphioxus have strickingly different brightness, yet only few (but key) molecular differences
To be Published
2OTC
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BU of 2otc by Molmil
ORNITHINE TRANSCARBAMOYLASE COMPLEXED WITH N-(PHOSPHONACETYL)-L-ORNITHINE
分子名称: N-(PHOSPHONOACETYL)-L-ORNITHINE, ORNITHINE CARBAMOYLTRANSFERASE
著者Ha, Y, Allewell, N.M.
登録日1997-06-15
公開日1998-06-17
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Substrate-induced conformational change in a trimeric ornithine transcarbamoylase.
Proc.Natl.Acad.Sci.USA, 94, 1997
4E13
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Substrate-directed dual catalysis of dicarbonyl compounds by diketoreductase
分子名称: Diketoreductase, GLYCEROL, NICOTINAMIDE-ADENINE-DINUCLEOTIDE, ...
著者Lu, M, White, M.A, Huang, Y, Wu, X, Liu, N, Cheng, X, Chen, Y.
登録日2012-03-05
公開日2012-11-14
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.08 Å)
主引用文献Dual catalysis mode for the dicarbonyl reduction catalyzed by diketoreductase
Chem.Commun.(Camb.), 48, 2012
2KCE
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BU of 2kce by Molmil
BINDING OF THE ANTICANCER DRUG ZD1694 TO E. COLI THYMIDYLATE SYNTHASE: ASSESSING SPECIFICITY AND AFFINITY
分子名称: 2'-DEOXYURIDINE 5'-MONOPHOSPHATE, THYMIDYLATE SYNTHASE, TOMUDEX
著者Rutenber, E.E, Stroud, R.M.
登録日1997-06-09
公開日1997-11-19
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Binding of the anticancer drug ZD1694 to E. coli thymidylate synthase: assessing specificity and affinity.
Structure, 4, 1996
2KAU
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BU of 2kau by Molmil
THE CRYSTAL STRUCTURE OF UREASE FROM KLEBSIELLA AEROGENES AT 2.2 ANGSTROMS RESOLUTION
分子名称: NICKEL (II) ION, UREASE (ALPHA CHAIN), UREASE (BETA CHAIN), ...
著者Jabri, E, Carr, M.B, Hausinger, R.P, Karplus, P.A.
登録日1995-02-16
公開日1995-07-10
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献The crystal structure of urease from Klebsiella aerogenes.
Science, 268, 1995
2LBD
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LIGAND-BINDING DOMAIN OF THE HUMAN RETINOIC ACID RECEPTOR GAMMA BOUND TO ALL-TRANS RETINOIC ACID
分子名称: RETINOIC ACID, RETINOIC ACID RECEPTOR GAMMA
著者Renaud, J.-P, Rochel, N, Ruff, M, Moras, D, Structural Proteomics in Europe (SPINE)
登録日1997-08-19
公開日1997-11-12
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.06 Å)
主引用文献Crystal structure of the RAR-gamma ligand-binding domain bound to all-trans retinoic acid.
Nature, 378, 1995

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