4DEB
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![BU of 4deb by Molmil](/molmil-images/mine/4deb) | Aurora A in complex with RK2-17-01 | 分子名称: | 1,2-ETHANEDIOL, 4-[(4-{[3-(trifluoromethyl)phenyl]amino}pyrimidin-2-yl)amino]benzamide, Aurora kinase A | 著者 | Martin, M.P, Zhu, J.-Y, Schonbrunn, E. | 登録日 | 2012-01-20 | 公開日 | 2012-08-22 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (3.05 Å) | 主引用文献 | Development of o-Chlorophenyl Substituted Pyrimidines as Exceptionally Potent Aurora Kinase Inhibitors. J.Med.Chem., 55, 2012
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2ISE
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4TMK
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4N7X
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4C2C
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![BU of 4c2c by Molmil](/molmil-images/mine/4c2c) | Crystal structure of the protease CtpB in an active state | 分子名称: | CARBOXY-TERMINAL PROCESSING PROTEASE CTPB, PEPTIDE1, PEPTIDE2 | 著者 | Mastny, M, Heuck, A, Kurzbauer, R, Clausen, T. | 登録日 | 2013-08-17 | 公開日 | 2013-12-04 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Ctpb Assembles a Gated Protease Tunnel Regulating Cell-Cell Signaling During Spore Formation in Bacillus Subtilis. Cell(Cambridge,Mass.), 155, 2013
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4SRN
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![BU of 4srn by Molmil](/molmil-images/mine/4srn) | STRUCTURAL CHANGES THAT ACCOMPANY THE REDUCED CATALYTIC EFFICIENCY OF TWO SEMISYNTHETIC RIBONUCLEASE ANALOGS | 分子名称: | RIBONUCLEASE A, SULFATE ION | 著者 | deMel, V.S.J, Martin, P.D, Doscher, M.S, Edwards, B.F.P. | 登録日 | 1991-05-20 | 公開日 | 1994-12-20 | 最終更新日 | 2019-08-14 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structural changes that accompany the reduced catalytic efficiency of two semisynthetic ribonuclease analogs. J.Biol.Chem., 267, 1992
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5NN9
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![BU of 5nn9 by Molmil](/molmil-images/mine/5nn9) | REFINED ATOMIC STRUCTURES OF N9 SUBTYPE INFLUENZA VIRUS NEURAMINIDASE AND ESCAPE MUTANTS | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, NEURAMINIDASE N9, ... | 著者 | Tulip, W.R, Varghese, J.N, Baker, A.T, Vandonkelaar, A, Laver, W.G, Webster, R.G, Colman, P.M. | 登録日 | 1991-03-28 | 公開日 | 1992-07-15 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Refined atomic structures of N9 subtype influenza virus neuraminidase and escape mutants. J.Mol.Biol., 221, 1991
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4ROM
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![BU of 4rom by Molmil](/molmil-images/mine/4rom) | Deoxyhemoglobin in complex with imidazolylacryloyl derivatives | 分子名称: | 4-{2-chloro-4-[3-(1H-imidazol-2-yl)propanoyl]phenoxy}butanoic acid, Hemoglobin subunit alpha, Hemoglobin subunit beta, ... | 著者 | Omar, A.M, Mahran, M.A, Ghatge, M.N, Chowdhury, N, Bamane, F.H.A, El-Araby, M.E, Abdulmalik, O, Safo, M.K. | 登録日 | 2014-10-28 | 公開日 | 2015-05-20 | 最終更新日 | 2015-06-10 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Identification of a novel class of covalent modifiers of hemoglobin as potential antisickling agents. Org.Biomol.Chem., 13, 2015
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4STD
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![BU of 4std by Molmil](/molmil-images/mine/4std) | HIGH RESOLUTION STRUCTURES OF SCYTALONE DEHYDRATASE-INHIBITOR COMPLEXES CRYSTALLIZED AT PHYSIOLOGICAL PH | 分子名称: | N-[1-(4-BROMOPHENYL)ETHYL]-5-FLUORO SALICYLAMIDE, Scytalone dehydratase | 著者 | Wawrzak, Z, Sandalova, T, Steffens, J.J, Basarab, G.S, Lundqvist, T, Lindqvist, Y, Jordan, D.B. | 登録日 | 1999-02-10 | 公開日 | 1999-12-29 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | 主引用文献 | High-resolution structures of scytalone dehydratase-inhibitor complexes crystallized at physiological pH. Proteins, 35, 1999
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4THI
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![BU of 4thi by Molmil](/molmil-images/mine/4thi) | THIAMINASE I FROM BACILLUS THIAMINOLYTICUS WITH COVALENTLY BOUND 4-AMINO-2,5-DIMETHYLPYRIMIDINE | 分子名称: | 2,5-DIMETHYL-PYRIMIDIN-4-YLAMINE, PROTEIN (THIAMINASE I), SULFATE ION | 著者 | Campobasso, N, Begley, T.P, Ealick, S.E. | 登録日 | 1998-10-05 | 公開日 | 1998-10-14 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Crystal structure of thiaminase-I from Bacillus thiaminolyticus at 2.0 A resolution. Biochemistry, 37, 1998
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4C2G
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![BU of 4c2g by Molmil](/molmil-images/mine/4c2g) | Crystal structure of CtpB(S309A) in complex with a peptide having a Val-Pro-Ala C-terminus | 分子名称: | CARBOXY-TERMINAL PROCESSING PROTEASE CTPB, PEPTIDE1 | 著者 | Mastny, M, Heuck, A, Kurzbauer, R, Clausen, T. | 登録日 | 2013-08-17 | 公開日 | 2013-12-04 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Ctpb Assembles a Gated Protease Tunnel Regulating Cell-Cell Signaling During Spore Formation in Bacillus Subtilis. Cell(Cambridge,Mass.), 155, 2013
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2I7N
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![BU of 2i7n by Molmil](/molmil-images/mine/2i7n) | Crystal structure of human PANK1 alpha: the catalytic core domain in complex with AcCoA | 分子名称: | ACETYL COENZYME *A, Pantothenate kinase 1 | 著者 | Hong, B.S, Wang, L, Tempel, W, Loppnau, P, Allali-Hassani, A, Arrowsmith, C.H, Edwards, A.M, Sundstrom, M, Weigelt, J, Bochkarev, A, Park, H.W. | 登録日 | 2006-08-31 | 公開日 | 2006-12-26 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Crystal structures of human pantothenate kinases. Insights into allosteric regulation and mutations linked to a neurodegeneration disorder. J.Biol.Chem., 282, 2007
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5MHT
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![BU of 5mht by Molmil](/molmil-images/mine/5mht) | TERNARY STRUCTURE OF HHAI METHYLTRANSFERASE WITH HEMIMETHYLATED DNA AND ADOHCY | 分子名称: | DNA (5'-D(*CP*CP*AP*TP*GP*(5CM)P*GP*CP*TP*GP*AP*C)-3'), DNA (5'-D(*GP*TP*CP*AP*GP*CP*GP*CP*AP*TP*GP*G)-3'), PROTEIN (HHAI METHYLTRANSFERASE), ... | 著者 | Cheng, X. | 登録日 | 1996-10-22 | 公開日 | 1997-07-23 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | A structural basis for the preferential binding of hemimethylated DNA by HhaI DNA methyltransferase. J.Mol.Biol., 263, 1996
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7PA0
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![BU of 7pa0 by Molmil](/molmil-images/mine/7pa0) | NaK C-DI F92A mutant with Rb+ and K+ | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, POTASSIUM ION, Potassium channel protein, ... | 著者 | Minniberger, S, Plested, A.J.R. | 登録日 | 2021-07-28 | 公開日 | 2022-08-10 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Asymmetry and Ion Selectivity Properties of Bacterial Channel NaK Mutants Derived from Ionotropic Glutamate Receptors. J.Mol.Biol., 435, 2023
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4SLI
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![BU of 4sli by Molmil](/molmil-images/mine/4sli) | LEECH INTRAMOLECULAR TRANS-SIALIDASE COMPLEXED WITH 2-PROPENYL-NEU5AC, AN INACTIVE SUBSTRATE ANALOGUE | 分子名称: | 2-propenyl-N-acetyl-neuraminic acid, INTRAMOLECULAR TRANS-SIALIDASE | 著者 | Luo, Y, Li, S.C, Li, Y.T, Luo, M. | 登録日 | 1998-10-04 | 公開日 | 1999-05-25 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | The 1.8 A structures of leech intramolecular trans-sialidase complexes: evidence of its enzymatic mechanism. J.Mol.Biol., 285, 1999
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2K9P
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6IZM
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![BU of 6izm by Molmil](/molmil-images/mine/6izm) | Crystal structure of the PPARgamma-LBD complexed with compound 1l | 分子名称: | 3-[[6-(2,6-dimethylpyridin-3-yl)oxy-1-methyl-benzimidazol-2-yl]methoxy]benzoic acid, Peptide from Peroxisome proliferator-activated receptor gamma coactivator 1-alpha, Peroxisome proliferator-activated receptor gamma | 著者 | Matsui, Y, Hanzawa, H. | 登録日 | 2018-12-20 | 公開日 | 2019-03-27 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Structure-Activity Relationship Studies of 3- or 4-Pyridine Derivatives of DS-6930. Acs Med.Chem.Lett., 10, 2019
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4RLA
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4DEE
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![BU of 4dee by Molmil](/molmil-images/mine/4dee) | Aurora A in complex with ADP | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, Aurora kinase A, MAGNESIUM ION | 著者 | Martin, M.P, Zhu, J.-Y, Schonbrunn, E. | 登録日 | 2012-01-20 | 公開日 | 2012-08-22 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Development of o-Chlorophenyl Substituted Pyrimidines as Exceptionally Potent Aurora Kinase Inhibitors. J.Med.Chem., 55, 2012
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4TPI
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![BU of 4tpi by Molmil](/molmil-images/mine/4tpi) | THE REFINED 2.2-ANGSTROMS (0.22-NM) X-RAY CRYSTAL STRUCTURE OF THE TERNARY COMPLEX FORMED BY BOVINE TRYPSINOGEN, VALINE-VALINE AND THE ARG15 ANALOGUE OF BOVINE PANCREATIC TRYPSIN INHIBITOR | 分子名称: | BOVINE PANCREATIC TRYPSIN INHIBITOR, CALCIUM ION, SULFATE ION, ... | 著者 | Bode, W, Walter, J. | 登録日 | 1985-06-11 | 公開日 | 1985-11-08 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | The refined 2.2-A (0.22-nm) X-ray crystal structure of the ternary complex formed by bovine trypsinogen, valine-valine and the Arg15 analogue of bovine pancreatic trypsin inhibitor Eur.J.Biochem., 144, 1984
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2H2K
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![BU of 2h2k by Molmil](/molmil-images/mine/2h2k) | Crystal Structure Analysis of Human S100A13 | 分子名称: | CALCIUM ION, Protein S100-A13 | 著者 | Li, M, Zhang, P.F, Zhang, J.P, Chang, W.R. | 登録日 | 2006-05-19 | 公開日 | 2007-05-22 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Crystal structure study on human S100A13 at 2.0 A resolution Biochem.Biophys.Res.Commun., 356, 2007
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4TWZ
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![BU of 4twz by Molmil](/molmil-images/mine/4twz) | Crystal Structure Analysis of E Coli. RecA Protein | 分子名称: | MAGNESIUM ION, Protein RecA | 著者 | Hikima, T, Hiraki, T, Furuse, M, Ikawa, S, Iwasaki, W, Shibata, T, Kamiya, N. | 登録日 | 2014-07-02 | 公開日 | 2015-07-08 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Loop L1 governs the DNA-binding specificity and order for RecA-catalyzed reactions in homologous recombination and DNA repair Nucleic Acids Res., 43, 2015
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6HBW
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4SKN
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![BU of 4skn by Molmil](/molmil-images/mine/4skn) | A NUCLEOTIDE-FLIPPING MECHANISM FROM THE STRUCTURE OF HUMAN URACIL-DNA GLYCOSYLASE BOUND TO DNA | 分子名称: | DNA (5'-D(*AP*AP*AP*GP*CP*CP*GP*CP*CP*C)-3'), DNA (5'-D(*TP*GP*GP*GP*(D1P)P*GP*GP*CP*TP*T)-3'), PROTEIN (URACIL-DNA GLYCOSYLASE), ... | 著者 | Slupphaug, G, Mol, C.D, Kavli, B, Arvai, A.S, Krokan, H.E, Tainer, J.A. | 登録日 | 1999-02-20 | 公開日 | 1999-02-26 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | A nucleotide-flipping mechanism from the structure of human uracil-DNA glycosylase bound to DNA. Nature, 384, 1996
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4C2F
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![BU of 4c2f by Molmil](/molmil-images/mine/4c2f) | Crystal structure of the CtpB R168A mutant present in an active conformation | 分子名称: | CARBOXY-TERMINAL PROCESSING PROTEASE CTPB, PEPTIDE1, PEPTIDE2 | 著者 | Mastny, M, Heuck, A, Kurzbauer, R, Clausen, T. | 登録日 | 2013-08-17 | 公開日 | 2013-12-04 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Ctpb Assembles a Gated Protease Tunnel Regulating Cell-Cell Signaling During Spore Formation in Bacillus Subtilis. Cell(Cambridge,Mass.), 155, 2013
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