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1LPG
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CRYSTAL STRUCTURE OF FXA IN COMPLEX WITH 79.
分子名称: Blood coagulation factor Xa, CALCIUM ION, [4-({[5-BENZYLOXY-1-(3-CARBAMIMIDOYL-BENZYL)-1H-INDOLE-2-CARBONYL]-AMINO}-METHYL)-PHENYL]-TRIMETHYL-AMMONIUM
著者Schreuder, H.A, Brachvogel, V, Liesum, A.
登録日2002-05-08
公開日2003-05-08
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Design and Quantitative Structure-Activity relationship of 3-amidinobenzyl-1H-indole-2-carboxamides as potent, nonchiral, and selective inhibitors of blood coagulation factor Xa.
J.Med.Chem., 45, 2002
1LPH
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LYS(B28)PRO(B29)-HUMAN INSULIN
分子名称: CHLORIDE ION, INSULIN, PHENOL, ...
著者Ciszak, E, Beals, J.M, Frank, B.H, Baker, J.C, Carter, N.D, Smith, G.D.
登録日1995-04-19
公開日1996-06-20
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Role of C-terminal B-chain residues in insulin assembly: the structure of hexameric LysB28ProB29-human insulin.
Structure, 3, 1995
1LPI
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HEW LYSOZYME: TRP...NA CATION-PI INTERACTION
分子名称: LYSOZYME, SODIUM ION
著者Wouters, J.
登録日1998-04-15
公開日1998-06-17
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Cation-pi (Na+-Trp) interactions in the crystal structure of tetragonal lysozyme.
Protein Sci., 7, 1998
1LPJ
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Human cRBP IV
分子名称: Retinol-binding protein IV, cellular
著者Calderone, V, Zanotti, G, Berni, R, Folli, C.
登録日2002-05-08
公開日2003-01-14
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Ligand binding and structural analysis of a human putative cellular retinol-binding protein
J.Biol.Chem., 277, 2002
1LPK
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CRYSTAL STRUCTURE OF FXA IN COMPLEX WITH 125.
分子名称: 1-(3-CARBAMIMIDOYL-BENZYL)-1H-INDOLE-2-CARBOXYLIC ACID 3-CARBAMIMIDOYL-BENZYLESTER, Blood coagulation factor Xa, CALCIUM ION
著者Schreuder, H.A, Loenze, P, Brachvogel, V, Liesum, A.
登録日2002-05-08
公開日2003-05-08
最終更新日2021-10-27
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Design and Quantitative Structure-Activity relationship of 3-amidinobenzyl-1H-indole-2-carboxamides as potent, nonchiral, and selective inhibitors of blood coagulation factor Xa
J.Med.Chem., 45, 2002
1LPL
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Structural Genomics of Caenorhabditis elegans: CAP-Gly domain of F53F4.3
分子名称: Hypothetical 25.4 kDa protein F53F4.3 in chromosome V
著者Li, S, Finley, J, Liu, Z.-J, Qiu, S.H, Luan, C.H, Carson, M, Tsao, J, Johnson, D, Lin, G, Zhao, J, Thomas, W, Nagy, L.A, Sha, B, DeLucas, L.J, Wang, B.-C, Luo, M, Southeast Collaboratory for Structural Genomics (SECSG)
登録日2002-05-08
公開日2002-05-22
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.77 Å)
主引用文献Crystal Structure of the Cytoskeleton-associated Protein Glycine-rich (CAP-Gly) Domain
J.Biol.Chem., 277, 2002
1LPM
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A STRUCTURAL BASIS FOR THE CHIRAL PREFERENCES OF LIPASES
分子名称: (1R)-MENTHYL HEXYL PHOSPHONATE GROUP, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Grochulski, P.G, Cygler, M.C.
登録日1995-01-06
公開日1995-04-20
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.18 Å)
主引用文献A Structural Basis for the Chiral Preferences of Lipases
J.Am.Chem.Soc., 116, 1994
1LPN
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ANALOGS OF REACTION INTERMEDIATES IDENTIFY A UNIQUE SUBSTRATE BINDING SITE IN CANDIDA RUGOSA LIPASE
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
著者Grochulski, P.G, Cygler, M.C.
登録日1995-01-11
公開日1995-04-20
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.18 Å)
主引用文献Analogs of reaction intermediates identify a unique substrate binding site in Candida rugosa lipase.
Biochemistry, 33, 1994
1LPO
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ANALOGS OF REACTION INTERMEDIATES IDENTIFY A UNIQUE SUBSTRATE BINDING SITE IN CANDIDA RUGOSA LIPASE
分子名称: 1-HEXADECANOSULFONIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Grochulski, P.G, Cygler, M.C.
登録日1995-01-13
公開日1995-04-20
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.18 Å)
主引用文献Analogs of reaction intermediates identify a unique substrate binding site in Candida rugosa lipase.
Biochemistry, 33, 1994
1LPP
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ANALOGS OF REACTION INTERMEDIATES IDENTIFY A UNIQUE SUBSTRATE BINDING SITE IN CANDIDA RUGOSA LIPASE
分子名称: 1-HEXADECANOSULFONIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Grochulski, P.G, Cygler, M.C.
登録日1995-01-17
公開日1995-04-20
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.18 Å)
主引用文献Analogs of reaction intermediates identify a unique substrate binding site in Candida rugosa lipase.
Biochemistry, 33, 1994
1LPQ
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Human DNA Topoisomerase I (70 Kda) In Non-Covalent Complex With A 22 Base Pair DNA Duplex Containing an 8-oxoG Lesion
分子名称: 5'-D(*AP*AP*AP*AP*AP*GP*AP*CP*TP*TP*(8OG)P*GP*AP*AP*AP*AP*AP*TP*TP*TP*TP*T)-3', 5'-D(*AP*AP*AP*AP*AP*TP*TP*TP*TP*TP*CP*CP*AP*AP*GP*TP*CP*TP*TP*TP*TP*T)-3', DNA topoisomerase I
著者Lesher, D.T, Pommier, Y, Stewart, L, Redinbo, M.R.
登録日2002-05-08
公開日2002-08-16
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (3.14 Å)
主引用文献8-Oxoguanine rearranges the active site of human topoisomerase I
Proc.Natl.Acad.Sci.USA, 99, 2002
1LPS
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A STRUCTURAL BASIS FOR THE CHIRAL PREFERENCES OF LIPASES
分子名称: (1S)-MENTHYL HEXYL PHOSPHONATE GROUP, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Grochulski, P.G, Cygler, M.C.
登録日1995-01-05
公開日1995-02-14
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.18 Å)
主引用文献A Structural Basis for the Chiral Preferences of Lipases
J.Am.Chem.Soc., 116, 1994
1LPU
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Low Temperature Crystal Structure of the Apo-form of the catalytic subunit of protein kinase CK2 from Zea mays
分子名称: BENZAMIDINE, Protein kinase CK2
著者Niefind, K, Puetter, M, Guerra, B, Issinger, O.-G, Schomburg, D.
登録日2002-05-08
公開日2002-05-29
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.86 Å)
主引用文献Inclining the purine base binding plane in protein kinase CK2 by exchanging the flanking side-chains generates a preference for ATP as a cosubstrate.
J.Mol.Biol., 347, 2005
1LPV
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DROSOPHILA MELANOGASTER DOUBLESEX (DSX), NMR, 18 STRUCTURES
分子名称: Doublesex protein, ZINC ION
著者Zhu, L, Wilken, J, Phillips, N, Narendra, U, Chan, G, Stratton, S, Kent, S, Weiss, M.A.
登録日2002-05-08
公開日2002-10-02
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Sexual dimorphism in diverse metazoans is regulated by a novel class of intertwined zinc fingers.
Genes Dev., 14, 2000
1LPW
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Solution structure of the yeast spliceosomal U2 snRNA-intron branch site helix featuring a conserved pseudouridine
分子名称: 5'-R(*GP*GP*UP*GP*(PSU)P*AP*GP*UP*A)-3', 5'-R(*UP*AP*CP*UP*AP*AP*CP*AP*CP*C)-3'
著者Newby, M.I, Greenbaum, N.L.
登録日2002-05-08
公開日2002-11-27
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Sculpting of the Spliceosomal Branch Site Recognition Motif by a Conserved Pseudouridine
Nat.Struct.Biol., 12, 2002
1LPY
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Multiple Methionine Substitutions in T4 Lysozyme
分子名称: BETA-MERCAPTOETHANOL, CHLORIDE ION, LYSOZYME, ...
著者Gassner, N.C, Baase, W.A, Mooers, B.H.M, Busam, R.D, Weaver, L.H, Lindstrom, J.D, Quillin, M.L, Matthews, B.W.
登録日2002-05-08
公開日2002-05-22
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Multiple methionine substitutions are tolerated in T4 lysozyme and have coupled effects on folding and stability.
Biophys.Chem., 100, 2003
1LPZ
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CRYSTAL STRUCTURE OF FXA IN COMPLEX WITH 41.
分子名称: 1-(3-carbamimidoylbenzyl)-N-(3,5-dichlorobenzyl)-4-methyl-1H-indole-2-carboxamide, Blood coagulation factor Xa, CALCIUM ION
著者Schreuder, H.A, Brachvogel, V, Liesum, A.
登録日2002-05-08
公開日2003-05-08
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Design and Quantitative Structure-Activity relationship of 3-amidinobenzyl-1H-indole-2-carboxamides as potent, nonchiral, and selective inhibitors of blood coagulation factor Xa
J.Biol.Chem., 45, 2002
1LQ0
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CRYSTAL STRUCTURE OF HUMAN CHITOTRIOSIDASE AT 2.2 ANGSTROM RESOLUTION
分子名称: CHITOTRIOSIDASE
著者Fusetti, F, Rozeboom, H.J, Dijkstra, B.W.
登録日2002-05-08
公開日2003-07-29
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structure of human chitotriosidase. Implications for specific inhibitor design and function of mammalian chitinase-like lectins
J.Biol.Chem., 277, 2002
1LQ1
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DNA Complexed Structure of the Key Transcription Factor Initiating Development in Sporulation Bacteria
分子名称: 5'-D(*AP*CP*AP*AP*AP*AP*TP*TP*CP*GP*AP*CP*AP*CP*GP*A)-3', 5'-D(*TP*TP*CP*GP*TP*GP*TP*CP*GP*AP*AP*TP*TP*TP*TP*G)-3', Stage 0 sporulation protein A
著者Zhao, H, Msadek, T, Zapf, J, Madhusudan, Hoch, J.A, Varughese, K.I.
登録日2002-05-08
公開日2002-08-23
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献DNA complexed structure of the key transcription factor initiating development in sporulating bacteria.
Structure, 10, 2002
1LQ2
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Crystal structure of barley beta-D-glucan glucohydrolase isoenzyme Exo1 in complex with gluco-phenylimidazole
分子名称: (5R,6R,7S,8S)-5-(HYDROXYMETHYL)-2-PHENYL-5,6,7,8-TETRAHYDROIMIDAZO[1,2-A]PYRIDINE-6,7,8-TRIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-6)-alpha-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-3)]2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Hrmova, M, De Gori, R, Smith, B.J, Vasella, A, Varghese, J.N, Fincher, G.B.
登録日2002-05-09
公開日2003-11-18
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Three-dimensional Structure of the Barley {beta}-D-Glucan Glucohydrolase in Complex with a Transition State Mimic.
J.Biol.Chem., 279, 2004
1LQ7
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De Novo Designed Protein Model of Radical Enzymes
分子名称: Alpha3W
著者Dai, Q.-H, Tommos, C, Fuentes, E.J, Blomberg, M, Dutton, P.L, Wand, A.J.
登録日2002-05-09
公開日2002-06-05
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Structure of a De Novo Designed Protein Model of Radical Enzymes
J.Am.Chem.Soc., 124, 2002
1LQ8
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Crystal structure of cleaved protein C inhibitor
分子名称: 2-acetamido-2-deoxy-alpha-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Huntington, J.A, Kjellberg, M, Stenflo, J.
登録日2002-05-09
公開日2003-02-11
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Crystal Structure of Protein C Inhibitor Provides Insights into Hormone Binding and Heparin Activation
Structure, 11, 2003
1LQ9
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Crystal Structure of a Monooxygenase from the Gene ActVA-Orf6 of Streptomyces coelicolor Strain A3(2)
分子名称: ACTVA-ORF6 MONOOXYGENASE, TETRAETHYLENE GLYCOL
著者Sciara, G, Kendrew, S.G, Miele, A.E, Marsh, N.G, Federici, L, Malatesta, F, Schimperna, G, Savino, C, Vallone, B.
登録日2002-05-09
公開日2003-01-14
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献The structure of ActVA-Orf6, a novel type of monooxygenase involved in actinorhodin biosynthesis
EMBO J., 22, 2003
1LQA
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TAS PROTEIN FROM ESCHERICHIA COLI IN COMPLEX WITH NADPH
分子名称: NADPH DIHYDRO-NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, Tas protein
著者Obmolova, G, Teplyakov, A, Khil, P.P, Howard, A.J, Camerini-Otero, R.D, Gilliland, G.L, Structure 2 Function Project (S2F)
登録日2002-05-09
公開日2003-07-08
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.604 Å)
主引用文献Crystal structure of the Escherichia coli Tas protein, an NADP(H)-dependent aldo-keto reductase
PROTEINS: STRUCT.,FUNCT.,GENET., 53, 2003
1LQB
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Crystal structure of a hydroxylated HIF-1 alpha peptide bound to the pVHL/elongin-C/elongin-B complex
分子名称: Elongin B, Elongin C, Hypoxia-inducible factor 1 ALPHA, ...
著者Hon, W.C, Wilson, M.I, Harlos, K, Claridge, T.D, Schofield, C.J, Pugh, C.W, Maxwell, P.H, Ratcliffe, P.J, Stuart, D.I, Jones, E.Y.
登録日2002-05-09
公開日2002-07-03
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural basis for the recognition of hydroxyproline in HIF-1 alpha by pVHL.
Nature, 417, 2002

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