3QLI
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2P3Z
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![BU of 2p3z by Molmil](/molmil-images/mine/2p3z) | Crystal structure of L-Rhamnonate dehydratase from Salmonella typhimurium | 分子名称: | L-rhamnonate dehydratase, SODIUM ION | 著者 | Malashkevich, V.N, Sauder, J.M, Dickey, M, Adams, J.M, Burley, S.K, Wasserman, S.R, Gerlt, J, Almo, S.C, New York SGX Research Center for Structural Genomics (NYSGXRC) | 登録日 | 2007-03-10 | 公開日 | 2007-03-20 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Crystal Structure of L-Rhamnonate Dehydratase from Salmonella Typhimurium Lt2 To be Published
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4KZC
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![BU of 4kzc by Molmil](/molmil-images/mine/4kzc) | Structure of PI3K gamma with Imidazopyridine inhibitors | 分子名称: | N-{6-[6-amino-5-(trifluoromethyl)pyridin-3-yl]imidazo[1,2-a]pyridin-2-yl}acetamide, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform, SULFATE ION | 著者 | Knapp, M.S, Elling, E.A. | 登録日 | 2013-05-29 | 公開日 | 2013-07-17 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (3.25 Å) | 主引用文献 | Structure guided optimization of a fragment hit to imidazopyridine inhibitors of PI3K. Bioorg.Med.Chem.Lett., 23, 2013
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3HHN
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![BU of 3hhn by Molmil](/molmil-images/mine/3hhn) | Crystal structure of class I ligase ribozyme self-ligation product, in complex with U1A RBD | 分子名称: | Class I ligase ribozyme, self-ligation product, MAGNESIUM ION, ... | 著者 | Shechner, D.M, Grant, R.A, Bagby, S.C, Bartel, D.P. | 登録日 | 2009-05-15 | 公開日 | 2009-11-24 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.987 Å) | 主引用文献 | Crystal structure of the catalytic core of an RNA-polymerase ribozyme. Science, 326, 2009
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4KZ9
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![BU of 4kz9 by Molmil](/molmil-images/mine/4kz9) | Crystal structure of AmpC beta-lactamase in complex with fragment 41 ((4R,4aS,8aS)-4-phenyldecahydroquinolin-4-ol) | 分子名称: | (4R,4aS,8aS)-4-phenyldecahydroquinolin-4-ol, Beta-lactamase, PHOSPHATE ION | 著者 | Eidam, O, Barelier, S, Fish, I, Shoichet, B.K. | 登録日 | 2013-05-29 | 公開日 | 2014-05-21 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.72 Å) | 主引用文献 | Increasing chemical space coverage by combining empirical and computational fragment screens. Acs Chem.Biol., 9, 2014
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3HI7
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![BU of 3hi7 by Molmil](/molmil-images/mine/3hi7) | Crystal structure of human diamine oxidase | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Amiloride-sensitive amine oxidase, CALCIUM ION, ... | 著者 | McGrath, A.P, Guss, J.M. | 登録日 | 2009-05-19 | 公開日 | 2009-10-20 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.799 Å) | 主引用文献 | Structure and inhibition of human diamine oxidase Biochemistry, 48, 2009
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4L06
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3HIW
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![BU of 3hiw by Molmil](/molmil-images/mine/3hiw) | Crystal structure of Saporin-L1 in complex with the cyclic tetranucleotide inhibitor, a transition state analogue | 分子名称: | 9,9'-{(2R,3R,3aR,5S,7aR,9R,10R,10aR,12S,23R,25aR,27R,28R,28aR,30S,32aR,35aR,37S,39aR)-9-(6-amino-9H-purin-9-yl)-34-[(4-amino-5H-pyrrolo[3,2-d]pyrimidin-7-yl)methyl]-5,12,23,30,37-pentahydroxy-3,10,28-trimethoxy-5,12,23,30,37-pentaoxidotetracosahydro-2H,7H,25H-trifuro[3,2-f:3',2'-l:3'',2''-x]pyrrolo[3,4-r][1,3,5,9,11,15,17,21,23,27,29,2,4,10,16,22,28]undecaoxazapentaphosphacyclopentatriacontine-2,27-diyl}bis(2-amino-3,9-dihydro-6H-purin-6-one), Vacuolar saporin | 著者 | Ho, M, Sturm, M.B, Almo, S.C, Schramm, V.L. | 登録日 | 2009-05-20 | 公開日 | 2009-12-08 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Transition state analogues in structures of ricin and saporin ribosome-inactivating proteins. Proc.Natl.Acad.Sci.USA, 106, 2009
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2P5S
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![BU of 2p5s by Molmil](/molmil-images/mine/2p5s) | RAB domain of human RASEF in complex with GDP | 分子名称: | GUANOSINE-5'-DIPHOSPHATE, RAS and EF-hand domain containing, UNKNOWN ATOM OR ION | 著者 | Zhu, H, Wang, J, Shen, Y, Tempel, W, Landry, R, Arrowsmith, C.H, Edwards, A.M, Sundstrom, M, Weigelt, J, Bochkarev, A, Park, H, Structural Genomics Consortium (SGC) | 登録日 | 2007-03-16 | 公開日 | 2007-03-27 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | 主引用文献 | RAB domain of human RASEF in complex with GDP To be Published
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2FE8
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![BU of 2fe8 by Molmil](/molmil-images/mine/2fe8) | SARS coronavirus papain-like protease: structure of a viral deubiquitinating enzyme | 分子名称: | BROMIDE ION, Replicase polyprotein 1ab, SULFATE ION, ... | 著者 | Ratia, K, Santarsiero, B.D, Mesecar, A.D. | 登録日 | 2005-12-15 | 公開日 | 2006-03-21 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Severe acute respiratory syndrome coronavirus papain-like protease: Structure of a viral deubiquitinating enzyme Proc.Natl.Acad.Sci.Usa, 103, 2006
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4L08
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![BU of 4l08 by Molmil](/molmil-images/mine/4l08) | Crystal structure of the maleamate amidase Ami(C149A) in complex with maleate from Pseudomonas putida S16 | 分子名称: | Hydrolase, isochorismatase family, MALEIC ACID | 著者 | Chen, D.D, Lu, Y, Zhang, Z, Wu, G, Xu, P. | 登録日 | 2013-05-31 | 公開日 | 2014-07-16 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2.66 Å) | 主引用文献 | Structural insights into the specific recognition of N-heterocycle biodenitrogenation-derived substrates by microbial amide hydrolases. Mol.Microbiol., 91, 2014
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2FGN
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2P71
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3QPZ
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![BU of 3qpz by Molmil](/molmil-images/mine/3qpz) | Crystal structure of the N59A mutant of the 3-deoxy-d-manno-octulosonate 8-phosphate synthase (KDO8PS) from Neisseria meningitidis | 分子名称: | 2-dehydro-3-deoxyphosphooctonate aldolase, CHLORIDE ION, GLYCEROL, ... | 著者 | Allison, T.M, Jameson, G.B, Parker, E.J, Cochrane, F.C. | 登録日 | 2011-02-14 | 公開日 | 2011-04-13 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Targeting the role of a key conserved motif for substrate selection and catalysis by 3-deoxy-D-manno-octulosonate 8-phosphate synthase Biochemistry, 50, 2011
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2FHX
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![BU of 2fhx by Molmil](/molmil-images/mine/2fhx) | Pseudomonas aeruginosa SPM-1 metallo-beta-lactamase | 分子名称: | 1,2-ETHANEDIOL, AZIDE ION, CHLORIDE ION, ... | 著者 | Murphy, T.A, Catto, L.E, Halford, S.E, Hadfield, A.T, Minor, W, Walsh, T.R, Spencer, J. | 登録日 | 2005-12-27 | 公開日 | 2006-01-17 | 最終更新日 | 2022-04-13 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Crystal Structure of Pseudomonas aeruginosa SPM-1 Provides Insights into Variable Zinc Affinity of Metallo-beta-lactamases. J.Mol.Biol., 357, 2006
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3Q6D
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![BU of 3q6d by Molmil](/molmil-images/mine/3q6d) | Xaa-Pro dipeptidase from Bacillus anthracis. | 分子名称: | CALCIUM ION, GLYCEROL, Proline dipeptidase | 著者 | Osipiuk, J, Makowska-Grzyska, M, Papazisi, L, Anderson, W.F, Joachimiak, A, Center for Structural Genomics of Infectious Diseases (CSGID) | 登録日 | 2010-12-31 | 公開日 | 2011-02-02 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.97 Å) | 主引用文献 | Xaa-Pro dipeptidase from Bacillus anthracis. To be Published
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2QLK
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![BU of 2qlk by Molmil](/molmil-images/mine/2qlk) | Adenovirus AD35 fibre head | 分子名称: | Fiber, GLYCEROL | 著者 | Liaw, Y.-C, Amiraslanov, I, Wang, H, Lieber, A. | 登録日 | 2007-07-13 | 公開日 | 2008-02-19 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.02 Å) | 主引用文献 | Identification of CD46 binding sites within the adenovirus serotype 35 fiber knob J.Virol., 81, 2007
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3Q7Z
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![BU of 3q7z by Molmil](/molmil-images/mine/3q7z) | CBAP-acylated BlaR1 sensor domain from Staphylococcus aureus | 分子名称: | (2R,4S)-2-[(1R)-1-{[(2'-carboxybiphenyl-2-yl)carbonyl]amino}-2-oxoethyl]-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid, Beta-lactamase regulatory protein BlaR1 | 著者 | Borbulevych, O.Y, Mobashery, S, Baker, B.M. | 登録日 | 2011-01-05 | 公開日 | 2011-07-06 | 最終更新日 | 2017-11-08 | 実験手法 | X-RAY DIFFRACTION (1.87 Å) | 主引用文献 | Lysine Nzeta-decarboxylation switch and activation of the beta-lactam sensor domain of BlaR1 protein of methicillin-resistant Staphylococcus aureus. J.Biol.Chem., 286, 2011
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4L4P
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![BU of 4l4p by Molmil](/molmil-images/mine/4l4p) | the mutant(E139A) structure in complex with xylotriose | 分子名称: | Endo-1,4-beta-xylanase, beta-D-xylopyranose-(1-4)-beta-D-xylopyranose-(1-4)-beta-D-xylopyranose | 著者 | An, J, Feng, Y, Wu, G. | 登録日 | 2013-06-08 | 公開日 | 2014-05-07 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Crystal structure of CbXyn10B from Caldicellulosiruptor bescii and its mutant(E139A) in complex with xylotriose To be Published
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2QQN
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3Q5R
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![BU of 3q5r by Molmil](/molmil-images/mine/3q5r) | Crystal structure of BmrR bound to Kanamycin | 分子名称: | 23 bp promoter DNA, KANAMYCIN A, Multidrug-efflux transporter 1 regulator | 著者 | Bachas, S, Eginton, C, Gunio, G, Wade, H. | 登録日 | 2010-12-29 | 公開日 | 2011-07-20 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (3.05 Å) | 主引用文献 | Structural contributions to multidrug recognition in the multidrug resistance (MDR) gene regulator, BmrR. Proc.Natl.Acad.Sci.USA, 108, 2011
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3Q96
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![BU of 3q96 by Molmil](/molmil-images/mine/3q96) | B-Raf kinase domain in complex with a tetrahydronaphthalene inhibitor | 分子名称: | (2S)-N-[3-(2-aminopropan-2-yl)-5-(trifluoromethyl)phenyl]-7-[(7-oxo-5,6,7,8-tetrahydro-1,8-naphthyridin-4-yl)oxy]-1,2,3,4-tetrahydronaphthalene-2-carboxamide, Serine/threonine-protein kinase B-raf | 著者 | Sintchak, M.D, Aertgeerts, K, Yano, J. | 登録日 | 2011-01-07 | 公開日 | 2011-03-23 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Design and optimization of potent and orally bioavailable tetrahydronaphthalene raf inhibitors. J.Med.Chem., 54, 2011
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3Q65
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![BU of 3q65 by Molmil](/molmil-images/mine/3q65) | Human Aldose Reductase in Complex with NADP+ in Space Group P212121 | 分子名称: | Aldose reductase, GLYCEROL, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ... | 著者 | Sawaya, M.R, Cascio, D, Balendiran, G.K. | 登録日 | 2010-12-30 | 公開日 | 2011-01-19 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.09 Å) | 主引用文献 | The role of Cys-298 in aldose reductase function. J.Biol.Chem., 286, 2011
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3HG9
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![BU of 3hg9 by Molmil](/molmil-images/mine/3hg9) | CRYSTAL STRUCTURE OF putative pilM protein from Pseudomonas aeruginosa 2192 | 分子名称: | NICKEL (II) ION, PilM | 著者 | Malashkevich, V.N, Toro, R, Sauder, J.M, Burley, S.K, Almo, S.C, New York SGX Research Center for Structural Genomics (NYSGXRC) | 登録日 | 2009-05-13 | 公開日 | 2009-05-26 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | CRYSTAL STRUCTURE OF putative pilM protein from Pseudomonas aeruginosa 2192 To be Published
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3Q9H
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![BU of 3q9h by Molmil](/molmil-images/mine/3q9h) | LVFFA segment from Alzheimer's Amyloid-Beta displayed on 42-membered macrocycle scaffold | 分子名称: | 1,4-BUTANEDIOL, Cyclic pseudo-peptide LVFFA(ORN)(HAO)LK(ORN), GLYCEROL, ... | 著者 | Liu, C, Sawaya, M.R, Eisenberg, D, Nowick, J.S, Cheng, P, Zheng, J. | 登録日 | 2011-01-07 | 公開日 | 2011-06-08 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Characteristics of Amyloid-Related Oligomers Revealed by Crystal Structures of Macrocyclic beta-Sheet Mimics. J.Am.Chem.Soc., 133, 2011
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