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7YSO
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BU of 7yso by Molmil
Tubulin heterodimer structure of GDP-1 state in solution
分子名称: GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, Tubulin alpha-1B chain, ...
著者Zhou, J, Wang, H.-W.
登録日2022-08-12
公開日2023-10-18
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献Structural insights into the mechanism of GTP initiation of microtubule assembly.
Nat Commun, 14, 2023
7YSN
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BU of 7ysn by Molmil
Tubulin heterodimer structure of GMPCPP state in solution
分子名称: GUANOSINE-5'-TRIPHOSPHATE, PHOSPHOMETHYLPHOSPHONIC ACID GUANYLATE ESTER, Tubulin alpha-1B chain, ...
著者Zhou, J, Wang, H.-W.
登録日2022-08-12
公開日2023-10-18
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献Structural insights into the mechanism of GTP initiation of microtubule assembly.
Nat Commun, 14, 2023
7YOP
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BU of 7yop by Molmil
Spiroplasma melliferum FtsZ bound to GMPPNP
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Cell division protein FtsZ, GUANOSINE-5'-DIPHOSPHATE, ...
著者Chakraborty, J, Pananghat, G.
登録日2022-08-01
公開日2023-08-16
実験手法X-RAY DIFFRACTION (2.20003128 Å)
主引用文献Structural basis of kinetic polarity of FtsZ from a cell wall-less bacterium Spiroplasma
To Be Published
7YLW
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BU of 7ylw by Molmil
yeast TRiC-plp2-tubulin complex at S3 closed TRiC state
分子名称: ADENOSINE-5'-DIPHOSPHATE, ALUMINUM FLUORIDE, GUANOSINE-5'-TRIPHOSPHATE, ...
著者Han, W.Y.
登録日2022-07-27
公開日2023-03-29
実験手法ELECTRON MICROSCOPY (3.39 Å)
主引用文献Structural basis of plp2-mediated cytoskeletal protein folding by TRiC/CCT.
Sci Adv, 9, 2023
7YHN
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BU of 7yhn by Molmil
ANTI-TUMOR AGENT Y48 IN COMPLEX WITH TUBULIN
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 4-methyl-3-[(4-methylphenyl)sulfonylamino]-~{N}-[(6-methylpyridin-3-yl)methyl]benzamide, GUANOSINE-5'-DIPHOSPHATE, ...
著者Du, T, Ji, M, Hou, Z, Lin, S, Zhang, J, Wu, D, Zhang, K, Lu, D, Xu, H, Chen, X.
登録日2022-07-14
公開日2023-07-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Optimization of Benzamide Derivatives as Potent and Orally Active Tubulin Inhibitors Targeting the Colchicine Binding Site.
J.Med.Chem., 65, 2022
7XR1
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BU of 7xr1 by Molmil
Crystal structure of T2R-TTL-3a complex
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 2-chloranyl-6-fluoranyl-N-(4-methoxyphenyl)-N-methyl-quinazolin-4-amine, CALCIUM ION, ...
著者Lun, T, Wu, C.Y.
登録日2022-05-09
公開日2023-05-17
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.81 Å)
主引用文献Crystal structure of T2R-TTL-3a complex
To Be Published
7XR0
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BU of 7xr0 by Molmil
Crystal structure of T2R-TTL-27a complex
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 2-chloranyl-5-fluoranyl-N-(4-methoxyphenyl)-N-methyl-quinazolin-4-amine, CALCIUM ION, ...
著者Lun, T, Wu, C.Y.
登録日2022-05-09
公開日2023-05-17
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Crystal structure of T2R-TTL-27a complex
To Be Published
7XQY
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BU of 7xqy by Molmil
Crystal structure of T2R-TTL-15 complex
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 2-chloranyl-N-(4-methoxyphenyl)-N-methyl-pyrido[3,2-d]pyrimidin-4-amine, CALCIUM ION, ...
著者Lun, T, ChengYong, W.
登録日2022-05-09
公開日2023-05-17
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Crystal structure of T2R-TTL-15 complex
To Be Published
7XQX
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BU of 7xqx by Molmil
Crystal structure of T2R-TTL-27a complex
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 2-chloranyl-7-fluoranyl-N-(4-methoxyphenyl)-N-methyl-quinazolin-4-amine, CALCIUM ION, ...
著者Lun, T, Wu, C.Y.
登録日2022-05-09
公開日2023-05-17
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (3.36 Å)
主引用文献Crystal structure of T2R-TT complex
To Be Published
7X4N
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BU of 7x4n by Molmil
Crystal Structure of C. elegans kinesin-4 KLP-12 complexed with tubulin and DARPin
分子名称: DARPin, GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, ...
著者Taguchi, S, Imasaki, T, Saijo-Hamano, Y, Sakai, N, Nitta, R.
登録日2022-03-03
公開日2022-09-21
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.88 Å)
主引用文献Structural model of microtubule dynamics inhibition by kinesin-4 from the crystal structure of KLP-12 -tubulin complex.
Elife, 11, 2022
7X0S
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BU of 7x0s by Molmil
Human TRiC-tubulin-S3
分子名称: ADENOSINE-5'-DIPHOSPHATE, ALUMINUM FLUORIDE, MAGNESIUM ION, ...
著者Cong, Y, Liu, C.X.
登録日2022-02-22
公開日2023-04-12
最終更新日2023-07-05
実験手法ELECTRON MICROSCOPY (3.1 Å)
主引用文献Pathway and mechanism of tubulin folding mediated by TRiC/CCT along its ATPase cycle revealed using cryo-EM.
Commun Biol, 6, 2023
7VMK
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BU of 7vmk by Molmil
Crystal structure of tubulin with 3
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, DI(HYDROXYETHYL)ETHER, ...
著者Jifa, Z, Lun, T.
登録日2021-10-08
公開日2022-10-19
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal structure of tubulin with 3
To Be Published
7VMJ
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BU of 7vmj by Molmil
Crystal structure of tubulin with 17a
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, CHLORIDE ION, ...
著者Jifa, Z, Lun, T.
登録日2021-10-08
公開日2022-10-19
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Crystal structure of tubulin with 17j
To Be Published
7VMG
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BU of 7vmg by Molmil
Crystal structure of tubulin with 17j
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, CHLORIDE ION, ...
著者Jifa, Z, Lun, T.
登録日2021-10-08
公開日2022-10-19
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.39 Å)
主引用文献Crystal structure of tubulin with 17a
To Be Published
7UNG
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BU of 7ung by Molmil
48-nm repeat of the human respiratory doublet microtubule
分子名称: Cilia- and flagella-associated protein 161, Cilia- and flagella-associated protein 20, Cilia- and flagella-associated protein 45, ...
著者Gui, M, Croft, J.T, Zabeo, D, Acharya, V, Kollman, J.M, Burgoyne, T, Hoog, J.L, Brown, A.
登録日2022-04-11
公開日2022-10-05
最終更新日2024-06-12
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献SPACA9 is a lumenal protein of human ciliary singlet and doublet microtubules.
Proc.Natl.Acad.Sci.USA, 119, 2022
7UN1
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BU of 7un1 by Molmil
8-nm repeat of the human sperm tip singlet microtubule
分子名称: GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, ...
著者Gui, M, Croft, J.T, Zabeo, D, Acharya, V, Kollman, J.M, Burgoyne, T, Hoog, J.L, Brown, A.
登録日2022-04-08
公開日2022-10-05
最終更新日2024-06-12
実験手法ELECTRON MICROSCOPY (6 Å)
主引用文献SPACA9 is a lumenal protein of human ciliary singlet and doublet microtubules.
Proc.Natl.Acad.Sci.USA, 119, 2022
7U0F
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BU of 7u0f by Molmil
HIV-1 Rev in complex with tubulin
分子名称: Protein Rev, Tubulin alpha-1A chain, Tubulin beta chain
著者Eren, E.
登録日2022-02-18
公開日2023-08-23
最終更新日2023-10-18
実験手法ELECTRON MICROSCOPY (3.53 Å)
主引用文献Structural basis of microtubule depolymerization by the kinesin-like activity of HIV-1 Rev.
Structure, 31, 2023
7TUB
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BU of 7tub by Molmil
The beta-tubulin folding intermediate IV
分子名称: ADENOSINE-5'-DIPHOSPHATE, ALUMINUM FLUORIDE, MAGNESIUM ION, ...
著者Zhao, Y, Frydman, J, Chiu, W.
登録日2022-02-02
公開日2022-12-28
最終更新日2024-06-12
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献Structural visualization of the tubulin folding pathway directed by human chaperonin TRiC/CCT.
Cell, 185, 2022
7TTT
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BU of 7ttt by Molmil
The beta-tubulin folding intermediate III
分子名称: ADENOSINE-5'-DIPHOSPHATE, ALUMINUM FLUORIDE, MAGNESIUM ION, ...
著者Zhao, Y, Frydman, J, Chiu, W.
登録日2022-02-01
公開日2022-12-28
最終更新日2024-06-12
実験手法ELECTRON MICROSCOPY (2.9 Å)
主引用文献Structural visualization of the tubulin folding pathway directed by human chaperonin TRiC/CCT.
Cell, 185, 2022
7TTN
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BU of 7ttn by Molmil
The beta-tubulin folding intermediate II
分子名称: ADENOSINE-5'-DIPHOSPHATE, ALUMINUM FLUORIDE, MAGNESIUM ION, ...
著者Zhao, Y, Frydman, J, Chiu, W.
登録日2022-02-01
公開日2022-12-28
最終更新日2024-06-12
実験手法ELECTRON MICROSCOPY (3.3 Å)
主引用文献Structural visualization of the tubulin folding pathway directed by human chaperonin TRiC/CCT.
Cell, 185, 2022
7TTF
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BU of 7ttf by Molmil
Tubulin-RB3_SLD in complex with compound 12k
分子名称: 7-methoxy-4-[2-(methylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl]-3,4-dihydroquinoxalin-2(1H)-one, GLYCEROL, GUANOSINE-5'-DIPHOSPHATE, ...
著者White, S.W, Yun, M.
登録日2022-02-01
公開日2023-04-12
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Design, Synthesis, and Biological Evaluation of Pyrimidine Dihydroquinoxalinone Derivatives as Tubulin Colchicine Site-Binding Agents That Displayed Potent Anticancer Activity Both In Vitro and In Vivo.
Acs Pharmacol Transl Sci, 6, 2023
7TTE
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BU of 7tte by Molmil
Tubulin-RB3_SLD in complex with compound 12j
分子名称: 4-[2-(cyclopropylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl]-7-methoxy-3,4-dihydroquinoxalin-2(1H)-one, GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, ...
著者White, S.W, Yun, M.
登録日2022-02-01
公開日2023-04-12
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Design, Synthesis, and Biological Evaluation of Pyrimidine Dihydroquinoxalinone Derivatives as Tubulin Colchicine Site-Binding Agents That Displayed Potent Anticancer Activity Both In Vitro and In Vivo.
Acs Pharmacol Transl Sci, 6, 2023
7TTD
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BU of 7ttd by Molmil
Tubulin-RB3_SLD in complex with compound 12e
分子名称: 7-methoxy-4-[2-(morpholin-4-yl)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl]-3,4-dihydroquinoxalin-2(1H)-one, GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, ...
著者White, S.W, Yun, M.
登録日2022-02-01
公開日2023-04-12
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.27 Å)
主引用文献Design, Synthesis, and Biological Evaluation of Pyrimidine Dihydroquinoxalinone Derivatives as Tubulin Colchicine Site-Binding Agents That Displayed Potent Anticancer Activity Both In Vitro and In Vivo.
Acs Pharmacol Transl Sci, 6, 2023
7TRG
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BU of 7trg by Molmil
The beta-tubulin folding intermediate I
分子名称: ADENOSINE-5'-DIPHOSPHATE, ALUMINUM FLUORIDE, MAGNESIUM ION, ...
著者Zhao, Y, Frydman, J, Chiu, W.
登録日2022-01-28
公開日2022-12-28
最終更新日2024-06-12
実験手法ELECTRON MICROSCOPY (3 Å)
主引用文献Structural visualization of the tubulin folding pathway directed by human chaperonin TRiC/CCT.
Cell, 185, 2022
7TR3
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BU of 7tr3 by Molmil
CaKip3[2-482] - AMP-PNP in complex with a dolastatin-10-stabilized tubulin ring
分子名称: GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, Kinesin-like protein, ...
著者Benoit, M.P.M.H, Asenjo, A.B, Hunter, B, Allingham, J.S, Sosa, H.
登録日2022-01-27
公開日2022-07-20
最終更新日2024-02-21
実験手法ELECTRON MICROSCOPY (3.9 Å)
主引用文献Kinesin-8-specific loop-2 controls the dual activities of the motor domain according to tubulin protofilament shape.
Nat Commun, 13, 2022

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件を2024-06-12に公開中

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