4H00
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![BU of 4h00 by Molmil](/molmil-images/mine/4h00) | The crystal structure of mon-Zn dihydropyrimidinase from Tetraodon nigroviridis | 分子名称: | ZINC ION, dihydropyrimidinase | 著者 | Hsieh, Y.C, Chen, M.C, Hsu, C.C, Chan, S.I, Yang, Y.S, Chen, C.J. | 登録日 | 2012-09-06 | 公開日 | 2013-09-11 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Lysine Carboxylation: Metal and Structural Requirements for Post-translational Modification To be Published
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4YD7
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8IAJ
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![BU of 8iaj by Molmil](/molmil-images/mine/8iaj) | Cryo-EM structure of the yeast SPT-ORM2 (ORM2-S3A) complex | 分子名称: | N-[(2S,3R,4E)-1,3-dihydroxyoctadec-4-en-2-yl]tetracosanamide, PYRIDOXAL-5'-PHOSPHATE, Protein ORM2, ... | 著者 | Xie, T, Gong, X. | 登録日 | 2023-02-08 | 公開日 | 2024-02-14 | 実験手法 | ELECTRON MICROSCOPY (3.1 Å) | 主引用文献 | Collaborative regulation of yeast SPT-Orm2 complex by phosphorylation and ceramide. Cell Rep, 43, 2024
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6WZM
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![BU of 6wzm by Molmil](/molmil-images/mine/6wzm) | LY3041658 Fab bound to CXCL8 | 分子名称: | 1,2-ETHANEDIOL, Interleukin-8, LY3041658 Fab heavy chain, ... | 著者 | Durbin, J.D, Druzina, Z. | 登録日 | 2020-05-14 | 公開日 | 2020-11-25 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.28 Å) | 主引用文献 | Discovery and characterization of a neutralizing pan-ELR+CXC chemokine monoclonal antibody. Mabs, 12
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4Z4S
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![BU of 4z4s by Molmil](/molmil-images/mine/4z4s) | Crystal structure of GII.10 P domain in complex with 150mM fucose | 分子名称: | 1,2-ETHANEDIOL, Capsid protein, NITRATE ION, ... | 著者 | Koromyslova, A.D, Leuthold, M.M, Hansman, G.S. | 登録日 | 2015-04-02 | 公開日 | 2015-05-27 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | The sweet quartet: Binding of fucose to the norovirus capsid. Virology, 483, 2015
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8IAM
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![BU of 8iam by Molmil](/molmil-images/mine/8iam) | Cryo-EM structure of the yeast SPT-ORM2 (ORM2-S3D) complex | 分子名称: | Chimera of Long chain base biosynthesis protein 1 and Serine palmitoyltransferase 1, N-[(2S,3R,4E)-1,3-dihydroxyoctadec-4-en-2-yl]tetracosanamide, PYRIDOXAL-5'-PHOSPHATE, ... | 著者 | Xie, T, Gong, X. | 登録日 | 2023-02-08 | 公開日 | 2024-02-14 | 実験手法 | ELECTRON MICROSCOPY (3.1 Å) | 主引用文献 | Collaborative regulation of yeast SPT-Orm2 complex by phosphorylation and ceramide. Cell Rep, 43, 2024
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6ZMB
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![BU of 6zmb by Molmil](/molmil-images/mine/6zmb) | Structure of the native tRNA-Monooxygenase enzyme MiaE | 分子名称: | 1-(2-METHOXY-ETHOXY)-2-{2-[2-(2-METHOXY-ETHOXY]-ETHOXY}-ETHANE, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CALCIUM ION, ... | 著者 | Carpentier, P, Atta, M. | 登録日 | 2020-07-02 | 公開日 | 2020-09-02 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Structural, biochemical and functional analyses of tRNA-monooxygenase enzyme MiaE from Pseudomonas putida provide insights into tRNA/MiaE interaction. Nucleic Acids Res., 48, 2020
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6WUW
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![BU of 6wuw by Molmil](/molmil-images/mine/6wuw) | Crystal structure of Human Serum Albumin complex with JMS-053 | 分子名称: | 1,2-ETHANEDIOL, 7-imino-2-phenylthieno[3,2-c]pyridine-4,6(5H,7H)-dione, MYRISTIC ACID, ... | 著者 | Czub, M.P, Cooper, D.R, Shabalin, I.G, Lazo, J.S, Minor, W, Center for Structural Genomics of Infectious Diseases (CSGID) | 登録日 | 2020-05-05 | 公開日 | 2020-05-20 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Structure of the Complex of an Iminopyridinedione Protein Tyrosine Phosphatase 4A3 Phosphatase Inhibitor with Human Serum Albumin. Mol.Pharmacol., 98, 2020
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4Z4V
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![BU of 4z4v by Molmil](/molmil-images/mine/4z4v) | Crystal structure of GII.10 P domain in complex with 19mM fucose | 分子名称: | 1,2-ETHANEDIOL, Capsid protein, NITRATE ION, ... | 著者 | Koromyslova, A.D, Leuthold, M.M, Hansman, G.S. | 登録日 | 2015-04-02 | 公開日 | 2015-05-27 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | The sweet quartet: Binding of fucose to the norovirus capsid. Virology, 483, 2015
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6NMQ
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![BU of 6nmq by Molmil](/molmil-images/mine/6nmq) | Hypoxia-Inducible Factor (HIF) Prolyl Hydroxylase 2 (PHD2) in Complex with the Carboxamide Analog JNJ43058171 | 分子名称: | Egl nine homolog 1, FE (II) ION, N-(4-oxo-1,4-dihydrocinnoline-3-carbonyl)glycine | 著者 | Bembenek, S.D, Mirzadegan, T. | 登録日 | 2019-01-11 | 公開日 | 2019-04-24 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (1.58 Å) | 主引用文献 | Beyond Traditional Structure-Based Drug Design: The Role of Iron Complexation, Strain, and Water in the Binding of Inhibitors for Hypoxia-Inducible Factor Prolyl Hydroxylase 2. Acs Omega, 4, 2019
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6ZQP
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![BU of 6zqp by Molmil](/molmil-images/mine/6zqp) | Structure of the Pmt2-MIR domain with bound ligands | 分子名称: | GLYCEROL, PMT2 isoform 1, SULFATE ION, ... | 著者 | Wild, K, Chiapparino, A, Hackmann, Y, Mortensen, S, Sinning, I. | 登録日 | 2020-07-10 | 公開日 | 2020-12-23 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Functional implications of MIR domains in protein O -mannosylation. Elife, 9, 2020
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7ZH8
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![BU of 7zh8 by Molmil](/molmil-images/mine/7zh8) | DYRK1a in Complex with a Bromo-Triazolo-Pyridine | 分子名称: | 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, 6-bromanyl-3H-[1,2,3]triazolo[4,5-b]pyridine, CHLORIDE ION, ... | 著者 | Dammann, M, Stahlecker, J, Stehle, T, Boeckler, F.M. | 登録日 | 2022-04-05 | 公開日 | 2022-11-09 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Screening of a Halogen-Enriched Fragment Library Leads to Unconventional Binding Modes. J.Med.Chem., 65, 2022
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4RTF
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![BU of 4rtf by Molmil](/molmil-images/mine/4rtf) | Crystal structure of molecular chaperone DnaK from Mycobacterium tuberculosis H37Rv | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, Chaperone protein DnaK, TETRAETHYLENE GLYCOL | 著者 | Filippova, E.V, Minasov, G, Kiryukhina, O, Endres, M, Babnigg, G, Rubin, E, Sacchettini, J, Joachimiak, A, Anderson, W.F, Midwest Center for Structural Genomics (MCSG), Structures of Mtb Proteins Conferring Susceptibility to Known Mtb Inhibitors (MTBI) | 登録日 | 2014-11-14 | 公開日 | 2014-12-10 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.77 Å) | 主引用文献 | Crystal structure of molecular chaperone DnaK from Mycobacterium tuberculosis H37Rv To be Published
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6NOV
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![BU of 6nov by Molmil](/molmil-images/mine/6nov) | A Fab derived from ixekizumab | 分子名称: | DODECAETHYLENE GLYCOL, Fab Heavy Chain, Fab Light Chain | 著者 | Durbin, J.D, Clawson, D.K, Lu, F, Tian, Y, Lu, J, Schmitt, M, Atwell, S. | 登録日 | 2019-01-16 | 公開日 | 2019-06-19 | 最終更新日 | 2019-08-14 | 実験手法 | X-RAY DIFFRACTION (2.14 Å) | 主引用文献 | Development of tibulizumab, a tetravalent bispecific antibody targeting BAFF and IL-17A for the treatment of autoimmune disease. Mabs, 11, 2019
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6NI4
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5L88
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![BU of 5l88 by Molmil](/molmil-images/mine/5l88) | AFAMIN ANTIBODY FRAGMENT, N14 FAB, L1- GLYCOSILATED, CRYSTAL FORM I, non-parsimonious model | 分子名称: | 3,6,9,12,15,18,21-HEPTAOXATRICOSANE-1,23-DIOL, Anti-afamin antibody N14, Fab fragment, ... | 著者 | Rupp, B, Naschberger, A. | 登録日 | 2016-06-07 | 公開日 | 2016-08-03 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.88 Å) | 主引用文献 | The N14 anti-afamin antibody Fab: a rare VL1 CDR glycosylation, crystallographic re-sequencing, molecular plasticity and conservative versus enthusiastic modelling. Acta Crystallogr D Struct Biol, 72, 2016
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5L9D
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![BU of 5l9d by Molmil](/molmil-images/mine/5l9d) | AFAMIN ANTIBODY FRAGMENT, N14 FAB, L1- GLYCOSYLATED, CRYSTAL FORM I, parsimonious model | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 3,6,9,12,15,18,21-HEPTAOXATRICOSANE-1,23-DIOL, DI(HYDROXYETHYL)ETHER, ... | 著者 | Rupp, B, Naschberger, A. | 登録日 | 2016-06-10 | 公開日 | 2016-08-03 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.88 Å) | 主引用文献 | The N14 anti-afamin antibody Fab: a rare VL1 CDR glycosylation, crystallographic re-sequencing, molecular plasticity and conservative versus enthusiastic modelling. Acta Crystallogr D Struct Biol, 72, 2016
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8AU8
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8AUM
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5KM9
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![BU of 5km9 by Molmil](/molmil-images/mine/5km9) | |
6ZQH
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![BU of 6zqh by Molmil](/molmil-images/mine/6zqh) | Yeast Uba1 in complex with ubiquitin | 分子名称: | BETA-MERCAPTOETHANOL, GLYCEROL, TETRAETHYLENE GLYCOL, ... | 著者 | Misra, M, Schindelin, H. | 登録日 | 2020-07-09 | 公開日 | 2020-11-04 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.032 Å) | 主引用文献 | Development of ADPribosyl Ubiquitin Analogues to Study Enzymes Involved in Legionella Infection. Chemistry, 27, 2021
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4Z4W
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![BU of 4z4w by Molmil](/molmil-images/mine/4z4w) | Crystal structure of GII.10 P domain in complex with 4.7mM fucose | 分子名称: | 1,2-ETHANEDIOL, Capsid protein, beta-L-fucopyranose | 著者 | Koromyslova, A.D, Leuthold, M.M, Hansman, G.S. | 登録日 | 2015-04-02 | 公開日 | 2015-05-27 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | The sweet quartet: Binding of fucose to the norovirus capsid. Virology, 483, 2015
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6NYX
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7U1Y
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![BU of 7u1y by Molmil](/molmil-images/mine/7u1y) | Structure of SPAC806.04c protein from fission yeast bound to AlF4 and Co2+ | 分子名称: | COBALT (II) ION, Damage-control phosphatase SPAC806.04c, POTASSIUM ION, ... | 著者 | Jacewicz, A, Sanchez, A.M, Shuman, S. | 登録日 | 2022-02-22 | 公開日 | 2022-06-01 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.81 Å) | 主引用文献 | Fission yeast Duf89 and Duf8901 are cobalt/nickel-dependent phosphatase-pyrophosphatases that act via a covalent aspartyl-phosphate intermediate. J.Biol.Chem., 298, 2022
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5ID7
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![BU of 5id7 by Molmil](/molmil-images/mine/5id7) | Crystal structure of human serum albumin in complex with phosphorodithioate derivative of myristoyl cyclic phosphatidic acid (cPA) | 分子名称: | (4S)-2-sulfanylidene-4-[(tetradecanoyloxy)methyl]-1,3,2lambda~5~-dioxaphospholane-2-thiolate, DI(HYDROXYETHYL)ETHER, Serum albumin, ... | 著者 | Sekula, B, Bujacz, A, Rytczak, P, Bujacz, G. | 登録日 | 2016-02-24 | 公開日 | 2016-05-11 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.26 Å) | 主引用文献 | Structural evidence of the species-dependent albumin binding of the modified cyclic phosphatidic acid with cytotoxic properties. Biosci.Rep., 36, 2016
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