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3MJR
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BU of 3mjr by Molmil
Human dCK complex with Acyclic Nucleoside
分子名称: 9-HYROXYETHOXYMETHYLGUANINE, Deoxycytidine kinase, URIDINE-5'-DIPHOSPHATE
著者Hazra, S, Lavie, A.
登録日2010-04-13
公開日2010-07-28
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献The Sugar Ring of the Nucleoside Is Required for Productive Substrate Positioning in the Active Site of Human Deoxycytidine Kinase (dCK): Implications for the Development of dCK-Activated Acyclic Guanine Analogues.
J.Med.Chem., 53, 2010
9QAJ
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BU of 9qaj by Molmil
Structure of the nucleosome-bound human BCL7A
分子名称: 601 DNA, Histone H2A, Histone H2B 1.1, ...
著者Martin, F, Bergamin, E.
登録日2025-02-28
公開日2025-04-23
実験手法ELECTRON MICROSCOPY (2.95 Å)
主引用文献Structure of the nucleosome-bound human BCL7A.
Nucleic Acids Res., 53, 2025
6BJ7
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BU of 6bj7 by Molmil
Crystal Structure of Purine Nucleoside Phosphorylase Isoform 2 from Schistosoma mansoni in complex with 4-chloro-6-methylpyrimidin-2-amine
分子名称: 4-chloro-6-methylpyrimidin-2-amine, DIMETHYL SULFOXIDE, Purine nucleoside phosphorylase
著者Faheem, M, Neto, J.B, Collins, P, Pearce, N.M, Valadares, N.F, Bird, L, Pereira, H.M, Delft, F.V, Barbosa, J.A.R.G.
登録日2017-11-05
公開日2018-11-07
最終更新日2024-10-30
実験手法X-RAY DIFFRACTION (1.56 Å)
主引用文献Crystal Structure of Purine Nucleoside Phosphorylase Isoform 2 from Schistosoma mansoni in complex with 4-chloro-6-methylpyrimidin-2-amine
To Be Published
6BJ6
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BU of 6bj6 by Molmil
Crystal Structure of Purine Nucleoside Phosphorylase Isoform 2 from Schistosoma mansoni in complex with 2-{[(S)-benzenesulfinyl]methyl}benzoic acid
分子名称: 2-{[(S)-phenylsulfinyl]methyl}benzoic acid, DIMETHYL SULFOXIDE, Purine nucleoside phosphorylase
著者Faheem, M, Neto, J.B, Collins, P, Pearce, N.M, Valadares, N.F, Bird, L, Pereira, H.M, Delft, F.V, Barbosa, J.A.R.G.
登録日2017-11-05
公開日2018-11-07
最終更新日2024-10-23
実験手法X-RAY DIFFRACTION (1.73 Å)
主引用文献Crystal Structure of Purine Nucleoside Phosphorylase Isoform 2 from Schistosoma mansoni in complex with 2-{[(S)-benzenesulfinyl]methyl}benzoic acid
To Be Published
6LD2
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BU of 6ld2 by Molmil
Zika NS5 polymerase domain
分子名称: (1S,2S,4S,5R)-2,4-dimethoxy-5-thiophen-2-yl-cyclohexane-1-carboxylic acid, RNA-directed RNA polymerase NS5, ZINC ION
著者El Sahili, A, Lescar, J.
登録日2019-11-20
公開日2020-08-12
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Non-nucleoside Inhibitors of Zika Virus RNA-Dependent RNA Polymerase.
J.Virol., 94, 2020
6LD1
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BU of 6ld1 by Molmil
Zika NS5 polymerase domain
分子名称: 1,2-ETHANEDIOL, RNA-directed RNA polymerase NS5, ZINC ION
著者El Sahili, A, Lescar, J.
登録日2019-11-20
公開日2020-08-12
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Non-nucleoside Inhibitors of Zika Virus RNA-Dependent RNA Polymerase.
J.Virol., 94, 2020
6LD5
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BU of 6ld5 by Molmil
Zika NS5 polymerase domain
分子名称: 2,4-dimethoxy-5-thiophen-2-yl-benzoic acid, RNA-directed RNA polymerase NS5, ZINC ION, ...
著者El Sahili, A, Lescar, J.
登録日2019-11-20
公開日2020-08-19
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.94 Å)
主引用文献Non-nucleoside Inhibitors of Zika Virus RNA-Dependent RNA Polymerase.
J.Virol., 94, 2020
6LD4
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BU of 6ld4 by Molmil
Zika NS5 polymerase domain
分子名称: 2,4-dimethoxy-5-thiophen-2-yl-benzoic acid, 3-methoxybenzenesulfonamide, RNA-directed RNA polymerase NS5, ...
著者El Sahili, A, Lescar, J.
登録日2019-11-20
公開日2020-08-19
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Non-nucleoside Inhibitors of Zika Virus RNA-Dependent RNA Polymerase.
J.Virol., 94, 2020
6LD3
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BU of 6ld3 by Molmil
Zika NS5 polymerase domain
分子名称: 2,4-dimethoxy-5-thiophen-2-yl-benzoic acid, RNA-directed RNA polymerase NS5, ZINC ION, ...
著者El Sahili, A, Lescar, J.
登録日2019-11-20
公開日2020-08-19
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Non-nucleoside Inhibitors of Zika Virus RNA-Dependent RNA Polymerase.
J.Virol., 94, 2020
6YTM
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BU of 6ytm by Molmil
Human Brd2(BD2) L383V mutant in complex with ET-JQ1-OMe
分子名称: (2S)-1-[3-{[(2R)-2-hydroxypropyl]oxy}-2,2-bis({[(2R)-2-hydroxypropyl]oxy}methyl)propoxy]propan-2-ol, Bromodomain-containing protein 2, methyl (2R)-2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.0^{2,6}]trideca-2(6),4,7,10,12-pentaen-9-yl]butanoate
著者Bond, A.G, Ciulli, A, Cowan, A.D.
登録日2020-04-24
公開日2020-05-27
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.56 Å)
主引用文献Stereoselective synthesis of allele-specific BET inhibitors.
Org.Biomol.Chem., 18, 2020
1E2I
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BU of 1e2i by Molmil
The nucleoside binding site of Herpes simplex type 1 thymidine kinase analyzed by X-ray crystallography
分子名称: 9-HYDROXYPROPYLADENINE, R-ISOMER, S-ISOMER, ...
著者Vogt, J, Scapozza, L, Schulz, G.E.
登録日2000-05-23
公開日2000-11-06
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Nucleoside Binding Site of Herpes Simplex Type 1 Thymidine Kinase Analyzed by X-Ray Crystallography
Proteins, 41, 2000
2DXE
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BU of 2dxe by Molmil
Crystal structure of nucleoside diphosphate kinase in complex with GDP
分子名称: CHLORIDE ION, GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ...
著者Kato-Murayama, M, Murayama, K, Terada, T, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2006-08-25
公開日2007-02-25
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Crystal structure of nucleoside diphosphate kinase in complex with GDP
To be Published
8UW1
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BU of 8uw1 by Molmil
Cryo-EM structure of DNMT3A1 UDR in complex with H2AK119Ub-nucleosome
分子名称: DNA (146-MER), DNA (cytosine-5)-methyltransferase 3A, Histone H2A, ...
著者Gretarsson, K, Abini-Agbomson, S, Armache, K.-J, Lu, C.
登録日2023-11-05
公開日2024-09-11
最終更新日2025-05-21
実験手法ELECTRON MICROSCOPY (2.88 Å)
主引用文献Cancer-associated DNA hypermethylation of Polycomb targets requires DNMT3A dual recognition of histone H2AK119 ubiquitination and the nucleosome acidic patch.
Sci Adv, 10, 2024
1E2J
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BU of 1e2j by Molmil
The nucleoside binding site of Herpes simplex type 1 thymidine kinase analyzed by X-ray crystallography
分子名称: SULFATE ION, THYMIDINE, THYMIDINE KINASE
著者Vogt, J, Scapozza, L, Schulz, G.E.
登録日2000-05-23
公開日2000-11-06
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Nucleoside Binding Site of Herpes Simplex Type 1 Thymidine Kinase Analyzed by X-Ray Crystallography
Proteins: Struct.,Funct., Genet., 41, 2000
1E2H
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BU of 1e2h by Molmil
The nucleoside binding site of Herpes simplex type 1 thymidine kinase analyzed by X-ray crystallography
分子名称: SULFATE ION, THYMIDINE KINASE
著者Vogt, J, Scapozza, L, Schulz, G.E.
登録日2000-05-23
公開日2000-11-06
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Nucleoside Binding Site of Herpes Simplex Type 1 Thymidine Kinase Analyzed by X-Ray Crystallography
Proteins: Struct.,Funct., Genet., 41, 2000
8WG5
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BU of 8wg5 by Molmil
Cryo-EM structure of USP16 bound to H2AK119Ub nucleosome
分子名称: DNA (147-MER), Histone H2A type 1-B/E, Histone H2B type 1-K, ...
著者Ai, H.S, He, Z.Z, Deng, Z.H, Liu, L.
登録日2023-09-20
公開日2023-12-27
最終更新日2024-11-27
実験手法ELECTRON MICROSCOPY (3.05 Å)
主引用文献Structural and mechanistic basis for nucleosomal H2AK119 deubiquitination by single-subunit deubiquitinase USP16.
Nat.Struct.Mol.Biol., 31, 2024
6BI9
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BU of 6bi9 by Molmil
Crystal Structure of Purine Nucleoside Phosphorylase Isoform 2 from Schistosoma mansoni in complex with 1,2,5-trimethyl-1H-pyrrole-3-carboxylic acid
分子名称: 1,2,5-trimethyl-1H-pyrrole-3-carboxylic acid, DIMETHYL SULFOXIDE, Purine nucleoside phosphorylase
著者Faheem, M, Neto, J.B, Collins, P, Pearce, N.M, Valadares, N.F, Bird, L, Pereira, H.M, Delft, F.V, Barbosa, J.A.R.G.
登録日2017-11-01
公開日2018-11-07
最終更新日2024-11-20
実験手法X-RAY DIFFRACTION (1.59 Å)
主引用文献Crystal Structure of Purine Nucleoside Phosphorylase Isoform 2 from Schistosoma mansoni in complex with 1,2,5-trimethyl-1H-pyrrole-3-carboxylic acid
To Be Published
6BI1
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BU of 6bi1 by Molmil
Crystal Structure of Purine Nucleoside Phosphorylase Isoform 2 from Schistosoma mansoni in complex with (2R)-2-amino-3-(benzyloxy)propan-1-ol
分子名称: DIMETHYL SULFOXIDE, O-benzyl-L-serine, Purine nucleoside phosphorylase
著者Faheem, M, Neto, J.B, Collins, P, Pearce, N.M, Valadares, N.F, Bird, L, Pereira, H.M, Delft, F.V, Barbosa, J.A.R.G.
登録日2017-10-31
公開日2018-11-07
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (1.42 Å)
主引用文献Crystal Structure of Purine Nucleoside Phosphorylase Isoform 2 from Schistosoma mansoni in complex with (2R)-2-amino-3-(benzyloxy)propan-1-ol
To Be Published
9II7
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BU of 9ii7 by Molmil
RNA polymerase II elongation complex stalled at SHL(-1) of the nucleosome containing histone variant H2A.B
分子名称: DNA (198-MER), DNA-directed RNA polymerase subunit, DNA-directed RNA polymerase subunit beta, ...
著者Akatsu, M, Kujirai, T, Rina, H, Ehara, H, Takizawa, Y, Sekine, S, Kurumizaka, H.
登録日2024-06-19
公開日2025-06-11
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献Structural basis of RNAPII transcription on the nucleosome containing histone variant H2A.B.
Embo J., 2025
5GAN
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BU of 5gan by Molmil
The overall structure of the yeast spliceosomal U4/U6.U5 tri-snRNP at 3.7 Angstrom
分子名称: 13 kDa ribonucleoprotein-associated protein, GUANOSINE-5'-TRIPHOSPHATE, Pre-mRNA-processing factor 31, ...
著者Nguyen, T.H.D, Galej, W.P, Bai, X.C, Oubridge, C, Scheres, S.H.W, Newman, A.J, Nagai, K.
登録日2015-12-15
公開日2016-01-27
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (3.7 Å)
主引用文献Cryo-EM structure of the yeast U4/U6.U5 tri-snRNP at 3.7 angstrom resolution.
Nature, 530, 2016
2DXD
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BU of 2dxd by Molmil
Crystal structure of nucleoside diphosphate kinase in complex with ATP analog
分子名称: ADENOSINE MONOPHOSPHATE, CHLORIDE ION, Nucleoside diphosphate kinase
著者Kato-Murayama, M, Murayama, K, Terada, T, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2006-08-25
公開日2007-02-25
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.77 Å)
主引用文献Crystal structure of nucleoside diphosphate kinase in complex with ATP analog
To be Published
2DYA
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BU of 2dya by Molmil
Crystal structure of complex between Adenine nucleotide and nucleoside diphosphate kinase
分子名称: ADENOSINE-5'-DIPHOSPHATE, CHLORIDE ION, MAGNESIUM ION, ...
著者Kato-Murayama, M, Murayama, K, Terada, T, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2006-09-08
公開日2007-03-08
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.77 Å)
主引用文献Crystal structure of complex between Adenine nucleotide and nucleoside diphosphate kinase
To be Published
2DXF
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BU of 2dxf by Molmil
Crystal structure of nucleoside diphosphate kinase in complex with GTP analog
分子名称: CHLORIDE ION, Nucleoside diphosphate kinase, PHOSPHOAMINOPHOSPHONIC ACID-GUANYLATE ESTER
著者Kato-Murayama, M, Murayama, K, Terada, T, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2006-08-25
公開日2007-02-25
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Crystal structure of nucleoside diphosphate kinase in complex with GTP analog
To be Published
2DY9
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BU of 2dy9 by Molmil
Crystal structure of nucleoside diphosphate kinase in complex with ADP
分子名称: ADENOSINE-5'-DIPHOSPHATE, CHLORIDE ION, MAGNESIUM ION, ...
著者Kato-Murayama, M, Murayama, K, Terada, T, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2006-09-08
公開日2007-03-08
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.01 Å)
主引用文献Crystal structure of nucleoside diphosphate kinase in complex with ADP
To be Published
9OAI
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BU of 9oai by Molmil
Crystal structure of nucleoside-diphosphate kinase from Cryptosporidium parvum in complex with thymidine-5'-phosphate
分子名称: ACETATE ION, THYMIDINE-5'-PHOSPHATE, nucleoside-diphosphate kinase
著者Seattle Structural Genomics Center for Infectious Disease, Seattle Structural Genomics Center for Infectious Disease (SSGCID)
登録日2025-04-21
公開日2025-04-30
実験手法X-RAY DIFFRACTION (1.51 Å)
主引用文献Crystal structure of nucleoside-diphosphate kinase Cryptosporidium parvum in complex with thymidine-5'-phosphate
To be published

238582

件を2025-07-09に公開中

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