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2FGI
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BU of 2fgi by Molmil
CRYSTAL STRUCTURE OF THE TYROSINE KINASE DOMAIN OF FGF RECEPTOR 1 IN COMPLEX WITH INHIBITOR PD173074
分子名称: 1-TERT-BUTYL-3-[6-(3,5-DIMETHOXY-PHENYL)-2-(4-DIETHYLAMINO-BUTYLAMINO)-PYRIDO[2,3-D]PYRIMIDIN-7-YL]-UREA, PROTEIN (FIBROBLAST GROWTH FACTOR (FGF) RECEPTOR 1)
著者Mohammadi, M, Froum, S, Hamby, J.M, Schroeder, M, Panek, R.L, Lu, G.H, Eliseenkova, A.V, Green, D, Schlessinger, J, Hubbard, S.R.
登録日1998-09-15
公開日1999-09-13
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal structure of an angiogenesis inhibitor bound to the FGF receptor tyrosine kinase domain.
EMBO J., 17, 1998
1PT5
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Crystal structure of gene yfdW of E. coli
分子名称: ACETYL COENZYME *A, Hypothetical protein yfdW
著者Gruez, A, Roig-Zamboni, V, Valencia, C, Campanacci, V, Cambillau, C.
登録日2003-06-23
公開日2003-09-09
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献The Crystal Structure of the Escherichia coli YfdW Gene Product Reveals a New Fold of Two Interlaced Rings Identifying a Wide Family of CoA Transferases
J.Biol.Chem., 278, 2003
3KE8
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BU of 3ke8 by Molmil
Crystal structure of IspH:HMBPP-complex
分子名称: 4-HYDROXY-3-METHYL BUTYL DIPHOSPHATE, 4-hydroxy-3-methylbut-2-enyl diphosphate reductase, IRON/SULFUR CLUSTER
著者Groll, M, Graewert, T, Span, I, Eisenreich, W, Bacher, A.
登録日2009-10-24
公開日2010-01-12
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Probing the reaction mechanism of IspH protein by x-ray structure analysis.
Proc.Natl.Acad.Sci.USA, 107, 2010
3GZF
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BU of 3gzf by Molmil
Structure of the C-terminal domain of nsp4 from Feline Coronavirus
分子名称: Replicase polyprotein 1ab, SULFATE ION
著者Manolaridis, I, Wojdyla, J.A, Panjikar, S, Snijder, E.J, Gorbalenya, A.E, Coutard, B, Tucker, P.A.
登録日2009-04-07
公開日2009-08-18
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.756 Å)
主引用文献Structure of the C-terminal domain of nsp4 from feline coronavirus
Acta Crystallogr.,Sect.D, 65, 2009
1QNX
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Ves v 5, an allergen from Vespula vulgaris venom
分子名称: SODIUM ION, VES V 5
著者Henriksen, A, Gajhede, M, Spangfort, M.D.
登録日1999-10-25
公開日2000-10-26
最終更新日2018-01-17
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Major Venom Allergen of Yellow Jackets, Ves V 5: Structural Characterization of a Pathogenesis-Related Protein Superfamily.
Proteins: Struct.,Funct., Genet., 45, 2001
3KYC
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Human SUMO E1 complex with a SUMO1-AMP mimic
分子名称: 5'-deoxy-5'-(sulfamoylamino)adenosine, SUMO-activating enzyme subunit 1, SUMO-activating enzyme subunit 2, ...
著者Lima, C.D.
登録日2009-12-05
公開日2010-02-16
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献Active site remodelling accompanies thioester bond formation in the SUMO E1.
Nature, 463, 2010
3LQQ
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BU of 3lqq by Molmil
Structure of the CED-4 Apoptosome
分子名称: ADENOSINE-5'-TRIPHOSPHATE, Cell death protein 4, MAGNESIUM ION
著者Qi, S, Pang, Y, Shi, Y, Yan, N, Liu, Q.
登録日2010-02-09
公開日2010-04-28
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (3.534 Å)
主引用文献Crystal structure of the Caenorhabditis elegans apoptosome reveals an octameric assembly of CED-4.
Cell(Cambridge,Mass.), 141, 2010
1HL3
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CtBP/BARS in ternary complex with NAD(H) and PIDLSKK peptide
分子名称: C-TERMINAL BINDING PROTEIN 3, NICOTINAMIDE-ADENINE-DINUCLEOTIDE, PRO-ILE-ASP-LEU-SER-LYS-LYS PEPTIDE
著者Nardini, M, Spano, S, Cericola, C, Pesce, A, Massaro, A, Millo, E, Luini, A, Corda, D, Bolognesi, M.
登録日2003-03-13
公開日2003-06-19
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Ctbp/Bars: A Dual-Function Protein Involved in Transcription Co-Repression and Golgi Membrane Fission
Embo J., 22, 2003
1QXK
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Monoacid-Based, Cell Permeable, Selective Inhibitors of Protein Tyrosine Phosphatase 1B
分子名称: 2-{4-[2-ACETYLAMINO-3-(4-CARBOXYMETHOXY-3-HYDROXY-PHENYL)-PROPIONYLAMINO]-BUTOXY}-6-HYDROXY-BENZOIC ACID METHYL ESTER, Protein-tyrosine phosphatase, non-receptor type 1
著者Xin, Z, Liu, G, Abad-Zapatero, C, Pei, Z, Szczepankiewick, B.G, Li, X, Zhang, T, Hutchins, C.W, Hajduk, P.J, Ballaron, S.J, Stashko, M.A, Lubben, T.H, Trevillyan, J.M, Jirousek, M.R.
登録日2003-09-08
公開日2003-10-28
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Identification of a Monoacid-Based, Cell Permeable, Selective Inhibitor of Protein Tyrosine Phosphatase 1B
BIOORG.MED.CHEM.LETT., 13, 2003
1QYA
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CRYSTAL STRUCTURE OF E. COLI PROTEIN YDDE
分子名称: HYPOTHETICAL PROTEIN yddE
著者Grassick, A, Sulzenbacher, G, Roig-Zamboni, V, Campanacci, V, Cambillau, C, Bourne, Y.
登録日2003-09-10
公開日2004-06-08
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal structure of E. coli yddE protein reveals a striking homology with diaminopimelate epimerase
Proteins, 55, 2004
1LVG
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Crystal structure of mouse guanylate kinase in complex with GMP and ADP
分子名称: ADENOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-MONOPHOSPHATE, Guanylate kinase, ...
著者Sekulic, N, Shuvalova, L, Spangenberg, O, Konrad, M, Lavie, A.
登録日2002-05-28
公開日2002-12-11
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Structural characterization of the closed conformation of mouse guanylate kinase.
J.Biol.Chem., 277, 2002
1LY4
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Analysis of quinazoline and PYRIDO[2,3D]PYRIMIDINE N9-C10 reversed bridge antifolates in complex with NADP+ and Pneumocystis carinii dihydrofolate reductase
分子名称: 2,4-DIAMINO-6-[N-(3',5'-DIMETHOXYBENZYL)-N-METHYLAMINO]PYRIDO[2,3-D]PYRIMIDINE, DIHYDROFOLATE REDUCTASE, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE
著者Cody, V, Galitsky, N, Luft, J.R, Pangborn, W, Queener, S.F, Gangjee, A.
登録日2002-06-06
公開日2002-08-28
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Analysis of quinazoline and pyrido[2,3-d]pyrimidine N9-C10 reversed-bridge antifolates in complex with NADP+ and Pneumocystis carinii dihydrofolate reductase.
Acta Crystallogr.,Sect.D, 58, 2002
1QMB
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BU of 1qmb by Molmil
Cleaved alpha-1-antitrypsin polymer
分子名称: ALPHA-1-ANTITRYPSIN
著者Huntington, J.A, Pannu, N.S, Hazes, B, Read, R.J, Lomas, D.A, Carrell, R.W.
登録日1999-09-24
公開日2000-02-06
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献A 2.6A Structure of a Serpin Polymer and Implications for Conformational Disease
J.Mol.Biol., 293, 1999
1LY3
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ANALYSIS OF QUINAZOLINE AND PYRIDOPYRIMIDINE N9-C10 REVERSED BRIDGE ANTIFOLATES IN COMPLEX WITH NADP+ AND PNEUMOCYSTIS CARINII DIHYDROFOLATE REDUCTASE
分子名称: 2,4-DIAMINO-6-[N-(2',5'-DIMETHOXYBENZYL)-N-METHYLAMINO]QUINAZOLINE, DIHYDROFOLATE REDUCTASE, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE
著者Cody, V, Galitsky, N, Luft, J.R, Pangborn, W, Queener, S.F, Gangjee, A.
登録日2002-06-06
公開日2002-08-28
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Analysis of quinazoline and pyrido[2,3-d]pyrimidine N9-C10 reversed-bridge antifolates in complex with NADP+ and Pneumocystis carinii dihydrofolate reductase.
Acta Crystallogr.,Sect.D, 58, 2002
2EBO
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BU of 2ebo by Molmil
CORE STRUCTURE OF GP2 FROM EBOLA VIRUS
分子名称: CHLORIDE ION, EBOLA VIRUS ENVELOPE GLYCOPROTEIN
著者Malashkevich, V.N, Schneider, B.J, Mcnally, M.L, Milhollen, M.A, Pang, J.X, Kim, P.S.
登録日1998-12-24
公開日1999-05-18
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Core structure of the envelope glycoprotein GP2 from Ebola virus at 1.9-A resolution.
Proc.Natl.Acad.Sci.USA, 96, 1999
2FGG
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Crystal Structure of Rv2632c
分子名称: Hypothetical protein Rv2632c/MT2708
著者Yu, M, Bursey, E.H, Radhakannan, T, Segelke, B.W, Lekin, T, Toppani, D, Kim, C.Y, Kaviratne, T, Woodruff, T, Terwilliger, T.C, Hung, L.W, TB Structural Genomics Consortium (TBSGC)
登録日2005-12-21
公開日2006-02-14
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal Structure of Rv2632c
To be Published
1MQM
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BU of 1mqm by Molmil
BHA/LSTa
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Hemagglutinin HA1 chain, ...
著者ha, y, steven, d.j, skehel, j.j, wiley, d.c.
登録日2002-09-16
公開日2003-08-26
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献X-ray structure of the hemagglutinin of a potential H3 avian progenitor of the 1968 Hong Kong pandemic influenza virus.
Virology, 309, 2003
2G4V
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anomalous substructure of proteinase K
分子名称: CALCIUM ION, CHLORIDE ION, POTASSIUM ION, ...
著者Mueller-Dieckmann, C, Weiss, M.S.
登録日2006-02-22
公開日2007-02-20
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.14 Å)
主引用文献On the routine use of soft X-rays in macromolecular crystallography. Part IV. Efficient determination of anomalous substructures in biomacromolecules using longer X-ray wavelengths.
Acta Crystallogr.,Sect.D, 63, 2007
2G4I
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Anomalous substructure of Concanavalin A
分子名称: CALCIUM ION, CHLORIDE ION, Concanavalin A, ...
著者Mueller-Dieckmann, C, Weiss, M.S.
登録日2006-02-22
公開日2007-02-20
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献On the routine use of soft X-rays in macromolecular crystallography. Part IV. Efficient determination of anomalous substructures in biomacromolecules using longer X-ray wavelengths.
Acta Crystallogr.,Sect.D, 63, 2007
5X9C
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Crystal structure of the cytosolic domain of human MiD51
分子名称: Mitochondrial dynamics protein MID51
著者Sun, F, Pang, X, Ma, J.
登録日2017-03-06
公開日2018-03-21
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献New interfaces on MiD51 for Drp1 recruitment and mitochondrial fission regulation
To Be Published
3EJC
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Full length Receptor Binding Protein from Lactococcal phage TP901-1
分子名称: Baseplate protein (BPP)
著者Spinelli, S, Lichiere, J, Blangy, S, Sciara, G, Cambillau, C, Campanacci, V.
登録日2008-09-18
公開日2009-10-06
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Structure and molecular assignment of lactococcal phage TP901-1 baseplate.
J.Biol.Chem., 285, 2010
3ELN
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A Putative Fe2+-bound Persulfenate Intermediate in Cysteine Dioxygenase
分子名称: Cysteine dioxygenase type 1, FE (II) ION, S-HYDROPEROXYCYSTEINE
著者Simmons, C.R, Stipanuk, M.H, Karplus, P.A.
登録日2008-09-22
公開日2008-10-21
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.42 Å)
主引用文献A putative Fe2+-bound persulfenate intermediate in cysteine dioxygenase.
Biochemistry, 47, 2008
3E4O
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Crystal structure of succinate bound state DctB
分子名称: C4-dicarboxylate transport sensor protein dctB, MAGNESIUM ION, SUCCINIC ACID
著者Zhou, Y.F, Nan, J, Nan, B.Y, Liang, Y.H, Panjikar, S, Su, X.D.
登録日2008-08-12
公開日2008-10-21
最終更新日2017-10-25
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献C4-dicarboxylates sensing mechanism revealed by the crystal structures of DctB sensor domain.
J.Mol.Biol., 383, 2008
1WQ3
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Escherichia coli tyrosyl-tRNA synthetase mutant complexed with 3-iodo-L-tyrosine
分子名称: 3-IODO-TYROSINE, Tyrosyl-tRNA synthetase
著者Kobayashi, T, Sakamoto, K, Nureki, O, Takimura, T, Kamata, K, Sekine, R, Nishimura, S, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2004-09-20
公開日2005-01-25
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural basis of nonnatural amino acid recognition by an engineered aminoacyl-tRNA synthetase for genetic code expansion
Proc.Natl.Acad.Sci.USA, 102, 2005
2TLX
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THERMOLYSIN (NATIVE)
分子名称: CALCIUM ION, DIMETHYL SULFOXIDE, LYSINE, ...
著者English, A.C, Done, S.H, Groom, C.R, Hubbard, R.E.
登録日1999-01-28
公開日2000-03-13
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Locating interaction sites on proteins: the crystal structure of thermolysin soaked in 2% to 100% isopropanol.
Proteins, 37, 1999

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