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7MQM
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AAC(3)-IIIa in complex with CoA and gentamicin
分子名称: Aminoglycoside N(3)-acetyltransferase III, COENZYME A, GLYCEROL, ...
著者Zielinski, M, Berghuis, A.M.
登録日2021-05-05
公開日2022-07-06
最終更新日2022-08-17
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structural elucidation of substrate-bound aminoglycoside acetyltransferase (3)-IIIa.
Plos One, 17, 2022
7MQL
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AAC(3)-IIIa in complex with CoA and neomycin
分子名称: Aminoglycoside N(3)-acetyltransferase III, COENZYME A, FORMIC ACID, ...
著者Zielinski, M, Berghuis, A.M.
登録日2021-05-05
公開日2022-07-06
最終更新日2022-08-17
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structural elucidation of substrate-bound aminoglycoside acetyltransferase (3)-IIIa.
Plos One, 17, 2022
3Q27
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Cyrstal structure of human alpha-synuclein (32-57) fused to maltose binding protein (MBP)
分子名称: GLYCEROL, Maltose-binding periplasmic protein/alpha-synuclein chimeric protein, SULFATE ION, ...
著者Zhao, M, Sawaya, M.R, Cascio, D, Eisenberg, D.
登録日2010-12-19
公開日2011-06-01
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.302 Å)
主引用文献Structures of segments of alpha-synuclein fused to maltose-binding protein suggest intermediate states during amyloid formation
Protein Sci., 20, 2011
4BBA
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Crystal structure of glucokinase regulatory protein complexed to phosphate
分子名称: GLUCOKINASE REGULATORY PROTEIN, PHOSPHATE ION
著者Pautsch, A, Stadler, N, Loehle, A, Lenter, M, Rist, W, Berg, A, Glocker, L, Nar, H, Reinhart, D, Heckel, A, Schnapp, G, Kauschke, S.G.
登録日2012-09-21
公開日2013-05-15
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.92 Å)
主引用文献Crystal Structure of Glucokinase Regulatory Protein.
Biochemistry, 52, 2013
3Q2X
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Structure of an amyloid forming peptide NKGAII (residues 27-32) from amyloid beta
分子名称: Amyloid beta A4 protein
著者Soriaga, A.B, Sawaya, M.R, Eisenberg, D.
登録日2010-12-20
公開日2011-10-12
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.451 Å)
主引用文献Molecular basis for amyloid-beta polymorphism.
Proc.Natl.Acad.Sci.USA, 108, 2011
4BG9
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Apo form of a putative sugar kinase MK0840 from Methanopyrus kandleri (orthorhombic space group)
分子名称: ACETATE ION, CHLORIDE ION, POTASSIUM ION, ...
著者Schacherl, M, Waltersperger, S.M, Baumann, U.
登録日2013-03-24
公開日2013-11-27
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.902 Å)
主引用文献Structural Characterization of the Ribonuclease H-Like Type Askha Superfamily Kinase Mk0840 from Methanopyrus Kandleri
Acta Crystallogr.,Sect.D, 69, 2013
4BLJ
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Galectin-3c in complex with Bisamido-thiogalactoside derivate 2
分子名称: Bis-(3-deoxy-3-(3-methoxy-benzamido)-b-D-galactopyranosyl)-sulfide, GALECTIN-3
著者Noresson, A.L, Oberg, C.T, Engstrom, O, Hakansson, M, Logan, D.T, Leffler, H, Nilsson, U.J.
登録日2013-05-03
公開日2014-05-14
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.2 Å)
主引用文献Controlling Protein Conformation Through Electronic Fine-Tuning of Arginine-Arene Interactions: Synthetic, Structural, and Biological Studies
To be Published
1UG3
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C-terminal portion of human eIF4GI
分子名称: eukaryotic protein synthesis initiation factor 4G
著者Bellsolell, L, Cho-Park, P.F, Poulin, F, Sonenberg, N, Burley, S.K.
登録日2003-06-11
公開日2005-03-22
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.24 Å)
主引用文献Two structurally atypical HEAT domains in the C-terminal portion of human eIF4G support binding to eIF4A and Mnk1
Structure, 14, 2006
1TOW
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Crystal structure of human adipocyte fatty acid binding protein in complex with a carboxylic acid ligand
分子名称: 4-(9H-CARBAZOL-9-YL)BUTANOIC ACID, Fatty acid-binding protein, adipocyte
著者Lehmann, F, Haile, S, Axen, E, Medina, C, Uppenberg, J, Svensson, S, Lundback, T, Rondahl, L, Barf, T.
登録日2004-06-15
公開日2004-08-24
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Discovery of inhibitors of human adipocyte fatty acid-binding protein, a potential type 2 diabetes target.
Bioorg.Med.Chem.Lett., 14, 2004
1TVZ
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Crystal structure of 3-hydroxy-3-methylglutaryl-coenzyme A synthase from Staphylococcus aureus
分子名称: 3-hydroxy-3-methylglutaryl-CoA synthase, SULFATE ION
著者Campobasso, N, Patel, M, Wilding, I.E, Kallender, H, Rosenberg, M, Gwynn, M.
登録日2004-06-30
公開日2004-08-31
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Staphylococcus aureus 3-hydroxy-3-methylglutaryl-CoA synthase: crystal structure and mechanism
J.Biol.Chem., 279, 2004
1TWG
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RNA polymerase II complexed with CTP
分子名称: CYTIDINE-5'-TRIPHOSPHATE, DNA-directed RNA polymerase II 13.6 kDa polypeptide, DNA-directed RNA polymerase II 14.2 kDa polypeptide, ...
著者Westover, K.D, Bushnell, D.A, Kornberg, R.D.
登録日2004-06-30
公開日2004-11-16
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献Structural basis of transcription: nucleotide selection by rotation in the RNA polymerase II active center.
Cell(Cambridge,Mass.), 119, 2004
3ZY1
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Crystal structure of the human p63 tetramerization domain
分子名称: TUMOR PROTEIN 63
著者Natan, E, Joerger, A.C.
登録日2011-08-16
公開日2011-11-30
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Structure and Kinetic Stability of the P63 Tetramerization Domain.
J.Mol.Biol., 415, 2012
3ZYH
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CRYSTAL STRUCTURE OF PA-IL LECTIN COMPLEXED WITH GALBG0 AT 1.5 A RESOLUTION
分子名称: 3-(beta-D-galactopyranosylthio)propanoic acid, CALCIUM ION, PA-I galactophilic lectin
著者Kadam, R.U, Bergmann, M, Hurley, M, Garg, D, Cacciarini, M, Swiderska, M.A, Nativi, C, Sattler, M, Smyth, A.R, Williams, P, Camara, M, Stocker, A, Darbre, T, Reymond, J.-L.
登録日2011-08-23
公開日2011-09-21
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.501 Å)
主引用文献A Glycopeptide Dendrimer Inhibitor of the Galactose Specific Lectin Leca and of Pseudomonas Aeruginosa Biofilms
Angew.Chem.Int.Ed.Engl., 50, 2011
3ZYB
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CRYSTAL STRUCTURE OF PA-IL LECTIN COMPLEXED WITH GALAG0 AT 2.3 A RESOLUTION
分子名称: CALCIUM ION, GALA-LYS-PRO-LEUNH2, P-HYDROXYBENZOIC ACID, ...
著者Kadam, R.U, Bergmann, M, Hurley, M, Garg, D, Cacciarini, M, Swiderska, M.A, Nativi, C, Sattler, M, Smyth, A.R, Williams, P, Camara, M, Stocker, A, Darbre, T, Reymond, J.-L.
登録日2011-08-19
公開日2011-09-21
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.29 Å)
主引用文献A Glycopeptide Dendrimer Inhibitor of the Galactose-Specific Lectin Leca and of Pseudomonas Aeruginosa Biofilms.
Angew.Chem.Int.Ed.Engl., 50, 2011
3ZYF
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CRYSTAL STRUCTURE OF PA-IL LECTIN COMPLEXED WITH NPG AT 1.9 A RESOLUTION
分子名称: 4-nitrophenyl beta-D-galactopyranoside, CALCIUM ION, PA-I GALACTOPHILIC LECTIN
著者Kadam, R.U, Bergmann, M, Hurley, M, Garg, D, Cacciarini, M, Swiderska, M.A, Nativi, C, Sattler, M, Smyth, A.R, Williams, P, Camara, M, Stocker, A, Darbre, T, Reymond, J.-L.
登録日2011-08-22
公開日2011-09-21
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.944 Å)
主引用文献A Glycopeptide Dendrimer Inhibitor of the Galactose-Specific Lectin Leca and of Pseudomonas Aeruginosa Biofilms.
Angew.Chem.Int.Ed.Engl., 50, 2011
3NI3
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54-Membered ring macrocyclic beta-sheet peptide
分子名称: 54-membered ring macrocyclic beta-sheet peptide, ISOPROPYL ALCOHOL
著者Sawaya, M.R, Eisenberg, D, Nowick, J.S, Korman, T.P, Khakshoor, O.
登録日2010-06-15
公開日2010-09-15
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.34 Å)
主引用文献X-ray crystallographic structure of an artificial beta-sheet dimer.
J.Am.Chem.Soc., 132, 2010
1TBP
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BU of 1tbp by Molmil
CRYSTAL STRUCTURE OF YEAST TATA-BINDING PROTEIN AND MODEL FOR INTERACTION WITH DNA
分子名称: TATA-BINDING PROTEIN
著者Chasman, D.I, Flaherty, K.M, Sharp, P.A, Kornberg, R.D.
登録日1993-08-02
公開日1994-01-31
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Crystal structure of yeast TATA-binding protein and model for interaction with DNA.
Proc.Natl.Acad.Sci.USA, 90, 1993
1TOK
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Maleic acid-bound structure of SRHEPT mutant of E. coli aspartate aminotransferase
分子名称: Aspartate aminotransferase, MALEIC ACID
著者Chow, M.A, McElroy, K.E, Corbett, K.D, Berger, J.M, Kirsch, J.F.
登録日2004-06-14
公開日2004-10-05
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Narrowing substrate specificity in a directly evolved enzyme: the A293D mutant of aspartate aminotransferase
Biochemistry, 43, 2004
3ZC3
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FERREDOXIN-NADP REDUCTASE (MUTATION S80A) COMPLEXED WITH NADP BY COCRYSTALLIZATION
分子名称: FERREDOXIN-NADP REDUCTASE, FLAVIN-ADENINE DINUCLEOTIDE, GLYCEROL, ...
著者Martinez-Julvez, M, Hurtado-Guerrero, R, Herguedas, B, Sanchez-Azqueta, A, Hervas, M, Navarro, J.A, Medina, M.
登録日2012-11-15
公開日2013-11-20
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献A Hydrogen Bond Network in the Active Site of Anabaena Ferredoxin-Nadp(+) Reductase Modulates its Catalytic Efficiency.
Biochim.Biophys.Acta, 1837, 2013
1TOJ
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Hydrocinnamic acid-bound structure of SRHEPT mutant of E. coli aspartate aminotransferase
分子名称: Aspartate aminotransferase, HYDROCINNAMIC ACID
著者Chow, M.A, McElroy, K.E, Corbett, K.D, Berger, J.M, Kirsch, J.F.
登録日2004-06-14
公開日2004-10-05
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Narrowing substrate specificity in a directly evolved enzyme: the A293D mutant of aspartate aminotransferase
Biochemistry, 43, 2004
1TOO
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Interleukin 1B Mutant F146W
分子名称: Interleukin-1 beta
著者Adamek, D.H, Guerrero, L, Caspar, D.L.
登録日2004-06-14
公開日2004-12-07
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Structural and energetic consequences of mutations in a solvated hydrophobic cavity.
J.Mol.Biol., 346, 2005
1TP0
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Triple mutation in interleukin 1 beta cavity:replacement of phenylalanines with tryptophan.
分子名称: Interleukin-1 beta
著者Adamek, D.H, Guerrero, L, Caspar, D.L.
登録日2004-06-15
公開日2005-02-08
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structural and energetic consequences of mutations in a solvated hydrophobic cavity.
J.Mol.Biol., 346, 2005
3PPD
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GGVLVN segment from Human Prostatic Acid Phosphatase Residues 260-265, involved in Semen-Derived Enhancer of Viral Infection
分子名称: ACETIC ACID, GGVLVN peptide, amyloid forming segment, ...
著者Zhao, A, Sawaya, M.R, Eisenberg, D.
登録日2010-11-24
公開日2011-06-29
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Structure-based design of non-natural amino-acid inhibitors of amyloid fibril formation.
Nature, 475, 2011
1TR7
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FimH adhesin receptor binding domain from uropathogenic E. coli
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, CACODYLATE ION, FimH protein, ...
著者Bouckaert, J, Berglund, J, Schembri, M, De Genst, E, Cools, L, Wuhrer, M, Hung, C.S, Pinkner, J, Slattegard, R, Zavialov, A, Choudhury, D, Langermann, S, Hultgren, S.J, Wyns, L, Klemm, P, Oscarson, S, Knight, S.D, De Greve, H.
登録日2004-06-21
公開日2005-05-03
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Receptor binding studies disclose a novel class of high-affinity inhibitors of the Escherichia coli FimH adhesin
Mol.Microbiol., 55, 2005
3ZUO
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OMCI in complex with leukotriene B4
分子名称: COMPLEMENT INHIBITOR, LEUKOTRIENE B4
著者Roversi, P, Maillet, I, Togbe, D, Couillin, I, Quesniaux, V.F.J, Teixeira, M, Ahmat, N, Lissina, O, Boland, W, Ploss, K, Caesar, J.J.E, Leonhartsberger, S, Ryffel, B, Lea, S.M, Nunn, M.A.
登録日2011-07-19
公開日2012-08-01
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.86 Å)
主引用文献Bifunctional Lipocalin Ameliorates Murine Immune Complex-Induced Acute Lung Injury.
J.Biol.Chem., 288, 2013

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