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3OBP
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Anaerobic complex of urate oxidase with uric acid
分子名称: SODIUM ION, URIC ACID, Uricase
著者Gabison, L, Chopard, C, Colloc'h, N, El Hajji, M, Castro, B, Chiadmi, M, Prange, T.
登録日2010-08-08
公開日2011-06-22
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献X-ray, ESR, and quantum mechanics studies unravel a spin well in the cofactor-less urate oxidase.
Proteins, 79, 2011
3M9S
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BU of 3m9s by Molmil
Crystal structure of respiratory complex I from Thermus thermophilus
分子名称: FE2/S2 (INORGANIC) CLUSTER, FLAVIN MONONUCLEOTIDE, IRON/SULFUR CLUSTER, ...
著者Efremov, R.G, Baradaran, R, Sazanov, L.A.
登録日2010-03-22
公開日2010-05-26
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (4.5 Å)
主引用文献The architecture of respiratory complex I
Nature, 465, 2010
4CI2
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BU of 4ci2 by Molmil
Structure of the DDB1-CRBN E3 ubiquitin ligase bound to lenalidomide
分子名称: DNA DAMAGE-BINDING PROTEIN 1, PROTEIN CEREBLON, S-Lenalidomide, ...
著者Fischer, E.S, Boehm, K, Thoma, N.H.
登録日2013-12-05
公開日2014-07-16
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (2.95 Å)
主引用文献Structure of the Ddb1-Crbn E3 Ubiquitin Ligase in Complex with Thalidomide.
Nature, 512, 2014
3P3P
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Factor inhibiting HIF-1 Alpha in complex with Notch 1 fragment mouse notch (1997-2016) peptide
分子名称: 2-OXOGLUTARIC ACID, FE (II) ION, GLYCEROL, ...
著者McDonough, M.A, Schofield, C.J.
登録日2010-10-05
公開日2010-11-24
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Asparaginyl hydroxylation of the Notch ankyrin repeat domain by factor inhibiting hypoxia-inducible factor
J.Biol.Chem., 282, 2007
4DUS
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BU of 4dus by Molmil
Structure of Bace-1 (Beta-Secretase) in complex with N-((2S,3R)-1-(4-fluorophenyl)-3-hydroxy-4-((6'-neopentyl-3',4'-dihydrospiro[cyclobutane-1,2'-pyrano[2,3-b]pyridin]-4'-yl)amino)butan-2-yl)acetamide
分子名称: Beta-secretase 1, GLYCEROL, IODIDE ION, ...
著者Sickmier, E.A.
登録日2012-02-22
公開日2012-10-10
最終更新日2014-07-02
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献A Potent and Orally Efficacious, Hydroxyethylamine-Based Inhibitor of beta-Secretase.
ACS Med Chem Lett, 3, 2012
3P3N
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Factor inhibiting HIF-1 Alpha in complex with Notch 1 fragment mouse notch (1930-1949) peptide
分子名称: 2-OXOGLUTARIC ACID, FE (II) ION, GLYCEROL, ...
著者McDonough, M.A, Schofield, C.J.
登録日2010-10-05
公開日2010-11-24
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Asparaginyl hydroxylation of the Notch ankyrin repeat domain by factor inhibiting hypoxia-inducible factor
J.Biol.Chem., 282, 2007
4ER4
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BU of 4er4 by Molmil
HIGH-RESOLUTION X-RAY ANALYSES OF RENIN INHIBITOR-ASPARTIC PROTEINASE COMPLEXES
分子名称: ENDOTHIAPEPSIN, H-142
著者Foundling, S.I, Watson, F.E, Szelke, M, Blundell, T.L.
登録日1991-01-05
公開日1991-04-15
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献High resolution X-ray analyses of renin inhibitor-aspartic proteinase complexes.
Nature, 327, 1987
3MWE
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BU of 3mwe by Molmil
Truncated Human ATP-Citrate Lyase with Tartrate Bound
分子名称: ATP-citrate synthase, L(+)-TARTARIC ACID, MAGNESIUM ION
著者Fraser, M.E, Sun, T.
登録日2010-05-05
公開日2010-06-16
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Identification of the citrate-binding site of human ATP-citrate lyase using X-ray crystallography.
J.Biol.Chem., 285, 2010
4ER1
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THE ACTIVE SITE OF ASPARTIC PROTEINASES
分子名称: ENDOTHIAPEPSIN, N-[(1R,2R,4R)-1-(cyclohexylmethyl)-2-hydroxy-6-methyl-4-{[(2R)-2-methylbutyl]carbamoyl}heptyl]-3-(1H-imidazol-3-ium-4-yl)-N~2~-[3-naphthalen-1-yl-2-(naphthalen-1-ylmethyl)propanoyl]-L-alaninamide
著者Quail, J.W, Cooper, J.B, Szelke, M, Blundell, T.L.
登録日1990-10-14
公開日1991-01-15
最終更新日2017-11-29
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献The active site of aspartic proteinases
FEBS Lett., 174, 1984
4F0H
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UNACTIVATED RUBISCO with OXYGEN BOUND
分子名称: OXYGEN MOLECULE, PHOSPHATE ION, Ribulose bisphosphate carboxylase large chain, ...
著者Stec, B.
登録日2012-05-04
公開日2012-11-14
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.96 Å)
主引用文献Structural mechanism of RuBisCO activation by carbamylation of the active site lysine.
Proc.Natl.Acad.Sci.USA, 109, 2012
3MWD
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Truncated Human ATP-Citrate Lyase with Citrate Bound
分子名称: ATP-citrate synthase, CITRIC ACID
著者Fraser, M.E, Sun, T.
登録日2010-05-05
公開日2010-06-16
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Identification of the citrate-binding site of human ATP-citrate lyase using X-ray crystallography.
J.Biol.Chem., 285, 2010
4F0M
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UNACTIVATED RUBISCO with MAGNESIUM AND A WATER MOLECULE BOUND
分子名称: CHLORIDE ION, GLYCEROL, MAGNESIUM ION, ...
著者Stec, B.
登録日2012-05-04
公開日2012-11-14
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Structural mechanism of RuBisCO activation by carbamylation of the active site lysine.
Proc.Natl.Acad.Sci.USA, 109, 2012
4C39
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Structure of rat neuronal nitric oxide synthase heme domain in complex with 6-((((3S, 5R)-5-(((6-amino-4-methylpyridin-2-yl)methoxy) methyl)pyrrolidin-3-yl)oxy)methyl)-4-methylpyridin-2-amine
分子名称: 5,6,7,8-TETRAHYDROBIOPTERIN, 6-((((3S, 5R)-5-(((6-amino-4-methylpyridin-2-yl)methoxy)methyl)pyrrolidin-3-yl)oxy)methyl)-4-methylpyridin-2-amine, ...
著者Li, H, Poulos, T.L.
登録日2013-08-22
公開日2014-04-02
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.98 Å)
主引用文献An Accessible Chiral Linker to Enhance Potency and Selectivity of Neuronal Nitric Oxide Synthase Inhibitors.
Acs Med.Chem.Lett., 5, 2014
4F0K
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UNACTIVATED RUBISCO with MAGNESIUM AND CARBON DIOXIDE BOUND
分子名称: CARBON DIOXIDE, CHLORIDE ION, GLYCEROL, ...
著者Stec, B.
登録日2012-05-04
公開日2012-11-14
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Structural mechanism of RuBisCO activation by carbamylation of the active site lysine.
Proc.Natl.Acad.Sci.USA, 109, 2012
4CI1
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Structure of the DDB1-CRBN E3 ubiquitin ligase bound to thalidomide
分子名称: DNA DAMAGE-BINDING PROTEIN 1, PROTEIN CEREBLON, S-Thalidomide, ...
著者Fischer, E.S, Boehm, K, Thoma, N.H.
登録日2013-12-05
公開日2014-07-16
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (2.98 Å)
主引用文献Structure of the Ddb1-Crbn E3 Ubiquitin Ligase in Complex with Thalidomide.
Nature, 512, 2014
4FQM
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Structure of B/Brisbane/60/2008 Influenza Hemagglutinin
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Hemagglutinin HA1, ...
著者Dreyfus, C, Laursen, N.S, Wilson, I.A.
登録日2012-06-25
公開日2012-08-22
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (3.45 Å)
主引用文献Highly conserved protective epitopes on influenza B viruses.
Science, 337, 2012
4ER2
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BU of 4er2 by Molmil
The active site of aspartic proteinases
分子名称: ENDOTHIAPEPSIN, PEPSTATIN, SULFATE ION
著者Bailey, D, Veerapandian, B, Cooper, J.B, Blundell, T.L.
登録日1990-10-20
公開日1991-01-15
最終更新日2017-11-29
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献The active site of aspartic proteinases
FEBS Lett., 174, 1984
3NB3
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BU of 3nb3 by Molmil
The host outer membrane proteins OmpA and OmpC are packed at specific sites in the Shigella phage Sf6 virion as structural components
分子名称: Outer membrane protein A, Outer membrane protein C
著者Zhao, H, Sequeira, R.D, Galeva, N.A, Tang, L.
登録日2010-06-02
公開日2011-02-16
最終更新日2024-02-21
実験手法ELECTRON MICROSCOPY (19 Å)
主引用文献The host outer membrane proteins OmpA and OmpC are associated with the Shigella phage Sf6 virion.
Virology, 409, 2011
3N7Z
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BU of 3n7z by Molmil
Crystal structure of acetyltransferase from Bacillus anthracis
分子名称: Acetyltransferase, GNAT family, SODIUM ION
著者Chang, C, Wu, R, Gornicki, P, Zhang, R, Joachimiak, A, Midwest Center for Structural Genomics (MCSG)
登録日2010-05-27
公開日2010-06-16
最終更新日2017-11-08
実験手法X-RAY DIFFRACTION (2.75 Å)
主引用文献Biochemical and Structural Analysis of an Eis Family Aminoglycoside Acetyltransferase from Bacillus anthracis.
Biochemistry, 54, 2015
4FQL
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Influenza B HA Antibody (Fab) CR8033
分子名称: monoclonal antibody CR8033 heavy chain, monoclonal antibody CR8033 light chain
著者Dreyfus, C, Laursen, N.S, Wilson, I.A.
登録日2012-06-25
公開日2012-08-22
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.898 Å)
主引用文献Highly conserved protective epitopes on influenza B viruses.
Science, 337, 2012
4FQV
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BU of 4fqv by Molmil
Crystal structure of broadly neutralizing antibody CR9114 bound to H7 influenza hemagglutinin
分子名称: Antibody CR9114 heavy chain, Antibody CR9114 light chain, Hemagglutinin HA1, ...
著者Ekiert, D.C, Dreyfus, C, Wilson, I.A.
登録日2012-06-25
公開日2012-08-22
最終更新日2018-01-31
実験手法X-RAY DIFFRACTION (5.75 Å)
主引用文献Highly conserved protective epitopes on influenza B viruses.
Science, 337, 2012
3NF1
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BU of 3nf1 by Molmil
Crystal structure of the TPR domain of kinesin light chain 1
分子名称: Kinesin light chain 1
著者Tong, Y, Tempel, W, Shen, L, Shen, Y, Nedyalkova, L, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Weigelt, J, Bochkarev, A, Park, H, Structural Genomics Consortium (SGC)
登録日2010-06-09
公開日2011-05-25
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Crystal structure of the TPR domain of kinesin light chain 1
to be published
4FQH
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Crystal Structure of Fab CR9114
分子名称: 1,2-ETHANEDIOL, NITRATE ION, antibody CR9114 heavy chain, ...
著者Dreyfus, C, Wilson, I.A.
登録日2012-06-25
公開日2012-08-22
最終更新日2018-01-31
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Highly conserved protective epitopes on influenza B viruses.
Science, 337, 2012
3PWH
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Thermostabilised Adenosine A2A Receptor
分子名称: 4-{2-[(7-amino-2-furan-2-yl[1,2,4]triazolo[1,5-a][1,3,5]triazin-5-yl)amino]ethyl}phenol, Adenosine receptor A2a
著者Dore, A.S, Robertson, N, Errey, J.C, Ng, I, Tehan, B, Hurrell, E, Magnani, F, Tate, C.G, Weir, M, Marshall, F.H.
登録日2010-12-08
公開日2011-09-07
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (3.296 Å)
主引用文献Structure of the adenosine A(2A) receptor in complex with ZM241385 and the xanthines XAC and caffeine
Structure, 19, 2011
3OFK
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Crystal structure of N-methyltransferase NodS from Bradyrhizobium japonicum WM9 in complex with S-adenosyl-l-homocysteine (SAH)
分子名称: Nodulation protein S, S-ADENOSYL-L-HOMOCYSTEINE
著者Cakici, O, Sikorski, M, Stepkowski, T, Bujacz, G, Jaskolski, M.
登録日2010-08-15
公開日2010-10-27
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Crystal Structures of NodS N-Methyltransferase from Bradyrhizobium japonicum in Ligand-Free Form and as SAH Complex.
J.Mol.Biol., 404, 2010

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