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1M2S
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Solution Structure of A New Potassium Channels Blocker from the Venom of Chinese Scorpion Buthus martensi Karsch
分子名称: Toxin BmTX3
著者Wang, Y, Li, M, Zhang, N, Wu, G, Hu, G, Wu, H.
登録日2002-06-25
公開日2004-04-06
最終更新日2022-02-23
実験手法SOLUTION NMR
主引用文献The solution structure of BmTx3B, a member of the scorpion toxin subfamily alpha-KTx 16
Proteins, 58, 2005
1HP2
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BU of 1hp2 by Molmil
SOLUTION STRUCTURE OF A TOXIN FROM THE SCORPION TITYUS SERRULATUS (TSTX-K ALPHA) DETERMINED BY NMR.
分子名称: TITYUSTOXIN K ALPHA
著者Ellis, K.C, Tenenholz, T.C, Gilly, W.F, Blaustein, M.P, Weber, D.J.
登録日2000-12-12
公開日2001-06-13
最終更新日2022-02-23
実験手法SOLUTION NMR
主引用文献Interaction of a toxin from the scorpion Tityus serrulatus with a cloned K+ channel from squid (sqKv1A).
Biochemistry, 40, 2001
6WHG
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BU of 6whg by Molmil
PI3P and calcium bound full-length TRPY1 in detergent
分子名称: (2R)-1-(butanoyloxy)-3-{[(R)-hydroxy{[(1S,2S,3S,4S,5S,6R)-2,3,4,6-tetrahydroxy-5-(phosphonooxy)cyclohexyl]oxy}phosphoryl]oxy}propan-2-yl hexadecanoate, CALCIUM ION, Calcium channel YVC1
著者Ahmed, T, Moiseenkova-Bell, V.Y.
登録日2020-04-08
公開日2021-04-21
最終更新日2024-05-29
実験手法ELECTRON MICROSCOPY (3.1 Å)
主引用文献Structure of the ancient TRPY1 channel from Saccharomyces cerevisiae reveals mechanisms of modulation by lipids and calcium.
Structure, 30, 2022
2N6O
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BU of 2n6o by Molmil
Structure of spider-venom peptide Hm1a
分子名称: Kappa-theraphotoxin-Hm1a
著者Undheim, E.A.B, King, G.F, Mobli, M.
登録日2015-08-27
公開日2016-09-07
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Structure of spider-venom peptide Hm1a
To be Published
6PZB
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BU of 6pzb by Molmil
Cryo-EM structure of the pancreatic beta-cell SUR1 Apo state
分子名称: ATP-binding cassette sub-family C member 8
著者Shyng, S.L, Yoshioka, C, Martin, G.M, Sung, M.W.
登録日2019-07-31
公開日2019-08-14
最終更新日2020-10-07
実験手法ELECTRON MICROSCOPY (4.55 Å)
主引用文献Mechanism of pharmacochaperoning in a mammalian K ATP channel revealed by cryo-EM.
Elife, 8, 2019
6PZI
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BU of 6pzi by Molmil
Cryo-EM structure of the pancreatic beta-cell SUR1 bound to ATP only
分子名称: ADENOSINE-5'-TRIPHOSPHATE, ATP-binding cassette sub-family C member 8
著者Shyng, S.L, Yoshioka, C, Martin, G.M, Sung, M.W.
登録日2019-07-31
公開日2019-08-14
最終更新日2020-10-07
実験手法ELECTRON MICROSCOPY (4.5 Å)
主引用文献Mechanism of pharmacochaperoning in a mammalian K ATP channel revealed by cryo-EM.
Elife, 8, 2019
6PZC
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BU of 6pzc by Molmil
Cryo-EM structure of the pancreatic beta-cell SUR1 bound to carbamazepine
分子名称: ATP-binding cassette sub-family C member 8
著者Shyng, S.L, Yoshioka, C, Martin, G.M, Sung, M.W.
登録日2019-07-31
公開日2019-08-14
最終更新日2024-03-20
実験手法ELECTRON MICROSCOPY (4.34 Å)
主引用文献Mechanism of pharmacochaperoning in a mammalian K ATP channel revealed by cryo-EM.
Elife, 8, 2019
5W3S
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BU of 5w3s by Molmil
Cryo-electron microscopy structure of a TRPML3 ion channel
分子名称: 1,2-Distearoyl-sn-glycerophosphoethanolamine, CHOLESTEROL HEMISUCCINATE, Mucolipin-3 isoform 1, ...
著者Hirschi, M, Herzik, M.A, Wie, J, Suo, Y, Borschel, W.F, Ren, D, Lander, G.C, Lee, S.Y.
登録日2017-06-08
公開日2017-10-11
最終更新日2024-03-13
実験手法ELECTRON MICROSCOPY (2.94 Å)
主引用文献Cryo-electron microscopy structure of the lysosomal calcium-permeable channel TRPML3.
Nature, 550, 2017
6AFZ
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BU of 6afz by Molmil
Proton pyrophosphatase-E225H mutant
分子名称: 2-(2-{2-[2-(2-METHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHANOL, MAGNESIUM ION, PHOSPHATE ION, ...
著者Tsai, J.-Y, Li, K.-M, Sun, Y.-J.
登録日2018-08-08
公開日2019-04-10
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.483 Å)
主引用文献Roles of the Hydrophobic Gate and Exit Channel in Vigna radiata Pyrophosphatase Ion Translocation.
J. Mol. Biol., 431, 2019
6AFW
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BU of 6afw by Molmil
Proton pyrophosphatase-T228D mutant
分子名称: 2-(2-{2-[2-(2-METHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHANOL, MAGNESIUM ION, PHOSPHATE ION, ...
著者Tsai, J.-Y, Li, K.-M, Sun, Y.-J.
登録日2018-08-08
公開日2019-04-10
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.185 Å)
主引用文献Roles of the Hydrophobic Gate and Exit Channel in Vigna radiata Pyrophosphatase Ion Translocation.
J. Mol. Biol., 431, 2019
6AFV
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BU of 6afv by Molmil
Proton pyrophosphatase-L555K mutant
分子名称: 2-(2-{2-[2-(2-METHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHANOL, MAGNESIUM ION, PHOSPHATE ION, ...
著者Tsai, J.-Y, Li, K.-M, Sun, Y.-J.
登録日2018-08-08
公開日2019-04-10
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.701 Å)
主引用文献Roles of the Hydrophobic Gate and Exit Channel in Vigna radiata Pyrophosphatase Ion Translocation.
J. Mol. Biol., 431, 2019
6AFT
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BU of 6aft by Molmil
Proton pyrophosphatase - E301Q
分子名称: 2-(2-{2-[2-(2-METHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHANOL, MAGNESIUM ION, PHOSPHATE ION, ...
著者Tsai, J.-Y, Tang, K.-Z, Sun, Y.-J.
登録日2018-08-08
公開日2019-04-10
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.492 Å)
主引用文献Roles of the Hydrophobic Gate and Exit Channel in Vigna radiata Pyrophosphatase Ion Translocation.
J. Mol. Biol., 431, 2019
6AFU
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BU of 6afu by Molmil
Proton pyrophosphatase-L555M mutant
分子名称: 2-(2-{2-[2-(2-METHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHANOL, MAGNESIUM ION, PHOSPHATE ION, ...
著者Tsai, J.-Y, Li, K.-M, Sun, Y.-J.
登録日2018-08-08
公開日2019-04-10
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.798 Å)
主引用文献Roles of the Hydrophobic Gate and Exit Channel in Vigna radiata Pyrophosphatase Ion Translocation.
J. Mol. Biol., 431, 2019
6AFY
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BU of 6afy by Molmil
Proton pyrophosphatase-E225S mutant
分子名称: 2-(2-{2-[2-(2-METHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHANOL, MAGNESIUM ION, PHOSPHATE ION, ...
著者Tsai, J.-Y, Li, K.-M, Sun, Y.-J.
登録日2018-08-08
公開日2019-04-10
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.401 Å)
主引用文献Roles of the Hydrophobic Gate and Exit Channel in Vigna radiata Pyrophosphatase Ion Translocation.
J. Mol. Biol., 431, 2019
6AFS
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BU of 6afs by Molmil
Proton pyrophosphatase - two phosphates-bound
分子名称: 2-(2-{2-[2-(2-METHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHANOL, MAGNESIUM ION, PHOSPHATE ION, ...
著者Tsai, J.-Y, Li, K.-M, Sun, Y.-J.
登録日2018-08-08
公開日2019-04-10
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.299 Å)
主引用文献Roles of the Hydrophobic Gate and Exit Channel in Vigna radiata Pyrophosphatase Ion Translocation.
J. Mol. Biol., 431, 2019
6AFX
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BU of 6afx by Molmil
Proton pyrophosphatase - E225A
分子名称: 2-(2-{2-[2-(2-METHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHANOL, MAGNESIUM ION, PHOSPHATE ION, ...
著者Tsai, J.-Y, Tang, K.-Z, Sun, Y.-J.
登録日2018-08-08
公開日2019-04-10
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.301 Å)
主引用文献Roles of the Hydrophobic Gate and Exit Channel in Vigna radiata Pyrophosphatase Ion Translocation.
J. Mol. Biol., 431, 2019
2K9E
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BU of 2k9e by Molmil
NMR Solution Structure for ShK-192: A Potent KV1.3-Specific Immunosuppressive Polypeptide
分子名称: Kappa-stichotoxin-She3a
著者Galea, C.A.
登録日2008-10-09
公開日2009-01-20
最終更新日2023-11-15
実験手法SOLUTION NMR
主引用文献Engineering a stable and selective peptide blocker of the Kv1.3 channel in T lymphocytes
Mol.Pharmacol., 75, 2009
4PDM
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BU of 4pdm by Molmil
Crystal Structure of K+ selective NaK mutant in rubidium
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, Potassium channel protein, RUBIDIUM ION
著者Lam, Y.
登録日2014-04-19
公開日2014-07-09
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.58 Å)
主引用文献High Resolution Structural Views of Rubidium, Cesium and Barium Binding within a Potassium Selective Channel Filter
To Be Published
4PDR
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BU of 4pdr by Molmil
Crystal Structure of a K+ selective NaK mutant in Barium and Sodium
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, BARIUM ION, Potassium channel protein, ...
著者Lam, Y, Zeng, W, Sauer, D.B, Jiang, Y.
登録日2014-04-21
公開日2014-07-09
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献High Resolution Structural Views of Rubidium, Cesium and Barium Binding within a Potassium Selective Channel Filter
To Be Published
4PDL
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BU of 4pdl by Molmil
Structure of K+ selective NaK mutant in caesium
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, CESIUM ION, HEXANE, ...
著者Lam, Y, Zeng, W, Sauer, D.B, Jiang, Y.
登録日2014-04-19
公開日2014-07-09
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献High Resolution Structural Views of Rubidium, Cesium and Barium Binding within a Potassium Selective Channel Filter
To Be Published
5WPT
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BU of 5wpt by Molmil
Cryo-EM structure of mammalian endolysosomal TRPML1 channel in nanodiscs in closed II conformation at 3.75 Angstrom resolution
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Mucolipin-1, SODIUM ION
著者Chen, Q, She, J, Guo, J, Bai, X, Jiang, Y.
登録日2017-08-07
公開日2017-10-18
最終更新日2023-04-05
実験手法ELECTRON MICROSCOPY (3.75 Å)
主引用文献Structure of mammalian endolysosomal TRPML1 channel in nanodiscs.
Nature, 550, 2017
5WPV
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BU of 5wpv by Molmil
Cryo-EM structure of mammalian endolysosomal TRPML1 channel in nanodiscs at 3.59 Angstrom resolution
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Mucolipin-1, SODIUM ION
著者Chen, Q, She, J, Guo, J, Bai, X, Jiang, Y.
登録日2017-08-07
公開日2017-10-18
最終更新日2023-04-05
実験手法ELECTRON MICROSCOPY (3.59 Å)
主引用文献Structure of mammalian endolysosomal TRPML1 channel in nanodiscs.
Nature, 550, 2017
2Q0A
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BU of 2q0a by Molmil
Structure and rearrangements in the carboxy-terminal region of SpIH channels
分子名称: CYCLIC GUANOSINE MONOPHOSPHATE, Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 2
著者Flynn, G.E, Black, K.D, Islas, L.D, Sankaran, B, Zagotta, W.N.
登録日2007-05-21
公開日2007-06-19
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Structure and rearrangements in the carboxy-terminal region of SpIH channels.
Structure, 15, 2007
5WPQ
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BU of 5wpq by Molmil
Cryo-EM structure of mammalian endolysosomal TRPML1 channel in nanodiscs in closed I conformation at 3.64 Angstrom resolution
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Mucolipin-1, SODIUM ION
著者Chen, Q, She, J, Guo, J, Bai, X, Jiang, Y.
登録日2017-08-07
公開日2017-10-18
最終更新日2023-04-05
実験手法ELECTRON MICROSCOPY (3.64 Å)
主引用文献Structure of mammalian endolysosomal TRPML1 channel in nanodiscs.
Nature, 550, 2017
4DEY
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BU of 4dey by Molmil
Crystal structure of the Voltage Dependent Calcium Channel beta-2 Subunit in Complex With The CaV1.2 I-II Linker.
分子名称: BROMIDE ION, Voltage-dependent L-type calcium channel subunit alpha-1C, Voltage-dependent L-type calcium channel subunit beta-2
著者Almagor, L, Hirsch, J.A.
登録日2012-01-22
公開日2012-06-13
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献The role of a voltage-dependent Ca2+ channel intracellular linker: a structure-function analysis.
J.Neurosci., 32, 2012

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