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8WTY
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BU of 8wty by Molmil
Cryo-EM structure of noradrenaline transporter in complex with ziprasidone
分子名称: 5-[2-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]ethyl]-6-chloranyl-1,3-dihydroindol-2-one, Sodium-dependent noradrenaline transporter
著者Zhao, Y, Hu, T, Yu, Z.
登録日2023-10-19
公開日2024-08-07
最終更新日2024-09-04
実験手法ELECTRON MICROSCOPY (3.2 Å)
主引用文献Transport and inhibition mechanisms of the human noradrenaline transporter.
Nature, 632, 2024
8WTX
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Cryo-EM structure of noradrenaline transporter in complex with bupropion
分子名称: (2~{R})-2-(~{tert}-butylamino)-1-(3-chlorophenyl)propan-1-one, Sodium-dependent noradrenaline transporter
著者Zhao, Y, Hu, T, Yu, Z.
登録日2023-10-19
公開日2024-08-07
最終更新日2024-09-04
実験手法ELECTRON MICROSCOPY (2.9 Å)
主引用文献Transport and inhibition mechanisms of the human noradrenaline transporter.
Nature, 632, 2024
2Q8U
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BU of 2q8u by Molmil
CRYSTAL STRUCTURE OF MRE11 FROM THERMOTOGA MARITIMA MSB8 (TM1635) AT 2.20 A RESOLUTION
分子名称: Exonuclease, putative
著者Joint Center for Structural Genomics (JCSG)
登録日2007-06-11
公開日2007-06-26
最終更新日2023-01-25
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Crystal structure of the first eubacterial Mre11 nuclease reveals novel features that may discriminate substrates during DNA repair.
J.Mol.Biol., 397, 2010
5TFV
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BU of 5tfv by Molmil
Crystal Structure of MT-I isolated from Bothrops asper venom.
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Basic phospholipase A2 myotoxin III
著者Salvador, G.H.M, dos Santos, J.I, Fontes, M.R.M.
登録日2016-09-26
公開日2017-10-04
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.54 Å)
主引用文献Crystal structure of a phospholipase A2 from Bothrops asper venom: Insights into a new putative "myotoxic cluster".
Biochimie, 133, 2017
4AP6
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BU of 4ap6 by Molmil
Crystal structure of human POFUT2 E54A mutant in complex with GDP- fucose
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, CHLORIDE ION, GDP-FUCOSE PROTEIN O-FUCOSYLTRANSFERASE 2, ...
著者Chen, C, Keusch, J.J, Klein, D, Hess, D, Hofsteenge, J, Gut, H.
登録日2012-03-30
公開日2012-08-08
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (3.401 Å)
主引用文献Structure of Human Pofut2: Insights Into Thrombospondin Type 1 Repeat Fold and O-Fucosylation.
Embo J., 31, 2012
7VSR
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BU of 7vsr by Molmil
Structure of McrBC (stalkless mutant)
分子名称: 5-methylcytosine-specific restriction enzyme B, MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-GUANYLATE ESTER, ...
著者Saikrishnan, K, Adhav, V.A, Bose, S, Kutti R, V.
登録日2021-10-27
公開日2023-02-15
最終更新日2024-06-26
実験手法ELECTRON MICROSCOPY (4.5 Å)
主引用文献Structure of McrBC (stalkless mutant)
To Be Published
8VUN
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BU of 8vun by Molmil
Human GluN1-2A With Fab 008-218
分子名称: 008-218 Heavy, 008-218 Light, Glutamate receptor ionotropic, ...
著者Michalski, K, Furukawa, H.
登録日2024-01-29
公開日2024-09-11
最終更新日2024-09-18
実験手法ELECTRON MICROSCOPY (4.01 Å)
主引用文献Structural and functional mechanisms of anti-NMDAR autoimmune encephalitis.
Nat.Struct.Mol.Biol., 2024
8VUQ
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BU of 8vuq by Molmil
Human GluN1-2A with Fab 008-218 Local refinement of ATD
分子名称: 008-218 Heavy, 008-218 Light, Glutamate receptor ionotropic, ...
著者Michalski, K, Furukawa, H.
登録日2024-01-29
公開日2024-09-11
最終更新日2024-09-18
実験手法ELECTRON MICROSCOPY (3.85 Å)
主引用文献Structural and functional mechanisms of anti-NMDAR autoimmune encephalitis.
Nat.Struct.Mol.Biol., 2024
8VVH
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BU of 8vvh by Molmil
rat GluN1a-2B Fab 003-102 local refinement
分子名称: 003-102 Heavy, 003-102 Light, Glutamate receptor ionotropic, ...
著者Michalski, K, Furukawa, H.
登録日2024-01-31
公開日2024-09-11
最終更新日2024-09-18
実験手法ELECTRON MICROSCOPY (3.95 Å)
主引用文献Structural and functional mechanisms of anti-NMDAR autoimmune encephalitis.
Nat.Struct.Mol.Biol., 2024
8VUL
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BU of 8vul by Molmil
Human GluN1-2A with Fab 003-102 Local refinement of ATD
分子名称: 003-102 Heavy, 003-102 Light, Glutamate receptor ionotropic, ...
著者Michalski, K, Furukawa, H.
登録日2024-01-29
公開日2024-09-11
最終更新日2024-09-18
実験手法ELECTRON MICROSCOPY (3.83 Å)
主引用文献Structural and functional mechanisms of anti-NMDAR autoimmune encephalitis.
Nat.Struct.Mol.Biol., 2024
8VUJ
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BU of 8vuj by Molmil
Human GluN1-2A with Fab 003-102
分子名称: 003-102 Heavy, 003-102 Light, Glutamate receptor ionotropic, ...
著者Michalski, K, Furukawa, H.
登録日2024-01-29
公開日2024-09-11
最終更新日2024-09-18
実験手法ELECTRON MICROSCOPY (3.92 Å)
主引用文献Structural and functional mechanisms of anti-NMDAR autoimmune encephalitis.
Nat.Struct.Mol.Biol., 2024
8VUT
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BU of 8vut by Molmil
Human GluN1-2A with IgG 008-218
分子名称: 008-218 Heavy, 008-218 Light, Glutamate receptor ionotropic, ...
著者Michalski, K, Furukawa, H.
登録日2024-01-29
公開日2024-09-11
最終更新日2024-09-18
実験手法ELECTRON MICROSCOPY (3.7 Å)
主引用文献Structural and functional mechanisms of anti-NMDAR autoimmune encephalitis.
Nat.Struct.Mol.Biol., 2024
8VUY
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BU of 8vuy by Molmil
Rat GluN1-2B with Fab 003-102
分子名称: 003-102 Heavy, 003-102 Light, Glutamate receptor ionotropic, ...
著者Michalski, K, Furukawa, H.
登録日2024-01-30
公開日2024-09-11
最終更新日2024-09-18
実験手法ELECTRON MICROSCOPY (3.81 Å)
主引用文献Structural and functional mechanisms of anti-NMDAR autoimmune encephalitis.
Nat.Struct.Mol.Biol., 2024
8VUS
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BU of 8vus by Molmil
Human GluN1-2A with IgG 007-168
分子名称: 007-168 Heavy, 007-168 Light, Glutamate receptor ionotropic, ...
著者Michalski, K, Furukawa, H.
登録日2024-01-29
公開日2024-09-11
最終更新日2024-09-18
実験手法ELECTRON MICROSCOPY (3.99 Å)
主引用文献Structural and functional mechanisms of anti-NMDAR autoimmune encephalitis.
Nat.Struct.Mol.Biol., 2024
3ZR8
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BU of 3zr8 by Molmil
Crystal structure of RxLR effector Avr3a11 from Phytophthora capsici
分子名称: AVR3A11, CHLORIDE ION, TRIETHYLENE GLYCOL
著者Boutemy, L.S, King, S.R.F, Win, J, Hughes, R.K, Clarke, T.A, Blumenschein, T.M.A, Kamoun, S, Banfield, M.J.
登録日2011-06-15
公開日2011-08-03
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (0.9 Å)
主引用文献Structures of Phytophthora Rxlr Effector Proteins: A Conserved But Adaptable Fold Underpins Functional Diversity.
J.Biol.Chem., 286, 2011
5WHR
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BU of 5whr by Molmil
Discovery of a novel and selective IDO-1 inhibitor PF-06840003 and its characterization as a potential clinical candidate.
分子名称: (3R)-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione, Indoleamine 2,3-dioxygenase 1, PROTOPORPHYRIN IX CONTAINING FE
著者Greasley, S.E, Kaiser, S.E, Feng, J.L, Stewart, A.
登録日2017-07-18
公開日2017-12-27
実験手法X-RAY DIFFRACTION (2.28 Å)
主引用文献Discovery of a Novel and Selective Indoleamine 2,3-Dioxygenase (IDO-1) Inhibitor 3-(5-Fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione (EOS200271/PF-06840003) and Its Characterization as a Potential Clinical Candidate.
J. Med. Chem., 60, 2017
4CEL
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BU of 4cel by Molmil
ACTIVE-SITE MUTANT D214N DETERMINED AT PH 6.0 WITH NO LIGAND BOUND IN THE ACTIVE SITE
分子名称: 1,4-BETA-D-GLUCAN CELLOBIOHYDROLASE I, 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION
著者Divne, C, Stahlberg, J, Jones, T.A.
登録日1996-08-24
公開日1997-03-12
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Activity studies and crystal structures of catalytically deficient mutants of cellobiohydrolase I from Trichoderma reesei.
J.Mol.Biol., 264, 1996
6MQF
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BU of 6mqf by Molmil
Myotoxin II from Bothrops moojeni complexed with Acetylsalicylic acid
分子名称: 2-(ACETYLOXY)BENZOIC ACID, Basic phospholipase A2 homolog 2, DIMETHYL SULFOXIDE
著者Salvador, G.H.M, Fontes, M.R.M.
登録日2018-10-09
公開日2019-03-20
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.693 Å)
主引用文献Search for efficient inhibitors of myotoxic activity induced by ophidian phospholipase A2-like proteins using functional, structural and bioinformatics approaches.
Sci Rep, 9, 2019
4LYO
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BU of 4lyo by Molmil
CROSS-LINKED CHICKEN LYSOZYME CRYSTAL IN NEAT ACETONITRILE, THEN BACK-SOAKED IN WATER
分子名称: LYSOZYME
著者Huang, Q, Wang, Z, Zhu, G, Qian, M, Shao, M, Jia, Y, Tang, Y.
登録日1998-03-11
公開日1998-05-27
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献X-ray studies on cross-linked lysozyme crystals in acetonitrile-water mixture.
Biochim.Biophys.Acta, 1384, 1998
4MHI
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BU of 4mhi by Molmil
Crystal structure of a H5N1 influenza virus hemagglutinin from A/goose/Guangdong/1/96
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Hemagglutinin HA1 chain, ...
著者Zhu, X, Wilson, I.A.
登録日2013-08-29
公開日2013-10-02
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.595 Å)
主引用文献A Unique and Conserved Neutralization Epitope in H5N1 Influenza Viruses Identified by an Antibody against the A/Goose/Guangdong/1/96 Hemagglutinin.
J.Virol., 87, 2013
2WB2
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BU of 2wb2 by Molmil
Drosophila Melanogaster (6-4) Photolyase Bound To double stranded Dna containing a T(6-4)C Photolesion
分子名称: 5'-D(*AP*CP*AP*GP*CP*GP*GP*64PP*ZP*GP*CP*AP *GP*GP*T)-3', 5'-D(*TP*AP*CP*CP*TP*GP*CP*GP*AP*CP*CP*GP*CP*TP*G)-3', FLAVIN-ADENINE DINUCLEOTIDE, ...
著者Glas, A.F, Schneider, S, Maul, M.J, Hennecke, U, Carell, T.
登録日2009-02-20
公開日2009-03-17
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.95 Å)
主引用文献Crystal Structure of the T(6-4)C Lesion in Complex with a (6-4) DNA Photolyase and Repair of Uv- Induced (6-4) and Dewar Photolesions.
Chemistry, 15, 2009
4HTQ
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BU of 4htq by Molmil
Mitigation of X-ray damage in macromolecular crystallography by submicrometer line focusing; total dose 6.70 x 10e+11 X-ray photons
分子名称: 1,2-ETHANEDIOL, CHLORIDE ION, Lysozyme C, ...
著者Duke, N.E.C, Finfrock, Y.Z, Stern, E.Z, Alkire, R.W, Lazarski, K, Joachimiak, A.
登録日2012-11-01
公開日2013-05-15
最終更新日2017-11-15
実験手法X-RAY DIFFRACTION (1.399 Å)
主引用文献Mitigation of X-ray damage in macromolecular crystallography by submicrometre line focusing.
Acta Crystallogr.,Sect.D, 69, 2013
3VX6
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BU of 3vx6 by Molmil
Crystal structure of Kluyveromyces marxianus Atg7NTD
分子名称: E1
著者Yamaguchi, M, Matoba, K, Sawada, R, Fujioka, Y, Nakatogawa, H, Yamamoto, H, Kobashigawa, Y, Hoshida, H, Akada, R, Ohsumi, Y, Noda, N.N, Inagaki, F.
登録日2012-09-11
公開日2012-11-14
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Noncanonical recognition and UBL loading of distinct E2s by autophagy-essential Atg7.
Nat.Struct.Mol.Biol., 19, 2012
3VX7
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Crystal structure of Kluyveromyces marxianus Atg7NTD-Atg10 complex
分子名称: E1, E2
著者Yamaguchi, M, Matoba, K, Sawada, R, Fujioka, Y, Nakatogawa, H, Yamamoto, H, Kobashigawa, Y, Hoshida, H, Akada, R, Ohsumi, Y, Noda, N.N, Inagaki, F.
登録日2012-09-11
公開日2012-11-14
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Noncanonical recognition and UBL loading of distinct E2s by autophagy-essential Atg7.
Nat.Struct.Mol.Biol., 19, 2012
2VNJ
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BU of 2vnj by Molmil
X-RAY STRUCTURE OF THE FERREDOXIN-NADP(H) REDUCTASE FROM RHODOBACTER CAPSULATUS IN COMPLEX WITH NADP. FORM I AT 2.13 ANGSTROMS RESOLUTION
分子名称: FLAVIN-ADENINE DINUCLEOTIDE, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, NADPH:FERREDOXIN REDUCTASE, ...
著者Perez-Dorado, I, Hermoso, J.A.
登録日2008-02-05
公開日2008-11-11
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.13 Å)
主引用文献Coenzyme Binding and Hydride Transfer in Rhodobacter Capsulatus Ferredoxin/Flavodoxin Nadp(H) Oxidoreductase.
Biochim.Biophys.Acta, 1794, 2009

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件を2024-09-25に公開中

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