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5ZQ5
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BU of 5zq5 by Molmil
SidE-Ubi
分子名称: SidE, Ubiquitin
著者Wang, Y, Gao, A, Gao, P.
登録日2018-04-17
公開日2018-05-23
最終更新日2018-05-30
実験手法X-RAY DIFFRACTION (2.487 Å)
主引用文献Structural Insights into Non-canonical Ubiquitination Catalyzed by SidE.
Cell, 173, 2018
5LLI
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BU of 5lli by Molmil
pVHL:EloB:EloC in complex with VH298
分子名称: (2~{S},4~{R})-1-[(2~{S})-2-[(1-cyanocyclopropyl)carbonylamino]-3,3-dimethyl-butanoyl]-~{N}-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-oxidanyl-pyrrolidine-2-carboxamide, Transcription elongation factor B polypeptide 1, Transcription elongation factor B polypeptide 2, ...
著者Gadd, M.S, Soares, P, Galdeano, C, Ciulli, A.
登録日2016-07-27
公開日2016-11-09
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Potent and selective chemical probe of hypoxic signalling downstream of HIF-alpha hydroxylation via VHL inhibition.
Nat Commun, 7, 2016
6NXK
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BU of 6nxk by Molmil
Ubiquitin binding variants
分子名称: Anaphase-promoting complex subunit 2, Polyubiquitin-C
著者Miller, D.J, Watson, E.R.
登録日2019-02-08
公開日2020-01-15
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Protein engineering of a ubiquitin-variant inhibitor of APC/C identifies a cryptic K48 ubiquitin chain binding site.
Proc.Natl.Acad.Sci.USA, 116, 2019
6GMX
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BU of 6gmx by Molmil
pVHL:EloB:EloC in complex with 6-chlorothiochroman-4-one
分子名称: 6-chloranyl-2,3-dihydrothiochromen-4-one, ACETATE ION, Elongin-B, ...
著者Van Molle, I, Lucas, X, Ciulli, A.
登録日2018-05-28
公開日2018-08-08
最終更新日2018-09-05
実験手法X-RAY DIFFRACTION (2.533 Å)
主引用文献Surface Probing by Fragment-Based Screening and Computational Methods Identifies Ligandable Pockets on the von Hippel-Lindau (VHL) E3 Ubiquitin Ligase.
J. Med. Chem., 61, 2018
5ZBI
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BU of 5zbi by Molmil
Crystal structure of asparaginyl endopeptidases from Viola Canadensis
分子名称: Peptide asparaginyl ligase, SODIUM ION
著者Wong, Y.H, Lescar, J.
登録日2018-02-12
公開日2018-05-09
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.09 Å)
主引用文献Crystal structure of Peptide asparaginyl ligase from Viola canadensis
To Be Published
6GMQ
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BU of 6gmq by Molmil
pVHL:EloB:EloC in complex with (4-(1H-pyrrol-1-yl)phenyl)methanol
分子名称: (4-pyrrol-1-ylphenyl)methanol, ACETATE ION, Elongin-B, ...
著者Van Molle, I, Lucas, X, Ciulli, A.
登録日2018-05-28
公開日2018-08-22
最終更新日2018-09-05
実験手法X-RAY DIFFRACTION (2.755 Å)
主引用文献Surface Probing by Fragment-Based Screening and Computational Methods Identifies Ligandable Pockets on the von Hippel-Lindau (VHL) E3 Ubiquitin Ligase.
J. Med. Chem., 61, 2018
6N5M
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BU of 6n5m by Molmil
Crystal structure of ABIN-1 UBAN in complex with one M1-linked di-ubiquitin
分子名称: Polyubiquitin-C, TNFAIP3-interacting protein 1
著者Rahighi, S, Dikic, I, Wakatsuki, S.
登録日2018-11-22
公開日2019-07-17
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (3.01 Å)
主引用文献Molecular Recognition of M1-Linked Ubiquitin Chains by Native and Phosphorylated UBAN Domains.
J.Mol.Biol., 431, 2019
6GFY
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BU of 6gfy by Molmil
pVHL:EloB:EloC in complex with modified VH032 containing (3R,4S)-3-fluoro-4-hydroxyproline (ligand 14a)
分子名称: (2~{R},3~{R},4~{S})-1-[(2~{S})-2-acetamido-3,3-dimethyl-butanoyl]-3-fluoranyl-~{N}-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-oxidanyl-pyrrolidine-2-carboxamide, Elongin-B, Elongin-C, ...
著者Gadd, M.S, Testa, A, Ciulli, A.
登録日2018-05-02
公開日2018-07-11
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献3-Fluoro-4-hydroxyprolines: Synthesis, Conformational Analysis, and Stereoselective Recognition by the VHL E3 Ubiquitin Ligase for Targeted Protein Degradation.
J. Am. Chem. Soc., 140, 2018
5LRV
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BU of 5lrv by Molmil
Structure of Cezanne/OTUD7B OTU domain bound to Lys11-linked diubiquitin
分子名称: GLYCEROL, OTU domain-containing protein 7B, PHOSPHATE ION, ...
著者Mevissen, T.E.T, Kulathu, Y, Mulder, M.P.C, Geurink, P.P, Maslen, S.L, Gersch, M, Elliott, P.R, Burke, J.E, van Tol, B.D.M, Akutsu, M, El Oualid, F, Kawasaki, M, Freund, S.M.V, Ovaa, H, Komander, D.
登録日2016-08-22
公開日2016-10-19
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Molecular basis of Lys11-polyubiquitin specificity in the deubiquitinase Cezanne.
Nature, 538, 2016
6GMN
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BU of 6gmn by Molmil
pVHL:EloB:EloC in complex with methyl 4H-furo[3,2-b]pyrrole-5-carboxylate
分子名称: ACETATE ION, Elongin-B, Elongin-C, ...
著者Van Molle, I, Lucas, X, Ciulli, A.
登録日2018-05-27
公開日2018-08-08
最終更新日2018-09-05
実験手法X-RAY DIFFRACTION (1.94 Å)
主引用文献Surface Probing by Fragment-Based Screening and Computational Methods Identifies Ligandable Pockets on the von Hippel-Lindau (VHL) E3 Ubiquitin Ligase.
J. Med. Chem., 61, 2018
5ZQ7
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BU of 5zq7 by Molmil
SidE-Ubi-NAD
分子名称: ADENOSINE MONOPHOSPHATE, NICOTINAMIDE-ADENINE-DINUCLEOTIDE, SidE, ...
著者Wang, Y, Gao, A, Gao, P.
登録日2018-04-17
公開日2018-05-23
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.847 Å)
主引用文献Structural Insights into Non-canonical Ubiquitination Catalyzed by SidE.
Cell, 173, 2018
6FMI
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BU of 6fmi by Molmil
pVHL:EloB:EloC in complex with N-((S)-1-((2S,4R)-4-Hydroxy-2-((4-(4-methylthiazol-5-yl)benzyl)carbamothioyl) pyrrolidin-1-yl)-1-oxopropan-2-yl)acetamide (ligand 2)
分子名称: Elongin-B, Elongin-C, von Hippel-Lindau disease tumor suppressor, ...
著者Soares, P, Lucas, X, Ciulli, A.
登録日2018-01-31
公開日2018-04-11
最終更新日2018-06-20
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Thioamide substitution to probe the hydroxyproline recognition of VHL ligands.
Bioorg. Med. Chem., 26, 2018
6O49
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BU of 6o49 by Molmil
CRYSTAL STRUCTURE OF SMT FUSION PEPTIDYL-PROLYL CIS-TRANS ISOMERASE FROM BURKHOLDERIA PSEUDOMALLEI COMPLEXED WITH SF339
分子名称: (2~{S})-~{N}-[3-oxidanylidene-3-[(3,4,5-trimethoxyphenyl)amino]propyl]-1-(phenylmethyl)sulfonyl-piperidine-2-carboxamide, 1,2-ETHANEDIOL, CALCIUM ION, ...
著者Seattle Structural Genomics Center for Infectious Disease (SSGCID)
登録日2019-02-28
公開日2020-02-12
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献CRYSTAL STRUCTURE OF SMT FUSION PEPTIDYL-PROLYL CIS-TRANS ISOMERASE FROM BURKHOLDERIA PSEUDOMALLEI COMPLEXED WITH SF339
to be published
5ZQ6
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BU of 5zq6 by Molmil
SidE-Ubi-ADPr
分子名称: ADENOSINE-5'-DIPHOSPHATE, SidE, Ubiquitin
著者Wang, Y, Gao, A, Gao, P.
登録日2018-04-17
公開日2018-05-23
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (3.009 Å)
主引用文献Structural Insights into Non-canonical Ubiquitination Catalyzed by SidE.
Cell, 173, 2018
6FNO
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BU of 6fno by Molmil
Caldiarchaeum Subterraneum Ubiquitin:Rpn11-homolog complex, zinc soak
分子名称: 26S proteasome regulatory subunit N11-like protein, SULFATE ION, Ubiquitin-like protein, ...
著者Fuchs, A.C.D, Albrecht, R, Martin, J, Hartmann, M.D.
登録日2018-02-04
公開日2018-07-25
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Rpn11-mediated ubiquitin processing in an ancestral archaeal ubiquitination system.
Nat Commun, 9, 2018
5LRW
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BU of 5lrw by Molmil
Structure of Cezanne/OTUD7B OTU domain bound to ubiquitin
分子名称: GLYCEROL, OTU domain-containing protein 7B, Polyubiquitin-B
著者Mevissen, T.E.T, Kulathu, Y, Mulder, M.P.C, Geurink, P.P, Maslen, S.L, Gersch, M, Elliott, P.R, Burke, J.E, van Tol, B.D.M, Akutsu, M, El Oualid, F, Kawasaki, M, Freund, S.M.V, Ovaa, H, Komander, D.
登録日2016-08-22
公開日2016-10-19
最終更新日2017-09-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Molecular basis of Lys11-polyubiquitin specificity in the deubiquitinase Cezanne.
Nature, 538, 2016
5WFI
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BU of 5wfi by Molmil
X-ray structure of MHV PLP2 (Cys1716Ser) catalytic mutant in complex with free ubiquitin
分子名称: FORMIC ACID, GLYCEROL, Ubiquitin, ...
著者Mesecar, A.D, Chen, Y.
登録日2017-07-12
公開日2018-08-01
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.851 Å)
主引用文献X-ray structure of MHV PLP2 (Cys1716Ser) catalytic mutant in complex with free ubiquitin
To Be Published
5V1Z
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BU of 5v1z by Molmil
Crystal structure of the RPN13 PRU-RPN2 (932-953)-ubiquitin complex
分子名称: 26S proteasome non-ATPase regulatory subunit 1, Proteasomal ubiquitin receptor ADRM1, Ubiquitin
著者Hemmis, C.W, VanderLinden, R.T, Yao, T, Robinson, H, Hill, C.P.
登録日2017-03-02
公開日2017-05-03
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structure and energetics of pairwise interactions between proteasome subunits RPN2, RPN13, and ubiquitin clarify a substrate recruitment mechanism.
J. Biol. Chem., 292, 2017
6GMR
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BU of 6gmr by Molmil
pVHL:EloB:EloC in complex with (4-(1H-pyrrol-1-yl)phenyl)methanol
分子名称: (4-pyrrol-1-ylphenyl)methanol, Elongin-B, Elongin-C, ...
著者Van Molle, I, Lucas, X, Ciulli, A.
登録日2018-05-28
公開日2018-08-08
最終更新日2018-09-05
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Surface Probing by Fragment-Based Screening and Computational Methods Identifies Ligandable Pockets on the von Hippel-Lindau (VHL) E3 Ubiquitin Ligase.
J. Med. Chem., 61, 2018
6A43
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BU of 6a43 by Molmil
R1EN(5-225)-ubiquitin fusion
分子名称: ACETIC ACID, RNA-directed DNA polymerase homolog (R1),Polyubiquitin-C
著者Maita, N.
登録日2018-06-19
公開日2018-10-24
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Crystal Structure Determination of Ubiquitin by Fusion to a Protein That Forms a Highly Porous Crystal Lattice
J. Am. Chem. Soc., 140, 2018
5W8T
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BU of 5w8t by Molmil
Crystal structure of MERS-CoV papain-like protease in complex with the C-terminal domain of human ISG15
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, ORF1ab, Ubiquitin-like protein ISG15, ...
著者Daczkowski, C.M, Goodwin, O.Y, Dzimianski, J.V, Farhat, J.J, Pegan, S.D.
登録日2017-06-22
公開日2017-09-27
最終更新日2024-04-24
実験手法X-RAY DIFFRACTION (2.758 Å)
主引用文献Structurally Guided Removal of DeISGylase Biochemical Activity from Papain-Like Protease Originating from Middle East Respiratory Syndrome Coronavirus.
J. Virol., 91, 2017
6A44
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BU of 6a44 by Molmil
R1EN(5-227)-ubiquitin fusion
分子名称: ACETIC ACID, RNA-directed DNA polymerase homolog (R1),Polyubiquitin-C
著者Maita, N.
登録日2018-06-19
公開日2018-10-24
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Crystal Structure Determination of Ubiquitin by Fusion to a Protein That Forms a Highly Porous Crystal Lattice
J. Am. Chem. Soc., 140, 2018
6OI4
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BU of 6oi4 by Molmil
RPN13 (19-132)-RPN2 (940-952) pY950-Ub complex
分子名称: 1,2-ETHANEDIOL, 26S proteasome non-ATPase regulatory subunit 1, Proteasomal ubiquitin receptor ADRM1, ...
著者Hemmis, C.W, Hill, C.P.
登録日2019-04-08
公開日2019-05-15
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.76 Å)
主引用文献Phosphorylation of Tyr-950 in the proteasome scaffolding protein RPN2 modulates its interaction with the ubiquitin receptor RPN13.
J.Biol.Chem., 294, 2019
5W8U
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BU of 5w8u by Molmil
Crystal structure of MERS-CoV papain-like protease in complex with the C-terminal domain of human ISG15
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, ORF1ab, Ubiquitin-like protein ISG15, ...
著者Daczkowski, C.M, Goodwin, O.Y, Dzimianski, J.D, Pegan, S.D.
登録日2017-06-22
公開日2017-09-27
最終更新日2024-04-24
実験手法X-RAY DIFFRACTION (2.411 Å)
主引用文献Structurally Guided Removal of DeISGylase Biochemical Activity from Papain-Like Protease Originating from Middle East Respiratory Syndrome Coronavirus.
J. Virol., 91, 2017
6GLC
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BU of 6glc by Molmil
Structure of phospho-Parkin bound to phospho-ubiquitin
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, E3 ubiquitin-protein ligase parkin, GLYCEROL, ...
著者Gladkova, C, Maslen, S.L, Skehel, J.M, Komander, D.
登録日2018-05-23
公開日2018-06-13
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Mechanism of parkin activation by PINK1.
Nature, 559, 2018

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件を2024-06-12に公開中

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