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8GZ1
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Cryo-EM structure of human NaV1.6/beta1/beta2,apo state
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, SODIUM ION, Sodium channel protein type 8 subunit alpha, ...
著者Li, Y, Jiang, D.
登録日2022-09-24
公開日2023-03-08
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Structure of human Na V 1.6 channel reveals Na + selectivity and pore blockade by 4,9-anhydro-tetrodotoxin.
Nat Commun, 14, 2023
7JPL
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BU of 7jpl by Molmil
Rabbit Cav1.1 in the presence of 10 micromolar (S)-(-)-Bay K8644 in nanodiscs at 3.4 Angstrom resolution
分子名称: 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOETHANOLAMINE, CALCIUM ION, ...
著者Yan, N, Gao, S.
登録日2020-08-09
公開日2020-11-18
最終更新日2021-03-10
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Structural Basis of the Modulation of the Voltage-Gated Calcium Ion Channel Ca v 1.1 by Dihydropyridine Compounds*.
Angew.Chem.Int.Ed.Engl., 60, 2021
8ED9
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BU of 8ed9 by Molmil
cryo-EM structure of TRPM3 ion channel in the presence with PIP2 and PregS, state 2
分子名称: (3beta,14beta,17beta,25R)-3-[4-methoxy-3-(methoxymethyl)butoxy]spirost-5-en, 1,2-DIACYL-GLYCEROL-3-SN-PHOSPHATE, SODIUM ION, ...
著者Zhao, C, MacKinnon, R.
登録日2022-09-03
公開日2022-11-09
最終更新日2023-01-18
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Structural and functional analyses of a GPCR-inhibited ion channel TRPM3.
Neuron, 111, 2023
6NT3
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BU of 6nt3 by Molmil
Cryo-EM structure of a human-cockroach hybrid Nav channel.
分子名称: (7E,21R,24S)-27-amino-24-hydroxy-18,24-dioxo-19,23,25-trioxa-24lambda~5~-phosphaheptacos-7-en-21-yl (9Z,12E)-octadeca-9,12-dienoate, 1,2-DIPALMITOYL-PHOSPHATIDYL-GLYCEROLE, 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Clairfeuille, T, Rohou, A, Payandeh, J.
登録日2019-01-28
公開日2019-02-20
最終更新日2021-08-25
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Cryo-EM structures of a human-cockroach hybrid Nav channel in the presence and absence of the alpha-scorpion toxin AaH2.
Science, 2019
8SEQ
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BU of 8seq by Molmil
Cryo-EM Structure of RyR1 + AMP
分子名称: ADENOSINE MONOPHOSPHATE, Glutathione S-transferase class-mu 26 kDa isozyme,Peptidyl-prolyl cis-trans isomerase FKBP1B, Ryanodine receptor 1, ...
著者Cholak, S, Saville, J.W, Zhu, X, Berezuk, A.M, Tuttle, K.S, Haji-Ghassemi, O, Van Petegem, F, Subramaniam, S.
登録日2023-04-10
公開日2023-05-24
最終更新日2023-07-19
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Allosteric modulation of ryanodine receptor RyR1 by nucleotide derivatives.
Structure, 31, 2023
6GYN
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BU of 6gyn by Molmil
Structure of human HCN4 hyperpolarization-activated cyclic nucleotide-gated ion channel
分子名称: 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1,2-Distearoyl-sn-glycerophosphoethanolamine, Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 4
著者Shintre, C.A, Pike, A.C.W, Tessitore, A, Young, M, Bushell, S.R, Strain-Damerell, C, Mukhopadhyay, S, Burgess-Brown, N.A, Huiskonen, J.T, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Carpenter, E.P, Structural Genomics Consortium (SGC)
登録日2018-06-30
公開日2019-05-08
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Structure of human HCN4 hyperpolarization-activated cyclic nucleotide-gated ion channel
To Be Published
6NQ2
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BU of 6nq2 by Molmil
Cryo-EM structure of human TPC2 channel in the ligand-bound closed state
分子名称: (2R)-3-{[(S)-hydroxy{[(1S,2R,3R,4S,5S,6R)-2,4,6-trihydroxy-3,5-bis(phosphonooxy)cyclohexyl]oxy}phosphoryl]oxy}propane-1,2-diyl dioctanoate, Two pore calcium channel protein 2
著者She, J, Zeng, W, Guo, J, Chen, Q, Bai, X, Jiang, Y.
登録日2019-01-18
公開日2019-03-27
最終更新日2019-11-20
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Structural mechanisms of phospholipid activation of the human TPC2 channel.
Elife, 8, 2019
8H9X
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BU of 8h9x by Molmil
Crystal structure of voltage-gated sodium channel NavAb N49K/L176Q mutant in sodium ion condition
分子名称: 1,2-DIMYRISTOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, CHAPSO, DODECYL-BETA-D-MALTOSIDE, ...
著者Irie, K, Oda, Y.
登録日2022-10-25
公開日2023-07-26
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (3.4 Å)
主引用文献The structural basis of divalent cation block in a tetrameric prokaryotic sodium channel.
Nat Commun, 14, 2023
8H9Y
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BU of 8h9y by Molmil
Crystal structure of voltage-gated sodium channel NavAb N49K/L176Q mutant in calcium ion condition
分子名称: 1,2-DIMYRISTOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, CALCIUM ION, CHAPSO, ...
著者Irie, K, Oda, Y.
登録日2022-10-25
公開日2023-07-26
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (3.4 Å)
主引用文献The structural basis of divalent cation block in a tetrameric prokaryotic sodium channel.
Nat Commun, 14, 2023
6GYO
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BU of 6gyo by Molmil
Structure of human HCN4 hyperpolarization-activated cyclic nucleotide-gated ion channel in complex with cAMP
分子名称: 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOINOSITOL, 1,2-Distearoyl-sn-glycerophosphoethanolamine, ...
著者Shintre, C.A, Pike, A.C.W, Tessitore, A, Young, M, Bushell, S.R, Strain-Damerell, C, Mukhopadhyay, S, Burgess-Brown, N.A, Huiskonen, J.T, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Carpenter, E.P, Structural Genomics Consortium (SGC)
登録日2018-06-30
公開日2019-05-01
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Structure of human HCN4 hyperpolarization-activated cyclic nucleotide-gated ion channel
To Be Published
8EOI
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BU of 8eoi by Molmil
Structure of a human EMC:human Cav1.2 channel complex in GDN detergent
分子名称: (3beta,14beta,17beta,25R)-3-[4-methoxy-3-(methoxymethyl)butoxy]spirost-5-en, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Chen, Z, Mondal, A, Abderemane-Ali, F, Minor, D.L.
登録日2022-10-03
公開日2023-05-24
最終更新日2023-07-26
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献EMC chaperone-Ca V structure reveals an ion channel assembly intermediate.
Nature, 619, 2023
7JPV
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BU of 7jpv by Molmil
Rabbit Cav1.1 in the presence of 1 micromolar (S)-(-)-Bay K8644 in nanodiscs at 3.4 Angstrom resolution
分子名称: 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOETHANOLAMINE, CALCIUM ION, ...
著者Yan, N, Gao, S.
登録日2020-08-10
公開日2020-11-18
最終更新日2021-03-10
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Structural Basis of the Modulation of the Voltage-Gated Calcium Ion Channel Ca v 1.1 by Dihydropyridine Compounds*.
Angew.Chem.Int.Ed.Engl., 60, 2021
7FBS
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BU of 7fbs by Molmil
structure of a channel
分子名称: (3beta,14beta,17beta,25R)-3-[4-methoxy-3-(methoxymethyl)butoxy]spirost-5-en, 1-[2-[(2R)-2-oxidanyl-3-(propylamino)propoxy]phenyl]-3-phenyl-propan-1-one, 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Jiang, D.J, Catterall, W.A.
登録日2021-07-12
公開日2021-09-22
最終更新日2022-02-16
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Open-state structure and pore gating mechanism of the cardiac sodium channel.
Cell, 184, 2021
5WO8
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BU of 5wo8 by Molmil
Crystal Structure of Transient Receptor Potential (TRP) channel TRPV6*-Del1
分子名称: 6-(5-METHYL-2-OXO-IMIDAZOLIDIN-4-YL)-HEXANOIC ACID, CALCIUM ION, Transient receptor potential cation channel subfamily V member 6
著者Singh, A.K, Saotome, K, Sobolevsky, A.I.
登録日2017-08-01
公開日2017-09-13
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (3.4 Å)
主引用文献Swapping of transmembrane domains in the epithelial calcium channel TRPV6.
Sci Rep, 7, 2017
6C96
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BU of 6c96 by Molmil
Cryo-EM structure of mouse TPC1 channel in the apo state
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, SODIUM ION, ...
著者She, J, Guo, J, Chen, Q, Bai, X, Jiang, Y.
登録日2018-01-25
公開日2018-04-04
最終更新日2020-07-29
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Structural insights into the voltage and phospholipid activation of the mammalian TPC1 channel.
Nature, 556, 2018
6U8A
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BU of 6u8a by Molmil
CBD-bound full-length rat TRPV2 in nanodiscs, state 1
分子名称: Transient receptor potential cation channel subfamily V member 2, cannabidiol
著者Pumroy, R.A, Moiseenkova-Bell, V.Y.
登録日2019-09-04
公開日2019-10-16
最終更新日2024-03-20
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Molecular mechanism of TRPV2 channel modulation by cannabidiol.
Elife, 8, 2019
7YIE
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BU of 7yie by Molmil
Human KCNH5-closed state 2
分子名称: POTASSIUM ION, Potassium voltage-gated channel subfamily H member 5
著者Zhang, M.F.
登録日2022-07-16
公開日2023-04-05
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Mechanism underlying delayed rectifying in human voltage-mediated activation Eag2 channel.
Nat Commun, 14, 2023
7YID
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BU of 7yid by Molmil
Human KCNH5 closed state 1
分子名称: POTASSIUM ION, Potassium voltage-gated channel subfamily H member 5
著者Zhang, M.F.
登録日2022-07-16
公開日2023-04-05
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Mechanism underlying delayed rectifying in human voltage-mediated activation Eag2 channel.
Nat Commun, 14, 2023
7WSW
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BU of 7wsw by Molmil
Cryo-EM structure of the Potassium channel AKT1 from Arabidopsis thaliana
分子名称: PHOSPHATIDYLETHANOLAMINE, POTASSIUM ION, Potassium channel AKT1
著者Yang, G.H, Lu, Y.M, Zhang, Y.M, Jia, Y.T, Li, X.M, Lei, J.L.
登録日2022-02-02
公開日2022-11-09
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Structural basis for the activity regulation of a potassium channel AKT1 from Arabidopsis.
Nat Commun, 13, 2022
7W6N
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BU of 7w6n by Molmil
CryoEM structure of human KChIP1-Kv4.3 complex
分子名称: Isoform 2 of Potassium voltage-gated channel subfamily D member 3, Kv channel-interacting protein 1
著者Ma, D.M, Guo, J.T.
登録日2021-12-02
公開日2022-11-02
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Structural basis for the gating modulation of Kv4.3 by auxiliary subunits.
Cell Res., 32, 2022
7XSU
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BU of 7xsu by Molmil
Cardiac sodium channel in complex with LqhIII
分子名称: (3beta,14beta,17beta,25R)-3-[4-methoxy-3-(methoxymethyl)butoxy]spirost-5-en, 2-acetamido-2-deoxy-beta-D-glucopyranose, Alpha-like toxin Lqh3, ...
著者Jiang, D, Catterall, W.A.
登録日2022-05-15
公開日2023-11-29
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Structural Basis for Nav1.5 Opening Modulated by a Gating Modifier Toxin
To Be Published
5YUB
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BU of 5yub by Molmil
Crystal structure of voltage-gated sodium channel NavAb E32Q mutant
分子名称: CALCIUM ION, CHAPSO, DODECYL-BETA-D-MALTOSIDE, ...
著者Irie, K, Shimomura, T, Fujiyoshi, Y.
登録日2017-11-21
公開日2017-12-27
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (3.40004 Å)
主引用文献Structural insight on the voltage dependence of prokaryotic voltage gated sodium channel NavAb.
FEBS Lett., 2017
5YUC
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BU of 5yuc by Molmil
Crystal structure of voltage-gated sodium channel NavAb N49K mutant
分子名称: CALCIUM ION, CHAPSO, DODECYL-BETA-D-MALTOSIDE, ...
著者Irie, K, Shimomura, T, Fujiyoshi, Y.
登録日2017-11-21
公開日2017-12-27
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (3.40099168 Å)
主引用文献Structural insight on the voltage dependence of prokaryotic voltage gated sodium channel NavAb.
FEBS Lett., 2017
4MTO
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BU of 4mto by Molmil
Structural Basis for Ca2+ Selectivity of a Voltage-gated Calcium Channel
分子名称: 1,2-DIMYRISTOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, CALCIUM ION, Ion transport protein
著者Tang, L, Gamal El-Din, T.M, Payandeh, J, Martinez, G.Q, Heard, T.M, Scheuer, T, Zheng, N, Catterall, W.A.
登録日2013-09-19
公開日2013-11-27
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (3.402 Å)
主引用文献Structural basis for Ca2+ selectivity of a voltage-gated calcium channel.
Nature, 505, 2014
7LQZ
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BU of 7lqz by Molmil
Structure of squirrel TRPV1 in complex with RTX
分子名称: (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, Osm-9-like TRP channel 1, SODIUM ION, ...
著者Neuberger, A, Nadezhdin, K.D, Sobolevsky, A.I.
登録日2021-02-15
公開日2021-04-21
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (3.41 Å)
主引用文献Extracellular cap domain is an essential component of the TRPV1 gating mechanism.
Nat Commun, 12, 2021

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