6T9Y
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6TNK
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1IY7
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![BU of 1iy7 by Molmil](/molmil-images/mine/1iy7) | Crystal Structure of CPA and sulfamide-based inhibitor complex | 分子名称: | Carboxypeptidase A, PHENYLALANINE-N-SULFONAMIDE, ZINC ION | 著者 | Kim, S.J, Woo, J.R, Park, J.D, Kim, D.H, Ryu, S.E. | 登録日 | 2002-07-24 | 公開日 | 2003-01-28 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Sulfamide-Based Inhibitors for Carboxypeptidase A. Novel Type Transition State Analogue Inhibitors for Zinc Proteases J.Med.Chem., 45, 2002
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4GM5
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![BU of 4gm5 by Molmil](/molmil-images/mine/4gm5) | Carboxypeptidase T with Sulphamoil Arginine | 分子名称: | CALCIUM ION, Carboxypeptidase T, GLYCEROL, ... | 著者 | Kuznetsov, S.A, Timofeev, V.I, Akparov, V.K, Kuranova, I.P. | 登録日 | 2012-08-15 | 公開日 | 2013-08-21 | 実験手法 | X-RAY DIFFRACTION (1.39 Å) | 主引用文献 | Carboxypeptidase T with Sulphamoil Arginine To be Published
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4UEE
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![BU of 4uee by Molmil](/molmil-images/mine/4uee) | Crystal structure of the human CARBOXYPEPTIDASE A1 in complex with the PHOSPHINIC INHIBITOR Acetyl-Leu-Ala-Y(PO2CH2)-homoPhe-OH | 分子名称: | (2S)-2-{[(R)-{(1R)-1-[(N-acetyl-L-leucyl)amino]ethyl}(hydroxy)phosphoryl]methyl}-4-phenylbutanoic acid, CARBOXYPEPTIDASE A1, ZINC ION | 著者 | Gallego, P, Covaleda, G, Costenaro, L, Devel, L, Dive, V, Aviles, F.X, Reverter, D. | 登録日 | 2014-12-17 | 公開日 | 2016-01-20 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.27 Å) | 主引用文献 | Crystal Structure of the Human Carboxypeptidase A1 in Complex with Phosphinic Inhibitors To be Published
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4UEZ
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![BU of 4uez by Molmil](/molmil-images/mine/4uez) | Crystal structure of the human CARBOXYPEPTIDASE A1 in complex with the PHOSPHINIC INHIBITOR Acetyl-Leu-Phe-Y(PO2CH2)-Phe-OH | 分子名称: | (2S)-3-[(R)-{(1R)-1-[(N-acetyl-L-leucyl)amino]-2-phenylethyl}(hydroxy)phosphoryl]-2-benzylpropanoic acid, HUMAN CARBOXYPEPTIDASE A1, ZINC ION | 著者 | Gallego, P, Covaleda, G, Costenaro, L, Devel, L, Dive, V, Aviles, F.X, Reverter, D. | 登録日 | 2014-12-22 | 公開日 | 2016-01-20 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.29 Å) | 主引用文献 | Crystal Structure of the Human Carboxypeptidase A1 in Complex with Phosphinic Inhibitors To be Published
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4UIB
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![BU of 4uib by Molmil](/molmil-images/mine/4uib) | Crystal structure of 3p in complex with tafCPB | 分子名称: | (2S)-6-AMINO-2-[[(1R)-1-(CYCLOHEXYLMETHYL)-2-OXO-2-[[(2S)-1,7,7-TRIMETHYLNORBORNAN-2-YL]AMINO]ETHYL]ARBAMOYLAMINO]HEXANOIC ACID, ACETATE ION, CARBOXYPEPTIDASE B, ... | 著者 | Halland, N, Broenstrup, M, Czech, J, Czechtizky, W, Evers, A, Follmann, M, Kohlmann, M, Schiell, M, Kurz, M, Schreuder, H.A, Kallus, C. | 登録日 | 2015-03-27 | 公開日 | 2015-06-03 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (1.94 Å) | 主引用文献 | Novel Small Molecule Inhibitors of Activated Thrombin Activatable Fibrinolysis Inhibitor (Tafia) from Natural Product Anabaenopeptin. J.Med.Chem., 58, 2015
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4UIA
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![BU of 4uia by Molmil](/molmil-images/mine/4uia) | Crystal structure of 3a in complex with tafCPB | 分子名称: | (2S)-6-azanyl-2-[[(2R)-3-cyclohexyl-1-(3-methylbutylamino)-1-oxidanylidene-propan-2-yl]carbamoylamino]hexanoic acid, CARBOXYPEPTIDASE B, ZINC ION | 著者 | Halland, N, Broenstrup, M, Czech, J, Czechtizky, W, Evers, A, Follmann, M, Kohlmann, M, Schiell, M, Kurz, M, Schreuder, H.A, Kallus, C. | 登録日 | 2015-03-27 | 公開日 | 2015-06-03 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (2.18 Å) | 主引用文献 | Novel Small Molecule Inhibitors of Activated Thrombin Activatable Fibrinolysis Inhibitor (Tafia) from Natural Product Anabaenopeptin. J.Med.Chem., 58, 2015
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4IAV
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![BU of 4iav by Molmil](/molmil-images/mine/4iav) | G215S, A251G, T257A, D260G, T262D mutant of carboxypeptidase T from Thermoactinomyces vulgaris with N-Sulfamoyl-L-phenylalanine | 分子名称: | CALCIUM ION, Carboxypeptidase T, GLYCEROL, ... | 著者 | Timofeev, V.I, Kuznetsov, S.A, Akparov, V.K, Kuranova, I.P. | 登録日 | 2012-12-07 | 公開日 | 2013-12-11 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.35 Å) | 主引用文献 | G215S, A251G, T257A, D260G, T262D mutant of carboxypeptidase T from Thermoactinomyces vulgaris with N-Sulfamoyl-L-phenylalanine TO BE PUBLISHED
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4IK2
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![BU of 4ik2 by Molmil](/molmil-images/mine/4ik2) | G215S, A251G, T257A, D260G, T262D mutant of carboxypeptidase T from Thermoactinomyces vulgaris with N-BOC-L-Leu | 分子名称: | CALCIUM ION, Carboxypeptidase T, N-(tert-butoxycarbonyl)-L-leucine, ... | 著者 | Timofeev, V.I, Kuznetsov, S.A, Akparov, V.K, Kuranova, I.P. | 登録日 | 2012-12-25 | 公開日 | 2013-12-25 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | G215S, A251G, T257A, D260G, T262D mutant of carboxypeptidase T from Thermoactinomyces vulgaris with N-BOC-L-Leu To be published
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4IHM
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![BU of 4ihm by Molmil](/molmil-images/mine/4ihm) | G215S, A251G, T257A, D260G, T262D mutant of carboxypeptidase T from Thermoactinomyces vulgaris | 分子名称: | CALCIUM ION, Carboxypeptidase T, GLYCEROL, ... | 著者 | Timofeev, V.I, Kuznetsov, S.A, Akparov, V.K, Kuranova, I.P. | 登録日 | 2012-12-19 | 公開日 | 2013-12-25 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.29 Å) | 主引用文献 | G215S, A251G, T257A, D260G, T262D mutant of carboxypeptidase T from Thermoactinomyces vulgaris To be published
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2CTB
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![BU of 2ctb by Molmil](/molmil-images/mine/2ctb) | THE HIGH RESOLUTION CRYSTAL STRUCTURE OF THE COMPLEX BETWEEN CARBOXYPEPTIDASE A AND L-PHENYL LACTATE | 分子名称: | CARBOXYPEPTIDASE A, ZINC ION | 著者 | Teplyakov, A, Wilson, K.S, Orioli, P, Mangani, S. | 登録日 | 1993-04-02 | 公開日 | 1994-01-31 | 最終更新日 | 2017-11-29 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | High-resolution structure of the complex between carboxypeptidase A and L-phenyl lactate. Acta Crystallogr.,Sect.D, 49, 1993
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4DUK
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![BU of 4duk by Molmil](/molmil-images/mine/4duk) | Carboxypeptidase T with L-BENZYLSUCCINIC ACID | 分子名称: | CALCIUM ION, Carboxypeptidase T, GLYCEROL, ... | 著者 | Kuznetsov, S.A, Timofeev, V.I, Akparov, V.K, Kuranova, I.P. | 登録日 | 2012-02-22 | 公開日 | 2013-02-27 | 最終更新日 | 2015-09-30 | 実験手法 | X-RAY DIFFRACTION (1.57 Å) | 主引用文献 | Structural insights into the broad substrate specificity of carboxypeptidase T from Thermoactinomyces vulgaris. Febs J., 282, 2015
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2C1C
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![BU of 2c1c by Molmil](/molmil-images/mine/2c1c) | Structural basis of the resistance of an insect carboxypeptidase to plant protease inhibitors | 分子名称: | CARBOXYPEPTIDASE B, YTTRIUM ION, ZINC ION | 著者 | Bayes, A, Comellas-Bigler, M, Rodriguez de la Vega, M, Maskos, K, Bode, W, Aviles, F.X, Jongsma, M.A, Beekwilder, J, Vendrell, J. | 登録日 | 2005-09-12 | 公開日 | 2005-10-19 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structural Basis of the Resistance of an Insect Carboxypeptidase to Plant Protease Inhibitors. Proc.Natl.Acad.Sci.USA, 102, 2005
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4DJL
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![BU of 4djl by Molmil](/molmil-images/mine/4djl) | Carboxypeptidase T with N-sulfamoyl-L-phenylalanine | 分子名称: | CALCIUM ION, Carboxypeptidase T, GLYCEROL, ... | 著者 | Kuznetsov, S.A, Timofeev, V.I, Akparov, V.K, Kuranova, I.P. | 登録日 | 2012-02-02 | 公開日 | 2013-02-06 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Carboxypeptidase T with N-sulfamoyl-L-phenylalanine TO BE PUBLISHED
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1OBR
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![BU of 1obr by Molmil](/molmil-images/mine/1obr) | CARBOXYPEPTIDASE T | 分子名称: | CALCIUM ION, CARBOXYPEPTIDASE T, SULFATE ION, ... | 著者 | Teplyakov, A, Polyakov, K, Obmolova, G, Osterman, A. | 登録日 | 1996-06-22 | 公開日 | 1997-01-11 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Crystal structure of carboxypeptidase T from Thermoactinomyces vulgaris. Eur.J.Biochem., 208, 1992
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2CTC
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![BU of 2ctc by Molmil](/molmil-images/mine/2ctc) | THE HIGH RESOLUTION CRYSTAL STRUCTURE OF THE COMPLEX BETWEEN CARBOXYPEPTIDASE A AND L-PHENYL LACTATE | 分子名称: | ALPHA-HYDROXY-BETA-PHENYL-PROPIONIC ACID, CARBOXYPEPTIDASE A, ZINC ION | 著者 | Teplyakov, A, Wilson, K.S, Orioli, P, Mangani, S. | 登録日 | 1993-04-02 | 公開日 | 1994-01-31 | 最終更新日 | 2017-11-29 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | High-resolution structure of the complex between carboxypeptidase A and L-phenyl lactate. Acta Crystallogr.,Sect.D, 49, 1993
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3HLP
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3HUV
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3I1U
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5HXD
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![BU of 5hxd by Molmil](/molmil-images/mine/5hxd) | Crystal structure of murein-tripeptide amidase MpaA from Escherichia coli O157 | 分子名称: | CACODYLATE ION, Protein MpaA, ZINC ION | 著者 | Ma, Y, Bai, G, Zhang, X, Zhao, J, Yuan, Z, Kang, X, Li, Z, Mu, S, Liu, X. | 登録日 | 2016-01-30 | 公開日 | 2017-02-08 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Crystal Structure of Murein-Tripeptide Amidase MpaA from Escherichia coli O157 at 2.6 angstrom Resolution Protein Pept.Lett., 24, 2017
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5J1Q
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3KGQ
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![BU of 3kgq by Molmil](/molmil-images/mine/3kgq) | Carboxypeptidase A liganded to an organic small-molecule: conformational changes | 分子名称: | ACETONE, CITRIC ACID, Carboxypeptidase A1, ... | 著者 | Fernandez, D, Boix, E, Pallares, I, Aviles, F.X, Vendrell, J. | 登録日 | 2009-10-29 | 公開日 | 2010-10-27 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Structural and Functional Analysis of the Complex between Citrate and the Zinc Peptidase Carboxypeptidase A Enzyme Res, 2011, 2011
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5JC6
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1BAV
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