5KO6
| Crystal Structure of Isoform 2 of Purine Nucleoside Phosphorylase from Schistosoma mansoni in complex with cytosine and ribose-1-phosphate | 分子名称: | 1-O-phosphono-alpha-D-ribofuranose, 6-AMINOPYRIMIDIN-2(1H)-ONE, Purine nucleoside phosphorylase | 著者 | Torini, J.R, Romanello, L, Bird, L, Owens, R, Brandao-Neto, J, Pereira, H.M. | 登録日 | 2016-06-29 | 公開日 | 2017-08-09 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.42 Å) | 主引用文献 | The molecular structure of Schistosoma mansoni PNP isoform 2 provides insights into the nucleoside selectivity of PNPs. PLoS ONE, 13, 2018
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6NZO
| Set2 bound to nucleosome | 分子名称: | DNA (149-MER), Histone H2B 1.1, Histone H3, ... | 著者 | Halic, M, Bilokapic, S. | 登録日 | 2019-02-14 | 公開日 | 2019-08-28 | 最終更新日 | 2019-09-04 | 実験手法 | ELECTRON MICROSCOPY (3.8 Å) | 主引用文献 | Nucleosome and ubiquitin position Set2 to methylate H3K36. Nat Commun, 10, 2019
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5NRL
| Structure of a pre-catalytic spliceosome. | 分子名称: | 13 kDa ribonucleoprotein-associated protein, 23 kDa U4/U6.U5 small nuclear ribonucleoprotein component, 66 kDa U4/U6.U5 small nuclear ribonucleoprotein component, ... | 著者 | Plaschka, C, Lin, P.-C, Nagai, K. | 登録日 | 2017-04-24 | 公開日 | 2017-05-31 | 最終更新日 | 2023-05-24 | 実験手法 | ELECTRON MICROSCOPY (7.2 Å) | 主引用文献 | Structure of a pre-catalytic spliceosome. Nature, 546, 2017
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5TUS
| Potent competitive inhibition of human ribonucleotide reductase by a novel non-nucleoside small molecule | 分子名称: | 2-hydroxy-N'-[(Z)-(2-hydroxynaphthalen-1-yl)methylidene]benzohydrazide, MAGNESIUM ION, Ribonucleoside-diphosphate reductase large subunit, ... | 著者 | Mohammed, F.A, Alam, I, Dealwis, C.G. | 登録日 | 2016-11-07 | 公開日 | 2017-08-02 | 最終更新日 | 2024-10-16 | 実験手法 | X-RAY DIFFRACTION (2.66 Å) | 主引用文献 | Potent competitive inhibition of human ribonucleotide reductase by a nonnucleoside small molecule. Proc. Natl. Acad. Sci. U.S.A., 114, 2017
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5IFK
| Purine nucleoside phosphorylase | 分子名称: | HYPOXANTHINE, Purine nucleoside phosphorylase | 著者 | Thakur, K.G, Priyanka, A. | 登録日 | 2016-02-26 | 公開日 | 2017-03-01 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.967 Å) | 主引用文献 | Functional and Structural Characterization of Purine Nucleoside Phosphorylase from Kluyveromyces lactis and Its Potential Applications in Reducing Purine Content in Food PLoS ONE, 11, 2016
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5O9G
| Structure of nucleosome-Chd1 complex | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, BERYLLIUM TRIFLUORIDE ION, Chromo domain-containing protein 1, ... | 著者 | Farnung, L, Vos, S.M, Wigge, C, Cramer, P. | 登録日 | 2017-06-19 | 公開日 | 2017-10-11 | 最終更新日 | 2024-05-15 | 実験手法 | ELECTRON MICROSCOPY (4.8 Å) | 主引用文献 | Nucleosome-Chd1 structure and implications for chromatin remodelling. Nature, 550, 2017
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6F52
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6F4W
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6F5I
| Crystal structure of H. pylori purine nucleoside phosphorylase | 分子名称: | METHANOL, Purine nucleoside phosphorylase DeoD-type | 著者 | Stefanic, Z. | 登録日 | 2017-12-01 | 公開日 | 2018-02-14 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2.298 Å) | 主引用文献 | Helicobacter pylori purine nucleoside phosphorylase shows new distribution patterns of open and closed active site conformations and unusual biochemical features. FEBS J., 285, 2018
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7OOY
| Purine nucleoside phosphorylase(DeoD-type) from H. pylori with 6-benzylthio-2-chloropurine | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 6-benzylthio-2-chloropurine, GLYCEROL, ... | 著者 | Narczyk, M, Stefanic, Z. | 登録日 | 2021-05-28 | 公開日 | 2022-05-04 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Interactions of 2,6-substituted purines with purine nucleoside phosphorylase from Helicobacter pylori in solution and in the crystal, and the effects of these compounds on cell cultures of this bacterium. J Enzyme Inhib Med Chem, 37, 2022
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7OOZ
| Purine nucleoside phosphorylase(DeoD-type) from H. pylori with 6-benzyloxo-2-chloropurine | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 6-benzyloxo-2-chloropurine, GLYCEROL, ... | 著者 | Narczyk, M, Stefanic, Z. | 登録日 | 2021-05-28 | 公開日 | 2022-05-04 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Interactions of 2,6-substituted purines with purine nucleoside phosphorylase from Helicobacter pylori in solution and in the crystal, and the effects of these compounds on cell cultures of this bacterium. J Enzyme Inhib Med Chem, 37, 2022
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7OP9
| Purine nucleoside phosphorylase(DeoD-type) from H. pylori with 2,6-dichloropurine | 分子名称: | 2,6-bis(chloranyl)-7H-purine, IMIDAZOLE, MAGNESIUM ION, ... | 著者 | Narczyk, M, Stefanic, Z. | 登録日 | 2021-05-31 | 公開日 | 2022-05-04 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Interactions of 2,6-substituted purines with purine nucleoside phosphorylase from Helicobacter pylori in solution and in the crystal, and the effects of these compounds on cell cultures of this bacterium. J Enzyme Inhib Med Chem, 37, 2022
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7OPA
| Purine nucleoside phosphorylase(DeoD-type) from H. pylori with 6-benzylthiopurine | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 6-benzylthio-2-chloropurine, GLYCEROL, ... | 著者 | Narczyk, M, Stefanic, Z. | 登録日 | 2021-05-31 | 公開日 | 2022-05-04 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Interactions of 2,6-substituted purines with purine nucleoside phosphorylase from Helicobacter pylori in solution and in the crystal, and the effects of these compounds on cell cultures of this bacterium. J Enzyme Inhib Med Chem, 37, 2022
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6F5A
| Crystal structure of H. pylori purine nucleoside phosphorylase | 分子名称: | Purine nucleoside phosphorylase DeoD-type | 著者 | Stefanic, Z. | 登録日 | 2017-12-01 | 公開日 | 2018-02-14 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2.201 Å) | 主引用文献 | Helicobacter pylori purine nucleoside phosphorylase shows new distribution patterns of open and closed active site conformations and unusual biochemical features. FEBS J., 285, 2018
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6F4X
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5UGF
| Crystal structure of human purine nucleoside phosphorylase (F159Y) mutant complexed with DADMe-ImmG and phosphate | 分子名称: | 2-amino-7-{[(3R,4R)-3-hydroxy-4-(hydroxymethyl)pyrrolidin-1-yl]methyl}-3,5-dihydro-4H-pyrrolo[3,2-d]pyrimidin-4-one, PHOSPHATE ION, Purine nucleoside phosphorylase | 著者 | Harijan, R.K, Cameron, S.A, Bonanno, J.B, Almo, S.C, Schramm, V.L. | 登録日 | 2017-01-08 | 公開日 | 2017-06-21 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Catalytic-site design for inverse heavy-enzyme isotope effects in human purine nucleoside phosphorylase. Proc. Natl. Acad. Sci. U.S.A., 114, 2017
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1K2A
| Modified Form of Eosinophil-derived Neurotoxin | 分子名称: | SULFATE ION, eosinophil-derived neurotoxin | 著者 | Chang, C, Newton, D.L, Rybak, S.M, Wlodawer, A. | 登録日 | 2001-09-26 | 公開日 | 2002-04-03 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1 Å) | 主引用文献 | Crystallographic and functional studies of a modified form of eosinophil-derived neurotoxin (EDN) with novel biological activities. J.Mol.Biol., 317, 2002
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5TBU
| Crystal Structure of Isoform 2 of Purine Nucleoside Phosphorylase complexed with Hypoxanthine | 分子名称: | DIMETHYL SULFOXIDE, HYPOXANTHINE, Purine nucleoside phosphorylase | 著者 | Faheem, M, Torini, J.R, Romanello, L, Brandao-Neto, J, Pereira, H.M. | 登録日 | 2016-09-13 | 公開日 | 2017-10-11 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | The molecular structure of Schistosoma mansoni PNP isoform 2 provides insights into the nucleoside selectivity of PNPs. PLoS ONE, 13, 2018
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5TBS
| Crystal Structure of Isoform 2 of Purine Nucleoside Phosphorylase complexed with adenine | 分子名称: | ADENINE, DIMETHYL SULFOXIDE, Purine nucleoside phosphorylase | 著者 | Faheem, M, Torini, J.R, Romanello, L, Brandao-Neto, J, Pereira, H.M. | 登録日 | 2016-09-13 | 公開日 | 2017-10-11 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | The molecular structure of Schistosoma mansoni PNP isoform 2 provides insights into the nucleoside selectivity of PNPs. PLoS ONE, 13, 2018
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5TBT
| Crystal Structure of Isoform 2 of Purine Nucleoside Phosphorylase complexed with Cytidine | 分子名称: | 4-AMINO-1-BETA-D-RIBOFURANOSYL-2(1H)-PYRIMIDINONE, Purine nucleoside phosphorylase, SULFATE ION | 著者 | Faheem, M, Torini, J.R, Romanello, L, Brandao-Neto, J, Pereira, H.M. | 登録日 | 2016-09-13 | 公開日 | 2017-10-11 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.101 Å) | 主引用文献 | The molecular structure of Schistosoma mansoni PNP isoform 2 provides insights into the nucleoside selectivity of PNPs. PLoS ONE, 13, 2018
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7ZSO
| human purine nucleoside phosphorylase in complex with JS-554 | 分子名称: | GLYCEROL, Purine nucleoside phosphorylase, SODIUM ION, ... | 著者 | Djukic, S, Pachl, P, Rezacova, P. | 登録日 | 2022-05-07 | 公開日 | 2023-05-17 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Design, Synthesis, Biological Evaluation, and Crystallographic Study of Novel Purine Nucleoside Phosphorylase Inhibitors. J.Med.Chem., 66, 2023
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7ZSL
| human purine nucleoside phosphorylase in complex with JS-196 | 分子名称: | 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, Purine nucleoside phosphorylase, ... | 著者 | Djukic, S, Pachl, P, Rezacova, P. | 登録日 | 2022-05-07 | 公開日 | 2023-05-17 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Design, Synthesis, Biological Evaluation, and Crystallographic Study of Novel Purine Nucleoside Phosphorylase Inhibitors. J.Med.Chem., 66, 2023
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7ZSM
| human purine nucleoside phosphorylase in complex with JS-375 | 分子名称: | CHLORIDE ION, Purine nucleoside phosphorylase, SULFATE ION, ... | 著者 | Djukic, S, Pachl, P, Rezacova, P. | 登録日 | 2022-05-07 | 公開日 | 2023-05-17 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.65 Å) | 主引用文献 | Design, Synthesis, Biological Evaluation, and Crystallographic Study of Novel Purine Nucleoside Phosphorylase Inhibitors. J.Med.Chem., 66, 2023
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7ZSQ
| human purine nucleoside phosphorylase in complex with JS-555 | 分子名称: | 1,2-ETHANEDIOL, 6-tungstotellurate(VI), DI(HYDROXYETHYL)ETHER, ... | 著者 | Djukic, S, Pachl, P, Rezacova, P. | 登録日 | 2022-05-08 | 公開日 | 2023-05-17 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.77 Å) | 主引用文献 | Design, Synthesis, Biological Evaluation, and Crystallographic Study of Novel Purine Nucleoside Phosphorylase Inhibitors. J.Med.Chem., 66, 2023
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7ZSR
| purine nucleoside phosphorylase in complex with JS-379 | 分子名称: | ACETATE ION, Purine nucleoside phosphorylase, [(~{E})-2-[5-bromanyl-2-[(4-oxidanylidene-3,5-dihydropyrrolo[3,2-d]pyrimidin-7-yl)sulfanyl]phenyl]ethenyl]phosphonic acid | 著者 | Djukic, S, Pachl, P, Rezacova, P. | 登録日 | 2022-05-08 | 公開日 | 2023-05-17 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.97 Å) | 主引用文献 | Design, Synthesis, Biological Evaluation, and Crystallographic Study of Novel Purine Nucleoside Phosphorylase Inhibitors. J.Med.Chem., 66, 2023
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