7BHD
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![BU of 7bhd by Molmil](/molmil-images/mine/7bhd) | FimH in complex with alpha1,6 core-fucosylated oligomannose-3, crystallized in the trigonal space group | 分子名称: | NICKEL (II) ION, SULFATE ION, Type 1 fimbrin D-mannose specific adhesin, ... | 著者 | Bridot, C, Bouckaert, J, Krammer, E.-M. | 登録日 | 2021-01-11 | 公開日 | 2022-07-20 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | Structural insights into a cooperative switch between one and two FimH bacterial adhesins binding pauci- and high-mannose type N-glycan receptors. J.Biol.Chem., 299, 2023
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6P6D
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![BU of 6p6d by Molmil](/molmil-images/mine/6p6d) | HUMAN IGG1 FC FRAGMENT, C239 INSERTION MUTANT | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-3)-[2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, CYSTEINE, IgG1 Fc fragment | 著者 | Gallagher, D.T, Dimasi, N, McCullough, C. | 登録日 | 2019-06-03 | 公開日 | 2020-04-15 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.31 Å) | 主引用文献 | Structure and Dynamics of a Site-Specific Labeled Fc Fragment with Altered Effector Functions. Pharmaceutics, 11, 2019
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4Y76
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![BU of 4y76 by Molmil](/molmil-images/mine/4y76) | Factor Xa complex with GTC000401 | 分子名称: | CALCIUM ION, Coagulation factor X, N~2~-[(6-chloronaphthalen-2-yl)sulfonyl]-N~2~-{(3S)-1-[(2S)-1-(4-methyl-1,4-diazepan-1-yl)-1-oxopropan-2-yl]-2-oxopyrrolidin-3-yl}glycinamide | 著者 | Convery, M.A, Young, R.J, Senger, S, Hamblin, J.N, Chan, C, Toomey, J.R, Watson, N.S. | 登録日 | 2015-02-13 | 公開日 | 2015-09-30 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Factor Xa inhibitors: S1 binding interactions of a series of N-{(3S)-1-[(1S)-1-methyl-2-morpholin-4-yl-2-oxoethyl]-2-oxopyrrolidin-3-yl}sulfonamides. J. Med. Chem., 50, 2007
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4Y79
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![BU of 4y79 by Molmil](/molmil-images/mine/4y79) | Factor Xa complex with GTC000406 | 分子名称: | (E)-2-(4-chlorophenyl)-N-{(3S)-1-[(2S)-1-(morpholin-4-yl)-1-oxopropan-2-yl]-2-oxopyrrolidin-3-yl}ethenesulfonamide, CALCIUM ION, Coagulation factor X, ... | 著者 | Convery, M.A, Young, R.J, Senger, S, Hamblin, J.N, Chan, C, Toomey, J.R, Watson, N.S. | 登録日 | 2015-02-13 | 公開日 | 2015-09-30 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Factor Xa inhibitors: S1 binding interactions of a series of N-{(3S)-1-[(1S)-1-methyl-2-morpholin-4-yl-2-oxoethyl]-2-oxopyrrolidin-3-yl}sulfonamides. J. Med. Chem., 50, 2007
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4Y7B
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![BU of 4y7b by Molmil](/molmil-images/mine/4y7b) | Factor Xa complex with GTC000441 | 分子名称: | 6-chloro-N-{(3S)-1-[(2S)-1-{(1R,5S)-7-[2-(methylamino)ethyl]-3,7-diazabicyclo[3.3.1]non-3-yl}-1-oxopropan-2-yl]-2-oxopy rrolidin-3-yl}naphthalene-2-sulfonamide, CALCIUM ION, Coagulation factor X | 著者 | Convery, M.A, Young, R.J, Senger, S, Hamblin, J.N, Chan, C, Toomey, J.R, Watson, N.S. | 登録日 | 2015-02-13 | 公開日 | 2015-09-30 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.79 Å) | 主引用文献 | Factor Xa complex with GTC000441 to be published
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4Y71
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![BU of 4y71 by Molmil](/molmil-images/mine/4y71) | Factor Xa complex with GTC000398 | 分子名称: | 6-chloro-N-{(3S)-1-[(2S)-1-(4-methyl-5-oxo-1,4-diazepan-1-yl)-1-oxopropan-2-yl]-2-oxopyrrolidin-3-yl}naphthalene-2-sulf onamide, CALCIUM ION, Coagulation factor X | 著者 | Convery, M.A, Young, R.J, Senger, S, Hamblin, J.N, Chan, C, Toomey, J.R, Watson, N.S. | 登録日 | 2015-02-13 | 公開日 | 2015-09-30 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Factor Xa complex with GTC000398 To be Published
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4Y7A
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![BU of 4y7a by Molmil](/molmil-images/mine/4y7a) | Factor Xa complex with GTC000422 | 分子名称: | CALCIUM ION, Coagulation factor X, MAGNESIUM ION, ... | 著者 | Convery, M.A, Young, R.J, Senger, S, Hamblin, J.N, Chan, C, Toomey, J.R, Watson, N.S. | 登録日 | 2015-02-13 | 公開日 | 2015-09-30 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.99 Å) | 主引用文献 | Factor Xa complex with GTC000422 to be published
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7PNI
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![BU of 7pni by Molmil](/molmil-images/mine/7pni) | |
7PNH
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![BU of 7pnh by Molmil](/molmil-images/mine/7pnh) | |
1C1V
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![BU of 1c1v by Molmil](/molmil-images/mine/1c1v) | |
1C1W
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![BU of 1c1w by Molmil](/molmil-images/mine/1c1w) | |
1C1U
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![BU of 1c1u by Molmil](/molmil-images/mine/1c1u) | |
6TEA
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![BU of 6tea by Molmil](/molmil-images/mine/6tea) | Tail of native GTA particle computed with helical refinement, C6 symmetry | 分子名称: | Phage major tail protein, TP901-1 family | 著者 | Bardy, P, Fuzik, T, Hrebik, D, Pantucek, R, Beatty, J.T, Plevka, P. | 登録日 | 2019-11-11 | 公開日 | 2020-07-22 | 最終更新日 | 2024-05-22 | 実験手法 | ELECTRON MICROSCOPY (3.89 Å) | 主引用文献 | Structure and mechanism of DNA delivery of a gene transfer agent. Nat Commun, 11, 2020
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6TO8
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![BU of 6to8 by Molmil](/molmil-images/mine/6to8) | Neck of empty GTA particle computed with C12 symmetry | 分子名称: | Adaptor protein Rcc01688, Portal protein Rcc01684 | 著者 | Bardy, P, Fuzik, T, Hrebik, D, Pantucek, R, Beatty, J.T, Plevka, P. | 登録日 | 2019-12-11 | 公開日 | 2020-07-22 | 最終更新日 | 2024-05-22 | 実験手法 | ELECTRON MICROSCOPY (3.36 Å) | 主引用文献 | Structure and mechanism of DNA delivery of a gene transfer agent. Nat Commun, 11, 2020
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1C5L
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![BU of 1c5l by Molmil](/molmil-images/mine/1c5l) | STRUCTURAL BASIS FOR SELECTIVITY OF A SMALL MOLECULE, S1-BINDING, SUB-MICROMOLAR INHIBITOR OF UROKINASE TYPE PLASMINOGEN ACTIVATOR | 分子名称: | CALCIUM ION, Hirudin, SODIUM ION, ... | 著者 | Katz, B.A, Mackman, R, Luong, C, Radika, K, Martelli, A, Sprengeler, P.A, Wang, J, Chan, H, Wong, L. | 登録日 | 1999-12-22 | 公開日 | 2000-12-22 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.47 Å) | 主引用文献 | Structural basis for selectivity of a small molecule, S1-binding, submicromolar inhibitor of urokinase-type plasminogen activator. Chem.Biol., 7, 2000
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1C5N
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![BU of 1c5n by Molmil](/molmil-images/mine/1c5n) | STRUCTURAL BASIS FOR SELECTIVITY OF A SMALL MOLECULE, S1-BINDING, SUB-MICROMOLAR INHIBITOR OF UROKINASE TYPE PLASMINOGEN ACTIVATOR | 分子名称: | 4-IODOBENZO[B]THIOPHENE-2-CARBOXAMIDINE, CALCIUM ION, Hirudin, ... | 著者 | Katz, B.A, Mackman, R, Luong, C, Radika, K, Martelli, A, Sprengeler, P.A, Wang, J, Chan, H, Wong, L. | 登録日 | 1999-12-22 | 公開日 | 2000-12-22 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Structural basis for selectivity of a small molecule, S1-binding, submicromolar inhibitor of urokinase-type plasminogen activator. Chem.Biol., 7, 2000
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6TB9
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![BU of 6tb9 by Molmil](/molmil-images/mine/6tb9) | Capsid of native GTA particle computed with C5 symmetry | 分子名称: | Head spike base Rcc01079, Head spike fiber Rcc01080, Major capsid protein Rcc01687 | 著者 | Bardy, P, Fuzik, T, Hrebik, D, Pantucek, R, Beatty, J.T, Plevka, P. | 登録日 | 2019-11-01 | 公開日 | 2020-07-22 | 最終更新日 | 2024-07-10 | 実験手法 | ELECTRON MICROSCOPY (3.56 Å) | 主引用文献 | Structure and mechanism of DNA delivery of a gene transfer agent. Nat Commun, 11, 2020
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1C5O
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![BU of 1c5o by Molmil](/molmil-images/mine/1c5o) | STRUCTURAL BASIS FOR SELECTIVITY OF A SMALL MOLECULE, S1-BINDING, SUB-MICROMOLAR INHIBITOR OF UROKINASE TYPE PLASMINOGEN ACTIVATOR | 分子名称: | BENZAMIDINE, Hirudin, SODIUM ION, ... | 著者 | Katz, B.A, Mackman, R, Luong, C, Radika, K, Martelli, A, Sprengeler, P.A, Wang, J, Chan, H, Wong, L. | 登録日 | 1999-12-22 | 公開日 | 2000-12-22 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structural basis for selectivity of a small molecule, S1-binding, submicromolar inhibitor of urokinase-type plasminogen activator. Chem.Biol., 7, 2000
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6TSU
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![BU of 6tsu by Molmil](/molmil-images/mine/6tsu) | Capsid of empty GTA particle computed with C5 symmetry | 分子名称: | Major capsid protein Rcc01687, Uncharacterized protein | 著者 | Bardy, P, Fuzik, T, Hrebik, D, Pantucek, R, Beatty, J.T, Plevka, P. | 登録日 | 2019-12-21 | 公開日 | 2020-07-22 | 最終更新日 | 2024-07-10 | 実験手法 | ELECTRON MICROSCOPY (3.42 Å) | 主引用文献 | Structure and mechanism of DNA delivery of a gene transfer agent. Nat Commun, 11, 2020
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6TEH
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![BU of 6teh by Molmil](/molmil-images/mine/6teh) | Baseplate of native GTA particle computed with C3 symmetry | 分子名称: | IRON/SULFUR CLUSTER, Putative gene transfer agent protein | 著者 | Bardy, P, Fuzik, T, Hrebik, D, Pantucek, R, Beatty, J.T, Plevka, P. | 登録日 | 2019-11-12 | 公開日 | 2020-07-22 | 最終更新日 | 2024-05-22 | 実験手法 | ELECTRON MICROSCOPY (3.99 Å) | 主引用文献 | Structure and mechanism of DNA delivery of a gene transfer agent. Nat Commun, 11, 2020
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6TUI
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![BU of 6tui by Molmil](/molmil-images/mine/6tui) | Virion of empty GTA particle | 分子名称: | Adaptor protein Rcc01688, Phage major capsid protein, HK97 family, ... | 著者 | Bardy, P, Fuzik, T, Hrebik, D, Pantucek, R, Beatty, J.T, Plevka, P. | 登録日 | 2020-01-07 | 公開日 | 2020-10-14 | 最終更新日 | 2024-05-22 | 実験手法 | ELECTRON MICROSCOPY (10.47 Å) | 主引用文献 | Virion of empty GTA particle Nat Commun, 11, 2020
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6TSV
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![BU of 6tsv by Molmil](/molmil-images/mine/6tsv) | Tail of empty GTA particle computed with helical refinement, C6 symmetry | 分子名称: | Tail tube protein Rcc01691 | 著者 | Bardy, P, Fuzik, T, Hrebik, D, Pantucek, R, Beatty, J.T, Plevka, P. | 登録日 | 2019-12-21 | 公開日 | 2020-07-22 | 最終更新日 | 2024-05-22 | 実験手法 | ELECTRON MICROSCOPY (3.78 Å) | 主引用文献 | Structure and mechanism of DNA delivery of a gene transfer agent. Nat Commun, 11, 2020
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6E2B
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![BU of 6e2b by Molmil](/molmil-images/mine/6e2b) | Ubiquitin in complex with Pt(2-phenilpyridine)(PPh3) | 分子名称: | GLYCEROL, SULFATE ION, Ubiquitin, ... | 著者 | Zhemkov, V.A, Kim, M. | 登録日 | 2018-07-11 | 公開日 | 2018-11-14 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | Reactions of Cyclometalated Platinum(II) [Pt(N∧C)(PR3)Cl] Complexes with Imidazole and Imidazole-Containing Biomolecules: Fine-Tuning of Reactivity and Photophysical Properties via Ligand Design. Inorg Chem, 58, 2019
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6TSW
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![BU of 6tsw by Molmil](/molmil-images/mine/6tsw) | Isometric capsid of empty GTA particle computed with I4(I,n25r) symmetry | 分子名称: | Major capsid protein Rcc01687 | 著者 | Bardy, P, Fuzik, T, Hrebik, D, Pantucek, R, Beatty, J.T, Plevka, P. | 登録日 | 2019-12-21 | 公開日 | 2020-07-22 | 最終更新日 | 2024-05-22 | 実験手法 | ELECTRON MICROSCOPY (4.03 Å) | 主引用文献 | Structure and mechanism of DNA delivery of a gene transfer agent. Nat Commun, 11, 2020
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6TBA
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![BU of 6tba by Molmil](/molmil-images/mine/6tba) | Virion of native gene transfer agent (GTA) particle | 分子名称: | IRON/SULFUR CLUSTER, Phage major capsid protein, HK97 family, ... | 著者 | Bardy, P, Fuzik, T, Hrebik, D, Pantucek, R, Beatty, J.T, Plevka, P. | 登録日 | 2019-11-01 | 公開日 | 2020-07-22 | 最終更新日 | 2024-05-22 | 実験手法 | ELECTRON MICROSCOPY (4.54 Å) | 主引用文献 | Structure and mechanism of DNA delivery of a gene transfer agent. Nat Commun, 11, 2020
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