Loading
PDBj
メニューPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

1BWQ
DownloadVisualize
BU of 1bwq by Molmil
PROBING THE SUBSTRATE SPECIFICITY OF THE INTRACELLULAR BRAIN PLATELET-ACTIVATING FACTOR ACETYLHYDROLASE
分子名称: PLATELET-ACTIVATING FACTOR ACETYLHYDROLASE
著者Ho, Y.S, Sheffield, P.J, Masuyama, J, Arai, H, Li, J, Aoki, J, Inoue, K, Derewenda, U, Derewenda, Z.
登録日1998-09-27
公開日1999-05-18
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Probing the Substrate Specificity of the Intracellular Brain Platelet-Activating Factor Acetylhydrolase
Protein Eng., 12, 1999
1BX0
DownloadVisualize
BU of 1bx0 by Molmil
Ferredoxin:nadp+ oxidoreductase (ferredoxin reductase) mutant e312l
分子名称: FLAVIN-ADENINE DINUCLEOTIDE, PHOSPHATE ION, PROTEIN (FERREDOXIN:NADP+ OXIDOREDUCTASE), ...
著者Aliverti, A, Deng, Z, Ravasi, D, Piubelli, L, Karplus, P.A, Zanetti, G.
登録日1998-10-10
公開日1998-10-14
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Probing the function of the invariant glutamyl residue 312 in spinach ferredoxin-NADP+ reductase.
J.Biol.Chem., 273, 1998
7T0L
DownloadVisualize
BU of 7t0l by Molmil
HLA-B*27:05 in complex with the pan-HLA-Ia monoclonal antibody W6/32
分子名称: Beta-2-microglobulin, IgG2a heavy chain, Light chain kappa, ...
著者Vivian, J.P, Rossjohn, J.
登録日2021-11-29
公開日2022-12-07
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献HLA-B*27:05 in complex with the pan-HLA-Ia monoclonal antibody W6/32
To Be Published
6YF1
DownloadVisualize
BU of 6yf1 by Molmil
FKBP12 in complex with the BMP potentiator compound 8 at 1.12A resolution
分子名称: (1aR,3R,5S,6R,7S,9R,10R,17aS,20S,21R,22S,25R,25aR)-25-Ethyl-10,22-dihydroxy-20-{(1E)-1-[(1R,3R,4R)-4-hydroxy-3-methoxycyclohexyl]prop-1-en-2-yl}-5,7-dimethoxy-1a,3,9,21-tetramethyloctadecahydro-2H-6,10-epoxyoxireno[p]pyrido[2,1-c][1,4]oxazacyclotricosine-11,12,18,24(1aH,14H)-tetrone, Peptidyl-prolyl cis-trans isomerase FKBP1A
著者Kallen, J.
登録日2020-03-25
公開日2021-03-10
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.12 Å)
主引用文献Phenotypic screen identifies calcineurin-sparing FK506 analogs as BMP potentiators for treatment of acute kidney injury.
Cell Chem Biol, 28, 2021
6YF2
DownloadVisualize
BU of 6yf2 by Molmil
FKBP12 in complex with the BMP potentiator compound 6 at 1.03A resolution
分子名称: (1~{R},9~{S},12~{S},13~{R},14~{S},17~{R},18~{E},21~{S},23~{S},24~{R},25~{S},27~{R})-23,25-dimethoxy-12-[(~{E})-1-[(1~{R},3~{R},4~{R})-3-methoxy-4-oxidanyl-cyclohexyl]prop-1-en-2-yl]-13,19,21,27-tetramethyl-1,14-bis(oxidanyl)-17-(2-oxidanylidenepropyl)-11,28-dioxa-4-azatricyclo[22.3.1.0^{4,9}]octacos-18-ene-2,3,10,16-tetrone, CADMIUM ION, CHLORIDE ION, ...
著者Kallen, J.
登録日2020-03-25
公開日2021-03-10
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.03 Å)
主引用文献Phenotypic screen identifies calcineurin-sparing FK506 analogs as BMP potentiators for treatment of acute kidney injury.
Cell Chem Biol, 28, 2021
1BMR
DownloadVisualize
BU of 1bmr by Molmil
ALPHA-LIKE TOXIN LQH III FROM SCORPION LEIURUS QUINQUESTRIATUS HEBRAEUS, NMR, 25 STRUCTURES
分子名称: LQH III ALPHA-LIKE TOXIN
著者Krimm, I, Gilles, N, Sautiere, P, Stankiewicz, M, Pelhate, M, Gordon, D, Lancelin, J.-M.
登録日1998-07-24
公開日1999-02-16
最終更新日2022-02-16
実験手法SOLUTION NMR
主引用文献NMR structures and activity of a novel alpha-like toxin from the scorpion Leiurus quinquestriatus hebraeus.
J.Mol.Biol., 285, 1999
1BNA
DownloadVisualize
BU of 1bna by Molmil
STRUCTURE OF A B-DNA DODECAMER. CONFORMATION AND DYNAMICS
分子名称: DNA (5'-D(*CP*GP*CP*GP*AP*AP*TP*TP*CP*GP*CP*G)-3')
著者Drew, H.R, Wing, R.M, Takano, T, Broka, C, Tanaka, S, Itakura, K, Dickerson, R.E.
登録日1981-01-26
公開日1981-05-21
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structure of a B-DNA dodecamer: conformation and dynamics.
Proc.Natl.Acad.Sci.USA, 78, 1981
6YF0
DownloadVisualize
BU of 6yf0 by Molmil
FKBP12 in complex with the BMP potentiator compound 9 at 1.55 A resolution
分子名称: 18-HYDROXYASCOMYCIN, Peptidyl-prolyl cis-trans isomerase FKBP1A, SULFATE ION
著者Kallen, J.
登録日2020-03-25
公開日2021-03-10
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献Phenotypic screen identifies calcineurin-sparing FK506 analogs as BMP potentiators for treatment of acute kidney injury.
Cell Chem Biol, 28, 2021
6YF3
DownloadVisualize
BU of 6yf3 by Molmil
FKBP12 in complex with the BMP potentiator compound 10 at 1.00A resolution
分子名称: (1~{R},9~{S},12~{S},13~{R},14~{S},17~{R},18~{E},21~{S},23~{S},24~{R},25~{S},27~{R})-17-ethyl-25-methoxy-12-[(~{E})-1-[(1~{R},3~{R},4~{R})-3-methoxy-4-oxidanyl-cyclohexyl]prop-1-en-2-yl]-13,19,21,27-tetramethyl-1,14,23-tris(oxidanyl)-11,28-dioxa-4-azatricyclo[22.3.1.0^{4,9}]octacos-18-ene-2,3,10,16-tetrone, CADMIUM ION, CHLORIDE ION, ...
著者Kallen, J.
登録日2020-03-25
公開日2021-03-10
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1 Å)
主引用文献Phenotypic screen identifies calcineurin-sparing FK506 analogs as BMP potentiators for treatment of acute kidney injury.
Cell Chem Biol, 28, 2021
1BR3
DownloadVisualize
BU of 1br3 by Molmil
CRYSTAL STRUCTURE OF AN 82-NUCLEOTIDE RNA-DNA COMPLEX FORMED BY THE 10-23 DNA ENZYME
分子名称: DNA (10-23 DNA ENZYME), RNA (5'-R(*GP*GP*AP*CP*AP*GP*AP*UP*GP*GP*GP*AP*G)-3')
著者Nowakowski, J, Shim, P.J, Prasad, G.S, Stout, C.D, Joyce, G.F.
登録日1998-08-13
公開日1999-02-23
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Crystal structure of an 82-nucleotide RNA-DNA complex formed by the 10-23 DNA enzyme.
Nat.Struct.Biol., 6, 1999
7ODI
DownloadVisualize
BU of 7odi by Molmil
Crystal structure of bovine Hsc70(aa1-554)E213A/D214A in complex with methanesulfonamide
分子名称: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, GLYCEROL, Heat shock cognate 71 kDa protein, ...
著者Zehe, M, Grimm, C, Sotriffer, C.
登録日2021-04-29
公開日2022-06-01
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.83 Å)
主引用文献Combined In-Solution Fragment Screening and Crystallographic Binding-Mode Analysis with a Two-Domain Hsp70 Construct.
Acs Chem.Biol., 2024
1BZJ
DownloadVisualize
BU of 1bzj by Molmil
Human ptp1b complexed with tpicooh
分子名称: 6-(DIFLUORO-PHOSPHONO-METHYL)-NAPHTHALENE-2-CARBOXYLIC ACID, PROTEIN (PROTEIN-TYROSINE-PHOSPHATASE)
著者Groves, M.R, Yao, Z.-J, Barford Jr, D.T.B.
登録日1998-10-29
公開日1999-02-16
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Structural basis for inhibition of the protein tyrosine phosphatase 1B by phosphotyrosine peptide mimetics.
Biochemistry, 37, 1998
7ODB
DownloadVisualize
BU of 7odb by Molmil
Crystal structure of bovine Hsc70(aa1-554)E213A/D214A in complex with triazine-derivative
分子名称: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, 6-methyl-5-sulfanylidene-2H-1,2,4-triazin-3-one, GLYCEROL, ...
著者Zehe, M, Grimm, C, Sotriffer, C.
登録日2021-04-29
公開日2022-06-01
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.662 Å)
主引用文献Combined In-Solution Fragment Screening and Crystallographic Binding-Mode Analysis with a Two-Domain Hsp70 Construct.
Acs Chem.Biol., 2024
1BVX
DownloadVisualize
BU of 1bvx by Molmil
THE 1.8 A STRUCTURE OF GEL GROWN TETRAGONAL HEN EGG WHITE LYSOZYME
分子名称: PROTEIN (LYSOZYME)
著者Dong, J, Boggon, T.J, Chayen, N.E, Raftery, J, Bi, R.C, Helliwell, J.R.
登録日1998-09-18
公開日1998-09-23
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Bound-solvent structures for microgravity-, ground control-, gel- and microbatch-grown hen egg-white lysozyme crystals at 1.8 A resolution.
Acta Crystallogr.,Sect.D, 55, 1999
6Y6R
DownloadVisualize
BU of 6y6r by Molmil
Crystal structure of MINDY1 T335D mutant
分子名称: Ubiquitin carboxyl-terminal hydrolase MINDY-1
著者Abdul Rehman, S.A, Kulathu, Y.
登録日2020-02-27
公開日2021-03-31
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (3.32 Å)
主引用文献Mechanism of activation and regulation of deubiquitinase activity in MINDY1 and MINDY2.
Mol.Cell, 81, 2021
1C1H
DownloadVisualize
BU of 1c1h by Molmil
CRYSTAL STRUCTURE OF BACILLUS SUBTILIS FERROCHELATASE IN COMPLEX WITH N-METHYL MESOPORPHYRIN
分子名称: FERROCHELATASE, MAGNESIUM ION, N-METHYLMESOPORPHYRIN
著者Lecerof, D, Fodje, M, Hansson, A, Hansson, M, Al-Karadaghi, S.
登録日1999-07-22
公開日2000-03-17
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structural and mechanistic basis of porphyrin metallation by ferrochelatase.
J.Mol.Biol., 297, 2000
7ODD
DownloadVisualize
BU of 7odd by Molmil
Crystal structure of bovine Hsc70(aa1-554)E213A/D214A in complex with tricine
分子名称: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, GLYCEROL, Heat shock cognate 71 kDa protein, ...
著者Zehe, M, Grimm, C, Sotriffer, C.
登録日2021-04-29
公開日2022-06-01
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.984 Å)
主引用文献Combined In-Solution Fragment Screening and Crystallographic Binding-Mode Analysis with a Two-Domain Hsp70 Construct.
Acs Chem.Biol., 2024
1BIV
DownloadVisualize
BU of 1biv by Molmil
BOVINE IMMUNODEFICIENCY VIRUS TAT-TAR COMPLEX, NMR, 5 STRUCTURES
分子名称: TAR RNA, TAT PEPTIDE
著者Ye, X, Kumar, R.A, Patel, D.J.
登録日1996-06-12
公開日1996-12-23
最終更新日2024-04-10
実験手法SOLUTION NMR
主引用文献Molecular recognition in the bovine immunodeficiency virus Tat peptide-TAR RNA complex.
Chem.Biol., 2, 1995
9F1C
DownloadVisualize
BU of 9f1c by Molmil
Mammalian quaternary complex of a translating 80S ribosome, NAC, MetAP1 and NatA/E
分子名称: 18S rRNA, 28S rRNA, 40S ribosomal protein S11, ...
著者Yudin, D, Scaiola, A, Ban, N.
登録日2024-04-18
公開日2024-08-21
実験手法ELECTRON MICROSCOPY (3.78 Å)
主引用文献NAC guides a ribosomal multienzyme complex for nascent protein processing
Nature, 2024
9F1D
DownloadVisualize
BU of 9f1d by Molmil
Mammalian quaternary complex of a translating 80S ribosome, NAC, MetAP1 and NatA/E-HYPK
分子名称: 18S rRNA, 28S rRNA, 40S ribosomal protein S11, ...
著者Yudin, D, Scaiola, A, Ban, N.
登録日2024-04-18
公開日2024-08-21
実験手法ELECTRON MICROSCOPY (3.26 Å)
主引用文献NAC guides a ribosomal multienzyme complex for nascent protein processing
Nature, 2024
8XGM
DownloadVisualize
BU of 8xgm by Molmil
Cryo-EM structure of human GPR1 bound to chemerin
分子名称: CHOLESTEROL, G-protein coupled receptor 1, Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1, ...
著者Liu, A.J, Liu, Y.Z, Ye, R.D.
登録日2023-12-15
公開日2024-08-21
実験手法ELECTRON MICROSCOPY (3.29 Å)
主引用文献Cryo-EM structure of human GPR1 bound to chemerin
To Be Published
8YE4
DownloadVisualize
BU of 8ye4 by Molmil
The complex of TCR NYN-I and HLA-A24 bound to SARS-CoV-2 Spike448-456 peptide NYNYLYRLF
分子名称: Beta-2-microglobulin, MHC class I antigen precusor, Spike protein S1, ...
著者Deng, S.S, Jin, T.C, Xu, Z.H, Wang, M.H.
登録日2024-02-21
公開日2024-08-21
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Structural insights into immune escape at killer T cell epitope by SARS-CoV-2 Spike Y453F variants.
J.Biol.Chem., 300, 2024
7B0Z
DownloadVisualize
BU of 7b0z by Molmil
Crystal Structure of human monoamine oxidase B in complex with (E)-3-phenyl-1-(4-(trifluoromethyl)phenyl)prop-2-en-1-one
分子名称: (E)-3-phenyl-1-(4-(trifluoromethyl)phenyl)prop-2-en-1-one, Amine oxidase [flavin-containing] B, FLAVIN-ADENINE DINUCLEOTIDE, ...
著者Iacovino, L.G, Binda, C.
登録日2020-11-23
公開日2021-11-03
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Promising Non-cytotoxic Monosubstituted Chalcones to Target Monoamine Oxidase-B.
Acs Med.Chem.Lett., 12, 2021
6JAO
DownloadVisualize
BU of 6jao by Molmil
Crystal structure of ABC transporter alpha-glycoside-binding mutant protein R356A in complex with palatinose
分子名称: 1,2-ETHANEDIOL, ABC transporter, periplasmic substrate-binding protein, ...
著者Kanaujia, S.P, Chandravanshi, M, Gogoi, P.
登録日2019-01-24
公開日2019-10-30
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.77 Å)
主引用文献Structural and thermodynamic correlation illuminates the selective transport mechanism of disaccharide alpha-glycosides through ABC transporter.
Febs J., 287, 2020
6YJF
DownloadVisualize
BU of 6yjf by Molmil
Plasmoodium vivax phosphoglycerate kinase bound to nitrofuran inhibitor from PEGSmear at pH 6.5
分子名称: (2~{S})-2-(5-nitrofuran-2-yl)-2,3,5,6,7,8-hexahydro-1~{H}-[1]benzothiolo[2,3-d]pyrimidin-4-one, GLYCEROL, Phosphoglycerate kinase
著者Hyvonen, M, Brear, P, Blaszczyk, B.K.
登録日2020-04-03
公開日2021-04-14
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Phosphoglycerate Kinase as a potential target for antimalarial therapy
to be published

224004

件を2024-08-21に公開中

PDB statisticsPDBj update infoContact PDBjnumon