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3TO7
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BU of 3to7 by Molmil
Crystal structure of yeast Esa1 HAT domain bound to coenzyme A with active site lysine acetylated
分子名称: CACODYLIC ACID, COENZYME A, GLYCEROL, ...
著者Yuan, H, Ding, E.C, Marmorstein, R.
登録日2011-09-04
公開日2011-11-09
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献MYST protein acetyltransferase activity requires active site lysine autoacetylation.
Embo J., 31, 2011
3M31
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BU of 3m31 by Molmil
Structure of the C150A/C295A mutant of S. cerevisiae Ero1p
分子名称: 1-ETHYL-PYRROLIDINE-2,5-DIONE, CADMIUM ION, Endoplasmic oxidoreductin-1, ...
著者Heldman, N, Fass, D.
登録日2010-03-08
公開日2010-11-03
最終更新日2024-10-30
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Steps in reductive activation of the disulfide-generating enzyme Ero1p
Protein Sci., 19, 2010
1BIC
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BU of 1bic by Molmil
CRYSTALLOGRAPHIC ANALYSIS OF THR-200-> HIS HUMAN CARBONIC ANHYDRASE II AND ITS COMPLEX WITH THE SUBSTRATE, HCO3-
分子名称: BICARBONATE ION, CARBONIC ANHYDRASE II, METHYL MERCURY ION, ...
著者Xue, Y, Vidgren, J, Svensson, L.A, Liljas, A, Jonsson, B.-H, Lindskog, S.
登録日1992-09-01
公開日1993-10-31
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystallographic analysis of Thr-200-->His human carbonic anhydrase II and its complex with the substrate, HCO3-.
Proteins, 15, 1993
3LZX
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BU of 3lzx by Molmil
Crystal structure of ferredoxin-NADP+ oxidoreductase from Bacillus subtilis (FORM II)
分子名称: FLAVIN-ADENINE DINUCLEOTIDE, Ferredoxin--NADP reductase 2, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ...
著者Komori, H, Seo, D, Sakurai, T, Higuchi, Y.
登録日2010-03-02
公開日2010-12-08
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystal structure analysis of Bacillus subtilis ferredoxin-NADP(+) oxidoreductase and the structural basis for its substrate selectivity
Protein Sci., 19, 2010
8EIT
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BU of 8eit by Molmil
Structure of FFAR1-Gq complex bound to DHA
分子名称: A modified Guanine nucleotide-binding protein G(q) subunit alpha, DOCOSA-4,7,10,13,16,19-HEXAENOIC ACID, Free fatty acid receptor 1, ...
著者Kumari, P, Inoue, A, Chapman, K, Lian, P, Rosenbaum, D.M.
登録日2022-09-15
公開日2023-05-24
最終更新日2025-05-28
実験手法ELECTRON MICROSCOPY (2.8 Å)
主引用文献Molecular mechanism of fatty acid activation of FFAR1.
Proc.Natl.Acad.Sci.USA, 120, 2023
3BZK
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BU of 3bzk by Molmil
Crystal Structure of the Tex protein from Pseudomonas aeruginosa, crystal form 2
分子名称: Tex
著者Johnson, S.J, Close, D, Hill, C.P.
登録日2008-01-18
公開日2008-04-08
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal structure and RNA binding of the Tex protein from Pseudomonas aeruginosa.
J.Mol.Biol., 377, 2008
3U47
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BU of 3u47 by Molmil
Human Carbonic Anhydrase II V143L
分子名称: Carbonic anhydrase 2, GLYCEROL, ZINC ION
著者West, D, Mckenna, R.
登録日2011-10-07
公開日2012-10-10
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structural modification of the hydrophobic pocket of Human Carbonic Anhydrase II
To be Published
8EJK
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BU of 8ejk by Molmil
Structure of FFAR1-Gq complex bound to TAK-875 in a lipid nanodisc
分子名称: A modified Guanine nucleotide-binding protein G(q) subunit alpha, Free fatty acid receptor 1, Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, ...
著者Kumari, P, Inoue, A, Chapman, K, Lian, P, Rosenbaum, D.M.
登録日2022-09-17
公開日2023-05-24
最終更新日2024-10-30
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Molecular mechanism of fatty acid activation of FFAR1.
Proc.Natl.Acad.Sci.USA, 120, 2023
3U4C
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BU of 3u4c by Molmil
Crystal structure of YwfH, NADPH dependent reductase involved in Bacilysin biosynthesis
分子名称: Bacilysin biosynthesis oxidoreductase ywfH, NADPH DIHYDRO-NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE
著者Rajavel, M, Gopal, B.
登録日2011-10-07
公開日2013-03-06
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.03 Å)
主引用文献Structural insights into the role of Bacillus subtilis YwfH (BacG) in tetrahydrotyrosine synthesis
Acta Crystallogr.,Sect.D, 69, 2013
8EJC
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BU of 8ejc by Molmil
Structure of FFAR1-Gq complex bound to TAK-875
分子名称: A modified Guanine nucleotide-binding protein G(q) subunit alpha, Free fatty acid receptor 1, Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, ...
著者Kumari, P, Inoue, A, Chapman, K, Lian, P, Rosenbaum, D.M.
登録日2022-09-16
公開日2023-05-24
最終更新日2024-10-30
実験手法ELECTRON MICROSCOPY (3 Å)
主引用文献Molecular mechanism of fatty acid activation of FFAR1.
Proc.Natl.Acad.Sci.USA, 120, 2023
3U4H
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BU of 3u4h by Molmil
CD38 structure-based inhibitor design using the N1-cyclic inosine 5'-diphosphate ribose template
分子名称: 8-Amino-N1-Cyclic Inosine 5'-Diphosphoribose, ADP-ribosyl cyclase 1
著者Liu, Q, Hao, Q, Lee, H.C, Graeff, R.
登録日2011-10-08
公開日2012-10-10
最終更新日2024-10-30
実験手法X-RAY DIFFRACTION (1.878 Å)
主引用文献CD38 Structure-Based Inhibitor Design Using the N1-Cyclic Inosine 5'-Diphosphate Ribose Template
Plos One, 8, 2013
2GB1
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BU of 2gb1 by Molmil
A NOVEL, HIGHLY STABLE FOLD OF THE IMMUNOGLOBULIN BINDING DOMAIN OF STREPTOCOCCAL PROTEIN G
分子名称: PROTEIN G
著者Gronenborn, A.M, Clore, G.M.
登録日1991-05-15
公開日1993-04-15
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献A novel, highly stable fold of the immunoglobulin binding domain of streptococcal protein G.
Science, 253, 1991
3GSY
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BU of 3gsy by Molmil
Structure of berberine bridge enzyme in complex with dehydroscoulerine
分子名称: 2,9-dihydroxy-3,10-dimethoxy-5,6-dihydroisoquino[3,2-a]isoquinolinium, 2-acetamido-2-deoxy-beta-D-glucopyranose, FLAVIN-ADENINE DINUCLEOTIDE, ...
著者Winkler, A, Macheroux, P, Gruber, K.
登録日2009-03-27
公開日2009-06-30
最終更新日2024-11-06
実験手法X-RAY DIFFRACTION (1.63 Å)
主引用文献Berberine bridge enzyme catalyzes the six electron oxidation of (S)-reticuline to dehydroscoulerine.
Phytochemistry, 70, 2009
8FOB
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BU of 8fob by Molmil
Cryo-EM structure of human TRPV6 in the open state
分子名称: (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, CALCIUM ION, ...
著者Neuberger, A, Yelshanskaya, M.V, Nadezhdin, K.D, Sobolevsky, A.I.
登録日2022-12-30
公開日2023-05-24
最終更新日2024-06-19
実験手法ELECTRON MICROSCOPY (2.71 Å)
主引用文献Structural mechanism of human oncochannel TRPV6 inhibition by the natural phytoestrogen genistein.
Nat Commun, 14, 2023
3GTO
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BU of 3gto by Molmil
Backtracked RNA polymerase II complex with 15mer RNA
分子名称: DNA (28-MER), DNA (5'-D(*CP*TP*GP*CP*TP*TP*AP*TP*CP*GP*GP*TP*AP*G)-3'), DNA-directed RNA polymerase II subunit RPB1, ...
著者Wang, D, Bushnell, D.A, Huang, X, Westover, K.D, Levitt, M, Kornberg, R.D.
登録日2009-03-27
公開日2009-06-09
最終更新日2024-10-30
実験手法X-RAY DIFFRACTION (4 Å)
主引用文献Structural basis of transcription: backtracked RNA polymerase II at 3.4 angstrom resolution.
Science, 324, 2009
1PU9
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BU of 1pu9 by Molmil
Crystal Structure of Tetrahymena GCN5 with Bound Coenzyme A and a 19-residue Histone H3 Peptide
分子名称: COENZYME A, HAT A1, Histone H3
著者Clements, A, Poux, A.N, Lo, W.S, Pillus, L, Berger, S.L, Marmorstein, R.
登録日2003-06-24
公開日2003-09-23
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structural basis for histone and phospho-histone binding by the GCN5 histone acetyltransferase
Mol.Cell, 12, 2003
1PW6
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BU of 1pw6 by Molmil
Low Micromolar Small Molecule Inhibitor of IL-2
分子名称: 2-CYCLOHEXYL-N-(2-{4-[5-(2,3-DICHLORO-PHENYL)-2H-PYRAZOL-3-YL]-PIPERIDIN-1-YL}-2-OXO-ETHYL)-2-GUANIDINO-ACETAMIDE, Interleukin-2, SULFATE ION
著者Thanos, C.D, Randal, M, Wells, J.A.
登録日2003-06-30
公開日2004-01-13
最終更新日2024-11-20
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Potent small-molecule binding to a dynamic hot spot on IL-2.
J.Am.Chem.Soc., 125, 2003
3TJL
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BU of 3tjl by Molmil
Crystal Structure of a Novel OYE from the Xylose-fermenting Fungus P. stipitis
分子名称: FLAVIN MONONUCLEOTIDE, MALONIC ACID, NADPH dehydrogenase, ...
著者Pompeu, Y.A, Stewart, J.D.
登録日2011-08-24
公開日2012-07-11
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Structural and Catalytic Characterization of Pichia stipitis OYE 2.6, a Useful Biocatalyst for Asymmetric Alkene Reductions
Adv.Synth.Catal., 2012
3M98
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BU of 3m98 by Molmil
Crystal structure of human carbonic anhydrase isozyme II with 5-(1H-benzimidazol-1-ylacetyl)-2-chlorobenzenesulfonamide
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 5-(1H-benzimidazol-1-ylacetyl)-2-chlorobenzenesulfonamide, Carbonic anhydrase 2, ...
著者Grazulis, S, Manakova, E, Golovenko, D.
登録日2010-03-21
公開日2011-03-02
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Crystal structure of human carbonic anhydrase isozyme II with 5-(1H-benzimidazol-1-ylacetyl)-2-chlorobenzenesulfonamide
To be published
6JWP
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BU of 6jwp by Molmil
crystal structure of EGOC
分子名称: Ego2, GTP-binding protein GTR1, GTP-binding protein GTR2, ...
著者Zhang, T, Ding, J.
登録日2019-04-21
公開日2019-12-11
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Structural insights into the EGO-TC-mediated membrane tethering of the TORC1-regulatory Rag GTPases.
Sci Adv, 5, 2019
3U2C
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BU of 3u2c by Molmil
Aldose reductase in complex with NSAID-type inhibitor at 1.0 A resolution
分子名称: 1-METHOXY-2-[2-(2-METHOXY-ETHOXY]-ETHANE, Aldose reductase, CITRIC ACID, ...
著者Steuber, H.
登録日2011-10-03
公開日2011-11-02
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1 Å)
主引用文献An old NSAID revisited: crystal structure of aldose reductase in complex with sulindac at 1.0 A supports a novel mechanism for its anticancer and antiproliferative effects.
Chemmedchem, 6, 2011
5A7Y
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BU of 5a7y by Molmil
Crystal structure of Sulfolobus acidocaldarius Trm10 in complex with S-adenosylhomocysteine
分子名称: ACETATE ION, DI(HYDROXYETHYL)ETHER, S-ADENOSYL-L-HOMOCYSTEINE, ...
著者Van Laer, B, Roovers, M, Wauters, L, Kasprzak, J, Dyzma, M, Deyaert, E, Feller, A, Bujnicki, J, Droogmans, L, Versees, W.
登録日2015-07-10
公開日2016-01-13
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural and Functional Insights Into tRNA Binding and Adenosine N1-Methylation by an Archaeal Trm10 Homologue.
Nucleic Acids Res., 44, 2016
2BJY
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BU of 2bjy by Molmil
The X-ray crystal structure of Listeria innocua Dps H31G-H43G mutant.
分子名称: NON-HEME IRON-CONTAINING FERRITIN
著者Ilari, A, Stefanini, S, Chiancone, E.
登録日2005-02-08
公開日2005-02-10
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献The Unusual Intersubunit Ferroxidase Center of Listeria Innocua Dps is Required for Hydrogen Peroxide Detoxification But not for Iron Uptake. A Study with Site-Specific Mutants
Biochemistry, 44, 2005
3GYP
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BU of 3gyp by Molmil
Rtt106p
分子名称: BETA-MERCAPTOETHANOL, CHLORIDE ION, Histone chaperone RTT106
著者Liu, Y, Huang, H, Shi, Y, Teng, M.
登録日2009-04-04
公開日2009-12-08
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (2.406 Å)
主引用文献Structural analysis of Rtt106p reveals a DNA-binding role required for heterochromatin silencing
J.Biol.Chem., 285, 2010
3RG3
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BU of 3rg3 by Molmil
Crystal structure of the W5E mutant of human carbonic anhydrase II
分子名称: Carbonic anhydrase 2, ZINC ION
著者Domsic, J.F, Robbins, A.H, McKenna, R.
登録日2011-04-07
公開日2012-02-22
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.903 Å)
主引用文献Structure and catalysis by carbonic anhydrase II: role of active-site tryptophan 5.
Arch.Biochem.Biophys., 516, 2011

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